Chemical & Pharmaceutical Bulletin

Article	Citations
Development of Ethylcellulose Microparticles for Taste Masking of Fexofenadine	52
Advances in Preparation of Peptide and Protein Thioesters Aiming to Use in Medicinal Sciences	37
Concise and Highly Stereoselective Synthesis of <i>β</i>,<i>β</i>-Disubstituted <i>α</i>,<i>β</i>-Unsaturated Esters	21
Foreword	20
Leonurine Preconditioning Attenuates Ischemic Acute Kidney Injury in Rats by Promoting Nrf2 Nuclear Translocation and Suppressing TLR4/NF-κB Pathway	19
Errata for Chemical and Pharmaceutical Bulletin	18
Clinical Pipelines for Alzheimer’s Disease Psychosis and Agitation	18
<i>In Vitro</i> and <i>in Silico</i> Studies of Potential Coronavirus-Specific 3C-Like Protease Inhibitors	17
CBDPS 1.0: A Python GUI Application for Machine Learning Models to Predict Bitter-Tasting Children’s Oral Medicines	16
Design, Synthesis and Radioprotective Activity Evaluation of Novel <i>N</i>-Phenyl-2<i>H</i>-chromene-3-carboxamides Derived from Ex-RAD	15
2-Azanorbornane-Based Amino Amide Organocatalysts for Asymmetric Michael Addition of <i>β</i>-Keto Esters with Nitroolefins	15
Protective Effect of Apple Polyphenols on H<sub>2</sub>O<sub>2</sub>-Induced Oxidative Stress Damage in Human Colon Adenocarcinoma Caco-2 Cells	14
Design, Synthesis, and Biological Evaluation of Water-Soluble Prodrugs of C5-Curcuminoid GO-Y030 Based on Reversible Thia-Michael Reaction	14
Syntheses of Aryl Thioethers <i>via</i> Aromatic Substitution of Aryl Halides at 0 to 25 °C	13
Synthesis and Evaluation of Novel Triaryl Derivatives with Readthrough-Inducing Activity	12
Teleocidin Analogs Isolated from <i>Streptomyces eurocidicus</i> as Membrane-Vesicle-Regulated Natural Products	12
Site-Specific Tritium Labeling at the Predefined Internal Position of the Chemically-Modified RNA	11
Oxygen-Fueled Iterative Hydride Transfer Driven by a Rigid Planar Architecture	11
Effect of Two-Photon Excitation to 8-Azacoumarin Derivatives as Photolabile Protecting Groups	11
Viscosity-Induced Emission of 5-(Diarylmethylene)imidazolone with Extended Conjugation <i>via</i> Attachment of <i>N</i>-Methylpyrrole at the 2-Position	11
Development of Efficient Synthetic Reactions Using Enamines and Enamides Carrying Oxygen Atom Substituent on Nitrogen Atom	11
Rapid Determination of Dapagliflozin in Rat Plasma by UHPLC-Q-Orbitrap MS and Its Application to a Pharmacokinetic Study	11
<i>In Vitro</i> Study on Combined Effect of Drugs for Hyperphosphatemia on Phosphorus Adsorption Capacity	11
Functions, Structures, and Engineering of the Teleocidin Biosynthetic Enzymes	10
Natural Compounds with BMI1 Promoter Inhibitory Activity from <i>Mammea siamensis</i> and <i>Andrographis paniculata</i>	10

Optimization and Advantages of Molded Tablets Using Trehalose as a Binder	10
Effectively Determining Dopamine Based on Dopamine Self-polymerization through Fluorescent Method Using Silicon Quantum Dots as Probe	10
Design, Synthesis, and Characterization of 1-(Anthracen-9-ylmethyl)-1,5,9-triazacyclododecane (Ant-[12]aneN3) and Its DNA Photocleavage Activity	10
Elucidation of Degradation Behavior of Barbiturates in Artificial Gastric Juice: Study on Degradability of Drugs in Stomach (V)	9
Molecular Modeling, Synthesis, and Preliminary Cytotoxicity Evaluation of New Indole-Based Molecules as Possible Sirtuin Inhibitors	9
Substituent Effects at the <i>N</i>-Nitrosoaminophenol Moiety of a Photoinduced-Electron-Transfer-Driven Nitric Oxide Releaser	9
<i>p</i>-Methoxy- and 2,4-Dimethoxybenzyl <i>N</i>-Acetylcarbamate Potassium Salts: Versatile Reagents for <i>N</i>-Alkylacetamide and <i>p</i>-Methoxy-	9
Anti-hepatitis C Virus Activity of Juglorubin Derivatives	9
Bromine K-Edge X-Ray Absorption Near-Edge Structure Analysis on Hydrobromide-Salt Crystals and the Solid Dispersion of Active Pharmaceutical Ingredients	9
Synthesis of Coumarin-Conjugated Oligonucleotides <i>via</i> Knoevenagel Condensation to Prepare an Oligonucleotide Library	9
Aminoalkylation of Alkenes for Modular Pyrrolidine Synthesis <i>via</i> Electron Donor–Acceptor Complexes Generated from Alkenes and Amine-Tethered <i>N</i>-Hydroxyphthalimide	9
Near-Infrared Metabolic Profiling for Discrimination of Apricot and Peach Kernels	9
Unusual Enzymatic C–C Bond Formation and Cleavage Reactions during Natural Product Biosynthesis	9
Development of a Potential-Modulated Electrochemiluminescence Measurement System for Selective and Sensitive Determination of the Controlled Drug Codeine	9
Synthesis of 2-Substituted Indoles <i>via</i> Migration Reaction of 3-Substituted Indoles with Triflic Acid	9
Liquid Chromatographic Determination of <i>o</i>-Phosphoethanolamine in Human Plasma Using Fluorescent Derivatization	9
Development of Low Molecular Weight Ligands for Integrin α<sub>v</sub>β<sub>3</sub>	8
Palatability of Aripiprazole Gummies Prepared from Commercially Available Products: Pharmaceutical Formulation for Improving Patient Adherence	8
The Effect of Iontophoresis with and without Electroporation on the Penetration of High Molecular Compounds into the Stratum Corneum	8
Discovery of a Novel Lidocaine Metabolite by Human Liver Microsome and Identification of Microbial Species Which Produces the Same Metabolite	8
Solid Fat Content and Relaxation Time Measurement of Petrolatum Using Time-Domain NMR, and the Correlation with Viscosity and Crystallinity	8
Masking the Taste of Fixed-Dose Combination Drugs: Particular NSAIDs Can Efficiently Mask the Bitterness of Famotidine	8
Isolation and Structure Elucidation of JBIR-157, a Skeletally Novel Aromatic Polyketide Produced by the Heterologous Expression of a Cryptic Gene Cluster	8
Emerging Separation Techniques in Supercritical Fluid Chromatography	7
Rapid Structure Determination of Ranitidine Hydrochloride API in Two Crystal Forms Using Microcrystal Electron Diffraction	7
Total Synthesis of (+)-Silybin A	7
Two New Halimanes with a <i>γ</i>-Lactone from <i>Croton argyratus</i>	7
Toward the Synthesis of Strychnos Alkaloids: Effective Construction of Fused Cyclohexane and Pyrrolidine Portion of the Strychnos Skeleton <i>via</i> Domino Intermolecular and Intramolecul	7
Identification of a Functionally Efficient and Thermally Stable Outward Sodium-Pumping Rhodopsin (<i>Be</i>NaR) from a Thermophilic Bacterium	7
Enteric Microcapsules Encapsulation of Roxithromycin-PVP Composite Core Particles to Inhibit Drug Crystallization upon Fluidized Bed Method for Oral Administration	7
Transport Characteristics of Placenta-Derived Extracellular Vesicles and Their Relevance to Placenta-to-Maternal Tissue Communication	7
Chlorocyclization of Alkenoic Thioester	7
Estimation for Raw Material Plants of a Henna Product Using LC-High Resolution MS and Multivariate Analysis	7
Simultaneous Overcoming Approach for Poor Wettability and Low Stability in Stomach by Simple Methods; Formulation Design and Development of Monoacylglycerol Acyltransferase 2 Inhibitor, S-309309	7
Optimization of the Hydrothermal Activation Treatment with Sodium Hydroxide Solution for the Conversion of Coal Fly Ash to Zeolite and Its Adsorption Capability of Lead (II) Ions from the Liquid Phase	7
Evaluation of the Mechanism of Phosphate Removal Using Oyster Shell Powder in Aqueous Environments	7
Flip-Flop Promotion Mechanisms by Model Transmembrane Peptides	7
Dynamic Dialysis Method for Characterizing Ammonia-Driven Drug Release from Liposomal Doxorubicin: Applicability and Kinetic Modeling	7
8-Iodoisoquinolinone, a Conformationally Rigid Highly Reactive 2-Iodobenzamide Catalyst for the Oxidation of Alcohols by Hypervalent Iodine	7
Organocatalyzed Amine-Free <i>O</i>-Phosphorylation of Alcohols with 4-Methylpyridine <i>N</i>-Oxide	7
Magnetic Field-Responsive Pulsatile Drug Release Using A Magnetic Fluid	7
<i>N</i>-Nitrosodimethylamine (NDMA) Formation from Ranitidine Impurities: Possible Root Causes of the Presence of NDMA in Ranitidine Hydrochloride	6
A Tricyclic Aromatic Polyketide Isolated from the Marine-Derived Fungus <i>Curvularia aeria</i>	6
Application of Quantitative NMR (qHNMR) towards Establishment of Pharmaceutical Reference Standard; A Case of a Ticagrelor Process Impurity	6
Synthesis and Evaluation of DHMEQ Derivatives with Tertiary Hydroxyl Group Instead of Secondary Hydroxyl Group	6
A Review on the Foodomics Based on Liquid Chromatography Mass Spectrometry	6
Tantalum-Catalyzed Peptide Elongation of Unprotected Amino Acids Using <i>N</i>-Trimethylsilylimidazole	6
Novel Pharmaceutical Cocrystals and Solvate Crystals of Nobiletin, a Citrus Flavonoid with Potent Pharmacological Activity	6
Theoretical Study of the Substituent Effect on the Diradical Character of <i>α</i>-Substituted <i>α</i>,3-Didehydrotoluenes	6
Physical Properties for Novel Cilostazol Co-amorphous; Effect of Preparation Method and Molar Ratio on the Co-amorphous	6

First Total Syntheses of Natural Phenanthrene Alkaloids, Uvariopsamine, Noruvariopsamine, 8-Hydroxystephenanthrine, 8-Methoxyuvariopsine, Thalihazine, and Secophoebine, and Their Potential as Antimala	6
Foreword	6
Antiproliferative Activities of Diterpenes from Leaves of <i>Isodon trichocarpus</i> against Cancer Stem Cells	6
Site-Selective Molecular Transformation: Acylation of Hydroxy Groups and C–H Amination	6
Effects of Physicochemical Properties of Constituent Ions of Ionic Liquid on Its Permeation through a Silicone Membrane	6
Exosome-Hijacking Drug Delivery System with Branched Arginine Linker Effectively Deliver Antisense Oligonucleotides into Lung Adenocarcinoma Cells	6
Comparison of Phosphate and Bicarbonate Buffer Solutions as Dissolution Test Media for Predicting Bioequivalence of Febuxostat Formulation	6
Isosteric Replacement of Ester Linkage of Lysophospholipids with Heteroaromatic Rings Retains Potency and Subtype Selectivity	6
Self-assembly of Urea Derivatives into Supramolecular Gels	6
C21 Steroidal Glycosides from the Roots of <i>Oxypetalum caeruleum</i>	6
Effect of Solubility Improvement <i>via</i> Formation of an Amorphous Composite of Indomethacin and Sulindac on Membrane Permeability	5
Synthesis and Characterization of Novel Radioiodinated Triazole-Pyrolidine Derivative to Detect Orexin 2 Receptor in the Brain	5
Remarkable Solvent Effect of Fluorinated Alcohols on Azo–Ene Reactions	5
Lewis Acid-Conjugated Pyrene Photoredox Catalyst Promoting the Addition Reaction of α-Silyl Amines with Benzalmalononitriles	5
Development of Highly Sensitive Method for Sugar Determination in Herbal Medicine; Application of Monosaccharides and Oligosaccharides in Japanese Angelica Root and Rehmannia Root	5
Selective Synthesis of the Aminobutadiene Intermediate and Mechanistic Analysis of 1,4-Dihydropyridine Formation Reaction in Water	5
Sulfonate Derivatives Containing a Kakuol Moiety as Potential Fungicidal Candidates: Design, Synthesis and Antifungal Activity Evaluation	5
μ-Oxo-Hypervalent-Iodine-Catalyzed Oxidative C–H Amination for Synthesis of Benzolactam Derivatives	5
Cyclopsammocinamides A and B, Enantiomeric Cyclic Peptides of Cyclocinamide A, from the Marine Sponge <i>Psammocinia</i> sp.	5
Structural Characterization of Zinc(II)/Cobalt(II) Complexes of Chiral <i>N</i>-(Anthracen-9-yl)methyl-<i>N</i>,<i>N</i>-bis(2-picolyl)amine and Evaluation of DNA P	5
Cellular Uptake and Transport Characteristics of FL118 Derivatives in Caco-2 Cell Monolayers	5
Design, Synthesis and Cytotoxicity Evalufation of Substituted Benzimidazole Conjugated 1,3,4-Oxadiazoles	5
Comparison of Growth in <i>Hydrangea macrophylla</i> var. <i>thunbergii</i> Grown in Different Soil pH and Quantitative Analysis of Its Sweetness-Related Constituents	5
C–H▪▪▪S Hydrogen Bonds in Ampicillin and Amoxicillin Crystals Investigated by Sulfur K-Edge X-Ray Absorption Near-Edge Structure Spectroscopy and Single-Crystal X-Ray Structure Analysis	5
Synthesis, Duplex-Forming Ability, and Nuclease Resistance of Oligonucleotides Containing a Thymidine Derivative with a 1-Oxaspiro[4.5]decane Skeleton	5
Electrochemical Characterization of a Novel Organoelectrocatalyst, 7-Azabicyclo[2.2.1]heptan-7-ol (ABHOL), and Its Application to Electrochemical Sensors	5
Guided Isolation of Isopentenyl Flavonoids from <i>Daphne giraldii</i> Based on the Combination of GNPS and SMART	5
Synthetic Studies on Vitamin D Derivatives with Diverse but Selective Biological Activities	5
Errata for Chemical and Pharmaceutical Bulletin	5
Methylene Blue Removal from the Aqueous Phase Using a Magnetic-Calcined Bamboo Composite Adsorbent	5
New Candidate Preservative in Ophthalmic Solution Instead of Benzalkonium Chloride: 1,3-Didecyl-2-methyl Imidazolium Chloride	5
Effects of Membrane Cholesterol on Stability of Transmembrane Helix Associations	5
Synthesis of Novel Pseudo-Enantiomeric Phase-Transfer Catalysts from <i>Cinchona</i> Alkaloids and Application to the Hydrolytic Dynamic Kinetic Resolution of Racemic 3-Phenyl-2-oxetanone	4
Structure–Activity Relationships of UTX-121 Derivatives for the Development of Novel Matrix Metalloproteinase-2/9 Inhibitors	4
Five New Analogs of Streptogramin Antibiotic Viridogrisein Isolated from <i>Streptomyces niveoruber</i>	4
Novel Strategies for Enantio- and Site-Selective Molecular Transformations	4
Elucidating the Light-Emitting Species Generated from Aminoluciferin in Firefly/Beetle Bioluminescence	4
Protein Chemical Modification Using Highly Reactive Species and Spatial Control of Catalytic Reactions	4
Structure–Activity Relationships of Thiophene Carboxamide Annonaceous Acetogenin Analogs: Shortening the Alkyl Chain in the Tail Part Significantly Affects Their Growth Inhibitory Activity against Hum	4
Determination of the Absolute Configuration of 2′-Amino-3′-methylacetophenone Based on the Modified Mosher and Microcrystal Electron Diffraction Methods	4
Liquiritigenin Attenuated Collagen-Induced Arthritis and Cardiac Complication <i>via</i> Inflammation and Fibrosis Inhibition in Mice	4
Chemical Components in <i>Hedera rhombea</i> Leaves and Their Cytotoxicity	4
Triflimide-Promoted Nucleophilic <i>C</i>-Arylation of Halopurines to Access <i>N</i><sup>7</sup>-Substituted Purine Biaryls	4
Importance of the Azole Moiety of Cimetidine Derivatives for the Inhibition of Human Multidrug and Toxin Extrusion Transporter 1 (hMATE1)	4
Development of a Fluorescence Probe for Detecting Nitroreductase Activity Based on Steric Repulsion-Induced Twisted Intramolecular Charge Transfer (sr-TICT)	4
Effects of Substituting Disubstituted Amino Acids into the Amphipathic Cell Penetrating Peptide Pep-1	4
A New 1,2-Naphthoquinone Derivative with Anti-lung Cancer Activity	4
Effect of Cultivation Conditions on Components of <i>Ephedra</i> sp. Using Liquid Chromatography-Mass Spectrometry and Multivariate Analysis	4
Shanpanootols G and H, Diterpenoids from the Rhizomes of <i>Kaempferia pulchra</i> Collected in Myanmar and Their Vpr Inhibitory Activities	4
The New Delivery Strategy of Albumin Carrier Utilizing the Interaction with Albumin Receptors	4
Dissolution Profiles of Oral Disintegrating Tablet with Taste Masking Granule Polymer Coating in Biorelevant Bicarbonate Buffer	4
Development and Validation of an LC–MS/MS-Based Method for Quantifying Urinary Endogenous 6-Hydroxymelatonin	4
Improved Dissolution Properties of Co-amorphous Probucol with Atorvastatin Calcium Trihydrate Prepared by Spray-Drying	4
Development of Fluorescent Estrogen Receptor Ligands with pH Sensor Functionality	4
Exploring the Effectiveness of Carboxymethylated and Crosslinked <i>Albizia procera</i> Gum in Diltiazem Hydrochloride Matrix Tablets: A Comparative Analysis	4
Aqueous Dispersion Polymerization for the Development of Lamivudine-Polyacrylonitrile Nanoparticles through Quality by Design Approach	4
Uric Acid as a Photosensitizer in the Reaction of Deoxyribonucleosides with UV Light of Wavelength Longer than 300 nm: Identification of Products from 2′-Deoxycytidine	4
GMP-Compliant Automated Radiolabeling and Quality Controls of [<sup>68</sup>Ga]Ga-FAPI-46 for Fibroblast Activation Protein-Targeted PET Imaging in Clinical Settings	4
Effect of Particle Size of Powdered Cellulose Nanofibers as an Additive in the Production of Orally Disintegrating Mini-Tablets by Direct Powder Compression	4
Bivalent β-Carbolines Inhibit Colorectal Cancer Growth through Inducing Autophagy	4
Synthesis of Formononetin Derivatives and Cardioprotective Effects	4
Cyclosporin A Inhibits the Activation of Membrane-Bound Guanylate Cyclase GC-A of Atrial Natriuretic Factor <i>via</i> NAD(P)H Oxidase	4
Formulation of Biopharmaceutical Dry Powder Inhaler Using the Void Forming Index (VFI) to Detect and Avoid Powder Caking in Dry Powder Inhaler Formulations	4
2-Thioxothiazolidin-4-one Analogs as Pan-PIM Kinase Inhibitors	4
Insights on Molecular Interaction between Polymer and Poorly Water-Soluble Loratadine in Solid Dispersion from Molecular Dynamics and Experiments	4
An Amphipathic Structure of a Dipropylglycine-Containing Helical Peptide with Sufficient Length Enables Safe and Effective Intracellular siRNA Delivery	4
Synthesis and Evaluation of Quinone Derivatives for Activity against <i>Trypanosome cruzi</i>	4
Effect of Sample Concentration on Nanoparticle Tracking Analysis of Small Extracellular Vesicles and Liposomes Mimicking the Physicochemical Properties of Exosomes	4
Quantification of Risperidone Contained in Precipitates Produced by Tea Catechins Using Nuclear Magnetic Resonance	4
Effect of Equipment Parameters on Amount and Dispersion of Wetting Liquid in Planetary Centrifugal Granulation	4
Preparation and <i>in Vitro</i> Evaluation of Osmotic-Pump Lorcaserin-hydrochloride Controlled-Release Tablets	4
Development of an Artificial Nucleic Acid Skeleton Allowing for Unnatural-Type Triplex DNA Formation with Duplex DNA Having a TA Inversion Site	4
An Update Mini-Review on the Progress of Azanucleoside Analogues	4
Epigenetic Inhibitors as Alzheimer’s Disease Therapeutic Agents	4
Compounds Designs of CK2α Inhibitors Derived from Virtual Screening Hit Compounds by Computational Chemistry with Crystallography	4
Oxidative Functionalization of Catechol Derivatives Substituted with Electron-Withdrawing Groups	3
12,20-Epoxypregnane Glycosides from the Roots of <i>Oxypetalum caeruleum</i>	3
Development of a Standard-Free Analytical Quantitative Method Based on Liquid Chromatography Using Relative Molar Sensitivity for Chlorogenic Acid in Apple Juice	3
A Stereoselective Synthesis of Fused Carbocycles with a <i>cis</i>-1,2-Diol Moiety by Desymmetrization: SmI<sub>2</sub>-Mediated Pinacol Coupling of <i>meso</i>-Cyc	3
Palladium-Catalyzed C–H Arylation of [1,1′-Biphenyl]-2-ols with Chloroarenes	3

Crystalline Phase Transitions of 5′-<i>O</i>-Triethylsilyl-2′-deoxy-5-azacytidine under Varying Temperature and Humidity Conditions and Its Closed Storage Stability	3
Isolation and Identification of Three New Iridoid Glucosides from the Aerial Parts of <i>Paederia scandens</i>	3
Elucidating the Factors Affecting the Patient-Centric Usability of Blister Packs for Spherical Capsules	3
Synthesis of Tetrahydrofuro[2,3-<i>d</i>]oxazoles and Oxazoles by Hypervalent Iodine (III)-Promoted [2 + 2 + 1] Annulation	3
Study of Polymer Nanofilms Using for High-Throughput Screening in the Development of Transdermal Therapeutic System	3
Extremely Simple and Rapid HPLC Analysis of Tocilizumab in Human Serum with Selective Precipitation Using Alkylamine	3
Asymmetric Total Syntheses of Mitragynine, Speciogynine, and 7-Hydroxymitragynine	3
Functional Characterization of Late-Stage Biosynthetic and Transporter Genes within the Biosynthetic Gene Cluster of the Organoarsenic Natural Product Bisenarsan	3
Development of Highly Sensitive Chemiluminescence Enzyme Immunostaining Assay to Determine Glycyrrhizin Content Using Anti-glycyrrhizin Monoclonal Antibody	3
Ruthenium-on-Carbon-Catalyzed Facile Solvent-Free Oxidation of Alcohols: Efficient Progress under Solid–Solid (Liquid)–Gas Conditions	3
Bioequivalence Dissolution Test Criteria for Formulation Development of High Solubility-Low Permeability Drugs	3
Peptide Tool-Driven Functional Elucidation of Biomolecules Related to Endocrine System and Metabolism	3
Substrate Flexibilities of Norbelladine Synthase and Noroxomaritidine/Norcraugsodine Reductase for Hydroxylated and/or Methoxylated Aldehydes	3
Determination of the Solid Content of Active Pharmaceutical Ingredient Powders in Suspension-Type Pharmaceutical Oral Jelly Using Time-Domain NMR	3
Development of Drug Discovery Platforms Using Artificial Intelligence and Cheminformatics	3
Hyaluronan Tetrasaccharides Penetrate into the Skin by Passive Diffusion and Contribute to Skin Health	3
Development of Naturally Inspired Peptide and Protein Chemistry	3
Ion-Pair Extraction with Tetracyanocyclopentadienides: A Method for Estimating Extraction Efficiency	3
Synergistic Activation of TLR7 and 8 Mediated by Reduction of Electrostatic Repulsion	3
Construction of 2,2-Dimethyloxepane Frameworks from Ene-Diols Catalyzed by Metal Catalyst or Brønsted Acid <i>via</i> 7-<i>Endo</i>-<i>Trig</i> Cyclization	3
Bicarbonate Buffer Dissolution Test Using the Floating Lid Method: Inter-Laboratory Reproducibility of pH Maintenance	3
Development of an Antigen Delivery System for a B Cell-Targeted Vaccine as an Alternative to Dendritic Cell-Targeted Vaccines	3
Lipase-Catalyzed Kinetic Resolution of <i>C</i><sub>1</sub>-Symmetric Heterocyclic Biaryls	3
Highly Precise Anomaly Detection Using Multivariate Statistical Process Control with Appropriate Scaling of Input Variables in Pharmaceutical Continuous Manufacturing	3
Theoretical Framework for Novel Catalytic Biomolecules Composed of Multiple Peptides	3
Determination of Hardness of a Pharmaceutical Oral Jelly by Using <i>T</i><sub>2</sub> Relaxation Behavior Measured by Time-Domain NMR	3
Foreword	3
Chemical Constituents of the Leaves of <i>Thujopsis dolabrata</i> and Their Cytotoxicity	3
Evaluation of STAT3 Inhibition by Cancer Chemopreventive Trichothecenes Derived from Metabolites of <i>Trichothecium roseum</i>	3
P(III)-Mediated Formal Reductive N–H Bond Insertion Reaction of Hydrazones to α-Keto Esters	3
Analysis of Powder Properties of Pharmaceutical Excipients Using a Constant-Volume Shear Tester	3
Fragment Molecular Orbital Based Affinity Prediction toward Pyruvate Dehydrogenase Kinases: Insights into the Charge Transfer in Hydrogen Bond Networks	3
Foreword	3
Foreword	3
Evaluation of Time-Dependent Deformation Behavior of Pharmaceutical Excipients in the Tableting Process	3
Model Synthetic Study of Tutin, a Picrotoxane-Type Sesquiterpene: Stereoselective Construction of a <i>cis</i>-Fused 5,6-Ring Skeleton	3
Total Synthesis and Antibacterial Activity of 5-Geranyloxy-7-hydroxycoumarin and Murrayacoumarin A	3
Foreword	3
Prediction of Intra-individual Variability in Bioequivalence Studies of 278 Formulations: Comprehensive Analysis Using Physicochemical and Pharmacokinetic Parameters	3
Colloidal Particle in Suspensions of Maobushisaishinto Extract Granules Enhances Drug Intestinal Penetration	3
Structure Derivatization of IgG-Binding Peptides and Analysis of Their Secondary Structure by Circular Dichroism Spectroscopy	2
Copper-Catalyzed Aerobic C(<i>sp</i><sup>3</sup>)–H Oxidation of β-(Alkoxy)imino Carbonyl Compounds	2
Understanding the Manufacturing Process of Lipid Nanoparticles for mRNA Delivery Using Machine Learning	2
Probing Iodine Atom Interactions in 4-Iodo-L-phenylalanine Crystals by X-Ray Absorption Near-Edge Structure Spectroscopy	2
Electrochemical Analysis for Total Alkalinity of Water by the Measurement of Cathodic Prepeak of Quinone Caused by Surplus Acid	2
Substitution Effects of Alkene Dipeptide Isosteres on Adjacent Peptide Bond Rotation	2
Enhanced Physical Stability of L-Ascorbic Acid in an Ionic Liquid	2
Omphalines A–E: <i>ent</i>-Rosane-Type Diterpenoids from the Madagascar Endemic Plant, <i>Omphalea oppositifolia</i>	2
Bioinspired Total Synthesis of Polycyclic Natural Products	2
Pharmaceutical Food Science: Search for Bio-Functional Molecules Obtained from Natural Resources to Prevent and Ameliorate Lifestyle Diseases	2
<sup>1</sup>H-NMR-Based Metabolomics for the Classification of the Roots of <i>Paeonia lactiflora</i>, a Constituent of Kampo Medicines	2
Stereoselective Synthesis of Aromatic Polyketide Prealnumycin	2
Construction of Acyclic All-Carbon Quaternary Stereocenter Based on Asymmetric Michael Addition of Chiral Amine	2
A Data-Driven Approach to Predicting Tablet Properties after Accelerated Test Using Raw Material Property Database and Machine Learning	2
Development of Fast Disintegrating Tablets Containing Loxoprofen Sodium by HYDROFLASH Manufacturing Method	2
Development of a Water Soluble Self-assembling Analogue of Vizantin	2
Deciphering Glycan Dynamics through Nonlinear Correlation Analysis	2
Four Novel Pharmaceutical Cocrystals of Oxyresveratrol, Including a 2 : 3 Cocrystal with Betaine	2
Construction of Biosensing System for Glycated Albumin Using an Electron Transfer Peptide-Modified Protein Probe	2
Biosynthesis of Bioactive Natural Products Derived from Theonellidae Family Marine Sponges	2
Antiproliferative Activities of Cynaropicrin and Related Compounds against Cancer Stem Cells	2
Chemical Constituents from the Leaves of <i>Pachyrhizus erosus</i> Collected in Vietnam	2
Facile Synthesis of 1,2-Disubstituted Benzimidazoles as Potent Cytotoxic Agents	2
Experimental and DFT Studies of Intermolecular Interaction-Assisted Oxindole Cyclization Reaction of Di-<i>t</i>-butyl 2-Aminophenyl-2-methyl Malonate	2
Semisynthesis and <i>in Vitro</i> Anti-cancer Effect of New Magnolol Derivatives on the Cell Proliferation, Apoptosis, Migration, and Invasion of Human Hepatocellular Carcinoma SMMC-7721 C	2
Molecular Transformation for Self-reproducing Vesicles and Underlying Analysis Methods	2
Isolation of Natural Prodrug-Like Metabolite by Simulating Human Prodrug Activation in Filamentous Fungus	2
Research Progress on the Mechanism of Reducing Toxicity and Increasing the Efficacy of Sini Decoction Compatibility	2
Synthesis of 2,8-Dioxabicyclo[3.3.1]nonane Derivatives and Their Neuroprotective Activities	2
Elucidation of Complex Dynamic Intermolecular Interactions in Membranes	2
Structure–Activity Relationship of the Linker Moiety in Photoinduced Electron Transfer-Driven Nitric Oxide Releasers	2
Simultaneous Determination and Comprehensive Evaluation of Mineral Elements in Yellow Croaker Ear-Stone on Sale in China	2
Spiromeroterpenoids from the Higher Plants	2
Derivation of the Extended Kawakita Equation for Estimating the Yield State of Powder in Die	2
Secorubenine, a Monoterpenoid Indole Alkaloid Glycoside from <i>Adina rubescens</i>: Isolation, Structure Elucidation, and Enantioselective Total Synthesis	2
Rational Design of Amphipathic Antimicrobial Peptides with Alternating L-/D-Amino Acids That Form Helical Structures	2
Neuroimmune Dysfunction in Alzheimer’s Disease and Other Forms of Dementia	2
Structure–Signal Relationships of the <i>δ</i>-Opioid-Receptor (DOR)-Selective Agonist KNT-127—Part I: Impact of the Morphinan Skeleton on the G-Protein-Biased DOR Agonism	2
4-Dimethylaminopyridine (DMAP), A Superior Mediator for Morita–Balylis–Hillman Reaction-Triggered Annulative Condensation of Salicylaldehydes and Acrylonitrile to Form 3-Cyano-2<i>H</i>-ch	2
The Inhibitory Effect of Adenylic Acid on the Bitterness of the Antibacterial Combination Drug Trimethoprim/Sulfamethoxazole	2
Enthalpy–Entropy Compensation in the Structure-Dependent Effect of Nonsteroidal Anti-inflammatory Drugs on the Aqueous Solubility of Diltiazem	2
Elucidating Molecular State of Loxoprofen in Acrylic Adhesive Patches Which Could Relate Transdermal Drug Permeability	2
Functionalization of Siloxanes with Arynes Generated from <i>o</i>-Triazenylarylboronic Acids	2
Synthesis and Characterization of Hydroxyethylamino- and Pyridyl-Substituted 2-Vinyl Chromone Derivatives for Detection of Cerebral Abnormal Prion Protein Deposits	2
Selection of Short 5′-UTR of Chemically Synthesized mRNA to Improve Translation Efficiency	2
Astragaloside IV Inhibits the Pyroptosis in the Acute Kidney Injury through Targeting the SIRT1/FOXO3a Axis	2
A Fluorescence Biosensor for Tyrosinase Activity Analysis Based on Silicon-Doped Carbon Quantum Dots	2
Cyclic Phthalate Esters as Liver X Receptor Antagonists with Anti-hepatitis C Virus and Anti-severe Acute Respiratory Syndrome Coronavirus 2 Properties	2
Exploration and Development of Nitrone Chemistry	2
Correlation between Membrane Permeability and the Intracellular Degradation Activity of Proteolysis-Targeting Chimeras	2
Gummi Formulations Comprising Amenamevir Solid Dispersions with Polyvinyl Alcohol	2
Synthesis and Biological Evaluation of 2-Azolylmethylene-3-(2<i>H</i>)-benzofuranone Derivatives as Potent Monoamine Oxidases Inhibitors	2
Development of Novel Methodology Using Diazo Compounds and Metal Catalysts	2
Formation of pH-Responsive Supramolecular Hydrogels in Basic Buffers: Self-assembly of Amphiphilic Tris-Urea	2
Identification of Proteolysis Targeting Chimeras (PROTACs) for Lysine Demethylase 5 and Their Neurite Outgrowth-Promoting Activity	2