Journal of Heterocyclic Chemistry

Papers
(The median citation count of Journal of Heterocyclic Chemistry is 1. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2021-04-01 to 2025-04-01.)
ArticleCitations
Synthesis and biological evaluation of 3‐hydroxypyrazoles as aquaporin 9 inhibitors74
Synthesis and characterization of a highly fluorescent benzofuran dimer derived from estradiol54
Synthesis of new tetrahydropyridopyrazine derivatives via continuous flow chemistry approach and their spectroscopic characterizations52
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One‐pot effective synthesis of new heterocyclic system: Pyrano[4′,3′:4,5]pyrido[2,3‐d]pyrimidin‐6‐one34
One‐pot synthesis of new functionalized 4H‐chromen‐4‐ylidene derivatives33
Retraction statement: Facile synthesis of two oxocan derivatives using some chemical strategies30
Retraction statement: Design and synthesis of a bismethylsulfanyl‐steroid‐azetyl butanol derivative from 2‐nitroestradiol25
Synthesis, antioxidant, and antimicrobial activity of some novel N‐substituted derivatives of 3‐(benzo[b]thiophen‐2‐yl)‐5‐(3‐[trifluoromethyl]styryl)‐4,5‐dihydro‐1H‐pyrazole24
Synthesis of anthracene linked polycyclic pyridine derivatives fused with coumarin and pyrazole by one‐pot multicomponent strategy followed by oxidation23
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Deoxygenation of N‐heterocyclic N‐oxides with Selectfluor and disulfane22
Palladium‐catalyzed [4 + 2] cycloaddition of sulfamate‐derived cyclic imines with γ‐methylidene‐δ‐valerolactones/2‐methylidenetrimethylene carbonate21
Synthesis of various 1‐alkylbenzimidazole derivatives directly from 2‐alkylaminonitroarenes via a two‐step, one‐pot procedure20
NiO‐Nanoparticles as green catalyst for an efficient synthesis of 4‐iminopyrido[1,2‐a]pyrimidine fluorophores via one pot cyclization of α‐aminonicotinonitrile20
An improved microwave‐assisted facile one‐pot synthesis of novel pyrazolylphosphonates via Knoevenagel‐phospha‐Michael protocol20
Synthesis and characterization of degradation impurities of Flucloxacillin and Dicloxacillin20
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Synthesis and molecular modeling of some novel hydroxypyrone derivatives as antidermatophytic agents19
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Facile and environmentally benign synthetic approach to the selective mono‐chlorination and mono‐bromination of benzo[d]OXAZOL‐2(3H)‐ONES18
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Novel angularly substituted [1,4]thiazino[3,4‐a]isoquinoline carboxylic acids prepared by cyclic imine‐cyclic anhydride reaction17
Highly efficient synthesis and NMR features of novel fused pyrimidothiazinium trihalogenides16
Synthesis and microbial screening of 8‐(benzyloxy)‐5‐(2‐[1,3‐diphenyl‐1H‐pyrazol‐4‐yl]thiazol‐4‐yl)quinolin‐2(1H)‐one derivatives16
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A facile synthesis of pyrrolo[2,3‐j]phenanthridines via the cascade reaction of indoleanilines and aldehydes14
Green multicomponent approach to novel 5‐[(2H‐Pyran‐3‐yl)(aryl)methyl]‐1,3‐dimethylpyrimidines14
Base promoted CuFe2O4 catalyzed one‐pot synthesis of 3,5‐diaryl‐1H‐pyrazoles14
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One‐pot three‐component synthesis of novel chromeno[3,2‐c]pyridine‐1,9(2H)‐diones by using SnCl2⋅2H2O as catalyst14
Photoinduced 6π‐electrocyclization of 2,5‐dichlorothiophene containing benzofuranylacrylonitriles as efficient method for the generation of hydrogen chloride14
Amidate ion‐mediated intramolecular ring transformation of 2‐pyrones to 2‐pyridones13
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Thallium(III) p‐tosylate‐mediated oxidative [1,2] rearrangement of 2‐naphthyl and 2‐heteroarylchromanones13
Facile access to 2‐amino‐4‐aryl‐5H‐chromeno[4,3‐b]pyridine‐3‐carbonitriles through a strategy of one‐pot Michael/cyclization reaction13
A selective chromone‐based colorimetric chemosensor for detecting Cu2+ in near‐perfect aqueous solution and test kit13
Efficient access to some new pyrimidine derivatives and their antimicrobial evaluation13
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One pot synthesis of α‐N‐heteroaryl ketone derivatives from aryl ketones using aqueous NaICl213
Synthesis and characterization of novel hybrid compounds containing coumarin and benzodiazepine rings based on dye12
Synthesis of new 2‐pyridinone and thiazole derivatives containing coumarin moiety12
Unprecedented, catalyst‐free, and rapid one‐pot, three‐component green synthesis of substituted 3‐hydroxy‐2‐oxindoles in water12
Synthesis and characterization of 4(R)‐epimer impurities of zanamivir and laninamivir octanoate12
Pd/C‐catalyzed one‐potSuzuki‐Miyauracross‐coupling/hydrogenation of pyridine derivatives12
Novel oxadiazole functionalized pyridopyrimidine derivatives; their anticancer activity and molecular docking studies12
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Total synthesis of xylapeptide B [Cyclo‐(L‐Leu‐L‐Pro‐N‐Me‐Phe‐L‐Val‐D‐Ala)]12
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Regiospecific synthesis of novel spiro‐pyrimidobarbiturates with promising antibacterial activities12
Catalytic Sc(OTf)3 mediated direct asymmetric aldol reaction of (−)‐menthyl isothiocyanatoacetate with aldehydes by using (−)‐menthol as chiral auxiliary12
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Mild and efficient regioselective surfactant catalyzed deacylation of lipophilic 5‐substituted 4‐acyl‐2‐(acylamino)‐Δ2‐1,3,4‐thiadiazolines11
One‐pot synthesis of quinazolinones and quinazolines under visible light via decarboxylation of α‐hydroxy acids11
An efficient synthesis of novel isoxazole bearing pyrazole derivatives via [3 + 2] heteroannulation using cupric acetate11
Solvent‐free Darzens condensation of 3‐chlorooxindoles with aryl aldehydes for diastereoselective construction of spiro‐epoxyoxindoles by grinding11
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Direct synthesis of 3,5‐diaryl‐1,2,4‐oxadiazoles using 1‐(2‐oxo‐2‐arylethyl)pyridin‐1‐iums with benzamidines11
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Promoting decanoic acid unveils the transfigure aldehyde carbonyl activation for synthesizing bis(indolyl)methane derivatives11
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Arylpyrazole as selective anti‐enterococci; synthesis and biological evaluation of novel derivatives for their antimicrobial efficacy10
[3+2] cycloaddition synthesis of new (nicotinonitrile‐chromene)‐based bis(pyrazole) hybrids as potential acetylcholinesterase inhibitors10
BimetallicCoCeO2oxide nanoparticles: An efficient and reusable heterogeneous catalyst for the preparation of2‐amino‐3‐cyano‐4H‐pyran derivatives10
Sulfa drugs–based Norbornenyl imides and reductive Heck reactions: Synthesis and antimicrobial screening10
Novel ferrocene cyclopalladated compounds: Synthesis, and in‐vitro antitumor activity study10
Microwave‐ultrasonic assisted synthesis, and characterization of novel 3′‐(amino, hydrazino and hydrazide)‐6′‐bromo‐spiro(isobenzofuran‐1,2′‐quinazoline)‐3,4′‐dione derivatives as antimicrobial agents10
Catalyst‐free one‐pot synthesis of quinoline tethered α‐amino ketones by multicomponent reactions10
Synthesis and anticancer activity of some thiophene, thienyl‐thiazole, and thienyl‐benzofuran analogues9
A new synthesis of 3′‐deoxy‐3′‐fluoroadenosine, a key intermediate of cyclic dinucleotide9
N‐Carbamimidoyl‐2,2,2‐Trifluoro‐N′‐Arylacetimidamides as Important Intermediates for the Synthesis of 3‐Amino‐4‐Aryl‐5‐(Trifluoromethyl)‐1H‐1,2,4‐Triazoles9
Glycerol‐1,2‐carbonate: A mild reagent for the N‐glycerylation of pyrazolecarboxylates9
Regioselective alkylation reaction of purines under microwave irradiation9
Advances in the Synthesis of 3‐Acyl‐2‐Pyridones: Strategies and Methods for Accessing the Versatile Scaffold9
Synthesis of novel amide/amino acid functionalized pyrazolo[3,4‐b]pyridine derivatives; their anticancer activity and docking studies9
A convenient total synthesis of indolo[2,3‐b]carbazole‐6,12‐dione9
Unveiling a Novel Mechanistic Pathway: Thiol and DMSO‐Facilitated Synthesis of Pyrazole Amine Thioether9
Metal‐free ring opening of 5‐amino‐1,4‐diaryl‐1H‐pyrazoles: A facile access to 2‐aryl‐3‐arylazoacrylonitriles9
The applications of β‐keto amides for heterocycle synthesis9
Crystal structure and quantum chemical calculations of (E)1‐benzyl‐3‐((4‐methoxyphenyl)imino)‐5‐methylindolin‐2‐one9
Synthesis and biological assessment of some fused Pyran derivatives9
Design, synthesis, and biological evaluation of 1,4,7,8‐tetrahydro‐5H‐furo[3,4‐b]pyrazolo[4,3‐e]pyridin‐5‐one‐based azo dyes9
A quick and easy access to a series of thiocyanated enaminones and 2‐iminothiazolones using PIDA under mild conditions9
Application of diazonium chemistry in purine modifications: A focused review8
L‐proline‐based DES in Knoevenagel synthesis of arylidene rhodanines, thiazolidine‐2,4‐diones, and barbituric derivatives8
The Influence of the Isosteric Exchange of Benzene by Thiophene‐Core of Phthalocyanine: The Synthesis, Structure and Opto‐Electronic Behavior of π‐Conjugated Unit Blocks in Materials8
Synthesis of pyrazole tethered oxadiazole and their analogs as potent antioxidant agents8
Synthesis and anticancer activity of cinnoline sulphonamides and 4‐heteroyclic derivatives: Cross‐coupling approach8
Synthesis and antiviral screening of 2‐(propylthio)‐7‐substituted‐thiazolo[5,4‐d]pyrimidines as anti‐bovine viral diarrhea virus agents8
Ultrasound‐promoted1,3‐dipolarcycloaddition of azomethine yields for synthesis of dispiropyrrolidineoxindole derivatives in hexyltriphenylphosphonium bromide as an ionic liquid, 8
A review on advances in synthetic methodology and biological profile of spirothiazolidin‐4‐ones8
Concise total synthesis of antiarrhythmic drug dronedarone via a conjugate addition followed intramolecular heck cyclization8
Efficient synthesis of piperidine derivatives using dendrimer based catalytical pockets8
Synthesis, antioxidant, and antimicrobial activity of 3‐(1H‐indole‐3‐carbonyl)‐2H‐chromen‐2‐ones8
Synthesis of novel indole‐oxadiazole molecular hybrids by a regioselective C‐3 sulfenylation of indole with 1,3,4‐oxadiazole‐2‐thiols using iodine‐dimethyl sulfoxide and their anticancer properties8
Synthesis of new 1,4‐ and 1,5‐disubstituted N‐ethyl acetate and N‐α‐butyro‐γ‐lactone alkylimidazole derivatives as N‐acylhomoserine lactone analogs8
The synthesis of novel 2, 3‐disubstituted 1,6‐dihydropyrrolo[2,3‐g]indazole derivatives via one‐pot three component reactions7
Palladium‐Catalyzed Synthesis of Pyrrolo[1,2‐α]Pyrazines From N‐Phenacyl Pyrrole‐2‐Carbonitriles and Aryl Boronic Acids7
Methoxy‐activated indole‐7‐carbohydrazides; synthesis, antioxidant, and anticancer properties7
Hybrid of the 1,2,3‐triazole nucleus and sesquiterpene skeleton as a potential antitumor agent: Hemisynthesis, molecular structure, Hirshfeld surface analysis, density functional theory, and in vitro 7
Synthesis and characterization of impurities of Apixaban drug substance—An anticoagulant7
A regiospecific fischer indole reaction with 3‐oxo‐24‐nor‐allobetulin7
Synthesis of bioactive quinoline appended spiro pyrrolidines as antioxidants7
Light, metal‐free regioselectiveC6‐Halkylation of purines and purine nucleosides with alcohols7
Synthetic Approaches Toward Imidazo‐Fused Heterocycles: A Comprehensive Review7
Design, synthesis, biological evaluation of a new tricyclicthiazolopy‐rimidinone derivatives as acetylcholinesterase inhibitors7
Catalyst‐free one‐pot three‐component rapid synthesis of polysubstituted pyrroles by liquid‐assisted grinding7
Discovery of 4H‐thieno[3,2‐b]pyrrole derivatives as potential anticancer agents7
A synthetic strategy for the preparation of alkoxy‐functionalized bis‐1,2,4‐triazinyl‐2,6‐pyridines7
Arylation of 2‐Chloro‐3‐(4,6‐Diaryl‐1,3,5‐Triazin‐2‐yl) Quinolines: Formal Synthesis of 3‐(4,6‐Diaryl‐1,3,5‐Triazin‐2‐yl)‐2‐Substituted Quinolines by Suzuki–Miyaura Reaction7
One‐pot green synthesis, study of fluorescence properties, and biological activity of pyrano[3,2‐c]chromenes derivatives via mesoporous materialsMgO/SBA‐157
Pyranoquinolone derivatives: A potent multi‐targeted pharmacological scaffold7
Trifluorodiazoethane: A versatile building block to access trifluoromethylated heterocycles7
Synthesis of substituted 5‐aryl‐2,3‐dihydropyrazine 1,4‐dioxides based on condensation of N,N′‐(2,3‐dimethylbutane‐2,3‐diyl)bis(hydroxylamine) with various arylglyoxals7
Synthesis and herbicidal activity of pyrimidyl‐1,2,4‐triazole derivatives containing aryl sulfonyl moiety6
N‐Functionalization of 4‐amino‐2‐(trifluoromethyl)‐1H‐pyrroles: Synthesis of N‐alkyl derivatives and 1,2,3‐triazol‐4‐yl‐pyrrole scaffolds6
A search for antiinflammatory therapies: Synthesis, in silico investigation of the mode of action, and in vitro analyses of new quinazolin‐2,4‐dione derivatives targeting phosphodiesterase‐4 enzyme6
Synthesis, and reverse screening of 6‐(3,4,5‐trimethoxyphenyl)pyrimidine‐5‐carbonitrile derivatives as anticancer agents: Part‐II6
Imidazo[1,2‐a]pyridine as a promising scaffold for the development of antibacterial agents6
Novel tryptanthrin hybrids bearing aminothiazoles as potential EGFR inhibitors: Design, synthesis, biological screening, molecular docking studies, and ADME/T predictions6
Antioxidant and cytotoxic properties of some new dipeptide‐indole conjugates6
Synthetic Strategies for C‐Amino 1,2,3‐Triazoles and Their Oxides: A Review6
An eco‐friendly, sustainable, and greener approach to the synthesis of Dihydroquinazolin‐4(1H)‐ones using a deep eutectic solvent6
Hantzsch‐like reaction of isoquinoline‐1‐acetonitrile in synthesis of 4H‐pyrido[2,1‐a]isoquinolines with antibacterial evaluation6
Synthesis, antimicrobial activity, and molecular docking studies of new fused pyrimidinethiones6
Research progress of piperazine and morpholine derivatives in the discovery of agricultural chemicals6
Visible Light Mediated CO2 Fixation Reactions to Produce Carbamates and Carbonates: A Comprehensive Review6
Catalyst‐free, one‐pot three‐component synthesis of N,3‐diphenybenzo[d]imidazo[2,1‐b]thiazoles and oxybis(1‐phenyl‐2‐(phenylamino)ethanones)6
Combination of N‐amino‐1,2,4‐triazole and 4‐hydroxy‐3,5‐dinitropyrazole for the synthesis of high performing explosives6
Design, synthesis, and biological activity of sulfoximine derivatives6
Synthesis, insecticidal activities, and structure–activity relationships of 1,3,4‐oxadiazole‐ring‐containing pyridylpyrazole‐4‐carboxamides as novel insecticides of the anthranilic diamide family5
Catalyst‐free one‐pot synthesis of 2,4,5‐tri‐ and 1,2,4,5‐tetrasubstituted imidazoles5
Hantzsch‐like synthesis of isoquinolino[2,1‐a]quinoline‐12‐carbonitrile incorporating aryl or heteroaryl moieties at C‐135
One‐pot regioselective synthesis of new imidazo[4,5‐e]thiazolo[3,2‐b][1,2,4]triazines by reaction of imidazotriazines with propargyl bromide5
Synthesis of new derivatives of Alkylselanyl[1,2,4]triazolo[4,3‐a]pyrimidine asselenium‐containingheterocyclic system5
5‐Sulfosalicylicacid an organocatalyst for the synthesis of highly functionalized piperidines through the multicomponent reaction5
New metal free organic dyes incorporating heterocyclic Benzofuran core as conjugated spacer: Synthesis, Opto‐electrochemical, DFT and DSSC studies5
Palladium‐catalyzed synthesis of Benzoannulated spiroketal lactones derived from cholesterol: NMR characterization and crystal structures5
p‐Toluenesulfonic acid catalyzed, isocyanide‐free, Groebke–Blackburn–Bienayme (GBB) type multicomponent synthesis of 3‐anilino‐imdazo[1,2‐5
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Microwave assisted synthesis, acetylcholinesterase inhibition and molecular docking studies of furo[2,3‐d]pyrido[1,2‐a]pyrimidin‐4‐one derivatives5
Research progress of triazole derivatives in the discovery of agricultural chemicals5
Regioselective synthesis of fused pyrimidines and quinazolines linked to Phenoxy‐N‐arylacetamide moieties as novel hybrid molecules via Biginelli‐like reaction5
Cu‐catalyzed dehydrogenative CO arylation for the synthesis of 6‐methyl benzofuro[3,2‐c] quinoline derivatives5
A novel synthetic approach to Pyrazolooxazines. One‐pot synthesis of Pyrazolo[5,1‐c][1,4]oxazine derivatives from 2,2‐dichlorovinylacetophenones5
Fullerene‐C60/NH2: A recyclable heterogeneous catalyst for the green synthesis of chromene and pyrimidine derivatives and antibacterial evaluation5
Synthesis of 4‐imidoyl‐, 4‐oxiranyl‐ and 4‐propargyloxyphenyl‐substituted β‐lactam building blocks5
Synthetic attempts toward α‐tocopherol—An overview5
[Et3NH][HSO4] catalyzed solvent‐free synthesis of new 1,2,3‐triazolidene‐indolinone derivatives5
Synthesis of 5‐spirocycle camptothecin using ring‐closing metathesis strategy5
Role of aurone ligands in microwave enhanced Mn (II) and Co (II) catalyzed dehydrogenative coupling reaction: An efficient ligand for the synthesis of quinoline, pyridine, and py5
Chalcone derived benzoheterodiazepines for medicinal applications: A Two‐pot and one‐pot synthetic approach5
Concise Synthesis of Azaphenanthrene Alkaloid Eupolauramine Via Au(I)‐Catalyzed Cycloisomerization and Intramolecular Ullmann‐Type Coupling Reaction5
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3‐Aminothieno[2,3‐b]pyridine‐2‐carboxylate: Effective precursor for microwave‐assisted three components synthesis of new pyrido[3′,2′:4,5]thieno[3,2‐d]pyrimidin‐4(3H5
Organic Brønsted acid‐catalyzed cycloadditions of o‐quinone methides with 1, 3‐dicarbonlys: Facile access to xanthenones and chromanones5
Organocatalyzed cycloaddition reactions of azomethine imines—A lookback5
Facile synthesis, antimicrobial, and anti‐inflammatory activities of novel isoxazolyl imidazo[1,2‐b]isoxazoles5
Direct demonstration of tautomeric nature of 4‐bromo‐3(5)‐methylpyrazoles5
Tin (IV) chloride catalyzed one‐pot synthesis, characterization, and docking studies of 4‐aminoquinoline derivatives as Myt1 inhibitors5
Synthesis and evaluation of new phosphonated δ‐lactam and glutarimide derivatives as angiotensin converting enzyme inhibitors5
Diastereoselective construction of carbazole‐based spiropyrrolidines and spiropyrrolizidines via cycloaddition reaction5
Study on antitumor activity of parthenolide C‐14 derivatives5
Efficient synthesis of some novel pyrimido[4,5‐e][1,3]oxazine dione derivatives via one‐pot three‐component reaction under thermal and thermal microwave‐assisted conditions5
An approach for the diastereoselective synthesis of (R)‐(+)‐methyl pipecolate and (+)‐dextro‐erythrophacetoperane from (S)‐(−)‐methylbenzylamine5
Kojic acid aldol adduct with isatin as inhibitors of pyruvate dehydrogenase kinase5
Design, syntheses and antitumor activities evaluation of 1,5‐diaryl substituted pyrazole secnidazole ester derivatives4
New synthetic strategy for Friedlander condensation of 4‐amino‐2‐oxo‐2H‐chromene‐3‐carbaldehyde by heterogeneous catalysis4
Synthesis of 1,3‐oxazepine derivatives via tandem reaction of 5‐benzylidine Meldrum's acids with TosMIC in presence of potassium carbonate4
Synthesis, characterization, biological evaluation, and computational study of benzimidazole hybrid thiosemicarbazide derivatives4
One‐step synthesis of novel N1‐substituted benzimidazole derivatives: Experimental and theoretical investigations4
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Pesticidal Efficacy of Innovative Heterocyclic Tosyl Esters: Design, Synthesis, Biochemical Assessment, and DFT Calculation4
Synthesis and antitumor evaluation of some new thiazolopyridine, nicotinonitrile, pyrazolopyridine, and polyhydroquinoline derivatives using ceric ammonium nitrate as a green catalyst4
Iron‐catalyzed construction of cyanomethylated thiohydantoins by cross‐dehydrogenative C(sp3)‐C(sp3) coupling4
Late‐stage functionalization of Vouacapane derivatives from Caesalpinia platyloba by a Groebke−Blackburn−Bienaymé reaction4
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Visible Light Triggered, Catalyst‐Free Approach for the Click Synthesis of Imidazole‐Fused Nitrogen‐Bridgehead Nucleus in EtOH:H2O Medium4
A new synthetic route for synthesis of 3‐substituted imidazo[1,5‐a]pyridines4
A Brief Review on Different Reactions of Rhodanine4
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Potassium dihydrogen phosphate‐catalyzed synthesis of benzylpyrazolyl coumarin and pyrano [2,3‐c] pyrazole derivatives via cascade—One‐pot—Multicomponent reaction4
Visible light induced eco sustainable synthesis of quinolines catalyzed by eosin Y4
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Visible‐light photoredox catalyzed synthesis of tetrahydrobenzofuranone: Oxidative [3 + 2] cycloaddition of dicarbonyl and alkene4
Progress in the chemistry of functional aramids properties4
Regioselective synthesis and computational calculation studies of some new pyrazolyl‐pyridine and bipyridine derivatives4
A general palladium‐catalyzed carbonylation synthesis of aurones with aryl bromides using CO24
Green catalyst access to thieno [2, 3‐b] pyridines derivatives4
Catalyst free synthesis of 2‐Aryl‐2H‐benzo[b][1,4]oxazines and 3‐Aryl‐2H‐benzo[b][1,4]thiazin‐2‐ones: An ultrasonication‐assisted strategy4
Stereoselective synthesis and characterization of monocyclic cis‐β‐lactams containing 5‐methyl‐1,3,4‐thiadiazole‐2‐thiol moiety4
Microwave‐assisted synthesis of benzo[4,5]imidazo[1,2‐a]pyrimidines and pyrano[4,3‐b]pyrans catalyzed by L‐glutamine functionalized magnetic nanoparticles in water:ethanol mixture4
Efficient preparation of (S)‐2‐(3,5‐dimethylphenyl)pyrrolidine via a recycle process of resolution4
A Synthetic Route Towards Spiro Indanone Fused Pyrano[2,3‐c]Chromene Derivatives via Oxa–Diels–Alder Reaction: Computational Investigation, Antibacterial Evaluation and Molecular Docking Studie4
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Synthesis, anticancer evaluation and in silico studies of novel N‐substituted arylidenethiazolidine‐2,4‐dione derivatives as adenosine monophosphate‐activated protein kinase activators4
The reported formation of 5H‐dibenzo[b,e][1,4]diazepin‐11(10H)‐ones in the noncatalyzed, base‐promoted double arylation of anthranilami4
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Investigation and comparison of biological effects of regioselectively synthesized thiazole derivatives4
New edaravone analogs incorporated with N‐benzylthiazole moiety: Multistep chemical synthesis, in vitro cytotoxicity with pRIPK3 inhibitory activities, and molecular docking4
Identification, isolation, and characterization of two novel impurities from phenothiazine heterocycle derivative: Perphenazine and their control in the process4
Versatile imidazole synthesis via multicomponent reaction approach4
Microwave‐assisted decarboxylation of 2H‐Pyran‐3‐carboxylic acid derivatives under basic condition4
Highly efficient and diastereoselective construction of substituted pyrrolidines bearing a quaternary carbon center via 1,3‐dipolar cycloaddition4
Synthesis, antiinflammatory, and cytotoxic activity of novel pyrazolo[4,3‐c][2,1]benzothiazine 4,4‐dioxide derivatives4
Synthesis and evaluation of the biological activities of novel hybrid isoindol‐1,3‐dione containing an aziridine unit4
Efficient synthesis of 3‐sulfonyl‐1,2‐dihydroquinolines via tandem aza‐Michael addition/cyclizations of N‐acyl‐protected 2‐aminobenzaldehyde with vinyl sulfones4
T3P‐Promoted Synthesis of a Series of Novel 3‐Aryl‐2‐phenyl‐2,3,5,6‐tetrahydro‐4H‐1,3‐thiazin‐4‐ones4
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Copper‐Catalyzed Carboamination of Unactivated Alkenes to Synthesize β‐Lactams with Trichloroacetonitrile4
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Efficient domino strategy for synthesis of 3‐substituted 1,5‐dihydro‐4H‐pyrrolo[3,2‐c]pyridin‐4‐one derivatives4
New thieno[2,3‐d]pyrimidine derivatives as EGFRWT and EGFRT790M inhibitors: Design, synthesis, antiproliferative activities, docking studi4
Synthesis and odor characteristics of N‐substituted pyrrolyl ketones derived from N‐substituted acetylpyrroles and alcohols3
Synthesis, characterization and in vitro bioactivity studies of isoindolin‐1‐3‐phosophonate compounds3
Design, synthesis, and insecticidal activities of novel diamide derivatives with alpha‐amino acid subunits3
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Potential applications of Aggregation Induced Emission  active heterocyclic compounds3
Organocatalytic[3 + 2]Cycloaddition: Synthesis of Quinazoline Containing Sulfonyl 1,2,3‐Triazoles as Potent EGFR Targeting Anti‐Breast Cancer Agents3
Diastereomerically pure (S)‐verbenone‐isoxazoline hybrids: Synthesis, molecular structure, Hirshfeld surface analysis, density functional theory, cytotoxic effect, and apoptosis induction3
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Benzenediazonium Tetrafluoroborate‐Catalyzed Formal [3 + 3] Cyclization of 4‐Hydroxycoumarins With Propargylicalcohols3
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Synthesis of new 1H‐spiro[acridine‐9,3′‐indoline]‐1,2′(2H,10H)‐dione derivatives using aqueous ethanol as a reaction medium3
Research progress of oxazole derivatives in the discovery of agricultural chemicals3
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Unusual impurity formation during the process development of Olsalazine sodium leads to a new efficient and economical synthesis of tricaine mesylate3
Pyrazolo[3,4‐d]pyrimidine‐based scaffolds as antibacterial agents: Synthetic strategies, reactions, and in vitro biological evaluation3
Design, synthesis, antifungal activity, and molecular docking of novel trifluoromethyl pyrimidine derivatives containing 1,3,4‐oxadiazole and thioether moieties as potential succinate dehyd3
Novel fluoroquinolones containing 2‐arylamino‐2‐oxoethyl fragment: Design, synthesis, evaluation of antibacterial and antituberculosis activities and molecular modeling studies3
Synthesis of (s)‐1‐{3‐[4‐(4‐benzo[d]isothiazol‐3‐yl‐piperazin‐1‐yl)‐3‐fluoro‐phenyl]‐2‐oxo‐oxazolidin‐5‐ylmetyl}‐3‐substituted‐urea derivatives as antibacterial agents3
Retraction statement: Facile synthesis of two oxocan derivatives using some chemical strategies3
Synthesis of cyclopentane annulated δ‐lactams via diazomethane‐mediated CC bond cleavage of α‐ketoN,O‐hemiaminals3
Recent research progress of heterocyclic nematicidal active compounds3
N‐Methoxy Pyrazole‐4‐Carboxamide Derivatives: Synthesis, Spectral Analyses, Antifungal Activity, In Silico Molecular Docking, ADMET, and DFT Studies3
An efficient and scalable synthesis of Isodesmosine3
Total synthesis and antimicrobial evaluation of xylapeptide A3
Simple grinding for the synthesis of monomeric, dimeric, and trimeric pyridinium salts and its photophysical studies3
Synthesis of methyl 1,5‐diaryl‐1H‐pyrrole‐2‐carboxylates via acid‐catalyzed ring‐opening/ring‐closure sequence3
Synthesis of substituted 5,6,7,8‐tetrafluoro‐1H‐benzo[f]indol‐4,9‐diones based on the reaction of hexafluoro‐1,4‐napthoquinone with methyl 3‐aminocrotonates3
From 2011 to 2022: The development of pyrazole derivatives through the α,β‐unsaturated carbonyl compounds3
A solvent‐free manganese(II) ‐catalyzed Clauson‐Kaas protocol for the synthesis of N‐aryl pyrroles under microwave irradiation3
Chalcones: Versatile intermediates in heterocyclic synthesis3
Synthesis of 1‐(4‐hydroxybutyl)‐2‐benzoyl indoles from 2‐pyrrolidine benzaldehydes and α‐bromoacetophenones in deep eutectic solvent3
Investigation of some new main group metal complexes of hydrazine and 2‐mercaptopyridine‐3‐carboxylic acid mixed–ligands3
Synthesis and Cancer Cell Cytotoxicity of 6‐, 7‐, or 8‐Substituted 2‐(Hetero)aryl‐4‐(4‐(Hetero)aryl‐2‐Oxobut‐3‐en‐1‐Ylidene)Benzothiazepanes3
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Dimroth rearrangement in the row of new pyrano[3,4‐c][1,2,4]triazolo[4,3‐a][1,5‐a]pyridines and synthesis of new heterocyclic systems: Pyranopyrazolo[4,3‐e][1,2,4]triazolop3
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