Journal of Heterocyclic Chemistry

Article	Citations
	80
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Issue Information	58
Novel ferrocene cyclopalladated compounds: Synthesis, and in‐vitro antitumor activity study	44
Issue Information	36
Synthesis and molecular modeling of some novel hydroxypyrone derivatives as antidermatophytic agents	36
A quick and easy access to a series of thiocyanated enaminones and 2‐iminothiazolones using PIDA under mild conditions	35
The applications of β‐keto amides for heterocycle synthesis	32
Facile access to 2‐amino‐4‐aryl‐5H‐chromeno[4,3‐b]pyridine‐3‐carbonitriles through a strategy of one‐pot Michael/cyclization reaction	31
Synthesis, antimicrobial activity, and molecular docking studies of new fused pyrimidinethiones	25
Retraction statement: Facile synthesis of two oxocan derivatives using some chemical strategies	25
	24
Microwave‐Assisted One‐Pot Synthesis of 1,5‐Benzodiazepine Derivatives Using Novel ZnFe2O4.Cu(OH)2 Magnetic Nanocomposite as Heterogeneous Cataly	23
Introduction of the Acyl Group at the C7 Position of Indole via N ‐Acyl Indole Photo‐Fries Rearrangeme	22
Photoinduced 6π‐electrocyclization of 2,5‐dichlorothiophene containing benzofuranylacrylonitriles as efficient method for the generation of hydrogen chloride	22
New Corono Asymmetrical N‐Bis ‐Heterocyclic Bis ‐Imidazolium Macrocycle Salt, Preliminary Physicochemical	21
NiO‐Nanoparticles as green catalyst for an efficient synthesis of 4‐iminopyrido[1,2‐a]pyrimidine fluorophores via one pot cyclization of α‐aminonicotinonitrile	20
Synthetic Approaches Toward Imidazo‐Fused Heterocycles: A Comprehensive Review	20
Novel angularly substituted [1,4]thiazino[3,4‐a]isoquinoline carboxylic acids prepared by cyclic imine‐cyclic anhydride reaction	19
Unprecedented, catalyst‐free, and rapid one‐pot, three‐component green synthesis of substituted 3‐hydroxy‐2‐oxindoles in water	19
Synthesis of substituted 5‐aryl‐2,3‐dihydropyrazine 1,4‐dioxides based on condensation of N,N′‐(2,3‐dimethylbutane‐2,3‐diyl)bis(hydroxylamine) with various arylglyoxals	19
A regiospecific fischer indole reaction with 3‐oxo‐24‐nor‐allobetulin	19
Synthesis and biological assessment of some fused Pyran derivatives	19
Palladium‐Catalyzed Synthesis of Pyrrolo[1,2‐α]Pyrazines From N‐Phenacyl Pyrrole‐2‐Carbonitriles and Aryl Boronic Acids	19
Combination of N‐amino‐1,2,4‐triazole and 4‐hydroxy‐3,5‐dinitropyrazole for the synthesis of high performing explosives	18

Solvent‐free Darzens condensation of 3‐chlorooxindoles with aryl aldehydes for diastereoselective construction of spiro‐epoxyoxindoles by grinding	18
[3+2] cycloaddition synthesis of new (nicotinonitrile‐chromene)‐based bis(pyrazole) hybrids as potential acetylcholinesterase inhibitors	18
Synthesis of novel amide/amino acid functionalized pyrazolo[3,4‐b]pyridine derivatives; their anticancer activity and docking studies	18
Ultrasound‐promoted1,3‐dipolarcycloaddition of azomethine yields for synthesis of dispiropyrrolidineoxindole derivatives in hexyltriphenylphosphonium bromide as an ionic liquid,	17
A synthetic strategy for the preparation of alkoxy‐functionalized bis‐1,2,4‐triazinyl‐2,6‐pyridines	17
Catalyst‐free one‐pot three‐component rapid synthesis of polysubstituted pyrroles by liquid‐assisted grinding	17
Design, Synthesis, and Biological Evaluation of Some New Thiazole‐Based Compounds as Antioxidant and Antimicrobial Agents	17
Cycloaddition or Metathesis: Selectivity in a Series of Indole‐2,3‐Quinodimethane Derivatives	16
Retraction statement: Facile synthesis of two oxocan derivatives using some chemical strategies	16
Synthesis and evaluation of the biological activities of novel hybrid isoindol‐1,3‐dione containing an aziridine unit	16
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An approach for the diastereoselective synthesis of (R)‐(+)‐methyl pipecolate and (+)‐dextro‐erythrophacetoperane from (S)‐(−)‐methylbenzylamine	16
Iron‐catalyzed construction of cyanomethylated thiohydantoins by cross‐dehydrogenative C(sp3)‐C(sp3) coupling	15
Development of Biscoumarin Compounds With Quorum‐Quenching Potential: Synthetic, Biological, and In Silico Studies	15
A “One‐Pot” Metal‐Free Synthesis and Evaluation of Antiproliferative Activity of Diversely Functionalized Pyrrolidine‐2‐Ones	15
New metal free organic dyes incorporating heterocyclic Benzofuran core as conjugated spacer: Synthesis, Opto‐electrochemical, DFT and DSSC studies	15
Synthesis and characterizations of some new selenolo[2,3‐b]quinoxaline derivatives	15
Synthesis of 1,3‐oxazepine derivatives via tandem reaction of 5‐benzylidine Meldrum's acids with TosMIC in presence of potassium carbonate	15
Natural and Synthetic Decahydroquinolines: Synthesis Strategies and Biological Activity	15
New edaravone analogs incorporated with N‐benzylthiazole moiety: Multistep chemical synthesis, in vitro cytotoxicity with pRIPK3 inhibitory activities, and molecular docking	14
Discovery of Promising Sulfadiazine Derivatives With Anti‐Proliferative Activity Against Tumor Cell Lines	14
Thiazolidinedione‐Pyrimidine Hybrid as Potential Antidiabetic Agents and Their Cardioprotective Effect	14
An efficient organopromotor L‐arginine facilitated synthesis of thiazolo[3,2‐a]pyrimidine derivatives in EtOH:H2O solvent	14
Visible‐light photoredox catalyzed synthesis of tetrahydrobenzofuranone: Oxidative [3 + 2] cycloaddition of dicarbonyl and alkene	14
Efficient preparation of (S)‐2‐(3,5‐dimethylphenyl)pyrrolidine via a recycle process of resolution	14
Thermal [2+2] Cycloaddition of Dihydropyrroles and Dimethyl Acetylenedicarboxylate	13
Manipulating sensitivities of planar oxadiazole‐based high performing energetic materials	13
Synthesis of Novel 6H‐Furo[3,2‐e]Indole Derivatives via One‐Pot Three Component Reactions	13
Long alkoxy substituted N2S2 porphyrins for liquid crystalline property	13
Research progress of oxazole derivatives in the discovery of agricultural chemicals	12
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Overview of Hydroxychloroquine and Remdesivir on severe acute respiratory syndrome coronavirus 2 (SARS‐CoV‐2)	11
Synthesis and bioactivity evaluation of 5‐trifluoromethyl‐1H‐pyrazole‐4‐carboxamide derivatives as potential anticancer and antifungal agents	11
Design, synthesis, and pesticidal activities of novel pyrimidin‐4‐amine derivatives containing trifluoroethyl sulfide moiety	11
A Simple, Economical, and Green Protocol for the Synthesis of Benzyl‐Quinoline Analogues by Grinding	11
A Sequential One‐Pot Synthesis of Quinoline‐Fused Benzoxe(Aze)pines via Intramolecular Reductive Heck Cyclisation	11
Investigation of some new main group metal complexes of hydrazine and 2‐mercaptopyridine‐3‐carboxylic acid mixed–ligands	11
Design, synthesis, antimicrobial evaluation, and in‐silico studies of some 4‐thiazolidinone hybrids bearing coumarin and pyridine moieties	10
Synthesis and Application of Azide‐Incorporated Copper‐Chelating Peptides for Efficient Click Conjugation Reaction	10
Issue Information	10
Kilogram synthesis of pinoxaden	10
Synthesis and biological evaluation of baloxavir marboxil analogs for the treatment of influenza A (H1N1) virus	10
Imidazo[1,2,4]triazolone and fused imidazo[1,2,4]triazolone derivatives: Synthesis, in vitro anticancer screening, CDK2 inhibitory activity, and molecular modeling studies	10
Novel pyrazole‐biphenyl‐carboxamides for SARS‐CoV2 entry‐level restriction and microbial infections	10
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Synthesis, characterization and crystal structure of some novel partially hydrogenated isoquinolines and their fused heterocyclic systems	10
Toward understanding the regioselectivity of the one‐pot reaction of phenylene diamines with aldehydes and cyclopentadiene (Povarov reaction). Combined experimental and theoretical approaches	10
Saccharin‐catalyzed multicomponent cascade reactions for the synthesis of 1,2,3,4,6‐pentasubstituted piperidines	10

Issue Information	10
Reactivity of pyrimidinylphosphazenes with acetylenic esters: Competitive [4 + 2] and [2 + 2] tandem cycloaddition or retro‐cycloaddition approaches	10
Synthetic strategies of phenazine derivatives: A review	10
Convenient synthesis and antibacterial evaluation of new bipyrazolyl and pyrazolopyridazine derivatives utilizing 4‐acetyl‐5‐methyl‐N‐phenyl‐1‐(p‐tolyl)‐1H‐p	9
Synthesis of Alpha‐Acyloxy‐(1,2,5‐Oxadiazole‐2‐Oxide) Carboxamides via Passerini Multicomponent Reaction. Evaluation of Nitric Oxide‐Releasing and Anti‐Proliferative Properties	9
Regio Selective Synthesis of Pyrazole Derivatives of 5‐Chloro‐2‐Methoxy Phenyl Hydrazide and Their Biological Evaluation	9
Exploring the Ring–Ring Expansion and Pyrazole Substitution of Chlorophosphazenes [ PCl 2 N	9
Facile synthesis and antimicrobial activity of bis(fused 4H‐pyrans) incorporating piperazine as novel hybrid molecules: Michael's addition approach	9
Neat multicomponent assembly of highly functionalized Acenaphtho[1,2‐b]pyrroles, in vitro evaluation for antioxidant and cytotoxic activities	9
CuI–Zn(OAc)2 Catalyzed Selective CC Bond Cleavage of 1,3‐Diketones/β‐Ketoester for the Formation of Quinazolin‐4(3H)‐Ones: A Fast, Solvent‐Free, Syn	9
Arylhydrazine salt‐selenium: A novel and efficient reagent system for arylselenenylation of unprotected uracil and its derivatives	9
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Visible‐Light Induced Rose Bengal Photocatalyzed One‐Pot Environmentally Sustainable Multicomponent Synthesis of Substituted Pyrazolo[3,4‐b]Quinolin‐5‐Ones	8
Synthesis of Benzofuran‐Based Hybrid Molecules: Molecular Docking and Antibacterial Activity Against Pseudomonas aeruginosa	8
Ni‐Ferrite an efficient catalyst for synthesis of 3‐aryl substituted isoxazole‐5‐carboxylic acids via one‐pot multicomponent reaction	8
Synthesis, antimicrobial activity, and in silico studies of fluoroquinolones bearing 1,3,4‐oxadiazolyl‐triazole derivatives	8
Issue Information	8
Issue Information	8
Synthesis of Naphtho[2,3‐b][1,10]phenanthrolines and Benzo[6,7]chromeno[3,2‐f]quinolines: One‐Pot Three‐Component Reaction of 2‐Hydroxy‐1,4‐Naphthoquinone, Aryl Aldehydes, and 8‐Aminoqui	8
Synthesis, characterization, anti‐proliferative evaluation, and molecular docking study of some new N‐(1, 3‐dioxoisoindolin‐4‐yl)acetamide derivatives	8
Study on halogen promoted cyclization of 2‐alkynylthiobenzimidazoles	8
Synthesis and Cellular Evaluation of Some Oxepino‐ and Pyranoxanthone Derivatives as Antitumor Agents: A Comparative Study	8
Synthesis of new thiazine and thiazole derivatives via cyclization reactions; investigating their electronic properties and determination of antioxidant properties	8
Direct synthesis of β2,3‐amino acid from β‐hydroxycarbamides: Implication in the synthesis of azumamide analogs and conformational analysis	8
Design, Synthesis, In Vitro Evaluation of New Tetrahydrooxazolo [5′,4′:4,5]Pyrimido[1,2‐a]Azepinone Derivatives as Anticancer Agents	8
Oxidative cross dehydrogenative coupling directed carbamates synthesis using Cu(II) pincer complex as active catalyst under mild reaction condition	8
Formation of anti‐Bredt‐type azabicyclo[4.2.0]octene frameworks through photochemical intramolecular [2+2] cycloaddition between indole and a distal double bond of allene	8
Facile Access to Benzofuro‐Fused‐Azeto[1,2‐ a ]Benzimidazoles as Promising Inhibitors of M. tuberculosis <	8
Synthesis and Characterization of Benzo[6,7]Cyclohepta[1,2‐b]Pyrazolo[4,3‐e]Pyridines	8
An operationally simple, one‐pot, convenient synthesis, and in vitro anti‐inflammatory activity of some new spirotriazolotriazine derivatives	8
Efficient synthesis and biological evaluation of some new series of pyridine derivatives: Promising and potent new class of anticancer agents	7
Dimethyl‐1,4‐Dithiines From 2‐Chloroprop‐2‐Enylisothiouronium Salt in KOH/Hydrazine Hydrate Medium: Experiment and Quantum Chemical Study	7
N‐Azidoethyl azoles through N‐alkylation under highly harmonized reaction conditions: Synthesis, characterization, and complexation as energetic coordination compounds	7
An efficient synthesis of new 3,5‐bis(2‐arylthiazol‐4‐yl)‐1,2,4‐oxadiazole derivatives and their antimicrobial evaluation	7
Issue Information	7
Catalyst‐Free and Visible Light‐Promoted Perfluoroalkylation of Indoles	7
Synthesis, Reactions, and Biological Evaluation Potential of Coumarin Derivatives: Review	7
Magnetically Recoverable CuFe 2 O 4	7
Synthesis of Terminal Alkenylindolines via Rhodium‐Catalyzed Direct CH Alkenylation With Alkenyl Borates	7
An Improved Synthesis of a Key Intermediate for Glycosylation of Biopterin and Its Application for the First Synthesis of Microcystbiopterin B	7
Issue Information	7
Facile synthesis and anticancer activity of tetrazolyl‐benzothiazole derivatives	7
Multicomponent synthesis of spiro 1,3,4‐thiadiazolines with anticancer activity by using deep eutectic solvent under microwave irradiation	7
Synthesis a group of 5(6)‐substituted benzimidazole Zn(II) and Co(II) complexes and investigation their cytotoxic and antimicrobial activities	7
Green Construction of Novel 3‐(Benzo[d][1,3]dioxol‐5‐yl)‐1,8‐naphthyridin‐2‐yl)amino)quinazoline‐2,4(1H,3H)‐dione and Phenyl‐[1,2,4]triazolo[4,3‐a][1,8]naphthyridine and Their An	7
Polycyclic Dicationic Heteroaromatic Compounds From One‐Step Multiple Condensation Reactions: Synthesis and Reactivity	7
Recyclization of 3‐substituted‐6,8‐dimethylchromones with some heterocyclic enamines: Spectroscopic, quantum calculations (HOMO–LUMO, MEP, NLO), biological evaluation, and ADME investigation	7
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Radical synthesis of dihydropyrano[2,3‐c]pyrazoles using acridine yellow G as a photo‐induced electron transfer photocatalyst	7
BimetallicCoCeO2oxide nanoparticles: An efficient and reusable heterogeneous catalyst for the preparation of2‐amino‐3‐cyano‐4H‐pyran derivatives	6
Construction of Carbon‐Nitrogen Bond From Addition Reaction of Weak Nucleophilic Nitrogen Atom of Imides With Para ‐Quinone Methides	6
A selective chromone‐based colorimetric chemosensor for detecting Cu2+ in near‐perfect aqueous solution and test kit	6
Design, Synthesis of Novel Pyrimidine Derivatives Containing Alkenyl Moieties With Herbicidal Activities	6
Synthesis, Photophysical Properties and Cytotoxic Activities of Isoxazole‐Containing Difluoroboron Complexes	6
Synthesis and antiviral activity of novel imidazo[2,1‐b]thiazoles coupled with morpholine and thiomorpholines	6
A Comprehensive Report on Environmentally Benign Synthesis of 1, 8‐Dioxo‐Octahydroxanthene Derivatives	6
Retraction statement: Design and synthesis of a bismethylsulfanyl‐steroid‐azetyl butanol derivative from 2‐nitroestradiol	6
Hantzsch‐like reaction of isoquinoline‐1‐acetonitrile in synthesis of 4H‐pyrido[2,1‐a]isoquinolines with antibacterial evaluation	6
A review on advances in synthetic methodology and biological profile of spirothiazolidin‐4‐ones	6
Synthesis and anticancer activity of some thiophene, thienyl‐thiazole, and thienyl‐benzofuran analogues	6
The synthesis of novel 2, 3‐disubstituted 1,6‐dihydropyrrolo[2,3‐g]indazole derivatives via one‐pot three component reactions	6
Synthesis and anticancer activity of cinnoline sulphonamides and 4‐heteroyclic derivatives: Cross‐coupling approach	6
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Recent developments in synthetic strategies and pharmacological outcomes of synthetic xanthine oxidase inhibitors: A comprehensive review	6
Ultrasound promoted three‐component synthesis of dihydroindeno[1,2‐b]pyrrole derivatives	6
A simple and efficient approach for the clickability of super‐bulky aryl azides	6
Synthesis and Biological Activities of Pyrazoline Derivatives: A Comprehensive Review	6
Green multicomponent approach to novel 5‐[(2H‐Pyran‐3‐yl)(aryl)methyl]‐1,3‐dimethylpyrimidines	6
Design, Synthesis, and Structure–Activity Relationship of Some New Ciprofloxacin Hybrids as Antibacterial Agents	6
Design, synthesis, and biological evaluation of 1,4,7,8‐tetrahydro‐5H‐furo[3,4‐b]pyrazolo[4,3‐e]pyridin‐5‐one‐based azo dyes	6
Novel oxadiazole functionalized pyridopyrimidine derivatives; their anticancer activity and molecular docking studies	6
Catalyst‐free one‐pot synthesis of quinoline tethered α‐amino ketones by multicomponent reactions	6
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Chiral Squaramide‐Catalyzed Asymmetric Synthesis of N,O‐Acetals From Pyrazolinone Ketimines	6
An efficient and green synthesis of multi‐heteroatom heterocycles via a three components reaction in acetic acid/aqueous condition	6
Synthesis and biological evaluation of 3‐hydroxypyrazoles as aquaporin 9 inhibitors	6
Pyranoquinolone derivatives: A potent multi‐targeted pharmacological scaffold	6
Recent Advances in the Chemistry of Selenopheno[2,3‐ b &3,4‐ b &3,4‐ c	6
Crystal Structure and Quantum Chemical Calculations of 2‐(2′‐Oxospiro[1,3‐dioxolane‐2,3′‐indol]‐1′(2′H)‐yl) acetohydrazide	5

Design, enantioselective synthesis, and antiviral activities against potato virus Y of axially chiral thiazine derivatives	5
Issue Information	5
Substrate‐controlled chemoselective synthesis of 1‐sulfonylquinazoline‐2,4(1H,3H)‐diones and 2‐sulfonamidobenzonitriles	5
Organocatalytic Enantioselective Synthesis of Oxindole‐4‐Aminopyrazolone Derivatives via Mannich Reaction of 3‐Substituted Oxindoles With Pyrazolinone Ketimines	5
Pyrazolo[3,4‐d]pyrimidine‐based scaffolds as antibacterial agents: Synthetic strategies, reactions, and in vitro biological evaluation	5
Design, synthesis, antifungal activity, and molecular docking of novel trifluoromethyl pyrimidine derivatives containing 1,3,4‐oxadiazole and thioether moieties as potential succinate dehyd	5
Issue Information	5
Synthetic, spectroscopic, and computational investigations of readily accessible 2‐phenyl‐3‐alkylbenzoxazaboroles	5
Baylis–Hillmanadducts as an important synthon for the synthesis of α‐carbolinone and α‐carboline derivatives	5
Efficient Synthetic Strategies for Highly Functionalized Pyrazole Including an Amidine Skeleton Based on Trichloroacetamidine, Alkynes, and Hydrazonoyl Chlorides	5
A Green Approach for the Synthesis of 5,6‐Dihydropyrimido[4,5‐d]Pyrimidines From N‐Uracil Amidines in Water	5
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β‐Nitrostyrenes as a valuable precursor for the synthesis of β‐aryl‐γ‐lactam and 2‐oxo‐1,2‐dihydroquinoline derivatives	5
N‐Methoxy Pyrazole‐4‐Carboxamide Derivatives: Synthesis, Spectral Analyses, Antifungal Activity, In Silico Molecular Docking, ADMET, and DFT Studies	5
Green synthesis and biological activity investigation of new derivatives of spiroisatins	5
(±)‐cis‐4a‐alkyl‐1,3,4,4a,9,9a‐hexahydro‐2H‐carbazol‐2‐ones by domino nitro reduction‐aza‐Michael addition to enones	5
Practical synthesis of (S)‐pyroglutamic acid	5
Oriented synthesis and insecticidal activities of novel meta‐diamide scaffolds incorporating with 1,2,4‐triazole moiety	5
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Synthesis, anticancer evaluation and in silico studies of novel N‐substituted arylidenethiazolidine‐2,4‐dione derivatives as adenosine monophosphate‐activated protein kinase activators	5
Unusual impurity formation during the process development of Olsalazine sodium leads to a new efficient and economical synthesis of tricaine mesylate	5
Synthesis of novel pyrido[3,4‐d]pyrimidine‐thiazolidione‐1,2,4‐oxadiazoles as potent EGFR targeting anticancer agents	5
Regioselective synthesis of fused pyrimidines and quinazolines linked to Phenoxy‐N‐arylacetamide moieties as novel hybrid molecules via Biginelli‐like reaction	5
Issue Information	5
Study on antitumor activity of parthenolide C‐14 derivatives	5
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Synthesis and Cancer Cell Cytotoxicity of 6‐, 7‐, or 8‐Substituted 2‐(Hetero)aryl‐4‐(4‐(Hetero)aryl‐2‐Oxobut‐3‐en‐1‐Ylidene)Benzothiazepanes	5
New oxadiazol‐5‐ones derivatives and their performance as angiotensin‐converting enzyme (ACE) inhibitors	5
Synthesis, antiinflammatory, and cytotoxic activity of novel pyrazolo[4,3‐c][2,1]benzothiazine 4,4‐dioxide derivatives	5
One‐Pot, Multicomponent Synthesis of 1,3‐Oxazin‐One and Evaluation of Their Potential Antioxidant Activities	5
Imidazo[1,2‐a]Pyrazine Linked Benzimidazole, Tetrahydropyrimidine, and 1,3,4‐Oxadizoles as Anticancer Agents	5
New thieno[2,3‐d]pyrimidine derivatives as EGFRWT and EGFRT790M inhibitors: Design, synthesis, antiproliferative activities, docking studi	5
A Solvent‐Free One‐Pot Synthesis of Ethyl 4‐Oxo‐3,4‐Dihydro Quinazoline‐2‐Carboxylates Utilizing N ‐(2‐Aminobenzoyl) Benzotriazoles	5
Synthesis, physico‐chemical characterization and theoretical exploration of some 2,4,5‐triaryl imidazole derivatives	5
Reaction Condition Dependent Multicomponent Reaction for the Synthesis of Substituted and Fused Naphthoquinone Derivatives	5
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Discovery of novel heterocyclic derivatives containing oxadiazolone or pyrimidinone cores as DPP‐4 inhibitors	5
Issue Information	5
2‐Vinylaniline in the synthesis of heterocycles: Recent advances	5
Regioselective synthesis and computational calculation studies of some new pyrazolyl‐pyridine and bipyridine derivatives	5
Preparation of chiral DMAP derivatives and investigation on their enantioselective catalytic activity in benzazetidine synthesis and kinetic resolutions of alcohols	5