Journal of Heterocyclic Chemistry

Papers
(The TQCC of Journal of Heterocyclic Chemistry is 5. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2021-06-01 to 2025-06-01.)
ArticleCitations
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Ultrasound‐promoted1,3‐dipolarcycloaddition of azomethine yields for synthesis of dispiropyrrolidineoxindole derivatives in hexyltriphenylphosphonium bromide as an ionic liquid, 42
Novel ferrocene cyclopalladated compounds: Synthesis, and in‐vitro antitumor activity study42
Catalyst‐free one‐pot three‐component rapid synthesis of polysubstituted pyrroles by liquid‐assisted grinding39
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Synthesis of novel amide/amino acid functionalized pyrazolo[3,4‐b]pyridine derivatives; their anticancer activity and docking studies25
Retraction statement: Facile synthesis of two oxocan derivatives using some chemical strategies25
Synthesis and herbicidal activity of pyrimidyl‐1,2,4‐triazole derivatives containing aryl sulfonyl moiety25
One‐pot synthesis of new functionalized 4H‐chromen‐4‐ylidene derivatives24
Trifluorodiazoethane: A versatile building block to access trifluoromethylated heterocycles23
One‐pot three‐component synthesis of novel chromeno[3,2‐c]pyridine‐1,9(2H)‐diones by using SnCl2⋅2H2O as catalyst23
Hybrid of the 1,2,3‐triazole nucleus and sesquiterpene skeleton as a potential antitumor agent: Hemisynthesis, molecular structure, Hirshfeld surface analysis, density functional theory, and in vitro 23
Efficient synthesis of piperidine derivatives using dendrimer based catalytical pockets23
Synthesis, antimicrobial activity, and molecular docking studies of new fused pyrimidinethiones22
A quick and easy access to a series of thiocyanated enaminones and 2‐iminothiazolones using PIDA under mild conditions22
Novel angularly substituted [1,4]thiazino[3,4‐a]isoquinoline carboxylic acids prepared by cyclic imine‐cyclic anhydride reaction20
Photoinduced 6π‐electrocyclization of 2,5‐dichlorothiophene containing benzofuranylacrylonitriles as efficient method for the generation of hydrogen chloride19
Solvent‐free Darzens condensation of 3‐chlorooxindoles with aryl aldehydes for diastereoselective construction of spiro‐epoxyoxindoles by grinding19
NiO‐Nanoparticles as green catalyst for an efficient synthesis of 4‐iminopyrido[1,2‐a]pyrimidine fluorophores via one pot cyclization of α‐aminonicotinonitrile18
Synthesis and molecular modeling of some novel hydroxypyrone derivatives as antidermatophytic agents17
The applications of β‐keto amides for heterocycle synthesis17
[3+2] cycloaddition synthesis of new (nicotinonitrile‐chromene)‐based bis(pyrazole) hybrids as potential acetylcholinesterase inhibitors17
Combination of N‐amino‐1,2,4‐triazole and 4‐hydroxy‐3,5‐dinitropyrazole for the synthesis of high performing explosives16
Unprecedented, catalyst‐free, and rapid one‐pot, three‐component green synthesis of substituted 3‐hydroxy‐2‐oxindoles in water16
A synthetic strategy for the preparation of alkoxy‐functionalized bis‐1,2,4‐triazinyl‐2,6‐pyridines16
Synthetic Approaches Toward Imidazo‐Fused Heterocycles: A Comprehensive Review15
Facile access to 2‐amino‐4‐aryl‐5H‐chromeno[4,3‐b]pyridine‐3‐carbonitriles through a strategy of one‐pot Michael/cyclization reaction15
Discovery of Promising Sulfadiazine Derivatives With Anti‐Proliferative Activity Against Tumor Cell Lines15
New edaravone analogs incorporated with N‐benzylthiazole moiety: Multistep chemical synthesis, in vitro cytotoxicity with pRIPK3 inhibitory activities, and molecular docking15
Palladium‐Catalyzed Synthesis of Pyrrolo[1,2‐α]Pyrazines From N‐Phenacyl Pyrrole‐2‐Carbonitriles and Aryl Boronic Acids15
Synthesis and biological assessment of some fused Pyran derivatives15
Synthesis of substituted 5‐aryl‐2,3‐dihydropyrazine 1,4‐dioxides based on condensation of N,N′‐(2,3‐dimethylbutane‐2,3‐diyl)bis(hydroxylamine) with various arylglyoxals15
Retraction statement: Facile synthesis of two oxocan derivatives using some chemical strategies15
Efficient preparation of (S)‐2‐(3,5‐dimethylphenyl)pyrrolidine via a recycle process of resolution15
A regiospecific fischer indole reaction with 3‐oxo‐24‐nor‐allobetulin15
Synthesis, and reverse screening of 6‐(3,4,5‐trimethoxyphenyl)pyrimidine‐5‐carbonitrile derivatives as anticancer agents: Part‐II15
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An approach for the diastereoselective synthesis of (R)‐(+)‐methyl pipecolate and (+)‐dextro‐erythrophacetoperane from (S)‐(−)‐methylbenzylamine15
Synthesis and evaluation of the biological activities of novel hybrid isoindol‐1,3‐dione containing an aziridine unit14
Visible‐light photoredox catalyzed synthesis of tetrahydrobenzofuranone: Oxidative [3 + 2] cycloaddition of dicarbonyl and alkene14
Synthesis of 1,3‐oxazepine derivatives via tandem reaction of 5‐benzylidine Meldrum's acids with TosMIC in presence of potassium carbonate14
New metal free organic dyes incorporating heterocyclic Benzofuran core as conjugated spacer: Synthesis, Opto‐electrochemical, DFT and DSSC studies14
Iron‐catalyzed construction of cyanomethylated thiohydantoins by cross‐dehydrogenative C(sp3)‐C(sp3) coupling14
An efficient organopromotor L‐arginine facilitated synthesis of thiazolo[3,2‐a]pyrimidine derivatives in EtOH:H2O solvent14
Saccharin‐catalyzed multicomponent cascade reactions for the synthesis of 1,2,3,4,6‐pentasubstituted piperidines13
Synthesis and characterizations of some new selenolo[2,3‐b]quinoxaline derivatives13
Long alkoxy substituted N2S2 porphyrins for liquid crystalline property13
Synthesis of novel Schiff bases as stable enol‐imine‐containing diazene bonds and pyrimidines using trimethinium salts13
Synthesis and bioactivity evaluation of 5‐trifluoromethyl‐1H‐pyrazole‐4‐carboxamide derivatives as potential anticancer and antifungal agents13
Design, synthesis, antimicrobial evaluation, and in‐silico studies of some 4‐thiazolidinone hybrids bearing coumarin and pyridine moieties13
Synthesis of Novel 6H‐Furo[3,2‐e]Indole Derivatives via One‐Pot Three Component Reactions13
Overview of Hydroxychloroquine and Remdesivir on severe acute respiratory syndrome coronavirus 2 (SARS‐CoV‐2)13
Synthesis of arylidene‐based benzoxazine derivatives as promising antimicrobial materials13
Imidazo[1,2,4]triazolone and fused imidazo[1,2,4]triazolone derivatives: Synthesis, in vitro anticancer screening, CDK2 inhibitory activity, and molecular modeling studies12
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Synthesis and Application of Azide‐Incorporated Copper‐Chelating Peptides for Efficient Click Conjugation Reaction12
Utility of pyrrole‐2‐thioacetohydrazide in synthesis of new heterocyclic compounds with promising antimicrobial activities and molecular docking studies12
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Novel pyrazole‐biphenyl‐carboxamides for SARS‐CoV2 entry‐level restriction and microbial infections12
Design, synthesis, and pesticidal activities of novel pyrimidin‐4‐amine derivatives containing trifluoroethyl sulfide moiety12
Manipulating sensitivities of planar oxadiazole‐based high performing energetic materials12
Convenient synthesis and antibacterial evaluation of new bipyrazolyl and pyrazolopyridazine derivatives utilizing 4‐acetyl‐5‐methyl‐N‐phenyl‐1‐(p‐tolyl)‐1H‐p11
Research progress of oxazole derivatives in the discovery of agricultural chemicals11
Synthesis and biological evaluation of baloxavir marboxil analogs for the treatment of influenza A (H1N1) virus11
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Arylhydrazine salt‐selenium: A novel and efficient reagent system for arylselenenylation of unprotected uracil and its derivatives11
Investigation of some new main group metal complexes of hydrazine and 2‐mercaptopyridine‐3‐carboxylic acid mixed–ligands11
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Regio Selective Synthesis of Pyrazole Derivatives of 5‐Chloro‐2‐Methoxy Phenyl Hydrazide and Their Biological Evaluation10
Kilogram synthesis of pinoxaden10
Facile synthesis and antimicrobial activity of bis(fused 4H‐pyrans) incorporating piperazine as novel hybrid molecules: Michael's addition approach10
Synthesis of new thiazine and thiazole derivatives via cyclization reactions; investigating their electronic properties and determination of antioxidant properties10
Neat multicomponent assembly of highly functionalized Acenaphtho[1,2‐b]pyrroles, in vitro evaluation for antioxidant and cytotoxic activities10
Design, synthesis, biological evaluation, and molecular docking studies of some novel N,N‐dimethylaminopropoxy‐substituted aurones10
Toward understanding the regioselectivity of the one‐pot reaction of phenylene diamines with aldehydes and cyclopentadiene (Povarov reaction). Combined experimental and theoretical approaches10
Reactivity of pyrimidinylphosphazenes with acetylenic esters: Competitive [4 + 2] and [2 + 2] tandem cycloaddition or retro‐cycloaddition approaches10
Synthetic strategies of phenazine derivatives: A review10
Recent progress in the synthesis of azoles and related five‐membered ring heterocycles using silica‐supported heterogeneous catalysts9
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Synthesis, characterization and crystal structure of some novel partially hydrogenated isoquinolines and their fused heterocyclic systems9
Synthesis, antimicrobial activity, and in silico studies of fluoroquinolones bearing 1,3,4‐oxadiazolyl‐triazole derivatives9
An operationally simple, one‐pot, convenient synthesis, and in vitro anti‐inflammatory activity of some new spirotriazolotriazine derivatives9
Direct synthesis of β2,3‐amino acid from β‐hydroxycarbamides: Implication in the synthesis of azumamide analogs and conformational analysis9
Synthesis, crystal structure, and density functional theory study of a new compound 4‐(2‐chlorobenzyl)‐1‐(5‐fluoro‐2‐hydroxy‐3‐(thiomorpholinomethyl)phenyl [1,2,4]triazolo[4,3‐a]9
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CuI–Zn(OAc)2 Catalyzed Selective CC Bond Cleavage of 1,3‐Diketones/β‐Ketoester for the Formation of Quinazolin‐4(3H)‐Ones: A Fast, Solvent‐Free, Syn9
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Synthesis of Benzofuran‐Based Hybrid Molecules: Molecular Docking and Antibacterial Activity Against Pseudomonas aeruginosa8
A rapid and quantitative synthesis of xanthene derivatives using sulfonated graphitic carbon nitride under ball‐milling8
Design, Synthesis, In Vitro Evaluation of New Tetrahydrooxazolo [5′,4′:4,5]Pyrimido[1,2‐a]Azepinone Derivatives as Anticancer Agents8
Formation of anti‐Bredt‐type azabicyclo[4.2.0]octene frameworks through photochemical intramolecular [2+2] cycloaddition between indole and a distal double bond of allene8
Synthesis, characterization, anti‐proliferative evaluation, and molecular docking study of some new N‐(1, 3‐dioxoisoindolin‐4‐yl)acetamide derivatives8
Recyclization of 3‐substituted‐6,8‐dimethylchromones with some heterocyclic enamines: Spectroscopic, quantum calculations (HOMO–LUMO, MEP, NLO), biological evaluation, and ADME investigation8
Efficient synthesis and biological evaluation of some new series of pyridine derivatives: Promising and potent new class of anticancer agents8
Facile synthesis and anticancer activity of tetrazolyl‐benzothiazole derivatives8
Green Construction of Novel 3‐(Benzo[d][1,3]dioxol‐5‐yl)‐1,8‐naphthyridin‐2‐yl)amino)quinazoline‐2,4(1H,3H)‐dione and Phenyl‐[1,2,4]triazolo[4,3‐a][1,8]naphthyridine and Their An8
Study on halogen promoted cyclization of 2‐alkynylthiobenzimidazoles8
Ni‐Ferrite an efficient catalyst for synthesis of 3‐aryl substituted isoxazole‐5‐carboxylic acids via one‐pot multicomponent reaction8
Radical synthesis of dihydropyrano[2,3‐c]pyrazoles using acridine yellow G as a photo‐induced electron transfer photocatalyst8
Synthesis a group of 5(6)‐substituted benzimidazole Zn(II) and Co(II) complexes and investigation their cytotoxic and antimicrobial activities8
N‐Azidoethyl azoles through N‐alkylation under highly harmonized reaction conditions: Synthesis, characterization, and complexation as energetic coordination compounds8
Synthesis and Characterization of Benzo[6,7]Cyclohepta[1,2‐b]Pyrazolo[4,3‐e]Pyridines8
Synthesis of Terminal Alkenylindolines via Rhodium‐Catalyzed Direct CH Alkenylation With Alkenyl Borates8
Multicomponent synthesis of spiro 1,3,4‐thiadiazolines with anticancer activity by using deep eutectic solvent under microwave irradiation8
Oxidative cross dehydrogenative coupling directed carbamates synthesis using Cu(II) pincer complex as active catalyst under mild reaction condition8
Medicinal perspective of quinazolinone derivatives: Recent developments and structure–activity relationship studies8
Benzimidazole tethered thioureas as a new entry to elastase inhibition and free radical scavenging: Synthesis, molecular docking, and enzyme inhibitory kinetics7
Retraction statement: Design and synthesis of a bismethylsulfanyl‐steroid‐azetyl butanol derivative from 2‐nitroestradiol7
Highly efficient microwave‐assisted solvent free sequential one‐pot multicomponent synthesis of novel 2‐hydroxy indenopyridin‐5‐ones and mechanismic computational study7
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A simple and efficient approach for the clickability of super‐bulky aryl azides7
Synthesis and biological evaluation of 3‐hydroxypyrazoles as aquaporin 9 inhibitors7
An efficient synthesis of new 3,5‐bis(2‐arylthiazol‐4‐yl)‐1,2,4‐oxadiazole derivatives and their antimicrobial evaluation7
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Catalyst‐free one‐pot synthesis of quinoline tethered α‐amino ketones by multicomponent reactions7
Ultrasound promoted three‐component synthesis of dihydroindeno[1,2‐b]pyrrole derivatives7
An elegant and efficient synthesis of heterocycles integrated with bisN‐acyl pyrazoline and bis‐1, 2, 3‐triazole via a green synthetic methodology7
Synthesis and antiviral activity of novel imidazo[2,1‐b]thiazoles coupled with morpholine and thiomorpholines7
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Synthesis, Photophysical Properties and Cytotoxic Activities of Isoxazole‐Containing Difluoroboron Complexes7
Recent developments in synthetic strategies and pharmacological outcomes of synthetic xanthine oxidase inhibitors: A comprehensive review7
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Design, synthesis, and bioactivity evaluation of novel thiochromanone derivatives containing an oxime or oxime ether moiety7
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Design, Synthesis of Novel Pyrimidine Derivatives Containing Alkenyl Moieties With Herbicidal Activities7
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Synthesis of various functionalized 2H‐azirines: An updated library7
An efficient and green synthesis of multi‐heteroatom heterocycles via a three components reaction in acetic acid/aqueous condition7
A review on advances in synthetic methodology and biological profile of spirothiazolidin‐4‐ones6
A search for antiinflammatory therapies: Synthesis, in silico investigation of the mode of action, and in vitro analyses of new quinazolin‐2,4‐dione derivatives targeting phosphodiesterase‐4 enzyme6
Study on antitumor activity of parthenolide C‐14 derivatives6
New thieno[2,3‐d]pyrimidine derivatives as EGFRWT and EGFRT790M inhibitors: Design, synthesis, antiproliferative activities, docking studi6
Stereoselective synthesis and characterization of monocyclic cis‐β‐lactams containing 5‐methyl‐1,3,4‐thiadiazole‐2‐thiol moiety6
Synthesis and anticancer activity of cinnoline sulphonamides and 4‐heteroyclic derivatives: Cross‐coupling approach6
Hantzsch‐like reaction of isoquinoline‐1‐acetonitrile in synthesis of 4H‐pyrido[2,1‐a]isoquinolines with antibacterial evaluation6
The synthesis of novel 2, 3‐disubstituted 1,6‐dihydropyrrolo[2,3‐g]indazole derivatives via one‐pot three component reactions6
Novel oxadiazole functionalized pyridopyrimidine derivatives; their anticancer activity and molecular docking studies6
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N‐Methoxy Pyrazole‐4‐Carboxamide Derivatives: Synthesis, Spectral Analyses, Antifungal Activity, In Silico Molecular Docking, ADMET, and DFT Studies6
Progress in the chemistry of functional aramids properties6
Design, synthesis, antifungal activity, and molecular docking of novel trifluoromethyl pyrimidine derivatives containing 1,3,4‐oxadiazole and thioether moieties as potential succinate dehyd6
Synthesis of new 1,4‐ and 1,5‐disubstituted N‐ethyl acetate and N‐α‐butyro‐γ‐lactone alkylimidazole derivatives as N‐acylhomoserine lactone analogs6
Design, synthesis, and biological evaluation of 1,4,7,8‐tetrahydro‐5H‐furo[3,4‐b]pyrazolo[4,3‐e]pyridin‐5‐one‐based azo dyes6
Green multicomponent approach to novel 5‐[(2H‐Pyran‐3‐yl)(aryl)methyl]‐1,3‐dimethylpyrimidines6
Synthesis and anticancer activity of some thiophene, thienyl‐thiazole, and thienyl‐benzofuran analogues6
BimetallicCoCeO2oxide nanoparticles: An efficient and reusable heterogeneous catalyst for the preparation of2‐amino‐3‐cyano‐4H‐pyran derivatives6
Synthesis and Cancer Cell Cytotoxicity of 6‐, 7‐, or 8‐Substituted 2‐(Hetero)aryl‐4‐(4‐(Hetero)aryl‐2‐Oxobut‐3‐en‐1‐Ylidene)Benzothiazepanes6
Efficient domino strategy for synthesis of 3‐substituted 1,5‐dihydro‐4H‐pyrrolo[3,2‐c]pyridin‐4‐one derivatives6
Pyranoquinolone derivatives: A potent multi‐targeted pharmacological scaffold6
Base promoted CuFe2O4 catalyzed one‐pot synthesis of 3,5‐diaryl‐1H‐pyrazoles6
A selective chromone‐based colorimetric chemosensor for detecting Cu2+ in near‐perfect aqueous solution and test kit6
Baylis–Hillmanadducts as an important synthon for the synthesis of α‐carbolinone and α‐carboline derivatives5
Green synthesis and biological activity investigation of new derivatives of spiroisatins5
Synthesis, crystal structure, and DFT study of 4‐(2‐Chlorobenzyl)‐1‐(furan‐2‐yl)‐[1,2,4]triazolo[4,3‐a]quinazolin‐5(4H)‐one5
Proton‐ and halogen‐induced cyclizations of 2‐(3‐butenyl)quinazolin‐4(3H)‐ones in the synthesis of pyrrolo[2,1‐b]‐ and pyrrolo[1,2‐а]quinazolinone derivatives5
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Discovery of novel heterocyclic derivatives containing oxadiazolone or pyrimidinone cores as DPP‐4 inhibitors5
One‐Pot, Multicomponent Synthesis of 1,3‐Oxazin‐One and Evaluation of Their Potential Antioxidant Activities5
One‐pot three‐component reaction; synthesis of new symmetrically bridge 4,4′‐(1,4‐phenylene)di‐pyrimidines under solvent free conditions5
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Regioselective synthesis of fused pyrimidines and quinazolines linked to Phenoxy‐N‐arylacetamide moieties as novel hybrid molecules via Biginelli‐like reaction5
Substrate‐controlled chemoselective synthesis of 1‐sulfonylquinazoline‐2,4(1H,3H)‐diones and 2‐sulfonamidobenzonitriles5
Pyrazolo[3,4‐d]pyrimidine‐based scaffolds as antibacterial agents: Synthetic strategies, reactions, and in vitro biological evaluation5
β‐Nitrostyrenes as a valuable precursor for the synthesis of β‐aryl‐γ‐lactam and 2‐oxo‐1,2‐dihydroquinoline derivatives5
Practical synthesis of (S)‐pyroglutamic acid5
Preparation of chiral DMAP derivatives and investigation on their enantioselective catalytic activity in benzazetidine synthesis and kinetic resolutions of alcohols5
New oxadiazol‐5‐ones derivatives and their performance as angiotensin‐converting enzyme (ACE) inhibitors5
Synthesis and bioactivity evaluation of eugenol hybrids obtained by Mannich and 1,3 dipolar cycloaddition reactions5
Ultrasonic‐Assisted condensation of aromatic and aliphatic aldehydes with 3‐(Thiophen‐2‐yl)‐5‐Pyrazolone: Synthesis, characterization and Stereoselective application5
Design, synthesis, and evaluation of new 4(3H)‐quinazolinone derivatives containing a pyrazole carboxamide moiety5
Introducing new method for the synthesis of polycyclic compounds containing [1,3]dithiine derivatives, with anticancer and antibacterial activities against common bacterial strains between aquatic and5
A high‐yielding protocol for the synthesis of 4,5‐diarylpyrimidin‐2‐amine derivatives from chalcones5
Chemoselective direct amidation of fatty acids with furfurylamine without coupling reagents in reversed micellar microenvironment5
An efficient synthesis of 4,6‐diarylnicotinonitrile‐acetamide hybrids via 1,2,3‐triazole linker as multitarget microbial inhibitors5
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Synthesis, anticancer evaluation and in silico studies of novel N‐substituted arylidenethiazolidine‐2,4‐dione derivatives as adenosine monophosphate‐activated protein kinase activators5
A facile approach to [1,2,4]triazolo[3,4‐i]purine via PIDA oxidation ring‐closing reaction5
Synthesis of non‐toxic anticancer active forskolin‐indole‐triazole conjugates along with their in silico succinate dehydrogenase inhibition studies5
Synthetic, spectroscopic, and computational investigations of readily accessible 2‐phenyl‐3‐alkylbenzoxazaboroles5
Unusual impurity formation during the process development of Olsalazine sodium leads to a new efficient and economical synthesis of tricaine mesylate5
A convenient and efficient process for the synthesis of 9‐aryl‐6,9‐dihydro‐1H‐pyrazolo[3,4‐f] quinoline‐8‐carbonitrile and 1‐aryl‐1,4‐ dihydrobenzo[f]quinoline‐2‐carbon5
2‐Vinylaniline in the synthesis of heterocycles: Recent advances5
Regioselective synthesis and computational calculation studies of some new pyrazolyl‐pyridine and bipyridine derivatives5
An eco‐efficient new path of mortar pestle grinding approach for the construction of methanol and ethylthio substituted pyridines with in silico studies5
(±)‐cis‐4a‐alkyl‐1,3,4,4a,9,9a‐hexahydro‐2H‐carbazol‐2‐ones by domino nitro reduction‐aza‐Michael addition to enones5
Antimicrobial and antiproliferative study of chalcone clubbed 2,4‐dimethylpyrrole‐3‐carboxamide derivatives: Synthesis and in vitro evaluation5
Synthesis, physico‐chemical characterization and theoretical exploration of some 2,4,5‐triaryl imidazole derivatives5
Synthesis of novel pyrido[3,4‐d]pyrimidine‐thiazolidione‐1,2,4‐oxadiazoles as potent EGFR targeting anticancer agents5
Synthesis, antiinflammatory, and cytotoxic activity of novel pyrazolo[4,3‐c][2,1]benzothiazine 4,4‐dioxide derivatives5
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Synthesis, characterization, and photophysical properties of some new thieno[2,3‐b]pyridines bearing phenylethenyl moiety5
Design, enantioselective synthesis, and antiviral activities against potato virus Y of axially chiral thiazine derivatives5
Design, Synthesis, Antiproliferative Screening, and In Silico Studies of Some Pyridinyl‐Pyrimidine Candidates5
Oriented synthesis and insecticidal activities of novel meta‐diamide scaffolds incorporating with 1,2,4‐triazole moiety5
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