Journal of Organic Chemistry

Papers
(The TQCC of Journal of Organic Chemistry is 8. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2021-04-01 to 2025-04-01.)
ArticleCitations
Stereoselective Synthesis of Substituted (Z)-N-Allyl Sulfonamides via a Palladium-Catalyzed Three-Component Tandem Reaction93
Issue Publication Information87
Transient Directing Group-Assisted Palladium-Catalyzed C4-Alkynylation of Indoles82
Tetra-Dentate Cycloaddition Catalysts for Rapid Photopolymerization Reactions82
From Pseudocyclic to Macrocyclic Ionophores: Strategies toward the Synthesis of Cyclic Monensin Derivatives73
Sulfonyl Radical-Induced Regioselective Cyclization of Enamide–Olefin To Form Sulfonylated 6–7-Membered Cyclic Enamines69
Gold Self-Relay Catalysis Enabling Regioselective Bicyclization toward [5]Azahelicenes68
Synthesis of Carboxylic Acids Containing α-All-Carbon Quaternary Centers from Diazo Compounds and Trialkylboranes63
The Aqueous and Acetonitrile Bond Dissociation Free Energies of N-Hydroxyphthalimide61
Photocatalytic Generation of Germyl Radicals from Digermanes Enabling the Hydro/Deuteriogermylation of Alkenes61
Asymmetric Aza Friedel–Crafts Reaction of 3,4-Dihydroisoquinolines with 1-Naphthols Catalyzed by Chiral Phosphoric Acids58
Regiodivergent Desymmetrization of meso-4,5-Epoxycyclohex-1-ene58
Catalytic Asymmetric Synthesis of Bicyclic Isothioureas from a Common Enolizable Template55
Nickel/Iridium Metallaphotoredox Catalysis for Allylic C–H Bond Arylation of N-Allyl Heterocycles55
NHC-BH3-Mediated Reduction of Sulfonyl Hydrazides into Disulfides and Further Cross-Coupling with Chlorostibine and Bioactivities54
Computational Study of Hypervalent Chalcogen Bond Catalysis on the Hydroarylation of Styrene with Phenol: O-Activation vs π-Activation53
Visible Light-Induced C–H Alkylation of Azauracils with N-Hydroxyphthalimide Esters via Catalytic EDA Complex52
Copper-Catalyzed Domino Annulation of Isoselenocyanates: A Pathway to Structurally Diverse N, Se-Bis-Heterocyclic, and Fused Heterocyclic Compounds52
Indoles Oxidative Ring-Opening/Cyclization Cascade with the 1,2-Diaminoarenes: Direct Synthesis of 2-Aryl-3-(2-aminoaryl)quinoxalines50
Structure Revision of Heptacyclic Naphthoquinone Dimer Arnebidin Based on NMR Spectroscopic Analysis and X-ray Crystallography49
Surfactant-Dependent Partitioning of Organics in Aqueous–Organic Reaction Systems49
Temperature-Dependent Photoreactivity of 2-Azidomethylbenzophenone: Insights into the Triplet Imine Biradical Pathway48
Synthesis and Performance of l-Tryptophanamide and (S)-1-(Naphthalen-2′-yl)ethanamine-Based Marfey-Type Derivatives for Amino Acid Configurational Analysis: Diastereomeric Resolution47
Modeling Possible Biogenetic Pathways to the Isomeric Pyrano[2,3-g]indole and Pyrano[3,2-f]indole Cores of Certain Prenylated Indole Alkaloids Using Gold(I)-Catalyzed Intramolecular Hydr47
Hydrogen Bond-Controlled Site-Selective C(sp3)–H Alkylation of Sulfonanilides46
Visible-Light-Induced Sulfonylation Cyclization to Generate Indole-Fused Medium-Sized N-Heterocycles in 2-Me-THF46
g-C3N4-Based Heterogeneous Photocatalyzed Synthesis and Evaluation of Antitumor Activities of Fluoroalkylated 4H-Pyrido[1,2-a]pyrimidin-4-ones45
Synthesis of Triarylsulfonium Salts with Sterically Demanding Substituents and Their Alkaline Stability43
Visible-Light-Induced Secondary Benzylic C(sp3)–H Functionalization for Nucleophilic Substitution: An Intermolecular C–X (C–N, C–C, and C–Br) Bond Forming Reaction43
Aerobic Copper-Catalyzed Intramolecular Cascade Oxidative Isomerization/[4+4] Cyclization of 2,2′-Disubstituted Stilbenes43
Palladium-Catalyzed Dual C–H Carbonylation of Diarylamines Leading to Diversified Acridones under CO-Free Conditions42
Unsymmetrical Benzothieno-Fused BODIPYs as Efficient NIR Heavy-Atom-Free Photosensitizers41
Stereoselective Synthesis of β-S-Glycosides via Palladium Catalysis41
Anhydrous and Stereoretentive Fluoride-Enhanced Suzuki–Miyaura Coupling of Immunomodulatory Imide Drug Derivatives40
Water-Compatible Staudinger–Diels–Alder Ligation40
Continuous Flow Generation of Acylketene Intermediates via Nitrogen Extrusion40
HCl/DMSO/HFIP-Mediated Chlorination of Pyrrolo[2,1-a]isoquinolines and Other Electron-Rich Heteroarenes40
Visible-Light-Driven Thioesterification of Aryl Halides with Potassium Thiocarboxylates: Transition-Metal Catalyst-Free Incorporation of Sulfur Functionalities into an Aromatic Ring39
Palladium-Catalyzed Asymmetric Hydrogenation of Unprotected 3-Substituted Indoles39
Diversity in Heterocycle Synthesis Using α-Iminocarboxylic Acids: Decarboxylation Dichotomy39
Investigation of Peptide Labeling with ortho-Phthalaldehyde and 2-Acylbenzaldehyde39
para-Selective, Direct C(sp2)–H Alkylation of Electron-Deficient Arenes by the Electroreduction Process38
Catalytic Asymmetric Synthesis of Atropisomeric N-Aryl 1,2,4-Triazoles38
Transition-Metal-, Additive-, and Solvent-Free [3 + 3] Annulation of RCF2-Imidoyl Sulfoxonium Ylides with Cyclopropenones to Give Multifunctionalized CF3-Pyridones38
Alkali Carbonates Improve β,β-Diaryl Serine-Catalyzed Enantioselective α-Fluorination of β-Dicarbonyl Compounds37
Issue Publication Information37
Iron-Catalyzed Synthesis of Peroxylpyrrolo[2,1-a]isoquinolines through Oxidative Dearomatization37
Continuous Flow Synthesis of α-Trifluoromethylthiolated Esters and Amides from Carboxylic Acids: a Telescoped Approach36
Promoting Catalytic C-Selective Sulfonylation of Cyclopropanols against Conventional O-Sulfonylation Using Readily Available Sulfonyl Chlorides36
Cascade Aza-Prins/Friedel–Crafts Reaction of Homocinnamyloxycarbamate and Aromatic Aldehydes Yielding Aromatic Ring-Annulated Hydrocyclopenta-1,2-oxazinane36
Issue Publication Information36
Metal-Free Electrochemical Allylic C–H Aerobic Oxidation35
Silver-Catalyzed Cascade Radical Isonitrile Insertion/Defluorinative Cyclization: Direct Synthesis of 4-CF2H-2-Phosphinoyl-quinolines35
Visible Light-Induced Divergent Deoxygenation/Hydroxymethylation of Pyridine N-Oxides35
Divergent Synthesis of Axially Chiral 2-Pyranones and Fused 2-Pyridones via N-Heterocyclic Carbene-Catalyzed Atroposelective [3 + 3] Annulation35
ChemEASTry Europe, the Status of the Chemical Sciences in a Growing Region35
Synthesis of N6-dA Damaged DNAs to Probe the Replication Ability of Human Translesion Polymerases35
Copper-Catalyzed Radical Cascade Cyclization of N-Substituted Indole-3-Aldehydes with Aryl Alkenes: Access to Pyrrolo[1,2-a]indole Scaffolds35
MAdPHOS, a P-Stereogenic Aminodiphosphane Ligand with Adamantyl Groups: Synthesis, NH/PH Tautomerism, and Rhodium and Nickel Complexes35
Photooxidation and Cleavage of Ethynylated 9,10-Dimethoxyanthracenes with Acid-Labile Ether Bonds35
Electrochemical Cyclization–Desulfurization Approach for the Synthesis of 1,3-Benzoxazines Using Cascade C–O and C–N Bond Formation35
Cobalt(II)-Catalyzed Selective C2–H Heck Reaction of Native (N–H) Indoles Enabled by Salicylaldehyde Ligand35
Molecular Sensing of Chiral Carboxylic Acid Enantiomers Using CD Inductions in the Visible Light Region35
Synthesis and Resolution of 4′-Substituted Nucleosides with Potential Antiviral and Antisense Strategies35
Ex Situ Synthesis of N-Capped Peptides in the Solution Phase via Palladium-Catalyzed Aminocarbonylation Utilizing Chloroform-COware35
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Mechanism and Selectivities in Ru-Catalyzed Anti-Markovnikov Formal Hydroalkylation of 1,3-Dienes and Enynes: A Computational Study34
Photoinitiated Rearrangement of Aromatic Azides to 2-Aminonicotinates34
Cross-Coupling Reactions of 5-Bromo-1,2,3-triazine34
Metal-Free Stereoselective Synthesis of (E)- and (Z)-N-Monosubstituted β-Aminoacrylates via Condensation Reactions of Carbamates34
3-Substituted-1-(Trimethylsilylmethyl)cyclobutyl Cations: Stereochemistry of Solvent Capture of β-Trimethylsilyl Carbocations34
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Nitroacetonitrile and Its Synthetic Equivalents33
Stereoselective and Divergent Aza-Adenosine and Aza-Guanosine Syntheses from Xylofuranose, the Key Fragments of a STING Cyclic Dinucleotide Agonist33
Issue Editorial Masthead33
Correction to Transition-Metal-Free Cross-Coupling of Aryl Halides with Arylstannanes33
Biocatalytic Synthesis of Nitrile-Bearing All-Carbon Quaternary Stereocenters32
Cu-Catalyzed Tandem C–N and C–C Bond Formation Leading to 4(1H)-Quinolones: A Scaffold with Diverse Biological Properties from Totally New Raw Materials in a Single Step32
Revealing the Role of Noncovalent Interactions on the Conformation of the Methyl Group in Tricyclic Orthoamide31
Molecular Nanocarbons Add New Dimensions to Organic Chemistry31
Issue Editorial Masthead31
Equipping 1,4,7-Triazacyclononane with Substituents via Solid-Phase Synthesis31
Selective N-Alkylation of Aminobenzenesulfonamides with Alcohols for the Synthesis of Amino-(N-alkyl)benzenesulfonamides Catalyzed by a Metal–Ligand Bifunctional Ruthenium Catalyst31
Zinc 1,1,2,2-Tetrafluoroethanesulfinate: A Synthetically Useful Oxidative and Photoredox Source of the 1,1,2,2-Tetrafluoroethyl Radical31
MSTFA as an Effective TMS Source for the TMSOTf-Catalzyed Synthesis of Cyclic Acetals31
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Enantioselective Mannich Reaction between Cyclic N-Sulfonyl Ketimines and Isatin-Derived Ketimines31
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Heck Reaction of 2-Oxyacrylates with Aryl Bromides: A Common Route to Monoaryl Pyruvates and Ortho Ester-Protected Monoaryl Pyruvates30
Heteroatom-Assisted Regio- and Stereoselective Palladium-Catalyzed Carboxylation of 9-Allyl Adenine30
Preparation, Characterization, and Mechanistic Considerations for 1,1,1-Tri(thioacetyl)ethane and 1,1-Di(thioacetyl)ethene30
Metal Binding and Its Amelioration in Tetramates30
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Mechanistic Study on CpRh(III)-Catalyzed [3 + 2] Annulation of Aniline Derivatives with Vinylsilanes: A DFT Study30
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Examining the Scope of Deriving β-Aryl Enones from Enol Silanes as Ketone Equivalents via Pd(II)-Mediated Sequential Dehydrosilylation and Arylation29
Closing a Calix[6]arene-Based Funnel Zn2+ Complex at Its Large Rim Entrance: Consequences on Metal Ion Affinity and Host–Guest Properties29
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SO2F2-Mediated N-Alkylation of Imino-Thiazolidinones29
Photoredox-Catalyzed Phosphonocarboxylation of Allenes with Phosphine Oxides and CO229
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Ir-Catalyzed Synthesis of Functionalized Pyrrolidines and Piperidines Using the Borrowing Hydrogen Methodology29
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Correction to “NHC-Catalyzed Aza-Benzoin Condensation of N,N′-Dipyridin-2-yl Aminals with Aldehydes”28
Rhodium(III)-Catalyzed Coupling of Quinolin-8-carboxaldehydes with CF3–Imidoyl Sulfoxonium Ylides by Chelation-Assisted C(sp2)-H Bond Activation for the Synthesis of Trifluoromet28
A Toolbox of Reagents for Trifluoromethylthiolation: From Serendipitous Findings to Rational Design28
Chiral Counteranion-Directed Catalytic Asymmetric Methylene Migration Reaction of Ene-Aldimines28
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Gram Scalable Method to Synthesize Biscarbodiimides and Asymmetric Monocarbodiimides: A Platform to Access an Array of Phosphaguanidines, Amidines, and Guanidines28
Scandium-Catalyzed Skeleton Conversion of Lathyrane to Lathyranone-Type Euphorbia Diterpenes28
Merging Imidazolidines with a Trifluoromethylated Tetrasubstituted Carbon through Tungsten Catalyzed 1,3-Dipolar Cycloaddition28
Synthesis of γ-Sultam-Annelated δ-Lactams via the Castagnoli–Cushman Reaction of Sultam-Based Dicarboxylic Acids28
Issue Publication Information28
Hybrid Catalysts for Enantioselective Photo-Phosphoric Acid Catalysis28
Rapid Enantioselective and Diastereoconvergent Hybrid Organic/Biocatalytic Entry into the Oseltamivir Core28
TEMPO-Mediated Dehydrogenative Hydroxyfluoroalkylation of Arylamines with Polyfluorinated Alcohols28
Copper-Catalyzed One-Pot Synthesis of Quinazolinones from 2-Nitrobenzaldehydes with Aldehydes: Application toward the Synthesis of Natural Products28
The Application of Benziodazole-Type O2NO-I(III) Compound as a Nitrating Reagent for Nitration of Phenols and Anilines27
Electrochemical Synthesis of 2-Amino-1,3-benzoxazines via TBAI-mediated Desulfurative Cyclization of Isothiocyanates and 2-Aminobenzyl Alcohols27
Aryne Generation from o-Triazenylarylboronic Acids Induced by 1,2-Diols and 4-Nitrophenol27
Multicomponent Reaction for Diastereoselective Synthesis of Spiro[carbazole-3,4′-pyrazoles] and Spiro[carbazole-3,4′-thiazoles]27
Approaches to Construction of the Medium-Sized Ring Structure in Zetekitoxin AB by Ring-Closing Metathesis27
Synthesis of Isoxazoles via One-Pot Oxidation/Cyclization Sequence from Propargylamines27
Synthetic Studies on Poecillastrin C: Synthesis of the C14–C35 Segment of the Macrolide Ring Model27
Direct Cross-Couplings of Aryl Nonaflates with Aryl Bromides under Nickel Catalysis27
A Photo-Smiles Rearrangement: Mechanistic Investigation of the Formation of Blatter Radical Helicenes27
Lambert Salt-Initiated Development of Friedel–Crafts Reaction on Isatin to Access Distinct Derivatives of Oxindoles27
Selectfluor-Enabled C(sp3)–H Alkoxylation of 3-Methylfuranocoumarins27
Issue Editorial Masthead27
DP4+-Based Stereochemical Reassignment and Total Synthesis of Polyenic Macrolactam Muanlactam27
Intramolecular Halogenative-Arylation of Alkynes Using N-halosuccinimide (NXS) Reagents in the CH3CN-H2O System27
Total Synthesis of Waltherione Alkaloids: A Strategic Molecular Diversity Approach27
Robust Organocatalytic Three-Component Approach to 1,3-Diarylallylidene Pyrazolones via Consecutive Double Condensation Reactions27
A Metal-Free Direct Decarboxylative Fluoroacylation of Indole Carboxylic Acids with Fluorinated Acids27
Microwave-Promoted Synthesis of 1-Tetralones via Iminyl Radical-Mediated 1,5-Hydrogen Atom Transfer27
Visible-Light-Mediated Oxidative Cyclization of 2-Aminobenzyl Alcohols and Secondary Alcohols Enabled by an Organic Photocatalyst26
3-Trifluoroacetyl-quinolin-2(1H)-ones as Carbonyl and Acid Surrogates in the Passerini-/Ugi-Type Reaction26
One-Pot Multicomponent Synthesis of Fully Substituted 1,3-Thiazoles Appended with Naturally Occurring Lawsone26
The First Highly Enantioselective Synthesis of 3-Sulfinyl-Substituted Isoindolinones Having Adjacent Carbon and Sulfur Stereocenters26
Pyramidalization of sp2 Centers26
Sc(OTf)3-Mediated [4 + 2] Annulations of N-Carbonyl Aryldiazenes with Cyclopentadiene to Construct Cinnoline Derivatives: Azo-Povarov Reaction26
Synthesis of Benzoxazines by Heterogeneous Multicomponent Biochemo Multienzymes Cascade Reaction26
Base-Promoted Cascade Reactions for the Synthesis of 3,3-Dialkylated Isoindolin-1-ones and 3-Methyleneisoindolin-1-ones26
Issue Editorial Masthead26
Stereochemical Analysis of Trifluoroacetamide Derivatives Based on Through-Space 1H19F Spin–Spin Couplings26
Isoelectronic Push–Pull Fluorescent Difluoroborates: Halogen Bonding and Photophysical Properties26
AlCl3-Promoted Intramolecular Indolinone-Quinolone Rearrangement of Spiro[indoline-3,2′-quinoxaline]-2,3′-diones: Easy Access to Quinolino[3,4-b]quinoxalin-6-ones26
Mechanistic Insight into the Photoinduced Decarboxylative Radical Addition of Carboxylic Acid to Alkenes in a Two-Molecule Photoredox System26
Electrochemical Synthesis of β-Keto Sulfones from Enol Acetates and Sulfonyl Hydrazides26
Total Synthesis of Cryptoconcatone D via Construction of 1,3-Diol Units Using Chiral Horner–Wittig Reagents26
Molecular Insights on Solvent Effects in Organic Reactions as Obtained through Computational Chemistry Tools26
C19 Benzylisoquinoline Alkaloid with Unprecedented Architecture from Hypecoum erectum26
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Two Faces of Styrylsulfonium Salts: Domino Michael Addition/Cyclopropanation of 2-(2-Acylvinyl)indoles for the Synthesis of Cyclopropa[3,4]pyrrolo[1,2-a]indoles26
Assembly of Diverse Allenes via Activator-Free Palladium-Catalyzed Regioselective γ-Arylation of Propargylamines with Boronic Acids26
Controlling the Diradical Character of Thiele Like Compounds26
Oxyphosphorodithiolation of Vinyl Azides with P4S10 and Alcohols Leading to β-Keto Phosphorodithioates26
One-Step Regioselective Synthesis of N-1-Substituted Dihydrouracils: A Motif of Growing Popularity in the Targeted Protein Degradation Field26
β-Methylation of Primary Alcohols with Methanol Catalyzed by a Metal–Ligand Bifunctional Iridium Catalyst25
Electron-Deficient CpRh(III)-Catalyzed C–H Functionalization of N-2-Pyridylanilines: Branch-Selective Alkenylation with Alkenes and Annulation with Alkynes25
One-Pot Synthesis of Substituted 2-Amino Isonicotinic Acids: Reminiscent of the Guareschi–Thorpe Condensation25
Synthesis of Substituted 2-Pyridones via 6π-Electrocyclization of Dienyl Isocyanates25
Copper-Catalyzed Synthesis of Functionalized Aryl Sulfonamides from Sodium Sulfinates in Green Solvents25
Mechanism of Iron-Catalyzed Oxidative α-Amination of Ketones with Sulfonamides25
Aymmetric Aza-Friedel–Crafts Reaction of Isatin-Derived Ketimines with Indoles Catalyzed by a Chiral Phase-Transfer Catalyst25
Surmounting Byproduct Inhibition in an Intermolecular Catalytic Asymmetric Alkene Bromoesterification Reaction as Revealed by Kinetic Profiling25
Accessing the Cloke-Wilson Rearrangement via Conjugate Addition of Phosphoranes to Michael Acceptors: A Route to Cyclopropanes and 5-Membered Ring Heterocycles Investigated by Density Functional and <25
Functionalization of 1N-Protected Tetrazoles by Deprotonation with the Turbo Grignard Reagent25
Correction to “Copper-Catalyzed Azide–Alkyne Cycloaddition of Hydrazoic Acid Formed In Situ from Sodium Azide Affords 4-Monosubstituted-1,2,3-triazoles”25
Synthesis of Chiral Tertiary Allylic- and Propargylic Fluorides from Nonaflates of Chiral α-Fluorinated β-Keto Dicarbonyl Compounds25
Silver-Catalyzed Thio-Claisen Rearrangement of Aryl Sulfoxides with AIBN24
Synthesis of Caged HMG-CoA Reductase Substrates for the Elucidation of Cellular Pathways24
Iodine-Mediated C2,3–H Aminoheteroarylation of Indoles24
Continuous Flow Inter- and Intramolecular Macrolactonization under High Dilution Conditions24
Halogen Radical-Enabled Dearomatization of N-Arylpropiolamides via Photoinduced Sequential Halogenation/Spirocyclization/Oxidation Process24
Electrosynthesis of 2-Substituted Benzoxazoles via Intramolecular Shono-Type Oxidative Coupling of Glycine Derivatives24
Organocatalytic (Z/E)-Selective Synthesis of 3-Vinylnaphthofurans via a Formal (3 + 2) Cycloaddition24
A Pyridinium Ylide-Alkylation Strategy for the Structural Diversification of N-Carbamoylpyridinium Salts24
Brønsted Acid Catalyzed Friedel–Crafts Alkylation of Naphthols with In Situ Generated Naphthol-Derived ortho-Quinone Methides: Synthesis of Chiral and Achiral Xanthene Derivatives24
In the Chalcogenoxide Elimination Panorama: Systematic Insight into a Key Reaction24
Lewis Acid-Catalyzed Remote Site-Selective Ring Deconstruction of Cyclobuteno[a]naphthalene-4-ones to Access Unsymmetric 1,1-Diarylated Olefins24
A Pummerer Reaction-Enabled Modular Synthesis of Alkyl Quinoline-3-carboxylates and 3-Arylquinolines from Amino Acids24
Co(III) or Ru(II)-Catalyzed Selective C–H Alkynylation of 2-Pyridones and Their Derivatives with Bromoalkynes24
Amidation of Enones via Beckmann Rearrangement24
Organic Base-Facilitated Thiol–Thioalkyne Reaction with Exclusive Regio- and Stereoselectivity24
Investigation of a Highly Selective Asymmetric Synthesis Strategy for cis-2-Fluorocyclopropanecarboxylic Acid: The Key Component of Sitafloxacin24
ortho-Alkynyl Benzyl Alcohols as C6 Synthons in Regioselective Construction of Polysubstituted Naphthalenes24
Synthesis of Unsymmetric Thiosulfonates Starting from N-Substituted O-Thiocarbamates: Easy Access to the S–SO2 Bond24
Palladium-Catalyzed Aminocyclization–Coupling Cascades: Preparation of Dehydrotryptophan Derivatives and Computational Study24
Synthesis of 4-O-Alkylated N-Acetylneuraminic Acid Derivatives24
Phenothiazine-, Dihydroacridine-, and Acridone-Based Boron Difluoride Complexes: Synthesis and Structure–Property Relationships24
Catalyst-Free α-Allylation of Dihydroisoquinolines with Morita–Baylis–Hillman Carbonates and Its Applications in the Construction of Benzo[a]quinolizidines24
Application of β-Keto Acylpyrazoles as 2C Synthons in Asymmetric Cyclizations of ortho-Hydroxychalcones: Stereoselective Construction of trans-3,4-Dihydrocoumarins24
Synthesis of Spiro[furan-2,1′-isoindolin]-3′-ones from 2-(4-Hydroxybut-1-yn-1-yl)benzonitriles and Aryl Aldehydes under the Action of Triflic Acid23
Theoretical Insight into the Multiple Roles of the Silyl-Phenanthroline Ligand in Ir-Catalyzed C(sp3)–H Borylation23
Specific Noncovalent Association of Truncated exo-Functionalized Triangular Homochiral Isotrianglimines through Head-to-Head, Tail-to-Tail, and Honeycomb Supramolecular Motifs23
Electrophilic Reagents for the Direct Incorporation of Uncommon SCF2CF2H and SCF2CF3 Motifs23
Umpolung of N-Tosylhydrazones: Synthesis of N-Cyano Tosylhydrazones and Their [3,3]-Sigmatropic Rearrangement to 2-Aminoimidazoles23
Two Squares in a Barrel: An Axially Disubstituted Conformationally Rigid Aliphatic Binding Motif for Cucurbit[6]uril23
Cholinium Pyridinolate Ionic Pair-Catalyzed Fixation of CO2 into Cyclic Carbonates23
Can Side-Chain Conformation and Glycosylation Selectivity of Hexopyranosyl Donors Be Controlled with a Dummy Ligand?23
Electrochemical Oxidative 1,2-Dithiocyanation: Access to Functionalized Alkenes and Alkynes23
Water-Based Solid-Phase Peptide Synthesis without Hydroxy Side Chain Protection23
Pd-Catalyzed [2 + 2 + 2] Cyclization of Alkyne-cyclohexadienones and O-Akynyl Benzenesulfonamides for Construction of Fused Tricyclic Hydronaphthofurans23
Mechanistic Insights into Visible-Light-Driven Dearomative Fluoroalkylation Mediated by an Electron Donor–Acceptor Complex23
Synthesis of α-Tropolones through Autoxidation of Dioxole-Fused Cycloheptatrienes23
Catalytic Role of Methanol in Anodic Coupling Reactions Involving Alcohol Trapping of Cation Radicals23
Zn(OTf)2-Promoted Isocyanide-Based Three-Component Reaction: Direct Access to 2-Oxazolines and β-Amino Amides23
Asymmetric Catalytic Access to Piperazin-2-ones and Morpholin-2-ones in a One-Pot Approach: Rapid Synthesis of an Intermediate to Aprepitant23
Aryl/Heteroaryl Substituted Boron-Difluoride Complexes Bearing 2-(Isoquinol-1-yl)pyrrole Ligands Exhibiting High Luminescence Efficiency with a Large Stokes Shift23
DBU-Mediated Domino Annulation Reaction of 2-Amino-4H-chromen-4-ones and Aromatic Aldehydes for Synthesis of Polysubstituted 3-Hydroxy-5H-chromeno[2,3-b]pyridinones23
Isothiouronium-Mediated Conversion of Carboxylic Acids to Cyanomethyl Thioesters23
Tailoring the Energetic Properties of Pyrazole Hybrids through Functionalization with Dinitromethyl and N-Hydroxytetrazole23
Azobis(polynitrophenyl-1,2,5-oxadiazoles) as Heat-Resistant Friction-Insensitive Energetic Materials23
Rapid Synthesis of Luotonin A Derivatives via Synergistic Visible-Light Photoredox and Acid Catalysis23
Stereocontrolled Synthesis of C20S-C26 and C20R-C26 Fragments of Amphidinolide L23
Copper-Catalyzed [4+1+1] Annulation of Ammonium Salts and Anthranils: Synthesis of 2,3-Diaroylquinolines23
Unveiling the Selectivity of Ru(II)-Catalyzed C–H Activation for Defluorinative Cyclization of 2-Arylbenzimidazole and Trifluoromethyl Diazo: A DFT Study23
[4 + 2] Annulation of δ-Hydroxy/δ-Sulfonamido-α,β-Unsaturated Ketones with Azlactones for Diastereoselective Synthesis of Highly Substituted 3-Amino-δ-Lactones and 3-Amino-δ-Lactams23
Direct Synthesis of Fluorescent Oxazolo-phenoxazines by Copper-Catalyzed/Hypervalent Iodine(III)-Mediated Dimerization/Cyclization of 2-Benzylamino-phenols23
Tandem Dearomative/Rearomative (3 + 2) Annulation of Aroyl-Substituted Donor–Acceptor Cyclopropanes with Benzothiazoles23
Au-Catalyzed 5C Reaction of Type II Diene-Ynenes toward Dihydrosemibullvalenes: Reaction Development and Mechanistic Study23
Iodine-Catalyzed Annulation Reaction of Ortho-Formylarylketones with Indoles: A General Strategy for the Synthesis of Indolylbenzo[b]carbazoles23
Highly Regioselective Tandem Reaction of Ene-Yne-Oxazolones Induced by H-Phosphonates: Construction of Phosphinylindane Derivatives22
Direct Construction of 1,4-Dihydropyridazines and Pyrazoles via Annulation of Alkyl 2-Aroyl-1-chlorocyclopropanecarboxylates22
Annulation of Enals with Carbamoylpropiolates via NHC-Catalyzed Enolate Pathway: Access to Functionalized Maleimides/Iso-maleimides and Synthesis of Aspergillus FH-X-21322
TiO2-Catalyzed Direct Diazenylation of Active Methylene Compounds with Diazonium Salts22
Hydrogenation of Sugar Enol-Ethers Using Pd/Et3SiH Reagent System: A Route to Deoxy Sugars/Glycosides22
Alkali Metal Fluorides in Fluorinated Alcohols: Fundamental Properties and Applications to Electrochemical Fluorination22
Photoinduced Etherification of Less-Strained Cycloketoxime Esters Enabled by C–C Bond Cleavage22
Regioselective Coupling of Different Conjugate Esters by Magnesium Metal Reduction: A Route to Unsymmetrical Adipic Acid Esters22
Electrophotocatalytic Thiocyanation and Sulfonylation Cyclization of Unactivated Alkenes22
Computational Determination of the Mechanism of the Palladium-Catalyzed Domino Reaction of ortho-Iodostyrene, Oxanorbornadiene, and Phenylboronic Acid22
Stereoselective Domino Rearrangement peri-Annulation of Cinchona Alkaloid Derivatives with 8-Bromo-1-naphthyl Grignard22
Hybrid Palladium-Catalyzed Intramolecular Carboamination of Conjugated Dienes: Synthesis of Functionalized Pyrrolidines via Selective Trifluoromethylarene Defluorination22
A One-Pot Synthesis-Functionalization Strategy for Streamlined Access to 2,5-Disubstituted 1,3,4-Oxadiazoles from Carboxylic Acids22
Photoredox Ring Opening 1,2-Alkylarylation of Alkenes with Sulfonium Salts Toward Thioether-Substituted Oxindoles22
Divergent Protocol for the Synthesis of Isoquinolino[1,2-b]quinazolinone and Isoquinolino[2,1-a]quinazolinone Derivatives22
Palladium-Catalyzed Domino Carboetherification Reactions: Synthesis of Bis-Heterocycles Bearing Isoxazoline and Methyleneindole Motifs22
Enabling, Decagram-Scale Synthesis of Macrocyclic MCL-1 Inhibitor ABBV-46722
TMSN3 Initiated Electrochemical Mono-Dealkylation of Tertiary Amides22
3,6,13,16-Tetrapropylporphycene: Rational Synthesis, Complexation, and Halogenation22
Synthesis and Chiroptical Properties of a Chiral Isotopologue of syn-Cryptophane-B22
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