Journal of Labelled Compounds & Radiopharmaceuticals

Article	Citations
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A flow electrochemistry‐enabled synthesis of 2‐substituted N‐(methyl‐d)piperidines	31
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Automated radiolabeling and handling of 177Lu‐ and 225Ac‐PSMA‐617 using a robotic pipettor	10
Radiosynthesis and Evaluation of [18F]FEHSP990 as Novel PET Tracer for Hsp90 PET Imaging	8
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Applications of radiolabeled antibodies in neuroscience and neuro‐oncology	7
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Influence of Activated Carbon on Fate of 14C‐Sulfamethoxazole and 14C‐Acetaminophen in Soil	6
Fully Automated Radiosynthesis of No‐Carrier‐Added [11C]Butanol Using the GE FASTLab 2 Module	6
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Small‐scale two‐dimensional liquid chromatography for a preparative re‐purification of a highly labile tritium‐labeled compound	6
Synthesis of One Carbon‐14 Labelled [ 14 C‐ pyrazolo ]‐Ibrutinib	5
Synthesis and Preclinical Evaluation of 99 ᵐTc‐HYNIC–Finasteride: A Novel SPECT Radiotracer Targeting 5α‐Reductase in Prostate Cancer	5
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Luminescence enhancement by deuterium	5
Synthesis of BI 1584142 and BI 1810631 (Zongertinib), Two Potent HER2 Inhibitors, Labeled With Carbon‐14 and With Deuterium	4
Development of a Fully Automated FASTlab 2 Process for [ 18 F]AlF Radiolabelling of NOTA Peptide Conjugates	4
Synthesis and Characterization of 3‐Hydroxybupivacaine and Deuterated 3‐Hydroxybupivacaine for Use in Equine Medication Regulation	4
Synthesis of Psilocin, Psilocybin and 5‐MeO‐DMT Succinate, All Labelled With Carbon‐14 at the Indole 2‐Position	4

Synthesis of Carbon 14 and Deuterium‐Labelled Nerandomilast (BI 1015550)	4
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Fully Automated Cassette‐Based Synthesis of 2‐Deoxy‐2‐[18F]Fluorocellobiose Using Trasis AllInOne Module	4
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Preliminary Research of Radiolabeled Atezolizumab for the Noninvasive Evaluation of TNBC PD‐L1 Expression In Vivo	3
11C‐Carbonylation for PET Imaging and Drug Discovery	3
Carbon‐14 Labeling Synthesis of RORγt Inhibitor JNJ‐61803534	3
Simplified and accessible [18F]F‐AraG synthesis procedure for preclinical PET	3
Tritium and deuterium labelling of a kainate receptor antagonist and evaluation as a radioligand	3
Application of Microfluidic Devices for Automated Two‐Step Radiolabeling of Antibodies	3
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68Ga Radiolabeling of NODASA‐Functionalized Phage Display–Derived Peptides for Prospective Assessment as Tuberculosis‐Specific PET Radiotracers	3
Carbon 14 and stable isotope synthesis of two potent and selective phosphodiesterase type 4 inhibitors	3
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[18F]Fluoropyridine‐losartan: A new approach toward human Positron Emission Tomography imaging of Angiotensin II Type 1 receptors	2
14C‐radiolabeling of a new steroidal antiandrogen with a C‐18 angular methyl extension	2
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Synthesis and Evaluation of Radioiodinated [ 125 I]7‐Iodo‐5H‐Pyrido[4,3‐B]Indole ([ 125 I]CTAU) in	2
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Ultrasound‐Assisted Microcontinuous Process Facilitates the Selective Deuteration of Steroid Hormones	2
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Abstracts From the 30th International Isotope Society UK Meeting 15th November 2024	2
Photocatalyzed radiosynthesis of 11C‐phenylacetic acids	2
Synthesis of BI 894416 and BI 1342561, two potent and selective spleen tyrosine kinase inhibitors, labeled with carbon 14 and with deuterium	2
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RO6807936 as a novel positron emission tomography (PET) radiotracer for in vitro and in vivo visualization and quantification of beta‐site amyloid precursor protein cleaving enzyme (BACE1) in the rode	2
Nitrilase mediated mild hydrolysis of a carbon‐14 nitrile for the radiosynthesis of 4‐(7‐hydroxycarbamoyl‐[1‐14C‐heptanoyl]‐oxy)‐benzoic acid methyl ester, [14C]‐SHP‐141: A novel	2
Targeting VEGF With 99mTc‐Labeled Ranibizumab for Noninvasive Diagnosis of Non‐Small Cell Lung Cancer	2
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Improving Routine 89Zr‐Immuno‐PET Applications: Mild Iron Removal Can Favor the Use of Fe‐DFO‐N‐suc‐TFP Ester Over p‐NCS‐Bz‐DFO	2
Low‐scale syringe‐made synthesis of 15N‐labeled oligonucleotides	2
Total synthesis of [13C2]‐labeled phytosiderophores of the mugineic and avenic acid families	2
Synthesis of Two Versions of Carbon‐14‐Labeled ARV‐110: An Androgen Receptor PROTAC Degrader for Prostate Cancer	2
Automated radiosynthesis of [18F]CETO, a PET radiotracer for imaging adrenal glands, on Synthra RNplus	2
Fully Automated Cassette‐Based Production of [18F]Albumin Using the Trasis AllinOne Module	2
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Synthesis and spectroscopic characterization of 13C4‐labeled 4‐cyano‐2‐oxobutyraldehyde semicarbazone: A metabolite of nitrofurazone	2
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Synthesis of trifold‐labeled versatile reagent [3,5‐13C2,4‐15 N]4‐phenyl‐1,2,4‐triazoline‐3,5‐dione	1
Synthesis and preclinical evaluation of a selective MET kinase positron emission tomography tracer	1
Thank You, Bob!	1
Synthesis and Characterization of Deuterated Detomidine for Use in Equine Medication Regulation	1
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Automated radiosynthesis of mGluR5 PET tracer [18F]FPEB from aryl‐chloro precursor and validation for clinical application	1
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RETRACTION: Enhanced Control of Bacterial Wilt Disease in Tomato Plant via Transport and Penetration Tracking by Aid of 99m Tc‐Labeled	1
Formulation of patient dose of [177Lu]Lu‐Trastuzumab using in‐house developed freeze‐dried kit: A path forward for clinical translation	1
The impact of zirconium‐89 solution formulation on the efficiency of [89Zr]Zr‐deferoxamine synthesis	1

Synthesis and Imaging of Novel CDK19‐Targeted Tracers Incorporating an Albumin‐Binding Moiety	1
Carbon 14 synthesis of glycine transporter 1 inhibitor Iclepertin (BI 425809) and its major metabolites	1
Synthesis of Potent Vanin‐1 Inhibitors Labelled With Carbon‐14 and Deuterium	1
Development of a high‐performance liquid chromatography method for rapid radiochemical purity measurement of [18F]PSMA‐1007, a PET radiopharmaceutical for detection of prostate cancer	1
Radiolabeling of Trastuzumab With Technetium‐99m [99mTc] as a Radioligand for Screening Mentha pulegium	1
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Synthesis of 14C‐Labeled Polyethylene Terephthalate and Generation of 14C‐Nanoparticles for Fate and Disposition Studies	1
[11C]CO2 BOP fixation with amines to access 11C‐labeled ureas for PET imaging	1
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An improved synthesis of [18F]VAT and its precursor	1
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Radiolabeled Aptamers for Bioimaging Applications in Oncology and Infectious Diseases	1
The inverse electron demand Diels–Alder cycloaddition with carbon‐11 and fluorine‐18: A gateway to pretargeted imaging across the blood–brain barrier	1
Good manufacturing procedure production of [18F]SynVesT‐1, a radioligand for in vivo positron emission tomography imaging of synaptic vesicle glycoprotein 2A	1
Lead‐212/Bismuth‐212 In Vivo Generator Based on Ultrasmall Silver Telluride Nanoparticles	1
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Synthesis and Preclinical Evaluation of Peptide Dimer‐Based PET Tracers for Imaging VEGFR‐2 Expression in Tumors	1
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Hypoxia Inducible Factor‐1α Specific Probe for Tumor Hypoxia Positron Emission Tomography Imaging	1
Assessment of Stability Extrapolation for Carbon‐14 Labelled Compounds for the Determination of Extended Retest Periods	1
Preparation of Macrobicyclic Cryptands for Radiometal Complexation	1
Next Generation of Solid Target Radionuclide Antibody Conjugates for Tumor Immuno‐Therapy	1
Automated radiosynthesis of 1‐(2‐[18F]fluoroethyl)‐L‐tryptophan ([18F]FETrp) for positron emission tomography (PET) imaging of cancer in humans	0
RETRACTED: Enhanced Control of Bacterial Wilt Disease in Tomato Plant via Transport and Penetration Tracking by Aid of 99m Tc‐Labeled	0
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Automated Radiosynthesis of [18F]FMeNER‐D2 Using the Simplified One‐Pot 18F‐Fluoromethylation Method	0
An optimized radiosynthesis of [18F]DK222, a PET radiotracer for imaging PD‐L1	0
Synthesis of 18F‐Labeled FC‐119S and Its Tosyl Precursor	0
Carbon 14 and Carbon 13 Syntheses of Velagliflozin	0
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A practical approach to the optimization of positron emission tomography imaging agents for the central nervous system	0
Open‐source flow setup for rapid and efficient [18F]fluoride drying for automation of PET tracer syntheses	0
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A 64 Cu‐Labeled Oxopurine Derivative for Translocator Protein–Targeted Inflammation Imaging	0
Validation of a good manufacturing practice procedure for the production of [ 11 C]AZD4747, a CNS penetrant KRAS G12c	0
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Correction to Validation of a Good Manufacturing Practice Procedure for the Production of [ 11 C]A	0
Preparation, Characterization, and Radiolabeling of Anti‐HER2 scFv With Technetium Tricarbonyl and Stability Studies	0
Detailed radiosynthesis of [18F]mG4P027 as a positron emission tomography radiotracer for mGluR4	0
Improved Radiosynthesis and Automation of [11C]2‐(2,6‐Difluoro‐4‐((2‐(N‐methylphenylsulfonamido)ethyl)thio)phenoxy)acetamide ([11C]K2) for Positron Emission Tomography of	0
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Direct Multi‐Deuterium Labelling of Pirtobrutinib	0
Development of 11C‐labeled CRANAD‐102 for positron emission tomography imaging of soluble Aβ‐species	0
Abstracts From the 31st International Isotope Society UK Meeting 14th November 2025	0
99mTc‐SNW‐1 Nanoparticle Labeling and Its Biodistribution/Pathological Evaluations	0
25 Years of “Loop” Radiochemistry for PET Imaging	0
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Enzymatic synthesis of halogen derivatives of L‐phenylalanine and phenylpyruvic acid stereoselectively labeled with hydrogen isotopes in the side chain	0
Synthesis, Preclinical Characterizations and Imaging Studies of [18F]AlF‐Labeled NY104, a CAIX‐Targeting Diagnostic Agent	0
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Development and Validation of an HPLC Method to Determine Chemical and Radiochemical Purity of [18F]Florbetazine Injection	0
Development of radiotracers for riboflavin transporter 3 imaging in diseases—A brief overview	0
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A practical and environmentally friendly protocol for synthesis of α‐deuterated carboxylic acids	0
Design and Synthesis of a 18F‐Radiolabeled Pyrrolo[2,3‐d]pyrimidine Ligand as a CSF1R Receptor PET Imaging Agent	0
Dosimetric Development of Yttrium‐90 Resin Microspheres for Selective Internal Radiation Therapy: Current Status and Perspectives	0
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Synthesis of Florasulam Stable Isotopes to Enable Identification of Degradants by Mass Spectrometry for Re‐registration Studies	0
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A Novel 68Ga‐Labeled 2‐Azabicyclo[3.1.0]Hexane‐3‐Carbonitrile‐Based Fibroblast Activation Protein‐Targeted Tracer for Cancer Imaging With Positron Emission Tomography	0
Preliminary PET imaging of [11C]evobrutinib in mouse models of colorectal cancer, SARS‐CoV‐2, and lung damage: Radiosynthesis via base‐aided palladium‐NiXantphos‐mediated 11C‐car	0
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Preparation of [1′‐13C]citric acid as a probe in a breath test to evaluate tricarboxylic acid cycle flux	0
Abstracts From the 29th International Isotope Society UK Meeting 17th November 2023	0
Improved protocol for the radiosynthesis of [18F]FTC‐146: A potent and selective sigma‐1 receptor radioligand	0
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Antibody Drug Conjugate Formation Using 2‐ 14 C‐Iminothiolane: A Radiochemical Analysis of Sequential Lysine Conjugation, Uncloaking of a Phantom Dru	0
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C14‐Labelled Synthesis of Benalaxyl‐M and Its Two Soil Metabolites	0
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Towards Optimal Automated 68Ga‐Radiolabeling Conditions of the DOTA‐Bisphosphonate BPAMD Without Pre‐Purification of the Generator Eluate	0
Site‐specifically radiolabeled nanobodies for imaging blood‐brain barrier penetration and targeting in the brain	0

An improved radiosynthesis of [18F]FAraG, a PET radiotracer for imaging T‐cell activation	0
Synthesis and Characterization of 2‐Thiophenemethanamine‐ 2 H 5 Hydrochloride	0
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Synthesis and Evaluation of a Cathepsin B–Recognizing Trifunctional Chelating Agent to Improve Tumor Retention of Radioimmunoconjugates	0
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Evaluation and improvement of CuI‐mediated 11C‐cyanation	0
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Synthesis and Preclinical Evaluation of [18F]AlF‐NOTA‐Asp2‐PEG2‐Folate as a Novel Folate‐Receptor‐Targeted Tracer for PET Imaging	0
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Synthesis and Preliminary Evaluation of an In Vivo Stable 131I‐Labeled Deuterated Tropane for Mapping Dopamine Transporter	0
Automated Manufacturing of Carbon‐11 Radiopharmaceuticals Using Cassette‐Based Radiosynthesizers	0
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In vivo and in vitro binding of [125I]I‐R‐(+)‐TISCH: A dopamine D1 receptor ligand for studying pancreatic β‐cell mass	0
Highly effective liquid and solid phase extraction methods to concentrate radioiodine isotopes for radioiodination chemistry	0
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Preparation and evaluation of radiolabeled acetaminosalol microspheres: A new potential selective radiotracer for ulcerative colitis early diagnosis	0
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Evaluation of New‐Modelled Recombinant Human Insulin (rh‐Insulin) Analog Expressed in E. coli Using Radioiodination Technique Followed by In Vivo Biodistribution in Diabetes‐Induced Mice	0
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Peptides for trans‐blood–brain barrier delivery	0
A simplified protocol for the automated production of 2‐[18F]fluoro‐3‐[2‐((S)‐3‐pyrrolinyl)methoxy]pyridine ([18F]nifene) on an IBA Synthera® module	0
Current Advances in PARP1‐Targeted Theranostics	0
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A practical protocol for large‐scale copper‐mediated radioiodination of organoboronic precursors: Radiosynthesis of [123I]KX‐1 for Auger radiotherapy	0
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Synthesis of Radiolabeled and Stable‐Isotope Labeled Deucravacitinib (BMS‐986165)	0
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Carbon‐13 labeling of ibrutinib for human microdosing	0
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Synthesis of Deuterated Endochin‐Like Quinolones	0
Radiotheranostics With Nanoparticles: Precision Targeting in Receptor‐Overexpressing Tumors	0
Automated Radiolabeling and Evaluation of [18F]FPMBBG: A Novel Cardiac Neuronal PET Imaging Agent	0
Synthesis of [3H]Org24598 using in‐house prepared [3H]MeI	0
A facile synthesis of precursor for the σ‐1 receptor PET radioligand [18F]FTC‐146 and its radiofluorination	0
Synthesis of Radiolabeled [14C]Rimsulfuron and Stable Isotope Labeled Rimsulfuron‐[M + 3] to Support Crop Metabolism Studies for Reregistration	0
Preclinical Evaluation of [ 225 Ac]Ac–Sibrotuzumab Employing a PEG 4 –Macropa Site‐Specific Chelat	0
Efficient synthesis of carbon‐14 labeled metabolites of the strobilurin fungicide mandestrobin using biomimetic iron‐porphyrin catalyzed oxidation	0
A practical approach to the optimization of positron emission tomography imaging agents for the central nervous system	0
Synthesis and evaluation of 111In‐labeled tetrapeptide‐based compounds as single‐photon emission computed tomography imaging probes targeting granzyme B	0
[68Ga]Ga‐PentixaFor: Development of a fully automated in hospital production on the Trasis miniAllinOne synthesizer	0
Facile synthesis of 14C‐nitrofurazone from 14C‐urea	0
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Synthesis and analysis of isotopically stable labeled nitrosamines as mass spectrometry standards for drug impurity quality control	0
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Simplified Flow Photosynthesis of Deuterium‐Labeled Pyocyanin	0
Benzylic deuteration of alkylnitroaromatics via amine‐base catalysed exchange with deuterium oxide	0
Fully Automated Production of Multiple 11 C‐Labeled PET Tracers Using a Self‐Cleaning TracerMaker Radiosynthesizer	0
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Development and physicochemical characterization of a biodegradable microspheres formulation loaded with samarium‐153 and doxorubicin for chemo‐radioembolization of liver tumours	0
Practitioner Protocol for the Photoreduction of [ 14 C]CO 2 to [ 14	0
Development of an economical method to synthesize O‐(2‐[18F]fluoroethyl)‐L‐tyrosine (18FFET)	0
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18F‐Fluorination of a supported 2‐(aryl‐di‐tert‐butylsilyl)‐N‐methyl‐imidazole for indirect 18F‐labeling of a VHH single‐variable domain	0
Wiley Young Scientist Awards were handed over at the 14th International Symposium on the synthesis on the Synthesis and Applications of Isotopically Labelled Compounds in Raleigh, USA	0
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Synthesis and Application of D‐ and 13C‐Labelled tert‐Butyl Hoechst Dye	0
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Synthesis of Stable Isotope, Tritiated, and Carbon‐14 Labeled Balcinrenone	0
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Radiosynthesis and validation of [18F]fluoroestradiol in a Synthra plus research platform for use in routine clinical practice	0
The synthesis of deuteriated tri‐tert‐butyl phosphine	0
Highly selective catalytic transfer hydrodeuteration of cyclic alkenes	0
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Synthesis of Carbon‐13 and Carbon‐14 Labeled BI 690517 (Vicadrostat) and Its O ‐Glucuronide Metabolite BI 689875	0
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Stable isotope synthesis of glycine transporter 1 inhibitor Iclepertin (BI 425809) and its major metabolites	0
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An Improved HPLC Separation Method for TSPO Radioligand [11C]ER176 Clinical Production	0
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Applications of Isotopes in Forensic Science	0
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Synthesis, Radiochemical Characterization, and Biodistribution of a 188 Re Analogue of [ 131 I]mIB	0
Strategies for designing novel positron emission tomography (PET) radiotracers to cross the blood–brain barrier	0
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Synthesis of a Potent Bruton's Tyrosine Kinase Inhibitor Labelled With Carbon‐14 and Deuterium	0
Mild and selective hydrogen–deuterium exchange for aromatic hydrogen of amines	0
Synthesis of beta‐site amyloid precursor protein‐cleaving enzyme 1 inhibitors BI 1147560 and BI 1181181 labeled with carbon‐14 and deuterium	0
Imidazolium‐methylene‐trifluoroborate: A novel radioprosthetic group validated with preclinical 18F‐Positron Emission Tomography imaging of Prostate Specific Membrane Antigen in mice	0
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Recent Advances in 11 C‐Labeling With [ 11 C]CO 2	0
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A Brief Review of Radiolabelling Nucleic Acid‐Based Molecules for Tracking and Monitoring	0
Blood Brain Barrier – tactics and attributes in developing successful neuroimaging agents	0
Efficient Reductive N‐11C‐Methylation Using Arylamines or Alkylamines and In Situ–Generated [11C]Formaldehyde From [11C]Methyl Iodide	0
Novel synthesis of 11C‐labeled imidazolines via Pd(0)‐mediated 11C‐carbomethoxylation using [11C]CO and arylborons	0
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Synthesis of [3H]muscimol	0
Radioiodination, purification, and evaluation of antihuman tumor‐derived immunoglobulin G light chain monoclonal antibody in tumor‐bearing nude mice	0
Synthesis and radiolabeling of a polar [125I]I‐1,2,4,5‐tetrazine	0