Journal of Labelled Compounds & Radiopharmaceuticals

Article	Citations
Issue Information	19
Issue Information	17
	17
A flow electrochemistry‐enabled synthesis of 2‐substituted N‐(methyl‐d)piperidines	9
Automated radiolabeling and handling of 177Lu‐ and 225Ac‐PSMA‐617 using a robotic pipettor	9
Issue Information	9
Issue Information	8
	8
	6
Applications of radiolabeled antibodies in neuroscience and neuro‐oncology	6
Influence of Activated Carbon on Fate of 14C‐Sulfamethoxazole and 14C‐Acetaminophen in Soil	6
	5
	5
Fully Automated Radiosynthesis of No‐Carrier‐Added [11C]Butanol Using the GE FASTLab 2 Module	4
	4
	4
Small‐scale two‐dimensional liquid chromatography for a preparative re‐purification of a highly labile tritium‐labeled compound	4
Issue Information	4
Radiosynthesis and Evaluation of [18F]FEHSP990 as Novel PET Tracer for Hsp90 PET Imaging	4
Luminescence enhancement by deuterium	3
Synthesis of BI 1584142 and BI 1810631 (Zongertinib), Two Potent HER2 Inhibitors, Labeled With Carbon‐14 and With Deuterium	3
Synthesis of Psilocin, Psilocybin and 5‐MeO‐DMT Succinate, All Labelled With Carbon‐14 at the Indole 2‐Position	3
Synthesis and Characterization of 3‐Hydroxybupivacaine and Deuterated 3‐Hydroxybupivacaine for Use in Equine Medication Regulation	3
	3
Synthesis and Preclinical Evaluation of 99 ᵐTc‐HYNIC–Finasteride: A Novel SPECT Radiotracer Targeting 5α‐Reductase in Prostate Cancer	3

Issue Information	3
Synthesis of Carbon 14 and Deuterium‐Labelled Nerandomilast (BI 1015550)	3
Carbon‐14 Labeling Synthesis of RORγt Inhibitor JNJ‐61803534	3
Issue Information	3
Fully Automated Cassette‐Based Synthesis of 2‐Deoxy‐2‐[18F]Fluorocellobiose Using Trasis AllInOne Module	3
Synthesis of One Carbon‐14 Labelled [ 14 C‐ pyrazolo ]‐Ibrutinib	3
Issue Information	3
68Ga Radiolabeling of NODASA‐Functionalized Phage Display–Derived Peptides for Prospective Assessment as Tuberculosis‐Specific PET Radiotracers	3
Issue Information	3
	2
Novel developed HPLC analyses of [68Ga]Ga/[177Lu]Lu‐EDTMP and [68Ga]Ga/[177Lu]Lu‐DOTA‐Zoledronate	2
Application of Microfluidic Devices for Automated Two‐Step Radiolabeling of Antibodies	2
	2
Carbon 14 and stable isotope synthesis of two potent and selective phosphodiesterase type 4 inhibitors	2
Initial evaluation of 99mTc‐labeled anti‐carcinoembryonic antigen single‐chain fragment variable for micro‐single‐photon emission computed tomography imaging in mice with colorectal cancer	2
Issue Information	2
Photocatalyzed radiosynthesis of 11C‐phenylacetic acids	2
Automated radiosynthesis of [18F]CETO, a PET radiotracer for imaging adrenal glands, on Synthra RNplus	2
Total synthesis of [13C2]‐labeled phytosiderophores of the mugineic and avenic acid families	2
Tritium and deuterium labelling of a kainate receptor antagonist and evaluation as a radioligand	2
Preliminary Research of Radiolabeled Atezolizumab for the Noninvasive Evaluation of TNBC PD‐L1 Expression In Vivo	2
11C‐Carbonylation for PET Imaging and Drug Discovery	2
Low‐scale syringe‐made synthesis of 15N‐labeled oligonucleotides	2
Issue Information	2
	2
RO6807936 as a novel positron emission tomography (PET) radiotracer for in vitro and in vivo visualization and quantification of beta‐site amyloid precursor protein cleaving enzyme (BACE1) in the rode	2
Issue Information	2
Synthesis of Two Versions of Carbon‐14‐Labeled ARV‐110: An Androgen Receptor PROTAC Degrader for Prostate Cancer	2
Simplified and accessible [18F]F‐AraG synthesis procedure for preclinical PET	2
	2
14C‐radiolabeling of a new steroidal antiandrogen with a C‐18 angular methyl extension	2
Nitrilase mediated mild hydrolysis of a carbon‐14 nitrile for the radiosynthesis of 4‐(7‐hydroxycarbamoyl‐[1‐14C‐heptanoyl]‐oxy)‐benzoic acid methyl ester, [14C]‐SHP‐141: A novel	2
Synthesis of BI 894416 and BI 1342561, two potent and selective spleen tyrosine kinase inhibitors, labeled with carbon 14 and with deuterium	2
[18F]Fluoropyridine‐losartan: A new approach toward human Positron Emission Tomography imaging of Angiotensin II Type 1 receptors	2
Issue Information	1
	1
Good manufacturing procedure production of [18F]SynVesT‐1, a radioligand for in vivo positron emission tomography imaging of synaptic vesicle glycoprotein 2A	1
	1
Issue Information	1
Targeting VEGF With 99mTc‐Labeled Ranibizumab for Noninvasive Diagnosis of Non‐Small Cell Lung Cancer	1
Improving Routine 89Zr‐Immuno‐PET Applications: Mild Iron Removal Can Favor the Use of Fe‐DFO‐N‐suc‐TFP Ester Over p‐NCS‐Bz‐DFO	1
Ultrasound‐Assisted Microcontinuous Process Facilitates the Selective Deuteration of Steroid Hormones	1
Automated radiochemical synthesis of pharmaceutical grade [18F]FLT using 3‐N‐Boc‐5′‐O‐dimethoxytrityl‐3′‐O‐nosyl‐thymidine precursor and its Sep‐Pak® purification employing selective elutio	1
Next Generation of Solid Target Radionuclide Antibody Conjugates for Tumor Immuno‐Therapy	1
Preparation of Macrobicyclic Cryptands for Radiometal Complexation	1
Issue Information	1
Synthesis of trifold‐labeled versatile reagent [3,5‐13C2,4‐15 N]4‐phenyl‐1,2,4‐triazoline‐3,5‐dione	1
Issue Information	1
Thank You, Bob!	1
	1

Formulation of patient dose of [177Lu]Lu‐Trastuzumab using in‐house developed freeze‐dried kit: A path forward for clinical translation	1
	1
Synthesis and spectroscopic characterization of 13C4‐labeled 4‐cyano‐2‐oxobutyraldehyde semicarbazone: A metabolite of nitrofurazone	1
High‐yielding, automated radiosynthesis of [11C]martinostat using [11C]methyl triflate	1
Lead‐212/Bismuth‐212 In Vivo Generator Based on Ultrasmall Silver Telluride Nanoparticles	1
Automated synthesis of (R)‐[18F]MH.MZ on the iPhase Flexlab reaction platform	1
Development of a high‐performance liquid chromatography method for rapid radiochemical purity measurement of [18F]PSMA‐1007, a PET radiopharmaceutical for detection of prostate cancer	1
Synthesis of 14C‐Labeled Polyethylene Terephthalate and Generation of 14C‐Nanoparticles for Fate and Disposition Studies	1
Synthesis and Preclinical Evaluation of Peptide Dimer‐Based PET Tracers for Imaging VEGFR‐2 Expression in Tumors	1
Synthesis and preclinical evaluation of a selective MET kinase positron emission tomography tracer	1
	1
Issue Information	1
Hypoxia Inducible Factor‐1α Specific Probe for Tumor Hypoxia Positron Emission Tomography Imaging	1
Fully Automated Cassette‐Based Production of [18F]Albumin Using the Trasis AllinOne Module	1
Issue Information	1
	1
Determination of isotope abundance for deuterium‐labeled compounds by quantitative 1H NMR + 2H NMR	1
The inverse electron demand Diels–Alder cycloaddition with carbon‐11 and fluorine‐18: A gateway to pretargeted imaging across the blood–brain barrier	1
Issue Information	1
Automated radiosynthesis of mGluR5 PET tracer [18F]FPEB from aryl‐chloro precursor and validation for clinical application	1
Practical approaches to labelling terminal alkynes with deuterium	1
Issue Information	0
Correction to Validation of a Good Manufacturing Practice Procedure for the Production of [11C]AZD4747, a CNS Penetrant KRASG12c Inhibitor	0
	0
Synthesis of N‐acetyl‐l‐aspartyl‐l‐glutamic acid; [3H]NAAG	0
Peptides for trans‐blood–brain barrier delivery	0
Design and Synthesis of a 18F‐Radiolabeled Pyrrolo[2,3‐d]pyrimidine Ligand as a CSF1R Receptor PET Imaging Agent	0
Issue Information	0
	0
Synthesis of a dual carbon‐14‐labeled calcitonin gene‐related peptide receptor antagonist for use in a human absorption–distribution–metabolism–elimination study	0
Mild and selective hydrogen–deuterium exchange for aromatic hydrogen of amines	0
	0
Strategies for designing novel positron emission tomography (PET) radiotracers to cross the blood–brain barrier	0
Carbon 14 synthesis of glycine transporter 1 inhibitor Iclepertin (BI 425809) and its major metabolites	0
Preliminary PET imaging of [11C]evobrutinib in mouse models of colorectal cancer, SARS‐CoV‐2, and lung damage: Radiosynthesis via base‐aided palladium‐NiXantphos‐mediated 11C‐car	0
Issue Information	0
Novel synthesis of 11C‐labeled imidazolines via Pd(0)‐mediated 11C‐carbomethoxylation using [11C]CO and arylborons	0
The impact of zirconium‐89 solution formulation on the efficiency of [89Zr]Zr‐deferoxamine synthesis	0
Improved protocol for the radiosynthesis of [18F]FTC‐146: A potent and selective sigma‐1 receptor radioligand	0
Automated Manufacturing of Carbon‐11 Radiopharmaceuticals Using Cassette‐Based Radiosynthesizers	0
Recent Advances in 11 C‐Labeling With [ 11 C]CO 2	0
Development of an economical method to synthesize O‐(2‐[18F]fluoroethyl)‐L‐tyrosine (18FFET)	0
C14‐Labelled Synthesis of Benalaxyl‐M and Its Two Soil Metabolites	0
Carbon 14 and Carbon 13 Syntheses of Velagliflozin	0
Issue Information	0
Synthesis and Preliminary Evaluation of an In Vivo Stable 131I‐Labeled Deuterated Tropane for Mapping Dopamine Transporter	0
Synthesis of 18F‐Labeled FC‐119S and Its Tosyl Precursor	0
Development and Validation of an HPLC Method to Determine Chemical and Radiochemical Purity of [18F]Florbetazine Injection	0
Preparation and evaluation of radiolabeled acetaminosalol microspheres: A new potential selective radiotracer for ulcerative colitis early diagnosis	0
Meet the advisors ‐ Suzy Lapi	0
Comparison of three different methods in [68Ga]Ga‐PSMA11 radiolabeling	0
Automated radiosynthesis of 1‐(2‐[18F]fluoroethyl)‐L‐tryptophan ([18F]FETrp) for positron emission tomography (PET) imaging of cancer in humans	0
Issue Information	0
Blood Brain Barrier – tactics and attributes in developing successful neuroimaging agents	0
	0
Highly effective liquid and solid phase extraction methods to concentrate radioiodine isotopes for radioiodination chemistry	0
	0
Automated radiosynthesis of [11C]MTP38—a phosphodiesterase 7 imaging tracer—using [11C]hydrogen cyanide for clinical applications	0
Issue Information	0
Issue Information	0
Issue Information	0
Issue Information	0
A facile synthesis of precursor for the σ‐1 receptor PET radioligand [18F]FTC‐146 and its radiofluorination	0
Issue Information	0
A Novel 68Ga‐Labeled 2‐Azabicyclo[3.1.0]Hexane‐3‐Carbonitrile‐Based Fibroblast Activation Protein‐Targeted Tracer for Cancer Imaging With Positron Emission Tomography	0
	0
A practical protocol for large‐scale copper‐mediated radioiodination of organoboronic precursors: Radiosynthesis of [123I]KX‐1 for Auger radiotherapy	0
Issue Information	0
Issue Information	0
Synthesis of Deuterated Endochin‐Like Quinolones	0
	0
Current Advances in PARP1‐Targeted Theranostics	0
Benzylic deuteration of alkylnitroaromatics via amine‐base catalysed exchange with deuterium oxide	0
Synthesis of Stable Isotope, Tritiated, and Carbon‐14 Labeled Balcinrenone	0
	0
	0
Synthesis of [3H]muscimol	0
	0
Issue Information	0
Development and physicochemical characterization of a biodegradable microspheres formulation loaded with samarium‐153 and doxorubicin for chemo‐radioembolization of liver tumours	0

Issue Information	0
Issue Information	0
Issue Information	0
	0
A synthesis of [14C]formamidine acetate	0
An improved synthesis of [18F]VAT and its precursor	0
	0
	0
Issue Information	0
Issue Information	0
Synthesis of [2H5]baricitinib via [2H5]ethanesulfonyl chloride	0
A practical approach to the optimization of positron emission tomography imaging agents for the central nervous system	0
Issue Information	0
Issue Information	0
Preparation, Characterization, and Radiolabeling of Anti‐HER2 scFv With Technetium Tricarbonyl and Stability Studies	0
Issue Information	0
Exploring the enzyme‐catalyzed synthesis of isotope labeled cyclopropanes	0
Open‐source flow setup for rapid and efficient [18F]fluoride drying for automation of PET tracer syntheses	0
An optimized radiosynthesis of [18F]DK222, a PET radiotracer for imaging PD‐L1	0
	0
A Brief Review of Radiolabelling Nucleic Acid‐Based Molecules for Tracking and Monitoring	0
A practical approach to the optimization of positron emission tomography imaging agents for the central nervous system	0
Synthesis of [3H]Org24598 using in‐house prepared [3H]MeI	0
Abstracts From the 29th International Isotope Society UK Meeting 17th November 2023	0
Issue Information	0
Simplified Flow Photosynthesis of Deuterium‐Labeled Pyocyanin	0
	0
	0
Tritium hydrogen‐isotope exchange with electron‐poor tertiary benzenesulfonamide moiety; application in late‐stage labeling of T0901317	0
Development of 11C‐labeled CRANAD‐102 for positron emission tomography imaging of soluble Aβ‐species	0
Synthesis and automated fluorine‐18 radiolabeling of new PSMA‐617 derivatives with a CuAAC radiosynthetic approach	0
A practical and environmentally friendly protocol for synthesis of α‐deuterated carboxylic acids	0
Wiley Young Scientist Awards were handed over at the 14th International Symposium on the synthesis on the Synthesis and Applications of Isotopically Labelled Compounds in Raleigh, USA	0
Synthesis of 13C‐labeled parabens from isotopically enriched phenols using the Houben–Hoesch reaction	0
The synthesis of deuteriated tri‐tert‐butyl phosphine	0
Site‐specifically radiolabeled nanobodies for imaging blood‐brain barrier penetration and targeting in the brain	0
Synthesis of a Potent Bruton's Tyrosine Kinase Inhibitor Labelled With Carbon‐14 and Deuterium	0
	0
Radiolabeling and brain penetration of [11C]VU0071063, a ligand of type 1 sulfonylurea receptors for positron emission tomography imaging	0
Efficient synthesis of carbon‐14 labeled metabolites of the strobilurin fungicide mandestrobin using biomimetic iron‐porphyrin catalyzed oxidation	0
Facile synthesis of 14C‐nitrofurazone from 14C‐urea	0
Development of an automated production process of [64Cu][Cu (ATSM)] for positron emission tomography imaging and theranostic applications	0
	0
Synthesis and Application of D‐ and 13C‐Labelled tert‐Butyl Hoechst Dye	0
Radioiodination, purification, and evaluation of antihuman tumor‐derived immunoglobulin G light chain monoclonal antibody in tumor‐bearing nude mice	0
In vivo and in vitro binding of [125I]I‐R‐(+)‐TISCH: A dopamine D1 receptor ligand for studying pancreatic β‐cell mass	0
Improved Radiosynthesis and Automation of [11C]2‐(2,6‐Difluoro‐4‐((2‐(N‐methylphenylsulfonamido)ethyl)thio)phenoxy)acetamide ([11C]K2) for Positron Emission Tomography of	0
Issue Information	0
Automated radiosynthesis of the adenosine A2A receptor‐targeting radiotracer [18F]FLUDA	0
Synthesis of deuterium‐labeled CCR2 antagonist JNJ‐26131300, [4‐(1H‐indol‐ 3‐yl)‐piperidin‐1‐yl]‐{1‐[3‐(3,4,5‐trifluoro‐phenyl)‐acryloyl]‐piperidin‐4‐yl}‐acetic acid	0
[11C]CO2 BOP fixation with amines to access 11C‐labeled ureas for PET imaging	0
	0
Synthesis and evaluation of 111In‐labeled tetrapeptide‐based compounds as single‐photon emission computed tomography imaging probes targeting granzyme B	0
Synthesis, Preclinical Characterizations and Imaging Studies of [18F]AlF‐Labeled NY104, a CAIX‐Targeting Diagnostic Agent	0
	0
Synthesis of Radiolabeled [14C]Rimsulfuron and Stable Isotope Labeled Rimsulfuron‐[M + 3] to Support Crop Metabolism Studies for Reregistration	0
	0
Automated Radiolabeling and Evaluation of [18F]FPMBBG: A Novel Cardiac Neuronal PET Imaging Agent	0
Synthesis and Imaging of Novel CDK19‐Targeted Tracers Incorporating an Albumin‐Binding Moiety	0
Synthesis and analysis of isotopically stable labeled nitrosamines as mass spectrometry standards for drug impurity quality control	0
	0
99mTc‐SNW‐1 Nanoparticle Labeling and Its Biodistribution/Pathological Evaluations	0
A simplified protocol for the automated production of 2‐[18F]fluoro‐3‐[2‐((S)‐3‐pyrrolinyl)methoxy]pyridine ([18F]nifene) on an IBA Synthera® module	0
An improved radiosynthesis of [18F]FAraG, a PET radiotracer for imaging T‐cell activation	0
Issue Information	0
Synthesis and Preclinical Evaluation of [18F]AlF‐NOTA‐Asp2‐PEG2‐Folate as a Novel Folate‐Receptor‐Targeted Tracer for PET Imaging	0
Automated Radiosynthesis of [18F]FMeNER‐D2 Using the Simplified One‐Pot 18F‐Fluoromethylation Method	0
Evaluation of New‐Modelled Recombinant Human Insulin (rh‐Insulin) Analog Expressed in E. coli Using Radioiodination Technique Followed by In Vivo Biodistribution in Diabetes‐Induced Mice	0
	0
Synthesis of beta‐site amyloid precursor protein‐cleaving enzyme 1 inhibitors BI 1147560 and BI 1181181 labeled with carbon‐14 and deuterium	0
[68Ga]Ga‐PentixaFor: Development of a fully automated in hospital production on the Trasis miniAllinOne synthesizer	0
	0
Evaluation and improvement of CuI‐mediated 11C‐cyanation	0
Synthesis and Evaluation of a Cathepsin B–Recognizing Trifunctional Chelating Agent to Improve Tumor Retention of Radioimmunoconjugates	0
18F‐Fluorination of a supported 2‐(aryl‐di‐tert‐butylsilyl)‐N‐methyl‐imidazole for indirect 18F‐labeling of a VHH single‐variable domain	0
	0
An Improved HPLC Separation Method for TSPO Radioligand [11C]ER176 Clinical Production	0
Stable isotope synthesis of glycine transporter 1 inhibitor Iclepertin (BI 425809) and its major metabolites	0
Featured Cover	0
Radioiodination of balsalazide, bioevaluation, and characterization as a highly selective radiotracer for imaging of ulcerative colitis in mice	0
Imidazolium‐methylene‐trifluoroborate: A novel radioprosthetic group validated with preclinical 18F‐Positron Emission Tomography imaging of Prostate Specific Membrane Antigen in mice	0
Direct Multi‐Deuterium Labelling of Pirtobrutinib	0
Enzymatic synthesis of halogen derivatives of L‐phenylalanine and phenylpyruvic acid stereoselectively labeled with hydrogen isotopes in the side chain	0
	0
	0
Carbon‐13 labeling of ibrutinib for human microdosing	0
Issue Information	0
	0
Efficient Reductive N‐11C‐Methylation Using Arylamines or Alkylamines and In Situ–Generated [11C]Formaldehyde From [11C]Methyl Iodide	0
Issue Information	0
Issue Information	0
Radiosynthesis and validation of [18F]fluoroestradiol in a Synthra plus research platform for use in routine clinical practice	0
Preparation of [1′‐13C]citric acid as a probe in a breath test to evaluate tricarboxylic acid cycle flux	0
Synthesis and radiolabeling of a polar [125I]I‐1,2,4,5‐tetrazine	0
Towards Optimal Automated 68Ga‐Radiolabeling Conditions of the DOTA‐Bisphosphonate BPAMD Without Pre‐Purification of the Generator Eluate	0