Journal of Labelled Compounds & Radiopharmaceuticals

Article	Citations
Radiosynthesis and validation of [18F]fluoroestradiol in a Synthra plus research platform for use in routine clinical practice	15
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Efficient synthesis of carbon‐14 labeled metabolites of the strobilurin fungicide mandestrobin using biomimetic iron‐porphyrin catalyzed oxidation	10
A synthesis of [14C]formamidine acetate	9
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Formulation of patient dose of [177Lu]Lu‐Trastuzumab using in‐house developed freeze‐dried kit: A path forward for clinical translation	7
Meet our Special Issue Editor: Jessica Bridoux	6
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Meet our advisors: Mathew Thakur	5
Practical approaches to labelling terminal alkynes with deuterium	4
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Preclinical evaluation of anti‐VEGFR2 monoclonal antibody ramucirumab labelled with zirconium‐89 for tumour imaging	4
Abstracts From the 29th International Isotope Society UK Meeting 17th November 2023	4
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A comparative study on Suzuki‐type 11C‐methylation of aromatic organoboranes performed in two reaction media	3
Meet our advisors: Crist N. Filer	3
Synthesis and preclinical evaluation of a selective MET kinase positron emission tomography tracer	3
Meet our advisors: Bart Cornelissen	3
Highly effective liquid and solid phase extraction methods to concentrate radioiodine isotopes for radioiodination chemistry	3
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Comparison of three different methods in [68Ga]Ga‐PSMA11 radiolabeling	3
Meet our advisors: Neil Vasdev	3
Efficient Reductive N‐11C‐Methylation Using Arylamines or Alkylamines and In Situ–Generated [11C]Formaldehyde From [11C]Methyl Iodide	3
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Direct Multi‐Deuterium Labelling of Pirtobrutinib	2
Automated Radiolabeling and Evaluation of [18F]FPMBBG: A Novel Cardiac Neuronal PET Imaging Agent	2
Determination of isotope abundance for deuterium‐labeled compounds by quantitative 1H NMR + 2H NMR	2
Automated radiolabeling and handling of 177Lu‐ and 225Ac‐PSMA‐617 using a robotic pipettor	2
Synthesis of 14C‐Labeled Polyethylene Terephthalate and Generation of 14C‐Nanoparticles for Fate and Disposition Studies	2
Total synthesis of [13C2]‐labeled phytosiderophores of the mugineic and avenic acid families	2
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A flow electrochemistry‐enabled synthesis of 2‐substituted N‐(methyl‐d)piperidines	2
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Tritium hydrogen‐isotope exchange with electron‐poor tertiary benzenesulfonamide moiety; application in late‐stage labeling of T0901317	2
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Strategies for designing novel positron emission tomography (PET) radiotracers to cross the blood–brain barrier	2
Preparation of [1′‐13C]citric acid as a probe in a breath test to evaluate tricarboxylic acid cycle flux	2
Meet our advisors: Jordi Llop	2
14C‐radiolabeling of a new steroidal antiandrogen with a C‐18 angular methyl extension	1
Synthesis of 13C‐labelled ω‐hydroxy carboxylic acids of the general formula HO213C‐(CH2)n‐CH2OH or HO2C‐(CH2	1
Meet our advisors—Matteo Zanda	1
Synthesis of N‐acetyl‐l‐aspartyl‐l‐glutamic acid; [3H]NAAG	1
Development of a high‐performance liquid chromatography method for rapid radiochemical purity measurement of [18F]PSMA‐1007, a PET radiopharmaceutical for detection of prostate cancer	1
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Preparation and biological evaluation of radioiodine‐labeled triphenylphosphine derivatives as mitochondrial targeting probes	1
Synthesis of trifold‐labeled versatile reagent [3,5‐13C2,4‐15 N]4‐phenyl‐1,2,4‐triazoline‐3,5‐dione	1
Radiosynthesis of 3H‐ and 14C‐labeled Veliparib	1
Peptides for trans‐blood–brain barrier delivery	1
Preparation, Characterization, and Radiolabeling of Anti‐HER2 scFv With Technetium Tricarbonyl and Stability Studies	1
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Stable isotope synthesis of glycine transporter 1 inhibitor Iclepertin (BI 425809) and its major metabolites	1
Synthesis of BI 894416 and BI 1342561, two potent and selective spleen tyrosine kinase inhibitors, labeled with carbon 14 and with deuterium	1
The inverse electron demand Diels–Alder cycloaddition with carbon‐11 and fluorine‐18: A gateway to pretargeted imaging across the blood–brain barrier	1
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Evaluation of New‐Modelled Recombinant Human Insulin (rh‐Insulin) Analog Expressed in E. coli Using Radioiodination Technique Followed by In Vivo Biodistribution in Diabetes‐Induced Mice	1
Applications of radiolabeled antibodies in neuroscience and neuro‐oncology	1
Carbon 14 synthesis of glycine transporter 1 inhibitor Iclepertin (BI 425809) and its major metabolites	1
Research on preparation and in vitro evaluation of the dendrimer–peptide nuclear acid conjugate for amplification pretargeting	1
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Synthesis of deuterium‐labeled CCR2 antagonist JNJ‐26131300, [4‐(1H‐indol‐ 3‐yl)‐piperidin‐1‐yl]‐{1‐[3‐(3,4,5‐trifluoro‐phenyl)‐acryloyl]‐piperidin‐4‐yl}‐acetic acid	1
Development of 11C‐labeled CRANAD‐102 for positron emission tomography imaging of soluble Aβ‐species	1
Radioiodination of balsalazide, bioevaluation, and characterization as a highly selective radiotracer for imaging of ulcerative colitis in mice	1
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Current Advances in PARP1‐Targeted Theranostics	1
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Open‐source flow setup for rapid and efficient [18F]fluoride drying for automation of PET tracer syntheses	0
Improving Routine 89Zr‐Immuno‐PET Applications: Mild Iron Removal Can Favor the Use of Fe‐DFO‐N‐suc‐TFP Ester Over p‐NCS‐Bz‐DFO	0
Meet our advisors: An interview with John Katzenellenbogen	0
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Automated production of 11C‐labeled carboxylic acids and esters via “in‐loop” 11C‐carbonylation using GE FX synthesis modules	0
Automated radiosynthesis of [11C]MTP38—a phosphodiesterase 7 imaging tracer—using [11C]hydrogen cyanide for clinical applications	0
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Synthesis of Radiolabeled [14C]Rimsulfuron and Stable Isotope Labeled Rimsulfuron‐[M + 3] to Support Crop Metabolism Studies for Reregistration	0
High‐yielding, automated radiosynthesis of [11C]martinostat using [11C]methyl triflate	0
Development and physicochemical characterization of a biodegradable microspheres formulation loaded with samarium‐153 and doxorubicin for chemo‐radioembolization of liver tumours	0
Automated radiosynthesis of [18F]CETO, a PET radiotracer for imaging adrenal glands, on Synthra RNplus	0
Synthesis of Carbon 14 and Deuterium‐Labelled Nerandomilast (BI 1015550)	0
A simplified protocol for the automated production of 2‐[18F]fluoro‐3‐[2‐((S)‐3‐pyrrolinyl)methoxy]pyridine ([18F]nifene) on an IBA Synthera® module	0
Synthesis of carbon‐14 and stable isotope labeled Censavudine	0
Site‐specifically radiolabeled nanobodies for imaging blood‐brain barrier penetration and targeting in the brain	0
Copper‐mediated radioiodination reaction through aryl boronic acid or ester precursor and its application to direct radiolabeling of a cyclic peptide	0
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Synthesis of tritium labeled 30‐KDa PEG and conjugation to form [3H]Pegbelfermin	0
Meet our advisors: Bill Lockley	0
An improved synthesis of [18F]VAT and its precursor	0
Synthesis and Evaluation of a Cathepsin B–Recognizing Trifunctional Chelating Agent to Improve Tumor Retention of Radioimmunoconjugates	0
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Preparation of Macrobicyclic Cryptands for Radiometal Complexation	0
Simplified Flow Photosynthesis of Deuterium‐Labeled Pyocyanin	0
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Meet the advisors ‐ Suzy Lapi	0
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Application of Microfluidic Devices for Automated Two‐Step Radiolabeling of Antibodies	0
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Meet the editors: Danielle Vugts	0
RO6807936 as a novel positron emission tomography (PET) radiotracer for in vitro and in vivo visualization and quantification of beta‐site amyloid precursor protein cleaving enzyme (BACE1) in the rode	0
Synthesis of [13C6]‐ibrutinib	0
Synthesis of deuterium‐labeled cinnamic acids: Understanding the volatile benzenoid pathway in the flowers of the Japanese loquat Eriobotrya japonica	0
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Synthesis of Deuterated Endochin‐Like Quinolones	0
Meet the editorial staff—Interview series	0
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Facile synthesis of 14C‐nitrofurazone from 14C‐urea	0
Synthesis of [3H]Org24598 using in‐house prepared [3H]MeI	0
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Benzylic deuteration of alkylnitroaromatics via amine‐base catalysed exchange with deuterium oxide	0
Automated radiosynthesis of mGluR5 PET tracer [18F]FPEB from aryl‐chloro precursor and validation for clinical application	0
Highly selective catalytic transfer hydrodeuteration of cyclic alkenes	0
Detailed radiosynthesis of [18F]mG4P027 as a positron emission tomography radiotracer for mGluR4	0
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Synthesis of 13C‐labeled parabens from isotopically enriched phenols using the Houben–Hoesch reaction	0
An Improved HPLC Separation Method for TSPO Radioligand [11C]ER176 Clinical Production	0
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Low‐scale syringe‐made synthesis of 15N‐labeled oligonucleotides	0
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Radioiodination, purification, and evaluation of antihuman tumor‐derived immunoglobulin G light chain monoclonal antibody in tumor‐bearing nude mice	0
Next Generation of Solid Target Radionuclide Antibody Conjugates for Tumor Immuno‐Therapy	0
Exploring the enzyme‐catalyzed synthesis of isotope labeled cyclopropanes	0
Synthesis and spectroscopic characterization of 13C4‐labeled 4‐cyano‐2‐oxobutyraldehyde semicarbazone: A metabolite of nitrofurazone	0
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68Ga Radiolabeling of NODASA‐Functionalized Phage Display–Derived Peptides for Prospective Assessment as Tuberculosis‐Specific PET Radiotracers	0
Automated radiosynthesis of the adenosine A2A receptor‐targeting radiotracer [18F]FLUDA	0
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Synthesis and Preclinical Evaluation of Peptide Dimer‐Based PET Tracers for Imaging VEGFR‐2 Expression in Tumors	0
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Preparation and evaluation of radiolabeled acetaminosalol microspheres: A new potential selective radiotracer for ulcerative colitis early diagnosis	0
[68Ga]Ga‐PentixaFor: Development of a fully automated in hospital production on the Trasis miniAllinOne synthesizer	0
Automated radiosynthesis of 1‐(2‐[18F]fluoroethyl)‐L‐tryptophan ([18F]FETrp) for positron emission tomography (PET) imaging of cancer in humans	0
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Nitrilase mediated mild hydrolysis of a carbon‐14 nitrile for the radiosynthesis of 4‐(7‐hydroxycarbamoyl‐[1‐14C‐heptanoyl]‐oxy)‐benzoic acid methyl ester, [14C]‐SHP‐141: A novel	0

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An optimized radiosynthesis of [18F]DK222, a PET radiotracer for imaging PD‐L1	0
Towards Optimal Automated 68Ga‐Radiolabeling Conditions of the DOTA‐Bisphosphonate BPAMD Without Pre‐Purification of the Generator Eluate	0
An improved radiosynthesis of [18F]FAraG, a PET radiotracer for imaging T‐cell activation	0
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Simplified and accessible [18F]F‐AraG synthesis procedure for preclinical PET	0
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Automated radiochemical synthesis of pharmaceutical grade [18F]FLT using 3‐N‐Boc‐5′‐O‐dimethoxytrityl‐3′‐O‐nosyl‐thymidine precursor and its Sep‐Pak® purification employing selective elutio	0
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An efficient and general method for the synthesis of stable isotope deuterium labeled phthalate esters	0
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Synthesis, Preclinical Characterizations and Imaging Studies of [18F]AlF‐Labeled NY104, a CAIX‐Targeting Diagnostic Agent	0
Mild and selective hydrogen–deuterium exchange for aromatic hydrogen of amines	0
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Polyethylene oxide–polyacrylic acid–folic acid (PEO‐PAAc) nanogel as a99mTc targeting receptor for cancer diagnostic imaging	0
Radiolabeling and brain penetration of [11C]VU0071063, a ligand of type 1 sulfonylurea receptors for positron emission tomography imaging	0
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Luminescence enhancement by deuterium	0
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Meet our advisors: Dieter Muri	0
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Synthesis and Application of D‐ and 13C‐Labelled tert‐Butyl Hoechst Dye	0
Evaluation and improvement of CuI‐mediated 11C‐cyanation	0
18F‐Fluorination of a supported 2‐(aryl‐di‐tert‐butylsilyl)‐N‐methyl‐imidazole for indirect 18F‐labeling of a VHH single‐variable domain	0
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Good manufacturing procedure production of [18F]SynVesT‐1, a radioligand for in vivo positron emission tomography imaging of synaptic vesicle glycoprotein 2A	0
Novel synthesis of 11C‐labeled imidazolines via Pd(0)‐mediated 11C‐carbomethoxylation using [11C]CO and arylborons	0
Development of radiotracers for riboflavin transporter 3 imaging in diseases—A brief overview	0
Fully Automated Cassette‐Based Synthesis of 2‐Deoxy‐2‐[18F]Fluorocellobiose Using Trasis AllInOne Module	0
Preliminary PET imaging of [11C]evobrutinib in mouse models of colorectal cancer, SARS‐CoV‐2, and lung damage: Radiosynthesis via base‐aided palladium‐NiXantphos‐mediated 11C‐car	0
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Automated synthesis of (R)‐[18F]MH.MZ on the iPhase Flexlab reaction platform	0
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Synthesis and Characterization of 3‐Hydroxybupivacaine and Deuterated 3‐Hydroxybupivacaine for Use in Equine Medication Regulation	0
A practical approach to the optimization of positron emission tomography imaging agents for the central nervous system	0
Improved protocol for the radiosynthesis of [18F]FTC‐146: A potent and selective sigma‐1 receptor radioligand	0
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Synthesis and radiolabeling of a polar [125I]I‐1,2,4,5‐tetrazine	0
Carbon 14 and stable isotope synthesis of two potent and selective phosphodiesterase type 4 inhibitors	0
Evaluating N‐difluoromethyltriazolium triflate as a precursor for the synthesis of high molar activity [18F]fluoroform	0
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A facile synthesis of precursor for the σ‐1 receptor PET radioligand [18F]FTC‐146 and its radiofluorination	0
An improved one‐pot preparation of [18F]FMISO based on solid phase extraction purification: Pitfalls on the analytical method reported in the Ph.Eur.'s monograph	0
Synthesis of beta‐site amyloid precursor protein‐cleaving enzyme 1 inhibitors BI 1147560 and BI 1181181 labeled with carbon‐14 and deuterium	0
A Novel 68Ga‐Labeled 2‐Azabicyclo[3.1.0]Hexane‐3‐Carbonitrile‐Based Fibroblast Activation Protein‐Targeted Tracer for Cancer Imaging With Positron Emission Tomography	0
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Synthesis and automated fluorine‐18 radiolabeling of new PSMA‐617 derivatives with a CuAAC radiosynthetic approach	0
Carbon 14 and Carbon 13 Syntheses of Velagliflozin	0
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Design and Synthesis of a 18F‐Radiolabeled Pyrrolo[2,3‐d]pyrimidine Ligand as a CSF1R Receptor PET Imaging Agent	0
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Ultra‐fast liquid chromatography method coupled with ultraviolet detection to quantify dimethylsulfoxide, dimethylformamide and dimethylacetamide in short half‐lives radiopharmaceuticals	0
Novel developed HPLC analyses of [68Ga]Ga/[177Lu]Lu‐EDTMP and [68Ga]Ga/[177Lu]Lu‐DOTA‐Zoledronate	0
Synthesis and Imaging of Novel CDK19‐Targeted Tracers Incorporating an Albumin‐Binding Moiety	0
11C‐Carbonylation for PET Imaging and Drug Discovery	0
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Meet the advisors: An interview with Gunnar Antoni	0
A practical protocol for large‐scale copper‐mediated radioiodination of organoboronic precursors: Radiosynthesis of [123I]KX‐1 for Auger radiotherapy	0
Fully automated production of the fibroblast activation protein radiotracer [18F]FAPI‐74	0
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Applications of Isotopes in Forensic Science	0
Meet our advisors: Billy Kerr	0
[18F]Fluoropyridine‐losartan: A new approach toward human Positron Emission Tomography imaging of Angiotensin II Type 1 receptors	0
Review: Self‐radiolysis of compounds containing tritium and carbon‐14	0
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Validation of a good manufacturing practice procedure for the production of [11C]AZD4747, a CNS penetrant KRASG12c inhibitor	0
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Synthesis and evaluation of 111In‐labeled tetrapeptide‐based compounds as single‐photon emission computed tomography imaging probes targeting granzyme B	0
The synthesis of deuteriated tri‐tert‐butyl phosphine	0
Tritium and deuterium labelling of a kainate receptor antagonist and evaluation as a radioligand	0
Synthesis of [2H5]baricitinib via [2H5]ethanesulfonyl chloride	0
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A practical and environmentally friendly protocol for synthesis of α‐deuterated carboxylic acids	0
Blood Brain Barrier – tactics and attributes in developing successful neuroimaging agents	0
Enzymatic synthesis of halogen derivatives of L‐phenylalanine and phenylpyruvic acid stereoselectively labeled with hydrogen isotopes in the side chain	0
[11C]CO2 BOP fixation with amines to access 11C‐labeled ureas for PET imaging	0
Synthesis and Preclinical Evaluation of [18F]AlF‐NOTA‐Asp2‐PEG2‐Folate as a Novel Folate‐Receptor‐Targeted Tracer for PET Imaging	0
Initial evaluation of 99mTc‐labeled anti‐carcinoembryonic antigen single‐chain fragment variable for micro‐single‐photon emission computed tomography imaging in mice with colorectal cancer	0
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Photocatalyzed radiosynthesis of 11C‐phenylacetic acids	0
Development of an economical method to synthesize O‐(2‐[18F]fluoroethyl)‐L‐tyrosine (18FFET)	0
Carbon‐14 Labeling Synthesis of RORγt Inhibitor JNJ‐61803534	0
Wiley Young Scientist Awards were handed over at the 14th International Symposium on the synthesis on the Synthesis and Applications of Isotopically Labelled Compounds in Raleigh, USA	0
Preliminary Research of Radiolabeled Atezolizumab for the Noninvasive Evaluation of TNBC PD‐L1 Expression In Vivo	0
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Synthesis and analysis of isotopically stable labeled nitrosamines as mass spectrometry standards for drug impurity quality control	0