Archiv der Pharmazie

Papers
(The TQCC of Archiv der Pharmazie is 5. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2021-04-01 to 2025-04-01.)
ArticleCitations
Cover Picture: Arch Pharm (4/2024)213
1,2,3‐Triazole‐based esters and carboxylic acids as nonclassical carbonic anhydrase inhibitors capable of cathepsin B inhibition195
New antiproliferative agents derived from tricyclic 3,4‐dihydrobenzo[4,5]imidazo[1,2‐a][1,3,5]triazine scaffold: Synthesis and pharmacological effects73
Issue Information: Arch Pharm (2/2025)64
Indole clubbed 2,4‐thiazolidinedione linked 1,2,3‐triazole as a potent antimalarial and antibacterial agent against drug‐resistant strain and molecular modeling studies56
Silver–N‐heterocyclic carbene complexes‐catalyzed multicomponent reactions: Synthesis, spectroscopic characterization, density functional theory calculations, and antibacterial study48
Cover Picture: Arch Pharm (1/2022)46
Editorial Board: Arch Pharm (1/2022)45
Current scenario of indole hybrids with antibacterial potential against Acinetobacter baumannii pathogens: A mini‐review42
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The C‐terminally shortened analogs of a hexapeptide derived from Lingzhi hydrolysate with enhanced tyrosinase‐inhibitory activity38
hERG stereoselective modulation by mexiletine‐derived ureas: Molecular docking study, synthesis, and biological evaluation38
Indole derivatives targeting colchicine binding site as potential anticancer agents38
Citrus wastewater as a source of value‐added products: Quali‐quantitative analysis and in vitro screening on breast cancer cell lines37
Exploration of cytotoxicity of iodoquinazoline derivatives as inhibitors of both VEGFR‐2 and EGFRT790M: Molecular docking, ADMET, design, and syntheses36
Design and development of novel series of indole‐3‐sulfonamide ureido derivatives as selective carbonic anhydrase II inhibitors34
Aminoalkoxy‐substituted coumarins: Synthesis and evaluation for reactivation of inhibited human acetylcholinesterase34
Design, synthesis, and evaluation of 4′‐phosphonomethoxy pyrimidine ribonucleosides as potential anti‐influenza agents34
In vitro and in silico studies of fluorinated 2,3‐disubstituted thiazolidinone‐pyrazoles as potential α‐amylase inhibitors and antioxidant agents32
Sulfonamide‐incorporated bis(α‐aminophosphonates) as promising carbonic anhydrase inhibitors: Design, synthesis, biological evaluation, and X‐ray crystallographic studies32
Synthesis, characterization, and biological study of new synthetic opioid hemorphin‐4 peptides containing sterically restricted nonnatural amino acids27
What doesn't fit is made to fit: Pim‐1 kinase adapts to the configuration of stilbene‐based inhibitors26
Suppression of the TRIF‐dependent signaling pathway of TLRs by epoxomicin26
Design, synthesis, and characterization of PROTACs targeting the androgen receptor in prostate and lung cancer models25
Design, synthesis, in silico ADMET, docking, and antiproliferative evaluations of [1,2,4]triazolo[4,3‐c]quinazolines as classical DNA intercalators25
Chemistry of heterocycles as carbonic anhydrase inhibitors: A pathway to novel research in medicinal chemistry review25
Synthesis and biological evaluation of coumarin‐thiazole hybrids as selective carbonic anhydrase IX and XII inhibitors23
New 3‐(1H‐benzo[d]imidazol‐2‐yl)quinolin‐2(1H)‐one‐based triazole derivatives: Design, synthesis, and biological evaluation as antiproliferative and apoptosis‐inducing agents23
Structure‐guided identification of a selective sulfonamide‐based inhibitor targeting the human carbonic anhydrase VA isoform23
Design, synthesis, and evaluation of new benzimidazole‏ ‏‎thiourea ‎derivatives as antitumor agents23
Synthesis and in vitro antiproliferative activity of certain novel pyrazolo[3,4‐b]pyridines with potential p38α MAPK‐inhibitory activity21
Combating DC‐SIGN‐mediated SARS‐CoV‐2 dissemination by glycan‐mimicking polymers21
New 1,2,4‐oxadiazole/pyrrolidine hybrids as topoisomerase IV and DNA gyrase inhibitors with promising antibacterial activity21
Synthesis and screening of 6‐alkoxy purine analogs as cell type‐selective apoptotic inducers in Jurkat cells21
Synthesis and biological evaluation of new coumarin derivatives as cytotoxic agents20
In vitro and in vivo evaluation of a water‐in‐oil microemulsion of platycodin D20
Synthesis and biological profile of benzoxazolone derivatives20
The current landscape of coumarin hybrids with antibreast cancer therapeutic applications: An updated review19
Extracting binding energies and binding modes from biomolecular simulations of fragment binding to endothiapepsin19
Strategies in synthetic design and structure–activity relationship studies of novel heterocyclic scaffolds as aldose reductase‐2 inhibitors19
A decade's overview of 2‐aminothiophenes and their fused analogs as promising anticancer agents19
Synthesis of 1,2,3‐triazole‐1,3,4‐thiadiazole hybrids as novel α‐glucosidase inhibitors by in situ azidation/click assembly19
Multi‐functional tyrosinase inhibitors derived from kojic acid and hydroquinone‐like diphenols for treatment of hyperpigmentation: Synthesis and in vitro biological evaluation19
Unveiling new thiazole‐clubbed piperazine derivatives as multitarget anti‐AD: Design, synthesis, and in silico studies19
Synthesis and biological evaluation of salophen nickel(II) and cobalt(III) complexes as potential anticancer compounds19
Exploration of 1,2,3‐triazolo fused triterpenoids as inhibitors of human coronavirus 229E targeting the viral nsp15 protein18
N‐Substituted piperidine‐3‐carbohydrazide‐hydrazones against Alzheimer's disease: Synthesis and evaluation of cholinesterase, beta‐amyloid inhibitory activity, and antioxidant capacity18
Synthesis, antimycobacterial, cytotoxicity, anti‐inflammatory, in silico studies and molecular dynamics of pyrazole‐embedded thiazolidin‐4‐one hybrids18
Microwave‐induced one‐pot synthesis of 3‐imidazolyl indole clubbed 1,2,3‐triazole hybrids as antiproliferative agents and density functional theory study18
Pioneering first‐in‐class FAAH‐HDAC inhibitors as potential multitarget neuroprotective agents17
Triazole derivatives as potential xanthine oxidase inhibitors: Design, enzyme inhibition potential, and docking studies17
Synthesis and antimicrobial testing of 5‐fluorouracil derivatives16
Symmetrical 2,7‐disubstituted 9H‐fluoren‐9‐one as a novel and promising scaffold for selective targeting of SIRT216
Emerging green synthetic routes for thiazole and its derivatives: Current perspectives16
5‐Fluoro/(trifluoromethoxy)‐2‐indolinone derivatives with anti‐interleukin‐1 activity16
Synthesis of novel pyrimido[4,5‐b]quinoline derivatives as dual EGFR/HER2 inhibitors as anticancer agents15
Tail‐approach based design, synthesis, and molecular modeling of benzenesulfonamides carrying thiadiazole and urea moieties as novel carbonic anhydrase inhibitors15
Synthesis and evaluation of febrifugine derivatives as anticoccidial agents15
Design, synthesis, and activity evaluation of novel multitargeted l‐tryptophan derivatives with powerful antioxidant activity against Alzheimer's disease15
Natural flavonoids as promising lactate dehydrogenase A inhibitors: Comprehensive in vitro and in silico analysis14
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Archiv der Pharmazie—200 years14
Synthesis, biological activities, and structure–activity relationships of Morita–Baylis–Hillman adducts: An update14
Structure–activity relationship study to improve cytotoxicity and selectivity of lonafarnib against breast cancer cells14
Issue Information: Arch Pharm (5/2024)14
Analysis of histamine and sisomicin in gentamicin: Search for the causative agents of adverse effects14
Biosynthesized metallic nanoparticles: A new era in cancer therapy14
Recent green approaches for the synthesis of pyrazolo[3,4‐d]pyrimidines: A mini review14
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Editorial Board: Arch Pharm (9/2022)13
Cover Picture: Arch Pharm (1/2024)13
Synthesis of 3‐hydroxy‐2‐naphthohydrazide‐based hydrazones and their implications in diabetic management via in vitro and in silico approaches13
Editorial Board: Arch Pharm (1/2024)13
Implication of in silico studies in the search for novel inhibitors against SARS‐CoV‐213
Cover Picture: Arch Pharm (3/2022)13
Cover Picture: Arch Pharm (11/2023)13
Triazolo‐linked benzimidazoles as tubulin polymerization inhibitors and DNA intercalators: Design, synthesis, cytotoxicity, and docking studies12
Functional combination of resveratrol and tamoxifen to overcome tamoxifen‐resistance in breast cancer cells12
A novel class for carbonic anhydrases inhibitors and evaluation of their non‐zinc binding12
Isobavachalcone suppresses the TRIF‐dependent signaling pathway of Toll‐like receptors12
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Synthesis and evaluation of novel xanthene‐based thiazoles as potential antidiabetic agents12
Correction to: Ecofriendly synthesis of pyrano[2,3‐d]pyrimidine derivatives and related heterocycles with anti‐inflammatory activities12
Synthesis and in vitro cytotoxicity of benzoxazole‐based PPARα/γ antagonists in colorectal cancer cell lines12
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Synthesis and evaluation of carbamate derivatives as fatty acid amide hydrolase and monoacylglycerol lipase inhibitors12
New 1,3,4‐oxadiazole‐chalcone/benzimidazole hybrids as potent antiproliferative agents12
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Thiazole‐based SARS‐CoV‐2 protease (COV Mpro) inhibitors: Design, synthesis, enzyme inhibition, and molecular modeling simulations12
New hydrazide derivatives of N‐amino‐11‐azaartemisinin as promising epidermal growth factor receptor inhibitors for therapeutic development in triple‐negative breast cancer11
New pyrimidine/thiazole hybrids endowed with analgesic, anti‐inflammatory, and lower cardiotoxic activities: Design, synthesis, and COX‐2/sEH dual inhibition11
Absolute configuration of cytotoxic anthraquinones from a Brazilian cave soil‐derived fungus, Aspergillus sp. SDC2811
Isatin thiazoles as antidiabetic: Synthesis, in vitro enzyme inhibitory activities, kinetics, and in silico studies11
New [1,2,4]triazolo[4,3‐c]quinazoline derivatives as vascular endothelial growth factor receptor‐2 inhibitors and apoptosis inducers: Design, synthesis, docking, and antiproliferative evaluatio11
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Coumarin‐modified ruthenium complexes: Synthesis, characterization, and antiproliferative activity against human cancer cells11
Synthesis and biological evaluation of sulfonamide‐based compounds as inhibitors of carbonic anhydrase from Vibrio cholerae11
Discovery of novel α‐carboline derivatives as glycogen synthase kinase‐3β inhibitors for the treatment of Alzheimer's disease10
C5‐Iminosugar modification of casein kinase 1δ lead 3‐(4‐fluorophenyl)‐5‐isopropyl‐4‐(pyridin‐4‐yl)isoxazole promotes enhanced inhibitor affinity and selectivity10
Oxadiazole: A highly versatile scaffold in drug discovery10
Pyrazole scaffold‐based derivatives: A glimpse of α‐glucosidase inhibitory activity, SAR, and route of synthesis10
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Comparative analysis of apocarotenoids and phenolic constituents of Crocus sativus stigmas from 11 countries: Ecological impact10
An exploratory study on the effect of mechanical stress on particle formation in monoclonal antibody infusions10
Design, synthesis, cytotoxicity, and molecular docking studies of novel thiazolyl–hydrazone derivatives as histone lysine acetyl‐transferase inhibitors and apoptosis inducers10
Selective cytotoxicity of ent‐kaurene diterpenoids isolated from Baccharis lateralis and Baccharis retusa (Asteraceae)10
Anticancer activities, structure–activity relationship, and mechanism of action of 12‐, 14‐, and 16‐membered macrolactones10
SC‐560 and mofezolac isosteres as new potent COX‐1 selective inhibitors with antiplatelet effect10
Pyrazole/pyrazoline as an excellent pharmacophore in the design of carbonic anhydrase inhibitors (2018–2022)10
Novel substituted 5‐methyl‐4‐acylaminoisoxazoles as antimitotic agents: Evaluation of selectivity to LNCaP cancer cells10
Quinoxaline‐based efflux pump inhibitors restore drug susceptibility in drug‐resistant nontuberculous mycobacteria10
On the hunt for metalloenzyme inhibitors: Investigating the presence of metal‐coordinating compounds in screening libraries and chemical spaces10
Corrigendum: The medicinal perspective of 2,4‐thiazolidinediones based ligands as antimicrobial, antitumor and antidiabetic agents: A review10
Curcumin‐based bioactive heterocycles derived via multicomponent reactions10
Design and synthesis of pyridazin‐4‐one derivatives as necroptosis inhibitors9
Review on the pharmacological effects and pharmacokinetics of scutellarein9
Piperlongumine and its derivatives against cancer: A recent update and future prospective9
Benzotriazole scaffold: An overview of antiproliferative potential, mechanisms of action, and structure–activity relationships9
Development and in vitro antiviral activity of ivermectin liposomes as a potential drug carrier system9
Synthesis and examination of 1,2,4‐triazine‐sulfonamide hybrids as potential inhibitory drugs: Inhibition effects on AChE and GST enzymes in silico and in vitro conditions9
Novel 2‐substituted thioquinazoline‐benzenesulfonamide derivatives as carbonic anhydrase inhibitors with potential anticancer activity9
Biological functions of kojic acid and its derivatives in medicine, cosmetics, and food industry: Insights into health aspects9
Issue Information: Arch Pharm (8/2024)9
Novel isoxazoline‐linked 1,3,4‐thiadiazole hybrids as anticancer agents: Design, synthesis, biological evaluation, molecular docking, and molecular dynamics simulation9
Synthesis and biological evaluation of new 4‐oxo‐thiazolidin‐2‐ylidene derivatives as antimicrobial agents9
In vitro antiviral activity of favipiravir and its 6‐ and 3‐O‐substituted derivatives against coronavirus: Acetylation leads to improvement of antiviral activity9
Discovery of xanthone‐based nitric oxide donors targeting biofilm clearance9
Unveiling tomorrow: Carbonic anhydrase activators and inhibitors pioneering new frontiers in Alzheimer's disease8
The anti‐breast cancer therapeutic potential of 1,2,3‐triazole‐containing hybrids8
In‐vitro and in‐silico investigations of SLC‐0111 hydrazinyl analogs as human carbonic anhydrase I, II, IX, and XII inhibitors8
Evaluation of betanin‐loaded liposomal nanocarriers in AlCl3‐induced Alzheimer's disease in rats: Impact on cognitive function, neurodegeneration, and TREM2/ADAM10 pathways8
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Synthesis and antitumor evaluation of glycyrrhetinic acid‐dithiocarbamate hybrids8
Synthesis, density functional theory calculation, molecular docking studies, and evaluation of novel 5‐nitrothiophene derivatives for anticancer activity8
GOAT rs10096097 and CREB1 rs6740584 single nucleotide polymorphisms are associated with type 2 diabetes mellitus in Egyptians8
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Phthalimide derivatives as a new class of papain‐like protease inhibitors in SARS‐CoV‐28
A review of recent advances in anticancer activity and SAR of pyrazole derivatives8
Identification and study of new NF‐κB‐inducing kinase ligands derived from the imidazolone scaffold8
FDA‐approved drugs featuring macrocycles or medium‐sized rings8
Discovery of a novel 2,4‐thiazolidinedione derivative as dual inhibitor of β‐catenin/TCF4 interaction and tubulin polymerization in colon cancer cells8
Synthesis of new dihydropyrimidine derivatives and investigation of their antimicrobial and DNA gyrase inhibitory activities8
Vitamin D promotes anticancer effects of low‐concentration cisplatin‐treated non‐small cell lung cancer cells via inhibiting the JAK2/STAT3 and TGF‐β/SMAD4 pathways8
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Mono‐ and bis(steroids) containing a cyclooctane core: Synthesis, antiproliferative activity, and action on cell cytoskeleton microtubules7
Sulfonyl thioureas with a benzo[d]thiazole ring as dual acetylcholinesterase/butyrylcholinesterase and human monoamine oxidase A and B inhibitors: An in vitro and in silico study7
Uncovering chemical profiles, biological potentials, and protection effect against ECM destruction in H2O2‐treated HDF cells of the extracts of Stachys tundjeliensis7
Pharmacophore‐linked pyrazolo[3,4‐d]pyrimidines as EGFR‐TK inhibitors: Synthesis, anticancer evaluation, pharmacokinetics, and in silico mechanistic studies7
New benzimidazole–indole–amide derivatives as potent α‐glucosidase and acetylcholinesterase inhibitors7
Editorial Board: Arch Pharm (5/2022)7
Cover Picture: Arch Pharm (8/2023)7
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Editorial Board: Arch Pharm (7/2021)7
Editorial Board: Arch Pharm (10/2023)7
Issue Information: Arch Pharm (7/2024)7
Cover Picture: Arch Pharm (5/2024)7
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Fabrication of sulfobutylether‐β‐cyclodextrin/glabridin inclusion complex for promoting bioactivities7
Novel RP‐HPLC method for estimation of a newly developed combination of tizanidine and etoricoxib in rat plasma: Eight criteria for greens evaluation7
Discovery of novel potent PI3K/mTOR dual‐target inhibitors based on scaffold hopping: Design, synthesis, and antiproliferative activity7
Cover Picture: Arch Pharm (2/2024)7
Editorial Board: Arch Pharm (6/2022)7
Cover Picture: Arch Pharm (7/2023)7
Editorial Board: Arch Pharm (11/2022)7
Cover Picture: Arch Pharm (10/2023)7
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Anticancer perspectives of monocarbonyl analogs of curcumin: A decade (2014–2024) review7
Discovery of N,N'‐diarylurea molecules with activity against multidrug‐resistant Staphylococcus aureus7
Discovery of sulfadrug–pyrrole conjugates as carbonic anhydrase and acetylcholinesterase inhibitors7
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Editorial Board: Arch Pharm (5/2023)7
Cover Picture: Arch Pharm (9/2021)7
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Antiprotozoal agents: How have they changed over a decade?6
Chemical composition and biological activities of Cucurbita okeechobeensis extracts from its aerial parts, seeds, and fruit shells6
Benzimidazolone‐piperazine/triazole/thiadiazole/furan/thiophene conjugates: Synthesis, in vitro urease inhibition, and in silico molecular docking studies6
Replacing the oxidation‐sensitive triaminoaryl chemotype of problematic KV7 channel openers: Exploration of a nicotinamide scaffold6
Combining chemical profiles and biological abilities of different extracts from Tanacetum nitens (Boiss. & NoëGrierson using network pharmacology6
Novel therapeutic strategies and drugs for idiopathic pulmonary fibrosis6
Synthesis of new N‐(3‐oxo‐1‐thia‐4‐azaspiro[4.5]decan‐4‐yl)pyridine‐3‐carboxamide derivatives and evaluation of their anti‐influenza virus and antitubercular activities6
Synthesis of benzylated amine‐substituted xanthone derivatives and their antioxidant and anti‐inflammatory activities6
Benzenesulfonamides functionalized with triazolyl‐linked pyrazoles possess dual cathepsin B and carbonic anhydrase inhibitory action6
Cover Picture: Arch Pharm (12/2022)6
Exploration of 3‐aryl pyrazole‐tethered sulfamoyl carboxamides as carbonic anhydrase inhibitors6
Development and evaluation of 2,4‐disubstituted‐5‐aryl pyrimidine derivatives as antibacterial agents6
Synthesis of selenophene‐based chalcone analogs and assessment of their biological activity as anticancer agents6
Unlocking nitrogen compounds’ promise against malaria: A comprehensive review6
A comparative untargeted metabolomic analysis and assessment of antiplasmodial potential of nine Albizia species6
Editorial Board: Arch Pharm (2/2022)6
Pentathiepins are an understudied molecular prism of biological activities6
Novel benzothiazole/benzothiazole thiazolidine‐2,4‐dione derivatives as potential FOXM1 inhibitors: In silico, synthesis, and in vitro studies6
A review: Biological activities of novel cyanopyridine derivatives6
In silico characterization of ligand–receptor interactions for U‐47700, N,N‐didesmethyl‐U‐47700, U‐50488 at mu‐ and kappa‐opioid receptors6
Identification and assessment of new PIM2 inhibitors for treating hematologic cancers: A combined approach of energy‐based virtual screening and machine learning evaluation6
From dyes to drugs: The historical impact and future potential of dyes in drug discovery6
Discovery of 5‐alkyl‐2‐pyrazol‐oxazolidin‐4‐one derivatives as novel hepatitis B virus capsid assembly modulators6
Cyclization of acyl thiosemicarbazides led to new Helicobacter pylori α‐carbonic anhydrase inhibitors6
Morpholinodiazenyl chalcone blocks influenza A virus capsid uncoating by perturbing the clathrin‐mediated vesicular trafficking pathway6
New chimeric HDAC inhibitors for the treatment of colorectal cancer6
Novel hydrazide‐hydrazone containing 1,2,4‐triazole as potent inhibitors of antiapoptotic protein Bcl‐xL: Synthesis, biological evaluation, and docking studies6
Editorial Board: Arch Pharm (10/2022)6
The medicinal perspective of 2,4‐thiazolidinediones based ligands as antimicrobial, antitumor and antidiabetic agents: A review5
Therapeutic potential of d‐limonene in rheumatoid arthritis: Modulation of inflammatory, anti‐inflammatory cytokines, and prostaglandin E25
EGB761 ameliorates mild cognitive impairment by inhibiting the pyroptosis and apoptosis in both in vivo and in vitro experiments5
Design and synthesis of novel chalcone derivatives and evaluation of their inhibitory activities against acetylcholinesterase5
Liposomal formulation of model pentathiepin improves solubility and stability toward glutathione while preserving anticancer activity5
Pharmacophore‐based, rationale design, and efficient synthesis of novel tetrahydrobenzo[b]thiophene candidates as potential dual Topo I/II inhibitors and DNA intercalators5
New potent muscarinic receptor ligands bearing the 1,4‐dioxane nucleus: Investigation on the nature of the substituent in position 25
A comprehensive update on the structure and synthesis of potential drug targets for combating the coronavirus pandemic caused by SARS‐CoV‐25
Design, synthesis, α‐glucosidase inhibition, pharmacokinetic, and cytotoxic studies of new indole‐carbohydrazide‐phenoxy‐N‐phenylacetamide derivatives5
New azaaurone derivatives as potential multitarget agents in HIV‐TB coinfection5
Novel pyrazolo[3,4‐b]pyridine derivatives: Synthesis, structure–activity relationship studies, and regulation of the AMPK/70S6K pathway5
In vivo hepatoprotective and nephroprotective effects ofStenocarpus sinuatusleaf extract against ifosfamide‐induced toxicity in rats5
Nanocarriers for the treatment of glioblastoma multiforme: A succinct review of conventional and repositioned drugs in the last decade5
Fragment‐type 4‐azolylcoumarin derivatives with anticancer properties5
A sustainable RP‐HPLC method for concurrent estimation of capecitabine and celecoxib in liposomal formulation: Greenness and whiteness appraisal5
Green synthesis of novel antifungal 1,2,4‐triazoles effective against γ‐irradiated Candida parapsilosis5
Multitargeting in cardioprotection: An example of biaromatic compounds5
Insights into modulating the monastrol scaffold: Development of new pyrimidinones as Eg5 inhibitors with anticancer activity5
Flucytosine‐based prodrug activation by cold physical plasma5
Recent advances on quinoxalines as target‐oriented chemotherapeutic anticancer agents through apoptosis5
Optimization of 4‐amino‐pyridazin‐3(2H)‐one as a valid core scaffold for FABP4 inhibitors5
Exploring ibuprofen derivatives as α‐glucosidase and lipoxygenase inhibitors: Cytotoxicity and in silico studies5
4‐{3‐[(Pyridin‐4‐ylmethyl)amino]‐[1,2,4]triazolo[4,3‐b][1,2,4]triazin‐6‐yl}phenol: An improved anticancer agent in hepatocellular carcinoma and a selective MDR1/MRP modulator5
Design, synthesis, and α‐glucosidase‐inhibitory activity of phenoxy‐biscoumarin–N‐phenylacetamide hybrids5
Development of heterodimeric estrogen receptor alpha antagonists to target simultaneously the ligand and coactivator binding site5
3‐Aryl‐substituted imidazo[1,2‐a]pyridines as antituberculosis agents5
Hibiscus schizopetalus boosts wound healing via restoring redox balance and hindering inflammatory responses in rats: Insights on metabolome profiling and molecular docking5
Development of fluorinated nicotinonitriles and fused candidates as antimicrobial, antibiofilm, and enzyme inhibitors5
Novel substituted 1,8‐naphthyridines: Design, synthesis, radiolabeling, and evaluation of apoptosis and topoisomerase II inhibition5
Soft drug inhibitors for the epigenetic targets lysine‐specific demethylase 1 and histone deacetylases5
Design, synthesis, and biological evaluation of naphthalene imidazo[1,2‐b]pyridazine hybrid derivatives as VEGFR selective inhibitors5
Nanomolar potency of imidazo[2,1‐b]thiazole analogs as indoleamine 2,3‐dioxygenase inhibitors5
Valorization of Citrus peels: GC/MS‐based metabolites profiling, multivariate analysis, and antiaging potential5
Structure‐guided design of potent JAK1‐selective inhibitors based on 4‐amino‐7H‐pyrrolo[2,3‐d]pyrimidine with anti‐inflammatory efficacy5
Anticancer 5‐arylidene‐2‐(4‐hydroxyphenyl)aminothiazol‐4(5H)‐ones as tubulin inhibitors5
Benzothiazole‐based apoptosis inducers: A comprehensive overview and future prospective5
Design, synthesis, biological evaluation, and molecular modeling simulations of new phthalazine‐1,4‐dione derivatives as anti‐Alzheimer's agents5
Evaluation of in vitro SARS‐CoV‐2 inactivation by a new quaternary ammonium compound: Bromiphen bromide5
Thiophene‐containing compounds with antimicrobial activity5
Quality parameters for the medicinal plant Drosera rotundifolia L.: A new approach with established techniques5
Synthesis and molecular docking simulation of new benzimidazole–thiazole hybrids as cholinesterase inhibitors5
First‐in‐class pyrido[2,3‐d]pyrimidine‐2,4(1H,3H)‐diones against leishmaniasis and tuberculosis: Rationale, in vitro, ex vivo studies and mechanistic insights5
Synthesis of new 1,2,4‐triazole–(thio)semicarbazide hybrid molecules: Their tyrosinase inhibitor activities and molecular docking analysis5
Identification of 9H‐purin‐6‐amine derivatives as novel aldose reductase inhibitors for the treatment of diabetic complications5
Phenol—Benzoxazolone bioisosteres: Synthesis and biological evaluation of tricyclic GluN2B‐selective N‐methyl‐d‐aspartate receptor antagonists5
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