OOIR: Observatory of International Research

Papers

(The H4-Index of Bioorganic & Medicinal Chemistry Letters is 28. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2021-04-01 to 2025-04-01.)

Article	Citations
Graphical abstract TOC	150
Synthesis and SAR of novel GPR39 agonists and positive allosteric modulators	95
Graphical abstract TOC	84
Contents Continued	70
Editorial Board	64
Angucyclines containing β-ᴅ-glucuronic acid from Streptomyces sp. KCB15JA151	63
Discovery of 3-amino-4-{(3S)-3-[(2-ethoxyethoxy)methyl]piperidin-1-yl}thieno[2,3-b]pyridine-2-carboxamide (DS96432529): A potent and orally active bone anabolic agent	50
Editorial Board	49
Development of BET inhibitors as potential treatments for cancer: A new carboline chemotype	49
Design of 99mTc-labeled zinc-chelating imaging probe for SPECT imaging of the pancreas	42
A late-stage diversification via Heck-Matsuda arylation: Straightforward synthesis and cytotoxic/antiproliferative profiling of novel aryl-labdane-type derivatives	41
Synthesis and biological evaluation of cajanonic acid A derivatives as potential PPARγ antagonists	41
Graphical abstract TOC	36
Design, synthesis and analysis of novel sphingosine kinase-1 inhibitors to improve oral bioavailability	35
Discovery of GNE-502 as an orally bioavailable and potent degrader for estrogen receptor positive breast cancer	35
Design, synthesis and biological evaluation of 1,3,4-triazole-3-acetamide derivatives as potent neuraminidase inhibitors	34
Discovery of (2-phenylthiazol-4-yl)urea derivatives that induce neuronal differentiation from mesenchymal stem cells	33
Graphical abstract TOC	32
Graphical abstract TOC	32
Discovery of tricyclic HIV-1 integrase-LEDGF/p75 allosteric inhibitors by intramolecular direct arylation reaction	31
Graphical abstract TOC	30
Editorial Board	30
Design and synthesis of unique morphinan-type molecules: Their application to the search for the unexplored binding domain between opioid receptors and morphinan ligands	30
Identification of novel glucocerebrosidase chaperones by unexpected skeletal rearrangement reaction	29
Graphical abstract TOC	29

Green synthesis and anti-biofilm activities of 3,5-disubstituted isoxazoline/isoxazole-linked secondary sulfonamide derivatives on Pseudomonas aeruginosa	29
Graphical Abstract Contents Continued	28
Discovery of SHR5428 as a selective and noncovalent inhibitor of CDK7	28
Editorial Board	28