Bioorganic & Medicinal Chemistry Letters

Article	Citations
Design, synthesis and biological evaluation of tanshinone IIA derivatives as NLRP3 inflammasome inhibitors	107
Editorial Board	73
Pyrazolo-1-carbothioamides as EGR-1–DNA binding disruptors	54
Design, synthesis and characterizations of prodrugs of brexanolone	52
Discovery of TNG-6132, a potent, selective, and orally bioavailable USP1 inhibitor	50
Armeniaspirol analogues disrupt the electrical potential (ΔΨ) of the proton motive force	42
Editorial Board	37
Graphical Abstract TOC	37
Contents continued	33
Neuropilin 1-targeted near-infrared fluorescence probes for tumor diagnosis	33
Synthesis and biological evaluation of novel 1,2,3,4-tetrahydro-β-carboline derivatives as potential antibacterial agents	32
Design, synthesis and biological evaluation of alginate oligosaccharide derivatives	30
Design and evaluation of anaplastic lymphoma kinase degraders using a covalent fumarate handle	29
Studies on in vitro modulatory effects to base excision repair enzymes induced by small molecule binding to Deaminated CAG repeat hairpin	29
Enteroviral replication inhibition by N-Alkyl triazolopyrimidinone derivatives through a non-capsid binding mode	28
Design and synthesis of Tetrahydroindeno[4,5-c]chromen-4(3H)-one derivatives as antiproliferative agents for prostate Cancer cells	27
Discovery of multitargeting single agents as a novel route to the potential treatment of neurodegenerative diseases	27
Phytochemical investigation of Asarum sieboldii var. seoulense and the phenotypic profiles of its constituents against a Parkinson’s Disease olfactory cell line	26
Discovery of DS-1093a: An oral hypoxia-inducible factor prolyl hydroxylase inhibitor for the treatment of renal anemia	26
SARS-CoV-2 papain-like protease (PLpro) inhibitory and antiviral activity of small molecule derivatives for drug leads	26
Epigallocatechin and epigallocatechin-3-gallate are not inhibitors of tyrosinase	25
Improved synthesis and anticancer activity of a potent neuronal nitric oxide synthase inhibitor	24
Revisiting the dipeptidyl carboxypeptidase inhibitor captopril as a source of pan anti-trypanosomatid agents	24
Green synthesis and anti-biofilm activities of 3,5-disubstituted isoxazoline/isoxazole-linked secondary sulfonamide derivatives on Pseudomonas aeruginosa	24
Discovery of structural diverse reversible BTK inhibitors utilized to develop a novel in vivo CD69 and CD86 PK/PD mouse model	23

Development of a highly potent and selective degrader of LRRK2	23
Design and structural optimization of thiadiazole derivatives with potent GLS1 inhibitory activity	22
4′-O-methoxyethyl-2′-deoxy-uridine and cytidine ribonucleotides improve duplex stability, nuclease resistance, and elicit efficient knockdown of Bcl-2 expression	22
Synthesis and evaluation of novel oxanthrene scaffold-derived oxazolidinone antibiotics with potent antitubercular activity and low cellular toxicity	22
Discovery of a macrocyclic FAK inhibitor GZD-257 for treatment of glioblastoma	22
New class of fused [3,2-b][1,2,4]triazolothiazoles for targeting glioma in vitro	22
A PSMA-targeted doxorubicin small-molecule drug conjugate	21
A concise review on MDM2 inhibitors and recent progress in radiopharmaceutical development for imaging MDM2 expression in tumors with PET or SPECT	21
Recent progress in synthetic strategies to develop potent, HDAC8-selective, small-molecule inhibitors	21
Design and activity evaluation of new EGFR tyrosine kinase inhibitors containing cyclic polyamines	20
Contents continued	20
A simple yet multifaceted 90 years old, evergreen enzyme: Carbonic anhydrase, its inhibition and activation	20
Contents continued	20
Contents continued	20
Synthesis and evaluation of lipoic acid – donepezil hybrids for Alzheimer’s disease using a straightforward strategy	19
High-yield and high-purity amide bond formation using DMTMM PF6 for DNA-encoded libraries	19
Design, synthesis, and biological evaluation of 5ʹ-deoxy (N)-methanocarbanucleoside derivatives as A3 adenosine receptor ligands	19
DDD-028: A potent, neuroprotective, non-opioid compound for the treatment of diabetic neuropathy	19
Structure-based discovery of sulfamoyl-ethyl-4-oxo-3,4-dihydro-7H-pyrrolo[2,3-d]pyrimidine amides and sulfonamides as potent B-Cell Lymphoma 6 (BCL6)-BTB inhibitors	19
PEG-lipid-modified agonistic antibody against tumor necrosis factor receptor family elicits superior apoptosis-inducing activity against human carcinoma	18
Discovery of 3-phenyl-1H-5-pyrazolylamides as PLpro inhibitors through virtual screening and structure optimization	18
Pharmacokinetic analysis of 6-O-[18F]FEE for PET imaging of EGFR mutation	17
Graphical abstract TOC	17
Design, synthesis and properties of peptide inhibitors based on BRCA1856-871	17
Graphical abstract TOC	17
Stereochemical inversion at a 1,4-cyclohexyl PROTAC linker fine-tunes conformation and binding affinity	17
Design, synthesis and biological evaluation of novel cyano-cinnamate derivatives as mitochondrial pyruvate carrier inhibitors	17
Graphical abstract TOC	16
Exploratory study of oxatomide derivatives with high P2X7 receptor inhibitory activity	16
A photoactivatable self-localizing ligand with improved photosensitivity for chemo-optogenetic control of protein localization in living cells	16
Discovery of arylsulfonamides as a novel class of allosteric integrase inhibitors with antiviral activity	16
Graphical abstract TOC	16
Ultrasound-dependent RNAi using TatU1A-rose bengal conjugate	16
Editorial Board	16
Design, synthesis and biological evaluation of pteridine-7(8H)-one derivatives as potent and selective CDK4/6 inhibitors	16
Design and synthesis of novel fluorene derivatives as inhibitors of pyruvate dehydrogenase kinase	15
Retraction notice to “Preclinical metabolism of LB42908, a novel farnesyl transferase inhibitor, and its effects on the cytochrome P450 isozyme activities” [Bioorg. Med. Chem. Lett. 22(9) (2012) 3067–	15
Discovery and optimization of (2-naphthylthio)acetic acid derivative as selective Bfl-1 inhibitor	15
Rational design, synthesis and biological evaluation of novel HIV-1 protease inhibitors containing 2-phenylacetamide derivatives as P2 ligands with potent activity against DRV-Resistant HIV-1 variants	15
Photocrosslinking and capture for the analysis of carbohydrate-dependent interactions	15
Biocatalytic synthesis and evaluation of antioxidant and antibacterial activities of hydroxyequols	15
Design, synthesis, and evaluation of 1,3,4-oxadiazole-based EGFR inhibitors	15
Optimisation of momelotinib with improved potency and efficacy as pan-JAK inhibitor	15
Comparative analysis of p-terphenylquinone and seriniquinone derivatives as reactive oxygen species-modulating agents	15
nTZDpa (non-thiazolidinedione PPARγ partial agonist) derivatives retain antimicrobial activity without improving renal toxicity	15
11C-labeling of 20(S)-protopanaxadiol, an aglycon of ginsenoside, based on the use of Pd(0)-mediated rapid C-[11C]methylation of boronic precursors	14
Structure-activity relationship study of HIF-2α inhibitors with tricyclic scaffold	14
Synthesis and pharmacological characterization of multiply substituted 2H-chromene derivatives as P2Y6 receptor antagonists	14
Biological evaluation of newly synthesized α-benzil monoxime thiocarbohydrazide derivatives as an antimicrobial and anticancer agent: In vitro screening and ADMET predictions	14
An overview of cyclopropenone derivatives as promising bioactive molecules	14

Graphical abstract TOC	14
Synthesis and evaluation of 3-hydroxyquinolin-2(1H)-one derivatives as inhibitors of tyrosinase	14
Design, synthesis and biological evaluation of pyrimidine base hydroxamic acid derivatives as dual JMJD3 and HDAC inhibitors	14
α-Fluorination of tropane compounds and its impact on physicochemical and ADME properties	14
Discovery and optimization of 2,3-Dihydroindole derivatives as STING receptor allosteric agonists	14
Natural products targeting the NF-κB signaling pathway:Potential therapeutic drug candidates	13
Potent and selective carbonic anhydrase inhibition activities of pyrazolones bearing benzenesulfonamides	13
(E)-3-(3-([1,1′-Biphenyl]-4-yl)-1-phenyl-1H-pyrazol-4-yl)-1-phenylprop-2-en-1-ones inducing reactive oxygen species generation through glutathione depletion	13
Editorial Board	13
Syntheses and antitumor activities of neorautenol and shinpterocarpin analogs	13
Editorial Board	13
Neratinib derivative 7A induces apoptosis in colon cancer cells via the p53 pathway	13
Graphical abstract TOC	13
Graphical abstract TOC	13
Lysine-reactive tag system for cell-surface protein labeling via N-acyl-N-alkyl sulfonamide chemistry	13
Design, synthesis, and antitumor activity study of novel oleanolic acid structural derivatives targeting c-Kit	13
Structure-activity relationship of dual inhibitors containing maleimide and imidazole motifs against glutaminyl cyclase and glycogen synthase kinase-3β	13
Graphical abstract TOC	13
6-Aryl-quinazolines as novel GABAB receptor positive allosteric modulators	13
Structure–activity relationship of 2-aminodibenzothiophene pharmacophore and the discovery of aminobenzothiophenes as potent inhibitors of Mycobacterium smegmatis	13
Discovery of novel 4-aminobenzamide derivatives as small molecule CBX2 inhibitors	12
Identification of potent and selective inhibitors of PKR via virtual screening and traditional design	12
Study of the reversal of metallo-β-lactamase-mediated resistance in Gram-negative bacteria by EDTMP	12
Enzymatic reconstitution of salicylate formation in promysalin biosynthesis	12
Structure-activity relationship of dibenzylideneacetone analogs against the neglected disease pathogen, Trypanosoma brucei	12
Graphical abstract TOC	12
Discovery of triazenyl triazoles as Nav1.1 channel blockers for treatment of epilepsy	12
Design, synthesis, in silico studies, and antiproliferative evaluations of novel indolin-2-one derivatives containing 3-hydroxy-4-pyridinone fragment	12
Design, synthesis and anti-pneumonic activity evaluation of shikonin ester derivatives	12
Strengths and limitations of Ba/F3 cells in modelling FLT3-driven AML resistance	12
Graphical abstract TOC	12
Design, synthesis and evaluation of clickable photoaffinity probes for nuclear lamins	12
Discovery of sinomenine/8-Bis(benzylthio)octanoic acid hybrids as potential anti-leukemia drug candidate via mitochondrial pathway	12
Discovery of novel N-(1-benzyl-1H-imidazol-2-yl)amide derivatives as melanocortin 1 receptor agonists	12
Contents continued	12
Editorial Board	12
Design, synthesis and activity evaluation of Hedgehog inhibitor Itraconazole derivatives in A549 cells	11
Exploration of imidazothiazole and imidazopyrimidine carboxamides for enhanced antitubercular activity	11
Improving reactivity of naphthalimide-based GST probe by imparting TPP cation: Development and application for live cell imaging	11
Discovery of N-Ts-3-benzylidene-indolin-2-imines as potent anti-colorectal cancer agents through suppression of the PI3K-AKT pathway	11
Reinvestigation of clopidogrel bioactivation unveils new cytochrome P450-catalyzed thioester cleavage mechanism	11
Graphical abstract TOC	11
Discovery and characterization a new collagenase from Hathewaya massiliensis for effective subcutaneous adipolysis	11
Synthesis of a tricyclic hexapeptide –via two consecutive ruthenium-catalyzed macrocyclization steps– with a constrained topology to mimic vancomycin's binding properties toward D-Ala-D-Ala dipeptide	11
Design, synthesis and biological evaluation of cajanonic acid A analogues as potent PPAR γ antagonists	11
Recent advances and perspectives in therapeutics for mpox	11
Direct-to-biology platform: From synthesis to biological evaluation of SHP2 allosteric inhibitors	11
Phenyl urea based adjuvants for β-lactam antibiotics against methicillin resistant Staphylococcus aureus	11
Contents continued	11
Synthesis of dolutegravir derivatives modified by 1,2,3-triazole structure and their anti-inflammatory activity in LPS-induced BV2 cells	11
Synthesis of a new series of quinoline/pyridine indole-3-sulfonamide hybrids as selective carbonic anhydrase IX inhibitors	11
Investigation of the site 2 pocket of Grp94 with KUNG65 benzamide derivatives	11
Design, synthesis, and biological evaluation of polyphenol derivatives as DYRK1A inhibitors. The discovery of a potentially promising treatment for Multiple Sclerosis	11
Design, synthesis and biological evaluation of novel cationic liposomes loaded with melphalan for the treatment of cancer	11
Contents continued	11
Design, synthesis and evaluation of pterostilbene-indole hybrids as potential anticancer agents	11
Iodophenyl-conjugated closo-dodecaborate as a promising small boron molecule that binds to serum albumin and accumulates in tumor	10
A small molecule binding to TGGAA pentanucleotide repeats that cause spinocerebellar ataxia type 31	10
Editorial Board	10
Synthesis, modeling, and biological evaluation of anti-tubulin indole-substituted furanones	10
Hydrazinecarbonyl-thiazol-2-acetamides with pronounced apoptotic behavior: synthesis, in vitro/in vivo anti-proliferative activity and molecular modeling simulations	10
Discovery of a potent orally available pyrazolopyridone derivative as a novel selective bromodomain and extra-terminal domain (BET)-first bromodomain (BD1) inhibitor	10
The Pyrimidinyl Hydrazones: Selective for anti-Cancer cytotoxicity	10
Evaluation of an ester-linked immunosuppressive payload: A case study in understanding the stability and cleavability of ester-containing ADC linkers	10
Corrigendum to “Discovery of 4-aminopyrimidine analogs as highly potent dual P70S6K/Akt inhibitors” [Bioorgan. Med. Chem. Lett. 50 (2021) 128352]	10
Harnessing dual-mode RIPK1 ligands for cross-species anti-necroptosis inhibitor compounds	10
Design, synthesis and antitumor evaluation of a novel nectin-4 targeting bicyclic toxin conjugate	10
Synthesis of substrate peptides incorporating non-natural amino acids and screening study using BACE1	10
Permeation behavior of porphyrin derivatives with different functional group positions across cancer cell membranes	10
A guanidinium group is an effective mimic of the tertiary carbocation formed by isopentenyl diphosphate isomerase	10
Synthesis and functional evaluation of tetrahydroisoquinoline and polysubstituted benzylamine derivatives as sigma-2 receptor-targeted small-molecule probes	10
New diarylpentanoids and chalcones as potential antimicrobial adjuvants	10
Synthesis and biological evaluation of biotinylated ZJ-101	10
PSMA-targeted SMART molecules outfitted with SN38	10
A small-molecule pretargeting approach for PSMA-targeted conjugates	10
Novel drug discovery approaches for MMP-13 inhibitors in the treatment of osteoarthritis	10
Development of novel GI-centric prostaglandin E2 receptor type 4 (EP4) agonist prodrugs as treatment for ulcerative colitis and other intestinal inflammatory diseases	10
Synthesis of mizoribine prodrugs and their in vivo evaluation as immunosuppressive agents	10
Further structural optimization and SAR study of sungsanpin derivatives as cell-invasion inhibitors	10
Methyl N-(tert-butoxycarbonyl)pyridine-2-carbimidothioate: A new reagent for the synthesis of N-phenylpyridinecarboxamidine (“arylimidamide”) DNA-minor groove binders from poorly nucleophilic amines	10

Discovery of a proteolysis targeting chimera (PROTAC) as a potent regulator of FOXP3	10
Graphical abstract TOC	10
Graphical abstract TOC	10
Graphical abstract TOC	10
Discovery of 3-acyl-2-anilino-1,4-dihydroquinolin-4-one derivatives as potential inhibitors of methicillin-resistant Staphylococcus aureus	10
Zinc-dependent deacetylases (HDACs) as potential targets for treating Alzheimer’s disease	10
Design, synthesis, and bioevaluation of SOS1 PROTACs derived from pyrido[2,3-d]pyrimidin-7-one-based SOS1 inhibitor	9
Contents continued	9
Synthesis of esters and amides of 2-aryl-1-hydroxy-4-methyl-1H-imidazole-5-carboxylic acids and study of their antiviral activity against orthopoxviruses	9
Graphical abstract TOC	9
Synthesis, in vitro cytotoxicity evaluation and mechanism of 5′ monosubstituted chalcone derivatives as antitumor agents	9
Highly potent anti-inflammatory, analgesic and antioxidant activities of 3,5-disubstituted tetrahydro-2H-1,3,5-thiadiazine thiones	9
Design, synthesis and biological evaluation of novel indole-piperazine derivatives as antibacterial agents	9
Synthesis and preliminary immunologic properties of di-/trisaccharide-conjugates related to Bacillus anthracis	9
Conversion of oxadiazolo[3,4-b]pyrazines to imidazo[4,5-b]pyrazines via a tandem reduction-cyclization sequence generates new mitochondrial uncouplers	9
A FOXC2 inhibitor, MC-1-F2, as a therapeutic candidate for targeting EMT in castration-resistant prostate cancer	9
Design, synthesis, and biological evaluation of 2,4-diaminopyrimidine inhibitors of hematopoietic progenitor kinase 1	9
Discovery of a potent and subtype-selective TYK2 degrader based on an allosteric TYK2 inhibitor	9
Discovery of BI-9787, a potent zwitterionic ketohexokinase inhibitor with oral bioavailability	9
Cyano-Hydrol green derivatives: Expanding the 9-cyanopyronin-based resonance Raman vibrational palette	9
5-Fluoro-2′-deoxyuridine as an efficient 19F NMR reporter for G-quadruplex and i-motif structures	9
Photo-regulated PROTACs: A novel tool for temporal control of targeted protein degradation	9
Editorial Board	9
Discovery of an ellipticine derivative as TLR3 inhibitor against influenza A virus and SARS-CoV-2	9
Editorial Board	9
A potent and selective RORγ inhibitor for the treatment of autoimmune diseases	9
Synthesis of drimanyl indole fragments of drimentine alkaloids and their antibacterial activities	9
Synthesis of triazolopyrimidinone- and imidazotriazinone-based tankyrase inhibitors: Identification of Basroparib (STP1002) as a clinical candidate	9
Genipin derivative induced the apoptosis and inhibited the invasion and migration of A549 cancer cells via regulation of EGFR/JAK1/STAT3 signaling	9
Imidazo[2,1-b]thiazole based indoleamine-2,3-dioxygenase 1 (IDO1) inhibitor: Structure based design, synthesis, bio-evaluation and docking studies	9
Discovery of acyl ureas as highly selective small molecule CSF1R kinase inhibitors	9
Graphical abstract TOC	8
Discovery of novel imidazo[4,5-b]pyridine derivatives as noncovalent reversible Bruton’s tyrosine kinase inhibitors	8
Short synthesis of a broadly Reactive, cell permeable serine hydrolase Fluorophosphonate-Alkyne probe	8
Development of chromone-thiazolidine-2,4-dione Knoevenagel conjugates as apoptosis inducing agents	8
Graphical Abstract TOC	8
Graphical Abstract Contents Continued	8
Synthesis of proposed structure of ledebourin A	8
Discovery of a DCAF11-dependent cyanoacrylamide-containing covalent degrader of BET-proteins	8
An ascidian Polycarpa aurata-derived pan-inhibitor against coronaviruses targeting Mpro	8
Graphical abstract TOC	8
Graphical abstract TOC	8
Design, synthesis, and biological evaluation of novel HDAC inhibitors with a 3-(benzazol-2-yl)quinoxaline framework	8
SAR study of niclosamide derivatives for neuroprotective function in SH-SY5Y neuroblastoma	8
Synthesis, antiproliferative activity, and biological profiling of C-19 trityl and silyl ether andrographolide analogs in colon cancer and breast cancer cells	8
Recent developments of benzimidazole based analogs as potential tubulin polymerization inhibitors: A critical review	8
Graphical Abstract TOC	8
Design of cyclic peptides as novel inhibitors of ICOS/ICOSL interaction	8
Synthesis and properties of PNA containing a dicationic nucleobase based on N4-benzoylated cytosine	8
Exploration of inhibitors of the bacterial LexA repressor-protease	8
Design, synthesis and antitumor activity of novel 4-oxobutanamide derivatives	8
Synthesis and evaluation of catecholamine derivatives as amyloid-beta aggregation inhibitors	8
Multifaceted roles of HDAC7 in disease and the evolving chemical toolkit for its modulation	8
The structural modification and biological evaluation of tetrahydrothienopyridine derivatives as selective BChE inhibitors	8
Synthesis and antitumor activity of a series of novel N-aryl-5-(2,2,2-trifluoroethoxy)-1,5-dihydro-2H-pyrrol-2-ones derivatives	8
Sensitive and reliable gastric ulcer related MicroRNA detection by bridge catalytic hairpin assembly (bCHA) mediated primer exchange reaction	8
Diamino variants of piperazine-based tissue transglutaminase inhibitors	8
Design, synthesis and evaluation of the Brigatinib analogues as potent inhibitors against tertiary EGFR mutants (EGFRdel19/T790M/C797S and EGFRL858R/T790M/C797S)	8
Graphical abstract TOC	8
Multigram-scale total synthesis of (±)-ambreinolide by a diastereoselective polyene cyclization	8
Design, synthesis, and antibacterial activity evaluation of tryptanthrin derivatives	8
Thiamine analogues featuring amino-oxetanes as potent and selective inhibitors of pyruvate dehydrogenase	8
Targeted design, synthesis, molecular simulation, ADME-T and in-vitro anticancer assessment of phenyl-substituted-thioxo-tetrahydro-pyrimidin-benzenesulfonamide derivatives as potential BRAFV600E/WT i	8
Design, synthesis, and activity evaluation of Asiatic acid derivatives as Survivin inhibitors	8
Contents continued	8
Novel imidazo[1,5-a]quinoxaline derivatives: SAR, selectivity and modeling challenges en route to the identification of an α5-GABAA receptor NAM	8
Design, synthesis and antifungal activities of novel triazole derivatives with selenium-containing hydrophobic side chains	7
Discovery of benzimidazole-2-amide BNZ-111 as new tubulin inhibitor	7
Lipid bilayer membrane permeability mechanism of the K-Ras(G12D)-inhibitory bicyclic peptide KS-58 elucidated by molecular dynamics simulations	7
Recent advances of the respiratory syncytial virus inhibitors	7
Identification of small molecule activators targeting TYK2 pseudokinase domain	7
The potential of Rhein's aromatic amines for Parkinson's disease prevention and treatment: α-Synuclein aggregation inhibition and disaggregation of preformed fibers	7
Discovery of L15 as a novel Vif PROTAC degrader with antiviral activity against HIV-1	7
Identification of (−)-Epigallocateshin gallate derivatives promoting innate immune activation via 2′,3′-cyclic GMP-AMP-stimulator of interferon genes pathway	7
Siderophores: Chemical tools for precise antibiotic delivery	7
Identification of sugar-containing natural products that interact with i-motif DNA	7
A self-assembling peptide platform enables plasma membrane protein degradation	7
Editorial Board	7
Graphical abstract TOC	7
Modification of the phenyl ring B of phenyl 4-(2-oxoimidazolidin-1-yl)benzenesulfonates by pyridinyl moiety leads to novel antimitotics targeting the colchicine-binding site	7
Discovery of PFI-6, a small-molecule chemical probe for the YEATS domain of MLLT1 and MLLT3	7
Split luciferase-based estimation of cytosolic cargo concentration delivered intracellularly via attenuated cationic amphiphilic lytic peptides	7
Rational design, synthesis, antiproliferative activity against MCF-7, MDA-MB-231 cells, estrogen receptors binding affinity, and computational study of indenopyrimidine-2,5-dione analogs for the treat	7
The association between oxidized low-density lipoprotein and cancer: An emerging targeted therapeutic approach?	7
Discovery of EP300/CBP histone acetyltransferase inhibitors through scaffold hopping of 1,4-oxazepane ring	7
Thermal treatment affects aptamers’ structural profiles	7
Inhibition of glutathione S-transferases by photoactive calix[4]arene α-ketophosphonic acids	7
Synthesis and analysis of novel catecholic ligands as inhibitors of catechol-O-methyltransferase	7
A conformationally-locked p-hydroxybenzylidene imidazolinone derivative for detecting Aβ42 aggregation	7
Discovery of 5-methyl-1H-benzo[d]imidazole derivatives as novel P2X3 Receptor antagonists	7
Inhibitors for metallo-β-lactamases from the B1 and B3 subgroups provide an avenue to combat a major mechanism of antibiotic resistance	7
Discovery of the potent covalent inhibitor with an acrylate warhead for SARS-CoV-2 3CL protease	7
Diffusion of 1O2 along the PNA backbone diminishes the efficiency of photooxidation of PNA/DNA duplexes by biphenyl photosensitizer	7
Fragment-based discovery of novel phenyltriazolyl derivatives as allosteric type-I1/2 ALK inhibitors with promising antitumor effects	7
Discovery of 4-((quinolin-8-ylthio)methyl)benzamide derivatives as a new class of SARS-CoV-2 nsp13 inhibitors	7