Bioorganic & Medicinal Chemistry Letters

Article	Citations
Revisiting the dipeptidyl carboxypeptidase inhibitor captopril as a source of pan anti-trypanosomatid agents	157
Design, synthesis and biological evaluation of alginate oligosaccharide derivatives	86
Design, synthesis and biological evaluation of tanshinone IIA derivatives as NLRP3 inflammasome inhibitors	83
Studies on in vitro modulatory effects to base excision repair enzymes induced by small molecule binding to Deaminated CAG repeat hairpin	62
Discovery of DS-1093a: An oral hypoxia-inducible factor prolyl hydroxylase inhibitor for the treatment of renal anemia	59
Epigallocatechin and epigallocatechin-3-gallate are not inhibitors of tyrosinase	53
Editorial Board	46
Armeniaspirol analogues disrupt the electrical potential (ΔΨ) of the proton motive force	44
Pyrazolo-1-carbothioamides as EGR-1–DNA binding disruptors	38
Design of 99mTc-labeled zinc-chelating imaging probe for SPECT imaging of the pancreas	34
Non-alkylator anti-glioblastoma agents induced cell cycle G2/M arrest and apoptosis: Design, in silico physicochemical and SAR studies of 2-aminoquinoline-3-carboxamides	34
Discovery of structural diverse reversible BTK inhibitors utilized to develop a novel in vivo CD69 and CD86 PK/PD mouse model	33
Phytochemical investigation of Asarum sieboldii var. seoulense and the phenotypic profiles of its constituents against a Parkinson’s Disease olfactory cell line	31
Improved synthesis and anticancer activity of a potent neuronal nitric oxide synthase inhibitor	30
Design, synthesis and characterizations of prodrugs of brexanolone	28
Discovery of 3-amino-4-{(3S)-3-[(2-ethoxyethoxy)methyl]piperidin-1-yl}thieno[2,3-b]pyridine-2-carboxamide (DS96432529): A potent and orally active bone anabolic agent	28
Development of a highly potent and selective degrader of LRRK2	27
Design and structural optimization of thiadiazole derivatives with potent GLS1 inhibitory activity	26
Editorial Board	25
SARS-CoV-2 papain-like protease (PLpro) inhibitory and antiviral activity of small molecule derivatives for drug leads	24
Editorial Board	24
New class of fused [3,2-b][1,2,4]triazolothiazoles for targeting glioma in vitro	24
Enteroviral replication inhibition by N-Alkyl triazolopyrimidinone derivatives through a non-capsid binding mode	24
Synthesis and characterization of chiral 6-azaspiro[2.5]octanes as potent and selective antagonists of the M4 muscarinic acetylcholine receptor	24
Graphical Abstract TOC	23

Neuropilin 1-targeted near-infrared fluorescence probes for tumor diagnosis	22
Discovery of TNG-6132, a potent, selective, and orally bioavailable USP1 inhibitor	21
A PSMA-targeted doxorubicin small-molecule drug conjugate	20
Contents continued	20
Design and evaluation of anaplastic lymphoma kinase degraders using a covalent fumarate handle	20
A simple yet multifaceted 90 years old, evergreen enzyme: Carbonic anhydrase, its inhibition and activation	19
A fluorescent molecular rotor for the selective detection of the hybrid-conformation 22AG G-Quadruplex	19
Novel carbohydrate-based sulfonamide derivatives as selective carbonic anhydrase II inhibitors: Synthesis, biological and molecular docking analysis	19
Green synthesis and anti-biofilm activities of 3,5-disubstituted isoxazoline/isoxazole-linked secondary sulfonamide derivatives on Pseudomonas aeruginosa	19
Synthesis and evaluation of 3-hydroxyquinolin-2(1H)-one derivatives as inhibitors of tyrosinase	18
Design and activity evaluation of new EGFR tyrosine kinase inhibitors containing cyclic polyamines	18
Synthesis and biological evaluation of novel 1,2,3,4-tetrahydro-β-carboline derivatives as potential antibacterial agents	18
New bis- and tetrakis-1,2,3-triazole derivatives: Synthesis, DNA cleavage, molecular docking, antimicrobial, antioxidant activity and acid dissociation constants	18
Synthesis and evaluation of lipoic acid – donepezil hybrids for Alzheimer’s disease using a straightforward strategy	18
Contents continued	18
Synthesis and SAR of novel GPR39 agonists and positive allosteric modulators	18
Contents continued	18
Contents continued	18
Amyloidogenic immunoglobulin light chain kinetic stabilizers comprising a simple urea linker module reveal a novel binding sub-site	18
Design, synthesis, biological evaluation and molecular modeling of N-isobutyl-N-((2-(p-tolyloxymethyl)thiazol-4yl)methyl)benzo[d][1,3] dioxole-5-carboxamides as selective butyrylcholinesterase inhibit	18
PEG-lipid-modified agonistic antibody against tumor necrosis factor receptor family elicits superior apoptosis-inducing activity against human carcinoma	17
Design, synthesis, and biological evaluation of 5ʹ-deoxy (N)-methanocarbanucleoside derivatives as A3 adenosine receptor ligands	17
Design, synthesis and properties of peptide inhibitors based on BRCA1856-871	17
Retraction notice to “Preclinical metabolism of LB42908, a novel farnesyl transferase inhibitor, and its effects on the cytochrome P450 isozyme activities” [Bioorg. Med. Chem. Lett. 22(9) (2012) 3067–	17
Discovery of 3-phenyl-1H-5-pyrazolylamides as PLpro inhibitors through virtual screening and structure optimization	17
An overview of cyclopropenone derivatives as promising bioactive molecules	17
α-Fluorination of tropane compounds and its impact on physicochemical and ADME properties	17
Comparative analysis of p-terphenylquinone and seriniquinone derivatives as reactive oxygen species-modulating agents	16
Design and discovery of C2-fluoroalkyl iminothiazine dioxides as BACE inhibitors	16
Editorial Board	16
Exploratory study of oxatomide derivatives with high P2X7 receptor inhibitory activity	16
Biocatalytic synthesis and evaluation of antioxidant and antibacterial activities of hydroxyequols	16
Graphical abstract TOC	16
Design, synthesis and biological evaluation of pteridine-7(8H)-one derivatives as potent and selective CDK4/6 inhibitors	16
DDD-028: A potent, neuroprotective, non-opioid compound for the treatment of diabetic neuropathy	16
Graphical abstract TOC	16
Discovery and optimization of (2-naphthylthio)acetic acid derivative as selective Bfl-1 inhibitor	16
Identification and evaluation of 4-anilinoquin(az)olines as potent inhibitors of both dengue virus (DENV) and Venezuelan equine encephalitis virus (VEEV)	16
Graphical abstract TOC	16
nTZDpa (non-thiazolidinedione PPARγ partial agonist) derivatives retain antimicrobial activity without improving renal toxicity	15
Ultrasound-dependent RNAi using TatU1A-rose bengal conjugate	15
Discovery of arylsulfonamides as a novel class of allosteric integrase inhibitors with antiviral activity	15
A photoactivatable self-localizing ligand with improved photosensitivity for chemo-optogenetic control of protein localization in living cells	15
Graphical abstract TOC	15
Optimisation of momelotinib with improved potency and efficacy as pan-JAK inhibitor	15
Rational design, synthesis and biological evaluation of novel HIV-1 protease inhibitors containing 2-phenylacetamide derivatives as P2 ligands with potent activity against DRV-Resistant HIV-1 variants	15
Topoisomerase IIα inhibitory and antiproliferative activity of dihydroxylated 2,6-diphenyl-4-fluorophenylpyridines: Design, synthesis, and structure-activity relationships	15
Design, synthesis and biological evaluation of novel procaine derivatives for intravenous anesthesia	14
Design, synthesis and biological evaluation of pyrimidine base hydroxamic acid derivatives as dual JMJD3 and HDAC inhibitors	14
Structure-activity relationship of dual inhibitors containing maleimide and imidazole motifs against glutaminyl cyclase and glycogen synthase kinase-3β	14

Synthesis and evaluation of potent novel inhibitors of human sulfide:quinone oxidoreductase	14
Synthesis and pharmacological characterization of multiply substituted 2H-chromene derivatives as P2Y6 receptor antagonists	14
High-yield and high-purity amide bond formation using DMTMM PF6 for DNA-encoded libraries	14
Pharmacokinetic analysis of 6-O-[18F]FEE for PET imaging of EGFR mutation	14
Design, synthesis and biological evaluation of novel cyano-cinnamate derivatives as mitochondrial pyruvate carrier inhibitors	14
Design, synthesis, and evaluation of 1,3,4-oxadiazole-based EGFR inhibitors	14
Design and synthesis of novel fluorene derivatives as inhibitors of pyruvate dehydrogenase kinase	14
pH-responsive aggregates consisted of oligodeoxynucleotides bearing nitrophenol group that deliver drugs into acidic cells	14
Biological evaluation of newly synthesized α-benzil monoxime thiocarbohydrazide derivatives as an antimicrobial and anticancer agent: In vitro screening and ADMET predictions	14
Photocrosslinking and capture for the analysis of carbohydrate-dependent interactions	14
Editorial Board	14
Stereochemical inversion at a 1,4-cyclohexyl PROTAC linker fine-tunes conformation and binding affinity	14
Synthesis of a new series of quinoline/pyridine indole-3-sulfonamide hybrids as selective carbonic anhydrase IX inhibitors	13
A dual aurora and lim kinase inhibitor reduces glioblastoma proliferation and invasion	13
Synthesis of dolutegravir derivatives modified by 1,2,3-triazole structure and their anti-inflammatory activity in LPS-induced BV2 cells	13
Phenyl urea based adjuvants for β-lactam antibiotics against methicillin resistant Staphylococcus aureus	13
(E)-3-(3-([1,1′-Biphenyl]-4-yl)-1-phenyl-1H-pyrazol-4-yl)-1-phenylprop-2-en-1-ones inducing reactive oxygen species generation through glutathione depletion	13
Investigation of the site 2 pocket of Grp94 with KUNG65 benzamide derivatives	13
Design, synthesis and biological evaluation of cajanonic acid A analogues as potent PPAR γ antagonists	13
Graphical abstract TOC	13
Potent and selective carbonic anhydrase inhibition activities of pyrazolones bearing benzenesulfonamides	13
Rationalizing the binding and α subtype selectivity of synthesized imidazodiazepines and benzodiazepines at GABAA receptors by using molecular docking studies	13
Neratinib derivative 7A induces apoptosis in colon cancer cells via the p53 pathway	13
Graphical abstract TOC	12
Identification of potent and selective inhibitors of PKR via virtual screening and traditional design	12
Graphical abstract TOC	12
Improving reactivity of naphthalimide-based GST probe by imparting TPP cation: Development and application for live cell imaging	12
Reinvestigation of clopidogrel bioactivation unveils new cytochrome P450-catalyzed thioester cleavage mechanism	12
Graphical abstract TOC	12
A unified “top-down” approach for the synthesis of diverse lead-like molecular scaffolds	12
Direct-to-biology platform: From synthesis to biological evaluation of SHP2 allosteric inhibitors	12
Contents continued	12
Design, synthesis, in silico studies, and antiproliferative evaluations of novel indolin-2-one derivatives containing 3-hydroxy-4-pyridinone fragment	12
Editorial Board	12
Design, synthesis, and biological evaluation of polyphenol derivatives as DYRK1A inhibitors. The discovery of a potentially promising treatment for Multiple Sclerosis	12
Discovery of triazenyl triazoles as Nav1.1 channel blockers for treatment of epilepsy	11
6-Aryl-quinazolines as novel GABAB receptor positive allosteric modulators	11
Enzymatic reconstitution of salicylate formation in promysalin biosynthesis	11
Structure–activity relationship of 2-aminodibenzothiophene pharmacophore and the discovery of aminobenzothiophenes as potent inhibitors of Mycobacterium smegmatis	11
Graphical Abstract Contents Continued	11
Discovery of sinomenine/8-Bis(benzylthio)octanoic acid hybrids as potential anti-leukemia drug candidate via mitochondrial pathway	11
Editorial Board	11
Syntheses and antitumor activities of neorautenol and shinpterocarpin analogs	11
Structure-activity relationship of dibenzylideneacetone analogs against the neglected disease pathogen, Trypanosoma brucei	11
Synthesis of a tricyclic hexapeptide –via two consecutive ruthenium-catalyzed macrocyclization steps– with a constrained topology to mimic vancomycin's binding properties toward D-Ala-D-Ala dipeptide	11
Design, synthesis and biological evaluation of novel cationic liposomes loaded with melphalan for the treatment of cancer	11
Design, synthesis and activity evaluation of Hedgehog inhibitor Itraconazole derivatives in A549 cells	11
Graphical Abstract Continued	11
Discovery of novel N-(1-benzyl-1H-imidazol-2-yl)amide derivatives as melanocortin 1 receptor agonists	11
Photo-regulated PROTACs: A novel tool for temporal control of targeted protein degradation	10
Development of novel GI-centric prostaglandin E2 receptor type 4 (EP4) agonist prodrugs as treatment for ulcerative colitis and other intestinal inflammatory diseases	10
Strengths and limitations of Ba/F3 cells in modelling FLT3-driven AML resistance	10
Novel drug discovery approaches for MMP-13 inhibitors in the treatment of osteoarthritis	10
Discovery of a potent and subtype-selective TYK2 degrader based on an allosteric TYK2 inhibitor	10
Synthesis of mizoribine prodrugs and their in vivo evaluation as immunosuppressive agents	10
Design, synthesis, and bioevaluation of SOS1 PROTACs derived from pyrido[2,3-d]pyrimidin-7-one-based SOS1 inhibitor	10
Graphical abstract TOC	10
PSMA-targeted SMART molecules outfitted with SN38	10
Synthesis of esters and amides of 2-aryl-1-hydroxy-4-methyl-1H-imidazole-5-carboxylic acids and study of their antiviral activity against orthopoxviruses	10
Discovery of a proteolysis targeting chimera (PROTAC) as a potent regulator of FOXP3	10
A small-molecule pretargeting approach for PSMA-targeted conjugates	10
Contents continued	10
Discovery of 3-acyl-2-anilino-1,4-dihydroquinolin-4-one derivatives as potential inhibitors of methicillin-resistant Staphylococcus aureus	10
Graphical abstract TOC	10
A guanidinium group is an effective mimic of the tertiary carbocation formed by isopentenyl diphosphate isomerase	10
Synthesis, in vitro cytotoxicity evaluation and mechanism of 5′ monosubstituted chalcone derivatives as antitumor agents	10
Graphical abstract TOC	10
Graphical abstract TOC	10
Design, synthesis and antitumor evaluation of a novel nectin-4 targeting bicyclic toxin conjugate	10
Discovery of a potent orally available pyrazolopyridone derivative as a novel selective bromodomain and extra-terminal domain (BET)-first bromodomain (BD1) inhibitor	10
Cyano-Hydrol green derivatives: Expanding the 9-cyanopyronin-based resonance Raman vibrational palette	10
Contents continued	10
Harnessing dual-mode RIPK1 ligands for cross-species anti-necroptosis inhibitor compounds	10
Permeation behavior of porphyrin derivatives with different functional group positions across cancer cell membranes	10
Highly potent anti-inflammatory, analgesic and antioxidant activities of 3,5-disubstituted tetrahydro-2H-1,3,5-thiadiazine thiones	10
A small molecule binding to TGGAA pentanucleotide repeats that cause spinocerebellar ataxia type 31	10
Graphical abstract TOC	10
Evaluation of an ester-linked immunosuppressive payload: A case study in understanding the stability and cleavability of ester-containing ADC linkers	10
Synthesis of substrate peptides incorporating non-natural amino acids and screening study using BACE1	10
Synthesis and biological evaluation of biotinylated ZJ-101	9

Editorial Board	9
Contents continued	9
Discovery of an ellipticine derivative as TLR3 inhibitor against influenza A virus and SARS-CoV-2	9
Editorial Board	9
Identification of Plasmodium falciparum falcilysin inhibitors by a virtual screen	9
Thiamine analogues featuring amino-oxetanes as potent and selective inhibitors of pyruvate dehydrogenase	9
Design, synthesis and evaluation of the Brigatinib analogues as potent inhibitors against tertiary EGFR mutants (EGFRdel19/T790M/C797S and EGFRL858R/T790M/C797S)	9
5-Fluoro-2′-deoxyuridine as an efficient 19F NMR reporter for G-quadruplex and i-motif structures	9
Zinc-dependent deacetylases (HDACs) as potential targets for treating Alzheimer’s disease	9
SAR study of niclosamide derivatives for neuroprotective function in SH-SY5Y neuroblastoma	9
Design, synthesis, and biological evaluation of 2,4-diaminopyrimidine inhibitors of hematopoietic progenitor kinase 1	9
Iodophenyl-conjugated closo-dodecaborate as a promising small boron molecule that binds to serum albumin and accumulates in tumor	9
Synthesis, modeling, and biological evaluation of anti-tubulin indole-substituted furanones	9
New diarylpentanoids and chalcones as potential antimicrobial adjuvants	9
Synthesis and evaluation of catecholamine derivatives as amyloid-beta aggregation inhibitors	9
Hydrazinecarbonyl-thiazol-2-acetamides with pronounced apoptotic behavior: synthesis, in vitro/in vivo anti-proliferative activity and molecular modeling simulations	9
Graphical abstract TOC	9
Synthesis and properties of PNA containing a dicationic nucleobase based on N4-benzoylated cytosine	9
Synthesis, antiproliferative activity, and biological profiling of C-19 trityl and silyl ether andrographolide analogs in colon cancer and breast cancer cells	9
Design, synthesis and biological evaluation of sulfonylurea derivatives as NLRP3 inflammasome inhibitors	9
Editorial Board	9
Design, synthesis, and activity evaluation of Asiatic acid derivatives as Survivin inhibitors	9
Imidazo[2,1-b]thiazole based indoleamine-2,3-dioxygenase 1 (IDO1) inhibitor: Structure based design, synthesis, bio-evaluation and docking studies	9
An ascidian Polycarpa aurata-derived pan-inhibitor against coronaviruses targeting Mpro	9
Discovery of BI-9787, a potent zwitterionic ketohexokinase inhibitor with oral bioavailability	9
Corrigendum to “Discovery of 4-aminopyrimidine analogs as highly potent dual P70S6K/Akt inhibitors” [Bioorgan. Med. Chem. Lett. 50 (2021) 128352]	9
PES derivative PESA is a potent tool to globally profile cellular targets of PES	9
Further structural optimization and SAR study of sungsanpin derivatives as cell-invasion inhibitors	9
Conversion of oxadiazolo[3,4-b]pyrazines to imidazo[4,5-b]pyrazines via a tandem reduction-cyclization sequence generates new mitochondrial uncouplers	9
Diamino variants of piperazine-based tissue transglutaminase inhibitors	9
Synthesis of drimanyl indole fragments of drimentine alkaloids and their antibacterial activities	9
Synthesis and antitumor activity of a series of novel N-aryl-5-(2,2,2-trifluoroethoxy)-1,5-dihydro-2H-pyrrol-2-ones derivatives	9
Graphical abstract TOC	9
Design, synthesis, and biological evaluation of novel HDAC inhibitors with a 3-(benzazol-2-yl)quinoxaline framework	9
Design, synthesis and antitumor activity of novel 4-oxobutanamide derivatives	9
Graphical abstract TOC	9
Synthesis and preliminary immunologic properties of di-/trisaccharide-conjugates related to Bacillus anthracis	9
Design, synthesis and biological evaluation of novel indole-piperazine derivatives as antibacterial agents	9
Short synthesis of a broadly Reactive, cell permeable serine hydrolase Fluorophosphonate-Alkyne probe	9
Methyl N-(tert-butoxycarbonyl)pyridine-2-carbimidothioate: A new reagent for the synthesis of N-phenylpyridinecarboxamidine (“arylimidamide”) DNA-minor groove binders from poorly nucleophilic amines	9
Multigram-scale total synthesis of (±)-ambreinolide by a diastereoselective polyene cyclization	8
Graphical abstract TOC	8
Editorial Board	8
Graphical Abstract Contents Continued	8
Graphical abstract TOC	8
Recent developments of benzimidazole based analogs as potential tubulin polymerization inhibitors: A critical review	8
Structural basis of the C-terminal domain of SARS-CoV-2 N protein in complex with GMP reveals critical residues for RNA interaction	8
Synthesis of proposed structure of ledebourin A	8
Semisynthetic derivatives of the fungal metabolite eupenifeldin via targeting the tropolone hydroxy groups	8
A FOXC2 inhibitor, MC-1-F2, as a therapeutic candidate for targeting EMT in castration-resistant prostate cancer	8
Discovery of benzimidazole-2-amide BNZ-111 as new tubulin inhibitor	8
4-Oxooctahydroquinoline-1(2H)-carboxamides as hepatitis B virus (HBV) capsid core protein assembly modulators	8
Graphical Abstract Contents Continued	8
Graphical Abstract TOC	8
Graphical abstract TOC	8
Retraction notice to “Corrigendum to “Preclinical metabolism of LB42908, a novel farnesyl transferase inhibitor, and its effects on the cytochrome P450 isozyme activities” [Bioorg. Med. Chem. Lett. 22	8
Editorial Board	8
Structure-activity relationship study of antitrypanosomal analogues of gibbilimbol B using multivariate analysis and computation-aided drug design	8
Conformationally constrained potent inhibitors for enhancer of zeste homolog 2 (EZH2)	8
Development of chromone-thiazolidine-2,4-dione Knoevenagel conjugates as apoptosis inducing agents	8
Discovery of 4-((quinolin-8-ylthio)methyl)benzamide derivatives as a new class of SARS-CoV-2 nsp13 inhibitors	8
Exploration of inhibitors of the bacterial LexA repressor-protease	8
Discovery of the potent covalent inhibitor with an acrylate warhead for SARS-CoV-2 3CL protease	8
Novel imidazo[1,5-a]quinoxaline derivatives: SAR, selectivity and modeling challenges en route to the identification of an α5-GABAA receptor NAM	8
Sensitive and reliable gastric ulcer related MicroRNA detection by bridge catalytic hairpin assembly (bCHA) mediated primer exchange reaction	8
The lipidation and glycosylation enabling bioactivity enhancement and structural change of antibacterial peptide G3	8
Contents continued	8
Design and synthesis of novel orexin 2 receptor agonists based on naphthalene skeleton	8
Synthesis, radiolabeling, and evaluation of a potent β-site APP cleaving enzyme (BACE1) inhibitor for PET imaging of BACE1 in vivo	8
Editorial Board	8
Aiming to improve binding of porphyrin diphenyl guanidinium conjugates to guanine-quadruplexes: When size matters	8
Design, synthesis, and biological evaluation of novel aminopyrimidine derivatives as EGFR inhibitors	8
The structural modification and biological evaluation of tetrahydrothienopyridine derivatives as selective BChE inhibitors	8
Discovery of a DCAF11-dependent cyanoacrylamide-containing covalent degrader of BET-proteins	8
Diffusion of 1O2 along the PNA backbone diminishes the efficiency of photooxidation of PNA/DNA duplexes by biphenyl photosensitizer	8
Discovery of aryl aminothiazole γ-secretase modulators with novel effects on amyloid β-peptide production	8
Design of a ROS-responsive fluorescent probe for the diagnosis and imaging of breast cancer	8
Design of cyclic peptides as novel inhibitors of ICOS/ICOSL interaction	8
Discovery of acyl ureas as highly selective small molecule CSF1R kinase inhibitors	8
Graphical Abstract TOC	8
Synthesis and in vitro antifungal activity of new Michael-type amino derivatives of xanthatin, a natural sesquiterpene lactone from Xanthium strumarium L.	7
Synthesis of pyrrolo[3,2-d]pyrimidineone derivatives as novel FXa inhibitors	7
Regulation of CD28 binding to SH2 domains of Grb2 and PI3K by trisubstituted carboranes for T-cell activation	7
Targeting ATP-binding site of WRN Helicase: Identification of novel inhibitors through pocket analysis and Molecular Dynamics-Enhanced virtual screening	7
Editorial Board	7
Editorial Board	7
Discovery of 5-methyl-1H-benzo[d]imidazole derivatives as novel P2X3 Receptor antagonists	7
Graphical Abstract Contents Continued	7
Targeting G-quadruplexes to achieve antiviral activity	7
Editorial Board	7
Synthesis, anti-microbial, toxicity and molecular docking studies of N-nitroso-N-phenylhydroxylamine (cupferron) and its derivatives	7
Synthesis and preliminary biological evaluation of a novel 99mTc-labeled small molecule for PD-L1 imaging	7
Identification of novel glucocerebrosidase chaperones by unexpected skeletal rearrangement reaction	7
Evaluation of darunavir-derived HIV-1 protease inhibitors incorporating P2′ amide-derivatives: Synthesis, biological evaluation and structural studies	7
Synthesis and biological evaluation of 2,5-disubstituted furan derivatives containing 1,3-thiazole moiety as potential α‐glucosidase inhibitors	7