OOIR: Observatory of International Research

Papers

(The H4-Index of Bioorganic & Medicinal Chemistry is 28. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2021-08-01 to 2025-08-01.)

Article	Citations
Synthesis and antiproliferative activity of (−)-cleistenolide, (6S)-cleistenolide and 4-substituted cleistenolide analogues	110
Synthesis and biological evaluation of pyrazole-fused oleanolic acid derivatives as novel inhibitors of inflammatory and osteoclast differentiation	94
Production and synthesis of a novel 191Pt-labeled platinum complex and evaluation of its biodistribution in healthy mice	86
A DNA-encoded library special issue	81
Discovery of novel 2,8-diazaspiro[4.5]decan-1-one derivatives as potent RIPK1 kinase inhibitors	67
Discovery of 5-methylpyrimidopyridone analogues as selective antimycobacterial agents	62
Targeting prolidase. A survey of the literature data to depict a structure-activity relationship frame and to address future studies for drug development	47
Current Japanese pharmaceutical chemistry	45
Site-specific construction of triptolide-based antibody-drug conjugates	42
RNA-templated chemical synthesis of proapoptotic L- and d-peptides	39
Janus dendritic ionizable lipids with fine designed headgroup and tails to improve mRNA delivery efficiency	38
Contents continued	37
Graphical abstract TOC	37
Graphical abstract TOC	36
Editorial Board	35
Development of delivery carriers for plasmid DNA by conjugation of a helical template to oligoarginine	35
Diterpenoids from the whole plants of Croton yunnanensis and their bioactivities	35
Synthesis, bioevaluation and docking studies of new imidamide derivatives as nitric oxide synthase inhibitors	33
Exploring novel A2AAR antagonists: Design, synthesis, and evaluation of 2,6,9-trisubstituted purine derivatives as promising antifibrotic agents	33
Selective targeting of human TET1 by cyclic peptide inhibitors: Insights from biochemical profiling	32
Design, synthesis and antibacterial evaluation of oxazolidinone derivatives containing N-methylglycyl or quaternary ammonium salts	32
Crescent-shaped meta-substituted benzene derivatives as a new class of non-nucleoside ribonuclease A inhibitors	31
Design, synthesis and evaluation the bioactivities of novel 1,3-dimethyl-6-amino-1H-indazole derivatives as anticancer agents	30
Research progress of STAT3-based dual inhibitors for cancer therapy	30
Targeting m6A binding protein YTHDFs for cancer therapy	30

Sustainable electrochemical C(sp3) − H oxygenation using water as the oxygen source	29
Design, synthesis and validation of a new Crimped Head-Piece for DNA-Encoded libraries generation	29
Synthesis and medicinal chemistry of tetronamides: Promising agrochemicals and antitumoral compounds	29
Discovery of 3-hydroxymethyl-azetidine derivatives as potent polymerase theta inhibitors	28
Antimycobacterial and anti-inflammatory activities of thiourea derivatives focusing on treatment approaches for severe pulmonary tuberculosis	28