OOIR: Observatory of International Research

Papers

(The median citation count of Bioconjugate Chemistry is 3. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2021-06-01 to 2025-06-01.)

Article	Citations
Issue Editorial Masthead	244
Issue Publication Information	174
Functionalization of Biomimetic Polydopamine Shells Constructed onto Bismuth-Core Particles for pH-Mediated Drug Targeting to Heal Bacterial Infections	121
Issue Publication Information	120
Issue Editorial Masthead	91
Tyrosinase-Related Protein2 Peptide with Replacement of N-Terminus Residue by Cysteine Binds to H-2K^b and Induces Antigen-Specific Cytotoxic T Lymphocytes after Conjugation with CpG-DNA	66
Enolate–Azide [3 + 2]-Cycloaddition Reaction Suitable for DNA-Encoded Library Synthesis	60
Equimolar Cross-Coupling Using Reactive Coiled Coils for Covalent Protein Assemblies	58
Identification of a Novel Transasparaginase Activity of Bacillus subtilis (bTG) for Sequence-Specific Bioconjugation	50
Designing Functional Bionanoconstructs for Effective In Vivo Targeting	47
RGD-Modified Titanium as an Improved Osteoinductive Biomaterial for Use in Dental and Orthopedic Implants	46
Issue Editorial Masthead	45
Linker Chemistry and Connectivity Fine-Tune the Immune Response and Kinetic Solubility of Conjugated NOD2/TLR7 Agonists	43
Choice of an Optimal Modular Strategy for the Synthesis of DOTA-Containing Heterobivalent Agents Targeting PSMA and GRPr	41
Evaluation of Cellular Targeting by Fab′ vs Full-Length Antibodies in Antibody–Nanoparticle Conjugates (ANCs) Using CD4 T-cells	41
Drug Delivery Targeting Neuroinflammation to Treat Brain Diseases	37
Bioderived Lipoic Acid-Based Dynamic Covalent Nanonetworks of Poly(disulfide)s: Enhanced Encapsulation Stability and Cancer Cell-Selective Delivery of Drugs	37
Efficiency and Safety of Dextran-PAMAM/siMMP-9 Complexes for Decreasing Matrix Metalloproteinase-9 Expression and Promoting Wound Healing in Diabetic Rats	36
Solid-Phase Synthesis of Caged Luminescent Peptides via Side Chain Anchoring	36
A Series of Furimazine Derivatives for Sustained Live-Cell Bioluminescence Imaging and Application to the Monitoring of Myogenesis at the Single-Cell Level	35
Hollow Cobalt Sulfide Nanospheres with Highly Enzyme-like Antibacterial Activities to Accelerate Infected Wound Healing	35
Xylose Dehydrogenase Immobilized on Ferromagnetic Nanoparticles for Bioconversion of Xylose to Xylonic Acid	30
A Cysteine-Maleimide-Based Design for Hemostatic, Antibacterial, and Biodegradable Wound Dressing	29
Non-Genetic Generation of Antibody Conjugates Based on Chemoenzymatic Tyrosine Click Chemistry	28
Elucidating Critical Factors of Internalization and Drug Release of Antibody-Drug Conjugates (ADCs) Using Kinetic Parameters Evaluated by a Novel Tool Named TORCH	28

Easy Surface Functionalization and Bioconjugation of Peptides as Capture Agents of a Microfluidic Biosensing Platform for Multiplex Assay in Serum	28
PEGylation of anti-MerTK Antibody Modulates Ocular Biodistribution	28
In Silico-Driven THIOMAB Approach for Stable PROTAC Conjugates by Docking Payloads in Antibody Cavities	27
Targeting HER2 with DNA Aptamers for Efficient Anticancer Drug Delivery: A Combined Experimental and Computational Study	26
Modular Adapters Utilizing Binders of Different Molecular Types Expand Cell-Targeting Options for Adenovirus Gene Delivery	25
Engineering and Validation of a Peptide-Stabilized Poly(lactic-co-glycolic) Acid Nanoparticle for Targeted Delivery of a Vascular Disruptive Agent in Cancer Therapy	24
Dimeric Metal-Salphen Complexes Which Target Multimeric G-Quadruplex DNA	24
Bioorthogonal Chemistry and Its Applications	24
Biocatalytic Clusterzyme Patches Restore Lung Function via Immunomodulation and Mitochondria Protection	23
DNA Modifications Enabling Proximity Biotinylation	23
Receptor-Mediated Transmembrane Activation of Protein Folding in Synthetic Cells	23
Single Gold Nanostars Achieve Inherent Cascade Catalytic and Near-Infrared Photothermal Activities for Efficient Tumor Therapy	23
Multivalent Display of Erythropoietin on Quantum Dots Enhances Aquaporin-4 Expression and Water Transport in Human Astrocytes In Vitro	23
Targeted Polymersomes Enable Enhanced Delivery to Peripheral Nerves Post-Injury	23
Site-Specific Molecular Engineering of Nanobody–Glucoside Conjugates for Enhanced Brain Tumor Targeting	23
Effect of Lipidation on the Structure, Oligomerization, and Aggregation of Glucagon-like Peptide 1	23
Effect of PEGylation on Host Defense Peptide Complexation with Bacterial Lipopolysaccharide	22
Using Spectroscopy to Guide the Adaptation of Aptamers into Electrochemical Aptamer-Based Sensors	22
Computational Approaches for Antimicrobial Peptide Delivery	22
Luminescent Ruthenium(II) Complexes Used for the Detection of 8-Oxoguanine in the Human Telomeric Sequence	22
Exo-Enzymatic Cell-Surface Glycan Labeling for Capturing Glycan–Protein Interactions through Photo-Cross-Linking	22
A Universal and Modular Scaffold for Heparanase Activatable Probes and Drugs	22
A General Set of DNA-Compatible Reactions for Preparing DNA-Tagged Multisubstituted Pyrroles	22
Artificial Nanocage Formed via Self-Assembly of β-Annulus Peptide for Delivering Biofunctional Proteins into Cell Interiors	21
Revival of Bioengineered Proteins as Carriers for Nucleic Acids	21
Rational Design of a Dual-Targeting Natural Toxin-Like Bicyclic Peptide for Selective Bioenergetic Blockage in Cancer Cells	21
Multisite Labeling of Proteins Using the Ligand-Directed Reactivity of Triggerable Michael Acceptors	21
Dual-Function Antibody Conjugate-Enabled Photoimmunotherapy Complements Fluorescence and Photoacoustic Imaging of Head and Neck Cancer Spheroids	21
Squaramide Formation for DNA-Encoded Library Synthesis	21
Resveratrol Carbon Dots Disrupt Mitochondrial Function in Cancer Cells	20
MMP-2-Activatable Photoacoustic Tumor Imaging Probes Based on Al- and Si-Naphthalocyanines	20
Advances in the Treatment of Spinal Cord Injury with Nanozymes	20
Preparation, In Vitro Affinity, and In Vivo Biodistribution of Receptor-Specific ⁶⁸Ga-Labeled Peptides Targeting Vascular Endothelial Growth Factor Receptors	20
Introducing TAPY as a Versatile Alternative to TPP for Selective Mitochondrial Targeting in Cancer Cells	20
Redesigning Ibuprofen for Improved Oral Delivery and Reduced Side Effects	20
A Switch-On Affinity-Based Iridium(III) Conjugate Probe for Imaging Mitochondrial Glutathione S-Transferase in Breast Cancer Cells	19
Photoactivated Nanohybrid for Dual-Nuclei MR/US/PA Multimodal-Guided Photothermal Therapy	19
Bioconjugate Chemistry: Enabling Innovation and Fostering Community at the Nexus of Synthetic and Biological Research	19
Structure–Activity Relationships of Antibody-Drug Conjugates: A Systematic Review of Chemistry on the Trastuzumab Scaffold	19
Radiotracers for Nuclear Imaging of Reactive Oxygen Species: Advances Made So Far	19
7-Deaza-2′-deoxyisoguanosine, a Noncanonical Nucleoside for Nucleic Acid Code Expansion and New DNA Constructs: Nucleobase Functionalization of Inverse Watson–Crick and Purine–Purine Base Pairs	18
Rapid Copper-free Click Conjugation to Lipid-Shelled Microbubbles for Ultrasound Molecular Imaging of Murine Bowel Inflammation	18
Issue Editorial Masthead	18
Comparison of Quenching Efficiencies in Long Triple-Labeled and Double-Labeled TaqMan Oligodeoxynucleotide Probes	18
A New Class of Tunable Acid-Sensitive Linkers for Native Drug Release Based on the Trityl Protecting Group	18
Tyrosinase-Mediated Conjugation for Antigen Display on Ferritin Nanoparticles	18
A Genetically Encoded Photocaged Cysteine for Facile Site-Specific Introduction of Conjugation-Ready Thiol Residues in Antibodies	18
Polyfluoroalkyl Tag Decoration Enables Significantly Enhanced Tumor Penetration Ability of a PTK7 Targeting Aptamer	17
Rapid Access to Potent Bispecific T Cell Engagers Using Biogenic Tyrosine Click Chemistry	17
Discovery of a Novel ADC for Multifunctional Theranostics: From Vascular Normalization to Synergistic Therapy	17

Protein Corona Formation on Lipid Nanoparticles Negatively Affects the NLRP3 Inflammasome Activation	17
Rational Design of Targeted Gold Nanoclusters with High Affinity to Integrin αvβ3 for Combination Cancer Therapy	17
Lysine-Derived Charge-Altering Releasable Transporters: Targeted Delivery of mRNA and siRNA to the Lungs	17
Recent Advances in Nanoimmunotherapy by Modulating Tumor-Associated Macrophages for Cancer Therapy	17
Targeted Protein Degradation (TPD) for Immunotherapy: Understanding Proteolysis Targeting Chimera-Driven Ubiquitin-Proteasome Interactions	17
A Novel Family of Acid-Cleavable Linker Based on Cyclic Acetal Motifs for the Production of Antibody-Drug Conjugates with High Potency and Selectivity	17
Poly(malic acid) Nanoconjugates of Pyrazinoic Acid for Lung Delivery in the Treatment of Tuberculosis	17
NIR II Luminescence Imaging for Sentinel Lymph Node and Enhanced Chemo-/Photothermal Therapy for Breast Cancer	17
Cytokine Biopharmaceuticals with “Activity-on-Demand” for Cancer Therapy	17
Azide-Functionalized Naphthoxyloside as a Tool for Glycosaminoglycan Investigations	16
Issue Publication Information	16
Fluorescence-Based Simple and Practical Assay Method for DNA Damage Analysis in DNA-Encoded Library Synthesis	16
Development of a Decafluorobiphenyl Cyclized Peptide Targeting the NEMO–IKKα/β Interaction that Enhances Cell Penetration and Attenuates Lipopolysaccharide-Induced Acute Lung Injury	16
pH-Responsive Amphiphilic Triblock Fluoropolymers as Assemble Oxygen Nanoshuttles for Enhancing PDT against Hypoxic Tumor	16
Synthetic and Computational Design Insights toward Mimicking Protein Binding of Phosphate	16
Issue Editorial Masthead	16
NIR-Triggered On-Demand Nitric Oxide Release for Enhanced Synergistic Phototherapy of Hypoxic Tumor	16
Noninvasive Analysis of Peptidoglycan from Living Animals	16
Light-Activated Molecular Purification (LAMP) of Recombinant Proteins	16
Lectin-Functionalized Chitosan Nanoparticle-Based Biosensor for Point-of-Care Detection of Bacterial Infections	16
Lipophilic Anchors that Embed Bioconjugates in Bilayer Membranes: A Review	16
Issue Publication Information	16
Novel Synthetic Strategies Enable the Efficient Development of Folate Conjugates for Cancer Radiotheranostics	15
Recent Progress of Surface Modified Nanomaterials for Scavenging Reactive Oxygen Species in Organism	15
Long-Acting Poly(ADP-ribose) Polymerase Inhibitor Prodrug for Humans	15
Zinc Triggered Release of Encapsulated Cargo from Liposomes via a Synthetic Lipid Switch	15
Asymmetry of Dual-Display DNA-Encoded Chemical Libraries	15
Bypassing the Need for Cell Permeabilization: Nanobody CDR3 Peptide Improves Binding on Living Bacteria	15
GB Tags: Small Covalent Peptide Tags Based on Protein Fragment Reconstitution	15
Bioorthogonal Chemistry and Bioconjugation: Synergistic Tools for Biology and Biomedicine	15
Mechanistic Characterization of the Potency of THIOMAB Antibody–Drug Conjugates Targeting Staphylococcus aureus and ETbR-Expressing Tumor Cells Using Quantitative LC-MS/MS Analysis of Intracell	15
Genetic Determinants of Surface Accessibility in Staphylococcus aureus	15
²¹¹At-Labeled Polymer Nanoparticles for Targeted Radionuclide Therapy of Glucose-Dependent Insulinotropic Polypeptide Receptor (GIPR)-Overexpressed Cancer	15
Precise Manipulation of the Site and Stoichiometry of Capsid Modification Enables Optimization of Functional Adeno-Associated Virus Conjugates	15
Sensitive Detection of the Human Epididymis Protein-4 (HE4) Ovarian Cancer Biomarker through a Sandwich-Type Immunoassay Method with Laser-Induced Breakdown Spectroscopy	15
Issue Publication Information	14
Click Chemistry Enables [⁸⁹Zr]Zr-DOTA Radioimmunoconjugation for Theranostic ⁸⁹Zr-immunoPET	14
Photoactivatable Liposomes for Blue to Deep Red Light-Activated Surface Drug Release: Application to Controlled Delivery of the Antitumoral Drug Melphalan	14
Miniaturized Synthetic Palmitoylation Motifs for Small-Molecule Localization in Living Cells	14
Modular Display of Plasmodium yoelii Circumsporozoite Surface Protein and Merozoite Surface Protein-1 on Norovirus-like Particles	14
Conceptualization and Preliminary Characterization of Poloxamer-Based Hydrogels for Biomedical Applications	14
Complex DNA Architectonics─Self-Assembly of Amphiphilic Oligonucleotides into Ribbons, Vesicles, and Asterosomes	14
Human Behavior-Inspired Linchpin-Directed Catalysis for Traceless Precision Labeling of Lysine in Native Proteins	14
Synthesis and Biological Evaluation of Bile Acid–Triclosan Conjugates: A Study on Antibacterial, Antibiofilm, and Molecular Docking	14
Metal-Free Click-Chemistry: A Powerful Tool for Fabricating Hydrogels for Biomedical Applications	14
Issue Publication Information	14
Correction to “Self-Assembling Nanoparticle Vaccines Displaying the Receptor Binding Domain of SARS-CoV-2 Elicit Robust Protective Immune Responses in Rhesus Monkeys”	14
Molecular Imaging-Guided Sonodynamic Therapy	13
Organotropic Targeting of Biomimetic Nanoparticles to Treat Lung Disease	13
Design, Synthesis, and Anticancer Activity of Triptycene–Peptide Hybrids that Induce Paraptotic Cell Death in Cancer Cells	13
Quantum Dot Erythropoietin Bioconjugates Enhance EPO-Receptor Clustering on Transfected Human Embryonic Kidney Cells	13
Mirror-Image Single-Domain Antibody for a Novel Nonimmunogenic Drug Scaffold	13
Radiation Cleaved Drug-Conjugate Linkers Enable Local Payload Release	13
Self-Assembly of the Tetraphenylethylene-Capped Diserine through a Hierarchical Assembly Process	13
Development of an Albumin–Polymer Bioconjugate via Covalent Conjugation and Supramolecular Interactions	13
Developing and Characterizing the Tumor-Targeting Efficiency of an Anti-EphA2-CD11b Bispecific Antibody	13
Issue Publication Information	13
Customizable Click Biochemistry Strategy for the Design and Preparation of Glucagon-like Peptide-1 Conjugates and Coagonists	13
Chemistry of DNA Nanotechnology Special Issue	13
A Simple and Versatile Strategy for Oriented Immobilization of His-Tagged Proteins on Magnetic Nanoparticles	13
Synergistic Experimental and Computational Investigation of the Bioorthogonal Reactivity of Substituted Aryltetrazines	13
Targeted NIR Fluorescent Mechanically Interlocked Molecules-Peptide Bioconjugate for Live Cancer Cells Submitochondrial Stimulated Emission Depletion Super-Resolution Microscopy	13
RGD and Scutellarin Conjugate (WK001) Targeting Platelet Glycoprotein IIb/IIIa Receptor Protects from Myocardial Ischemia/Reperfusion Injury: Synthesis, Characterization, and Bioactivity Evaluation	13
Matrix Metalloproteinase-Responsive Drug Delivery Systems	13
Synthetic Amine Linkers for Efficient Sortagging	12
Photochemical-Promoted Cross-Coupling Reaction of Alkyl Boronate Esters with DNA-Conjugated Aryl Bromides for DNA-Encoded Library Synthesis	12
Critical Evaluation of Different Lysosomal Labeling Methods Used to Analyze RNA Nanocarrier Trafficking in Cells	12
Bioreducible Amphiphilic Hyperbranched Polymer-Drug Conjugate for Intracellular Drug Delivery	12
Dual-Boronic Acid Reagents That Combine Dynamic and Covalent Bioconjugation	12
Issue Editorial Masthead	12
State-of-the-Art of Radiometal-based Bioconjugates for Molecular Imaging and Radiotherapy	12
Crossing the Solubility Rubicon: 15-Crown-5 Facilitates the Preparation of Water-Soluble Sulfo-NHS Esters in Organic Solvents	12
A Multifunctional Contrast Agent for ¹⁹F-Based Magnetic Resonance Imaging	12
Synergism of ⁶⁴Cu-Labeled RGD with Anti-PD-L1 Immunotherapy for the Long-Acting Antitumor Effect	12
A Photoacoustic Contrast Agent for miR-21 via NIR Fluorescent Hybridization Chain Reaction	12
Poly(hydrophobic amino acid) Conjugates for the Delivery of Multiepitope Vaccine against Group A Streptococcus	12
Sustained Releasable Copper and Zinc Biogenic Ions Co-Assembled in Metal–Organic Frameworks Reinforced Bacterial Eradication and Wound Mitigation in Diabetic Mice	12
Sequestration and Removal of Multiple Small-Molecule Contaminants Using an Optimized Aptamer-Based Ultrafiltration System	12
One-Step Conversion of NHS Esters to Reagents for Site-Directed Labeling of IgG Antibodies	12
Engineering a High-Affinity Anti-Methoxy Poly(ethylene glycol) (mPEG) Antibody for Sensitive Immunosensing of mPEGylated Therapeutics and mPEG Molecules	12

Dynamic Catalysis Guided by Nucleic Acid Networks and DNA Nanostructures	12
Issue Publication Information	11
IgG-Binding Nanobody Capable of Prolonging Nanobody-Based Radiotracer Plasma Half-Life and Enhancing the Efficacy of Tumor-Targeted Radionuclide Therapy	11
Carbon Dots as Potential Therapeutic Agents for Treating Non-Alcoholic Fatty Liver Disease and Associated Inflammatory Bone Loss	11
Targeted Delivery of TLR7 Agonists to the Tumor Microenvironment Enhances Tumor Immunity via Activation of Tumor-Resident Myeloid Cells	11
Guest-Induced Planar-Chiral Pillar[5]arene Surface for Selectively Adsorbing Protein Based on Host–Guest Chemistry	11
Recent Advances in Bioorthogonal Click Chemistry for Biomedical Applications	11
Development of a Long-Acting Myeloid-Derived Growth Factor via Site-Specific PEGylation	11
Protein Modification via Mild Photochemical Isomerization of Triazenes to Release Aryl Diazonium Ions	11
Fluorophore Labeling of Proteins: a Versatile Trigger–Release–Conjugation Platform Based on the Quinone Methide Chemistry	11
High-Affinity Points of Interaction on Antibody Allow Synthesis of Stable and Highly Functional Antibody–Gold Nanoparticle Conjugates	11
Issue Publication Information	11
Rapid Production of Bispecific Antibodies from Off-the-Shelf IgGs with High Yield and Purity	11
Solid-Phase Collateral Cleavage System Based on CRISPR/Cas12 and Its Application toward Facile One-Pot Multiplex Double-Stranded DNA Detection	11
Point-of-Care Testing for Norovirus Typing Using CRISPR/Cas12a Combined with Reverse Transcription Recombinase Polymerase Amplification	11
Generation of Multivalent Nanobody-Based Proteins with Improved Neutralization of Long α-Neurotoxins from Elapid Snakes	11
Harnessing DNA Nanotechnology and Chemistry for Applications in Photonics and Electronics	11
Issue Publication Information	11
Correction to “Oral Delivery of Peptide Drugs Using Nanoparticles Self-Assembled by Poly(γ-glutamic acid) and a Chitosan Derivative Functionalized by Trimethylation”	11
Issue Publication Information	10
New Triazacycloalkane Derivatives as Cytotoxic Agents for CLL Treatment: From Proof of Concept to the Targeting Biomolecule	10
Covalent and Oriented Immobilization of Antibodies through Systematic Modification of Photoactivatable RNA Hybrid Aptamers	10
iFLinkC-X: A Scalable Framework to Assemble Bespoke Genetically Encoded Co-polymeric Linkers of Variable Lengths and Amino Acid Composition	10
Issue Editorial Masthead	10
Impact of Drug Conjugation on Thermal and Metabolic Stabilities of Aglycosylated and N-Glycosylated Antibodies	10
Formal [4 + 2] Cycloadditions of Maleimides on Duplex DNA	10
Tumor-Derived PD-L1⁺ Exosomes with Natural Inflammation Tropism for Psoriasis-Targeted Treatment	10
Design and Optimization of an α-Helical Bundle Dimer Cell-Penetrating Peptide for In Vivo Drug Delivery	10
Issue Publication Information	10
Issue Editorial Masthead	10
Light-Activated Nanodiamond-Based Drug Delivery Systems for Spatiotemporal Release of Antisense Oligonucleotides	10
Rapid Covalent Labeling of Membrane Proteins on Living Cells Using a Nanobody–Epitope Tag Pair	10
Carbonic Anhydrase IX Targeting Mn(II)-Based Magnetic Resonance Molecular Imaging Probe for Hypoxia Tumors	10
Peptide Amphiphile Hydrogels Based on Homoternary Cucurbit[8]uril Host-Guest Complexes	10
Optimization of Enzymolysis Clearance Strategy To Enhance Renal Clearance of Radioligands	10
Cyclopentadiene as a Multifunctional Reagent for Normal- and Inverse-Electron Demand Diels–Alder Bioconjugation	10
Modular PET Agent Construction Strategy through Strain-Promoted Double-Click Reagent with Efficient Photoclick Step	10
In Situ Visualizing Nascent RNA by Exploring DNA-Templated Oxidative Amination of 4-Thiouridine	10
Linker and Conjugation Site Synergy in Antibody–Drug Conjugates: Impacts on Biological Activity	10
Mitigating Cannabidiol’s Non-Selective Cytotoxicity via Subcellular Organelle Targeting: Exploring Mitochondrial Targeting Potential	10
Multivalent Cucurbituril Dendrons for Cell Membrane Engineering with Supramolecular Receptors	10
Human CD47-Derived Cyclic Peptides Enhance Engulfment of mAb-Targeted Melanoma by Primary Macrophages	10
Synthesis and Evaluation of Three Azide-Modified Disaccharide Oxazolines as Enzyme Substrates for Single-Step Fc Glycan-Mediated Antibody-Drug Conjugation	10
Azobenzene-Based Amino Acids for the Photocontrol of Coiled-Coil Peptides	10
Issue Editorial Masthead	10
Live-Cell Mitochondrial Targeted NIR Fluorescent Covalent Labeling of Specific Proteins Using a Dual Localization Effect	10
Aptamer- vs Fab-Conjugated Liposomes: A Comparative Study in Targeting Acute Myeloid Leukemia Cells	10
Click Chemistry: Reaction Rates and Their Suitability for Biomedical Applications	9
Thymidine Phosphodiester Chemiluminescent Probe for Sensitive and Selective Detection of Ectonucleotide Pyrophosphatase 1	9
The Base Pairs of Isoguanine and 8-Aza-7-deazaisoguanine with 5-Methylisocytosine as Targets for DNA Functionalization	9
Intravenous Hemostats: Foundation, Targeting, and Controlled-Release	9
Evolution of Lipo-Xenopeptide Carriers for siRNA Delivery: Interplay of Stabilizing Subunits	9
Linker Architectures as Steric Auxiliaries for Altering Enzyme-Mediated Payload Release from Bioconjugates	9
Issue Publication Information	9
Fast and Selective Reaction of 2-Benzylacrylaldehyde with 1,2-Aminothiol for Stable N-Terminal Cysteine Modification and Peptide Cyclization	9
SARS-CoV-2 Peptide Bioconjugates Designed for Antibody Diagnostics	9
Biofilm-Mediated Immobilization of a Multienzyme Complex for Accelerating Inositol Production from Starch	9
Cationic Micelles Outperform Linear Polymers for Delivery of Antisense Oligonucleotides in Serum: An Exploration of Polymer Architecture, Cationic Moieties, and Cell Addition Order	9
Lipid Nanoparticles for Brain Tumor Theranostics: Challenges and Status	9
AUNP-12 Near-Infrared Fluorescence Probes across NIR-I to NIR-II Enable In Vivo Detection of PD-1/PD-L1 Axis in the Tumor Microenvironment	9
Advancing the Utility of DNA Origami Technique through Enhanced Stability of DNA-Origami-Based Assemblies	9
Dynamics of DNA Origami Lattices	9
Targeted Association and Intracellular Delivery of Nanocargoes into Primary T Lymphocytes via Interleukin-2 Receptor-Mediated Endocytosis	9
H₃TPAN-Triazole-Bn-NH₂: Tripicolinate Clicked-Bifunctional Chelate for [²²⁵Ac]/[¹¹¹In] Theranostics	9
Binary Copolymer Blending Enhances pDNA Delivery Performance and Colloidal Shelf Stability of Quinine-Based Polyplexes	9
Construction of Self-Assembling Lipopeptide-Based Benign Nanovesicles to Prevent Amyloid Fibril Formation and Reduce Cytotoxicity of GxxxGxxxGxxxG Motif	9
Application of N-Terminal Site-Specific Biotin and Digoxigenin Conjugates to Clinical Anti-drug Antibody Assay Development	9
Gold Nanoclusters: Imaging, Therapy, and Theranostic Roles in Biomedical Applications	9
Transferrin Receptor-Targeted Aptamer–Drug Conjugate Overcomes Blood–Brain Barrier for Potent Glioblastoma Therapy	9
Delivery of Targeted Co(III)–DNA Inhibitors of Gli Proteins to Disrupt Hedgehog Signaling	9
Cucurbituril–Ferrocene: Host–Guest Based Pretargeted Positron Emission Tomography in a Xenograft Model	9
Synthesis of 5′-Thiol Functionalized Morpholino Oligo-Nucleotide and Subsequent Conjugation with IGT to Improve Delivery and Antisense Efficacy In Vitro	9
Superresolution Imaging with Single-Antibody Labeling	9
One-Pot, One-Step Synthesis of Drug-Loaded Magnetic Multimicelle Aggregates	9
Diligent Design Enables Antibody-ASO Conjugates with Optimal Pharmacokinetic Properties	9
Combined Endothelialization Promoting and Surface Binding Chimeric Conjugate with Low Thrombogenicity	9
Design of Neuraminidase-Targeted Imaging and Therapeutic Agents for the Diagnosis and Treatment of Influenza Virus Infections	9
Issue Publication Information	9
Issue Editorial Masthead	9
Large Protein Assemblies for High-Relaxivity Contrast Agents: The Case of Gadolinium-Labeled Asparaginase	9
Targeting Colon Cancer Cells with Enzyme-Triggered Casein-Gated Release of Cargo from Mesoporous Silica-Based Nanoparticles	9
Stearylated Macropinocytosis-Inducing Peptides Facilitating the Cellular Uptake of Small Extracellular Vesicles	9
HOCl-Activated Reactive Organic Selenium Delivery Platform for Alleviation of Inflammation	9
Site-Specific Conjugation Strategy for Dual Antibody–Drug Conjugates Using Aerobic Formylglycine-Generating Enzymes	9
Thiol-Specific Linkers for the Synthesis of Oligonucleotide Conjugates via Metal-Free Thiol–Ene Click Reaction	8
Applications of Synthetic Receptors in Bioanalysis and Drug Transport	8
Doxorubicin-Loaded Walnut-Shaped Polydopamine Nanomotor for Photothermal-Chemotherapy of Cancer	8
Toward Bifunctional Chelators for Thallium-201 for Use in Nuclear Medicine	8
On-DNA Alkyne Iodination and Acetylenic Coupling as a Useful Tool for DEL Synthesis	8
Surface Presentation of Hyaluronic Acid Modulates Nanoparticle–Cell Association	8
On-Strand Knoevenagel Insertion of a Hemicyanine Molecular Rotor Loop Residue for Turn-On Fluorescence Detection of Pb-Induced G-Quadruplex Rigidity	8
A pH-Sensitive cRGD-PEG-siRNA Conjugated Compound Targeting Glioblastoma	8
Oligodeoxynucleotides Modified with 2′-O-(Cysteinylaminobutyl)carbamoylethylribothymidine Residues for Native Chemical Ligation with Peptide at Internal Positions	8
Enhanced ASO-Mediated Gene Silencing with Lipophilic pH-Responsive Micelles	8
Issue Publication Information	8