Organic Letters

Article	Citations
Versatile Access to Tetrasubstituted 2-Amidoacroleins through Formal Silylformylation of Ynamides	83
Diversity-Oriented Synthesis of ERα Modulators via Mitsunobu Macrocyclization	78
Synthesis of α-Aryl Secondary Amides via Nickel-Catalyzed Reductive Coupling of Redox-Active Esters	78
Visible-Light-Induced Selective α-Fluoroarylation of Secondary N-Alkyl Anilines with Polyfluoroarenes via Direct C–H/C–F Coupling	77
Deciphering the δ-Lactam Formation and lron-Reducing Activity of Spinactins from Saccharopolyspora spinosa	76
Oxoammonium Salt-Mediated Regioselective Vicinal Dioxidation of Alkenes: Relying on Transient and Persistent Nitroxides	75
Dioxygen-Triggered Oxosulfonylation/Sulfonylation of Terminal Olefins toward β-Keto Sulfones/Sulfones	74
Photocatalytic Strecker-Type Reaction for the Synthesis of Primary α-Aminonitriles	71
Paired Electrocatalysis-Enabled Cross Coupling of Sulfinamides with Olefins toward the Synthesis of Vinyl Sulfoximines	69
Visible-Light-Induced Difunctionalization of 3-Butenoic Acid with Bromodifluoromethyl Heteroarylsulfones	69
Relay Annulation of Ammonium Ylides with Oxindole-Derived α,β-Unsaturated Ketimines: Catalytic Construction of Spiro-polycyclic Oxindoles	69
Nonactivated Aziridine Synthesis by Intermolecular Polarity-Mismatched Carboamination of Unactivated Alkenes with Unactivated Alkyl Halides	68
Solvent-Driven Room-Temperature Curtius Rearrangements to Access Nucleotides Bearing Substituted Fused Pyridones	68
Nickel-Catalyzed Deaminative Allenylation of Amino Acid Derivatives: Catalytic Activity Enhanced by an Amide-Type NN2 Pincer Ligand	68
Spirochrains A–D, Four Caged [5,6,5] Spirocyclic Amides from an Antarctic Fungus Aspergillus ochraceopetaliformis SCSIO 05702 with Anti-RSV Activities	67
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Isolation and Bioinspired Total Synthesis of Rugosiformisin A, A Skeleton-Rearranged Abietane-Type Diterpenoid from Isodon rugosiformis	65
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Dinickel-Catalyzed Asymmetric Allylic Alkylation of Cyclic Ketones with Allylic Amine Derivatives	60
Enantioselective Cobalt-Catalyzed Remote Hydroboration of Alkenylboronates	59
Asymmetric Synthesis of β-Aminoboronates via Copper-Catalyzed Reductive Coupling of Vinyl Boronates with Imines	59
Exo-Selective and Enantioselective Photoenolization/Diels–Alder Reaction	58
Gold-Catalyzed Regioselective Synthesis of Crowded Cyclopentadienes by Migratory Cycloisomerization of Vinylallenes	58
Base Metal-Controlled Chemodivergent Cyclization of Propargylamines for the Atom-Economic Synthesis of Nitrogen Heterocycles	56
Stereoselective Double Spirocyclization of 2-Benzyl-3-alkynyl Chromone with Nitrone via Gold-Catalyzed Cascade Reactions	56
Free Amine-Directed Redox Neutral Ruthenium(II) Catalysis toward Regioselective Synthesis of Heterobiaryls	56
Cope-Type Hydroamination of Vinylboronates	55
Kinetic Resolution of Sulfinamides via Asymmetric N-Allylic Alkylation	55
Environmentally Friendly Synthesis of Highly Substituted Phenols Using Enallenoates and Grignard Reagents	55
Multiselective Diels–Alder Reaction of α-Arylacroleins Catalyzed by Boron Tribromide-Assisted Chiral Phosphoric Acids	55
Tosylazide as N1-Synthon: Iron-Catalyzed Nitrogenative Dimerization of Indoles to p-Bisindolopyrazine Derivatives	54
Total Synthesis of (±)-Furanether A	53
Domino Semipinacol/Iterative Aldol/Iso-Nazarov Cyclization to Triaryl-cyclopentenone: Enantioselective Synthesis of Combretastatin A-4 Analogues	53
Total Synthesis of the Phenolic Steroid Myrmenaphthol A	53
Correction to “Access to 6-Deoxy-heptose Constructs by One Carbon Homologation of Hexoses with Malononitrile: Divergent Synthesis of Campylobacter jejuni Strain 81-176 Capsular Trisaccharide Re	53
Sequential One-Pot Transformation to R–CF2-Embedded 1,5-Diketones Enabled by Nickel: Access to 4-Perfluoroalkylpyridines	53
Photodissociation of the Product from a Transition-Metal Center Allows the Catalytic Cycle to Proceed: The Rhodium(I)-Catalyzed [2+2+1] Carbonylative Cycloaddition of Diynes	53
Computationally Assisted Analysis of NMR Chemical Shifts as a Tool in Conformational Analysis	52
Manipulating Crystal Packing and Self-Assembly by π-Extended and Isomeric Fused Strategies in Thiophene Ring-Terminated Polycyclic Aromatic Hydrocarbons	52
Synthesis of 1-Substituted Bicyclo[2.1.1]hexan-2-ones via a Sequential SmI2-Mediated Pinacol Coupling and Acid-Catalyzed Pinacol Rearrangement Reaction	52
DNA-Compatible Diversification of Indole π-Activated Alcohols via a Direct Dehydrative Coupling Strategy	52
Solid-Phase Total Synthesis of Plusbacin A3	52
Palladium-Catalyzed Chemo- and Regiocontrolled Tandem Cyclization/Cross-Coupling of 2-Benzyl-3-alkynyl Chromones with Aryl Iodides for the Synthesis of 4H-Furo[3,2-c]chromenes and Xantho	52
Collective Syntheses of Corynanthe Alkaloids Based on a Chirality-Tunable Structure Unit	52
Palladium-Catalyzed Domino Conversion of Aryl–Thianthreniums with Anhydrides: Rapidly Building Highly Functionalized Fluorenones	51
Photochemical Organocatalytic Aerobic Cleavage of C═C Bonds Enabled by Charge-Transfer Complex Formation	51
Photocatalytic Borylation of Imines and Alkenes via Decarboxylation of Trimethylamine Carboxyborane: A New Approach for Generating Boryl Radicals	50
Enantioselective Palladium-Catalyzed Domino Carbonylative Heck Esterification of o-Iodoalkenylbenzenes with Arylboronic Acids	50
Gold(I)-Catalyzed Oxidative Amination of β-Amino-ynones to Quaternary Ammonium-olate Salts: The Benefit of a P,N-Bidentate Ligand	50
Reversal of Regioselectivity in Nucleophilic Difluoroalkylation of α,β-Enones Employing In Situ-Formed Sterically Encumbered Silylium Catalyst	49
Construction of Oxo-Bridged Diazocines via Rhodium-Catalyzed (4+3) Cycloaddition of Carbonyl Ylides with Azoalkenes	49
Nickel-Catalyzed Cross-Electrophile Ring Opening/gem-Difluoroallylation of Aziridines	48
Rh-Catalyzed Carbonylative Cyclization of Propargylic Alcohols with Aryl Boronic Acids	48
Cobalt-Catalyzed Intramolecular [4 + 2] Cycloaddition of Cyclopropyl-Capped Dienes with Alkynes/Alkenes/Allene and Reaction Mechanism	48
Nickel/SKP-Catalyzed Markovnikov Regio- and Enantioselective Hydroamination of Vinylarenes with Hydroxylamines	48
Asymmetric Synthesis of CF3-Substituted β-Hydroxyketones and 1,3-Diols by Engineered Ketoreductases	48
Electrochemical Oxidative C3 Acyloxylation of Imidazo[1,2-a]pyridines with Hydrogen Evolution	48
Syntheses and Properties of Hole-Transporting Biindenofluorenes	48
Dichloromethyl(diaryl) Sulfonium Salts as gem-Dichlorocyclopropanation Reagents	48
Sequential Strategies to Trigger Mild Dearomative Diels–Alder Cyclizations	48
Regiochemical Switching in Ir-Catalyzed C–H Borylation by Altering Ligand Loadings of N,B-Type Diboron Species	48
Expanded Access to Fluoroformamidines via a Modular Synthetic Pathway	47
Systematic Route to Construct the 5–5–6 Tricyclic Core of Furanobutenolide-Derived Cembranoids and Norcembranoids	47
Lewis Acid-Catalyzed Annulations of Geminally Disubstituted Cyclopropanes with Aldehydes or 1,3,5-Triazinanes	47
Enantioselective Synthesis of γ-Oxycarbonyl Motifs by Conjugate Addition of Photogenerated α-Alkoxy Radicals	47
Protecting-Group Free Total Synthesis of β-Levantenolide through Late Stage Bromo-Spirocyclization	46
Synergistic [4 + 1] Spiroannulation and Selective Ring-Opening Strategy toward γ-Spirolactams	46
Regioselective Alkylacylation of 1,3-Dienes by Merging N-Heterocyclic Carbene Catalysis with Photoinduced Palladium Catalysis	46

Biocatalytically Generated Library of Chiral Building Blocks Containing a Quaternary Stereocenter	46
Borylative Cyclization of 1,6-Allenynes Driven by BCl3	46
Ir-Catalyzed Asymmetric Cascade Allylation/Spiroketalization Reaction for Stereoselective Synthesis of Oxazoline-Spiroketals	46
Enantioselective Organocatalytic Conjugate Addition of Malonates to β,β-Disubstituted β-Trifluoromethyl Enones under High Pressure	46
DalPhos/Nickel-Catalyzed C2–H Arylation of 1,3-Azoles Using a Dual-Base System	46
Chiral Squaramide Catalyzed Asymmetric Spiroketalization toward Aromatic [6,5] Spiroketals	46
Radical Alkynylthiolation with Visible-Light-Sensitive S-Alkynylthio Sulfonates	45
Divergent Access to Polycyclic N-Heterocyclic Compounds through Büchner-Type Dearomatization Enabled Cycloisomerization of Diynamides under Gold Catalysis	45
A Sterically Tuned 2-Fluoropyridinium Salt for the Catalyst-Free, Visible-Light-Mediated Deoxygenation of Alcohols via an Electron Donor–Acceptor Complex	45
Reductive Hydrodehalogenation of Halogenated Carboxylic Acid Derivatives Using a DMSO/HCOONa·2H2O System	45
Palladium-Catalyzed Asymmetric (3 + 2) Cycloaddition of 5-Allenyloxazolidine-2,4-Diones with Barbiturate-Derived Alkenes: Synthesis of Spirobarbiturate-γ-Lactams	45
Weak-Chelation Assisted Cobalt-Catalyzed C–H Bond Activation: An Approach Toward Regioselective Ethynylation of N-Aryl γ-Lactam	45
From Nitrogen to Sulfur: Investigating the Effect of Core Modification within Azaacene-Fused 21,23-Dithiaporphyrins	44
A Synthetic Strategy for the Preparation of Fused [5,6,5,5]-Tetracyclic Energetic Compounds	44
Staudinger Cleavages of Amides on Naphthalene for the Ipsilateral Effect of 1,8-Substituents	44
Synthesis of Tertiary Amines through Extrusive Alkylation of Carbamates	44
Ligand-Controlled Diastereodivergency in Propargylic Alkylation of Vinylogous Aza-Enamines: Construction of 1,3-Stereocenters	44
Nickel-Catalyzed Domino Reaction of α-Aryloxyacetonitriles with Arylboronic Acids: Synthesis of 2-Aroylbenzo[b]furans	44
Synthesis of Planar Chiral 2-Aryl Aroylferrocenes via Palladium-Catalyzed C–C Bond-Cleavage/Ring-Opening Reaction	44
Stereospecific Nickel-Catalyzed Reductive Cross-Coupling of Alkyl Tosylate and Allyl Alcohol Electrophiles	44
Nucleophile-Induced Rearrangement of 2H-Azirine-2-carbonyl Azides to 2-(1H-Tetrazol-1-yl)acetic Acid Derivatives	44
Light-Induced Activation of C–X Bond via Carbonate-Assisted Anion−π Interactions: Applications to C–P and C–B Bond Formation	44
Synergistic Copper/Enamine Catalysis for the Regio-, Stereo-, and Enantioselective Intermolecular α-Addition of Aldehydes to Allenamides	43
Tertiary Amine-Mediated Reductions of Phosphine Oxides to Phosphines	43
Domino Synthesis of Thioindirubin via Aldol Condensation/C–S Cross-Coupling/Cyclization Reaction Using Xanthate as a Sulfur Surrogate	43
Environmentally Responsible and Cost-Effective Synthesis of the Antimalarial Drug Pyronaridine	43
Synthesis of Dialkyl-Substituted Monofluoroalkenes via Palladium-Catalyzed Cross-Coupling of Alkyl Carbagermatranes	43
Palladium-Catalyzed Double ipso-Defluoroetherification of Allylic gem-Difluorides with Phenols or Alcohols	43
Deciphering Regulatory Proteins of Prenylated Protein via the FRET Technique Using Nitroso-Based Ene-Ligation and Sequential Azidation and Click Reaction	43
Strain-Release Glycosylation of Thio- and Selenoglycosides Enabled by Activation of Donor–Acceptor Oxiranes with Catalytic TfOH	43
Asymmetric Synthesis of Chiral Aza-macrodiolides via Iridium-Catalyzed Cascade Allylation/Macrolactonization	43
Stereoselective Synthesis of Conjugated Dienes via Aryl-to-Vinyl 1,4-Nickel Migration and Reductive Cross-Coupling	43
Visible-Light-Induced NHC-Catalyzed Carboacylation Reaction of Alkenes from Aryl Thianthrenium Salts and Aldehydes	43
1,3-Butadiene Dicarbofunctionalization Enabled by the Dual Role of Diaryl Ketone in Photo-HAT/Chromium Catalysis	42
Organocalcium-Complex-Catalyzed Dehydrogenative Silylation and Mono/Dihydrosilylation Tandem Reactions of Terminal Alkynes	42
Contractions of 1,4-Diazepines to Pyrroles Triggered by Valence Tautomerization: A One-Pot Approach and Mechanism	42
N-Heterocyclic Carbene Catalysis for Polycyclic Benzazepines Assembly: Regioselective Intramolecular Tandem Radical Cyclization	42
Transformation-Guided Genome Mining Provides Access to Brominated Lanthipeptides	41
Deprotonative Generation and Trapping of Haloaryllithium in a Batch Reactor	41
Photocatalytic Synthesis of α-Ketonyl Glycosyl Compounds from Glycosyl Thiols and Silyl Enol Ethers	41
Biocatalytic Synthesis of Metaxalone and Its Analogues	41
Kinetic Resolution of BINOLs and Biphenols by Atroposelective, Cu–H-Catalyzed Si–O Coupling with Hydrosilanes	41
Effect of Transition Metals on Chemodivergent Cross-Coupling of Acrylamides with Vinyl Acetate via C–H Activation	41
Formal Syntheses of (−)-Quinocarcinamide and (−)-Quinocarcin	41
Mild Installation of Piperidines on 4-Alkylpyridines	41
My Discovery of Science	41
Asymmetric Organocatalysis Enables Rapid Assembly of Portimine Precursor Chains	41
Exploiting Iminoquinones as Electrophilic at Nitrogen “N+” Synthons for C–N Bond Construction	41
Stereoretentive Decarboxylative Amidation of α,β-Unsaturated Carboxylic Acids to Access Enamides	41
Formation and Rearrangement of a Congested Spiropentane from the Trapping of Dibenzonorcarynyliden(e/oid) by Phencyclone	41
Photocatalytic Umpolung Strategy for the Synthesis of α-Amino Phosphine Oxides and Deuterated Derivatives	41
Enantioselective Annulation of α,β-Unsaturated N-Acyliminium Ions with β-Keto Ester Enolates via Cooperative Palladium and Brønsted Acid Catalysis	41
Gold-Catalyzed C–O Cross-Coupling Reactions of Aryl Iodides with Silver Carboxylates	40
Visible-Light-Promoted Reduction of Epoxides, Hydroxysulfonates, and Halohydrines with Alkyltitanium Alkoxides	40
Ligand- and Substrate-Controlled para C–H Borylation of Anilines at Room Temperature	40
Application of Ni/Zr-Mediated Ketone Coupling for the Scalable Synthesis of Homohalichondrin B	40
Diarylamine Synthesis via Desulfinylative Smiles Rearrangement	40
Correction to Phosphine-Catalyzed Cascade Michael Addition/[4+2] Cycloaddition Reaction of Allenoates and 2-Arylidene-1,3-indanediones	40
Preparation of 3,5-Methanobenzo[b]azepines: An sp3-Rich Quinolone Isostere	40
Organic Chemistry in Argentina and the Genesis of SAIQO	40
Synthesis of 3-Benzazepines via Cobalt-Catalyzed C–H Bond Functionalization with CaC2 as the Acetylene Source	40
Photocatalytic Regioselective Alkoxycarbonylation/Cyclization of 3-Aza-1,5-dienes: Access to Ester-Containing Pyrrolin-2-ones	40
Photocatalyzed Aerobic Cross-Dehydrogenative Coupling of Diarylphosphine Oxides with Alcohols and Phenols	40
Cobalt-Catalyzed Enantioselective Reductive Amination of Ketones with Hydrazides	40
Three-Component Couplings among Heteroarenes, Difluorocyclopropenes, and Water via C–H Activation	40
Charge-Enhanced Reactivity of Esters by a Cationic Substituent	40
Ring-Enlargement of in Situ Generated Cyclopropanones by the Reaction with Sulfonium Ylides: One-Pot Synthesis of Cyclobutanones	40
Isolation and Total Synthesis of Beru’amide, an Antitrypanosomal Polyketide from a Marine Cyanobacterium Okeania sp.	40
Solid-Phase Photochemical Decarboxylative Hydroalkylation of Peptides	39
C–C Bond Cleavage-Induced C- to N-Acyl Transfer for Synthesis of Amides	39
Asymmetric Synthesis of Axially Chiral Arylpyrazole via an Organocatalytic Arylation Reaction	39
Synthesis of γ-Butyrolactones with Chiral Quaternary–Tertiary Stereocenters via Catalytic Asymmetric Mukaiyama–Michael Addition	39
Discovery, Characterization, and Anti-XOD Activity of Calcium Metallophore from Coix lacryma-jobi	39
Photochemical Reduction of Quinolines with γ-Terpinene	39
Total Synthesis of (+)-Leucolusine and (−)-7-epi-Leucolusine	39
Amidophosphine Boranes as Hydroboration Reagents for Nitriles, Alkynes, and Carboxylic Acids	39
Electrochemical Cyanation of Alcohols Enabled by an Iodide-Mediated Phosphine P(V/III) Redox Couple	39
Iridium-Catalyzed Double Asymmetric Hydrogenation of 2,5-Dialkylienecyclopentanones for the Synthesis of Chiral Cyclopentanones	39
A Catalytic Enantioselective Suzuki Coupling for the Modular Construction of Axially Chiral BODIPYs with Bright Solid-State Emission	38
Aromatic Amine and Chiral Phosphoric Acid Synergistic Catalyzed Cascade Reaction of Alkynylnaphthols with Aldehydes	38

Vitamin B12 and Micellar Solution Enable Regioselective Ring Opening of Epoxides and Aziridines with Electrophilic Olefins	38
Chromium-Catalyzed Diastereoselective Synthesis of Conformationally Constrained Spirotetrahydroquinolines	38
Stereoselective Synthesis of Acyclic Tetrasubstituted Alkenes from Anilines by Dearomatization and Trimethylenemethane Cycloaddition	38
Electrochemical Desaturation and β-Thiocyanation of Cyclic Amides	38
Fluorous Phase-Enhanced Fluorescent Sensitivity for Enantioselective Recognition of Lysine	38
Enantioselective [3 + 3] Annulation–Deoxalation Strategy for Rapid Access to δ-Oxoesters via N-Heterocyclic Carbene Catalysis	38
Intramolecular Friedel–Crafts Reactions of Sulfamoyl Fluorides, Fluorosulfates, and Sulfuramidimidoyl Fluorides	38
Photoinduced Difluoromethylation Cyclization to Generate Medium-Sized Difluoro-benzo[b]azepines	38
Ruthenium(II)-Catalyzed C–H Activation/Annulation of 5-Phenyl-pyrroline-2-carboxylates with Alkynes: Synthesis of 2,3-Diphenylspiro-[indene-1,2′pyrrolidine]carboxylate Derivatives	38
Biomimetic Total Synthesis of Clavicipitic Acid: A DDQ-Mediated Intramolecular Cross-Dehydrogenative Coupling Approach	38
Synthesis of ortho-Phosphated (Hetero)Arylamines through Cascade Atherton–Todd Reaction/[3,3]-Rearrangement from Arylhydroxylamines and Dialkyl Phosphites	38
Cobalt/Rhodium-Catalyzed Diversified Amidation of Benzocyclobutenols via C–C Cleavage under Catalyst and Condition Control	38
Pd-Catalyzed Asymmetric Intramolecular Dearomatizing Reductive Heck Reaction of Indoles	38
Asymmetric Intramolecular Hydroamination to Construct Diverse N–N/C–N Indole Atropisomers via Cooperative Pd(0) and Chiral Phosphoric Acid Catalysis	38
Sc-Catalyzed Asymmetric [2 + 2] Annulation of 2-Alkynylnaphthols with Dienes to Access Cyclobutene Frameworks	38
Photocatalytic Bicyclization of Indole-Tethered 1,6-Enynes for Diastereoselective Synthesis of Pyrrolo[3,2,1-jk]carbazoles	38
Palladium-Catalyzed Synthesis of Esters from Arenes through C–H Thianthrenation	38
Bicyclic Bridgehead Phosphoramidite-Based Hybrid Diphosphorus Ligands: Design, Synthesis, and Application in Catalytic Asymmetric Hydrogenation	38
Hydrophilic Azide-Containing Amino Acid to Enhance the Solubility of Peptides for SPAAC Reactions	38
Pd-Catalyzed Asymmetric Allylic Substitution Cascade of Substituted 4-Hydroxy-2H-pyrones with meso-Allyl Dicarbonates	37
Minisci-Type Dehydrogenative Coupling of C(sp3)–H and N-Heteroaromatics Enabled by Photoelectrochemical Hydrogen Atom Transfer	37
Switchable Cobalt-Catalyzed α-Olefination and α-Alkylation of Nitriles with Primary Alcohols	37
Synthesis of Sulfur-Substituted Bicyclo[1.1.1]pentanes by Iodo-Sulfenylation of [1.1.1]Propellane	37
Biosynthesis of Dolastatin 10 in Marine Cyanobacteria, a Prototype for Multiple Approved Cancer Drugs	37
Rhodium(III)-Catalyzed Synthesis of Diverse Fluorescent Polycyclic Purinium Salts from 6-Arylpurine Nucleosides and Alkynes	37
A Donor–Acceptor 10-Cycloparaphenylene and Its Use as an Emitter in an Organic Light-Emitting Diode	37
P(O)Me2–Alkenes: From Synthesis to Applications	37
Heteroarylation of Ethers, Amides, and Alcohols with Light and O2	37
Nickel-Catalyzed Photoredox Allenylation of Alkyl Halides	37
Triflylpyridinium as Coupling Reagent for Rapid Amide and Ester Synthesis	36
Gold-Catalyzed Synthesis of Diaza-hexatrienes Via Diazo Attack at Vinylgold Carbenes: An Easy Access to 1H-Pyrazolo[4,3-b]pyridine-5-ones	36
Photochemical “Cut and Sew” Transformations of Ethynylbenziodoxolone Reagents and Diazo Compounds	36
Dithionite-Involved Multicomponent Coupling for Alkenyl and Alkyl Tertiary Sulfones	36
Intramolecular Appel Reaction of Trifluoromethylated β-Keto Diazos Enabling Assembly of Trifluoromethylpyrazoles	36
Electrochemical Allylic C(sp3)–H Isothiocyanation via [3,3]-Sigmatropic Rearrangement	36
Highly Contorted Rigid Nitrogen-Rich Nanographene with Four Heptagons	36
Boron-Catalyzed Michael Reaction of Donor–Acceptor Carboxylic Acid Pairs Enabling Direct Synthesis of 1,5-Dicarboxylic Acids	36
Supramolecular Polymerization of Biphenyl-Cyanostilbenes. Triggering Circularly Polarized Luminescence by Self-Assembly	36
Visible-Light-Induced Cascade Cyclization of 3-(2-(Ethynyl)phenyl)quinazolinones to Phosphorylated Quinolino[2,1-b]quinazolinones	36
Photocatalytic Activation of Elemental Sulfur Enables a Chemoselective Three-Component Thioesterification	36
Rhodium(III)-Catalyzed [4 + 2] Annulation of N-Arylbenzamidines with Propargyl Alcohols: Highly Regioselective Synthesis of 1-Aminoisoquinolines Controlled by Noncovalent Interaction	36
Visible-Light-Induced Three-Component Selenofunctionalization of Alkenes: An Aerobic Selenol Oxidation Approach	36
Synthesis and Structural Revision of the Cyclic Hexapeptide Dimers Antatollamides A and B	36
Diphenylsilylsilanolates Enable the Transfer of a Wide Range of Silyl Groups	36
DMSO as a C1 Source for [2 + 2 + 1] Pyrazole Ring Construction via Metal-Free Annulation with Enaminones and Hydrazines	36
Rhodium-Catalyzed Selective C(sp2)–H Activation/Annulation of tert-Butyl Benzoyloxycarbamates with 1,3-Diynes: A One Step Access to Alkynylated Isocoumarins and Bis-Isocoumari	36
Visible-Light-Induced Photocatalytic Deoxygenative Benzylation of Quinoxalin-2-(1H)-ones with Carboxylic Acid Anhydrides	36
Visible-Light-Driven C,N-Selective Heteroarylation of N-Fluoroalkyl Hydroxylamine Reagents with Quinoxalin-2(1H)-ones	36
Manganese-Catalyzed Regioselective C–H Lactonization and Hydroxylation of Fatty Acids with H2O2	36
Polysubstituted Indole Synthesis via Palladium/Norbornene Cooperative Catalysis of Oxime Esters	35
Copper-Catalyzed Asymmetric Propargylic [3 + 2] Cycloaddition: Synthesis of Enantioenriched Dihydrofuro[3,2-c]coumarins and its Quinolinone and Thiocoumarin Analogues	35
Chiral Brønsted Acid Catalyzed Enantioselective Synthesis of Spiro-Isoindolinone-Indolines via Formal [3 + 2] Cycloaddition	35
Bioorthogonal Fluoride-Responsive Azide and Alkynyl Pyridinium Click Cycloaddition in Vitro and in Live Cells	35
Cobalt(II)-Catalyzed Directed C–H Functionalization/[3+2] Annulation of N-Arylguanidines with Alkynes	35
Main Group-Catalyzed Cationic Claisen Rearrangements via Vinyl Carbocations	35
Photoredox-Catalyzed Synthesis of β-Amino Alcohols: Hydroxymethylation of Imines with α-Silyl Ether as Hydroxymethyl Radical Precursor	35
Electrochemical Synthesis of Fluorinated Ketones from Enol Acetates and Sodium Perfluoroalkyl Sulfinates	35
Dilithium Amides as a Modular Bis-Anionic Ligand Platform for Iron-Catalyzed Cross-Coupling	35
Dual Rh(II)/Pd(0) Relay Catalysis Involving Sigmatropic Rearrangement Using N-Sulfonyl Triazoles and 2-Hydroxymethylallyl Carbonates	35
Cobalt-Catalyzed Migration Isomerization of Dienes	35
Palladium-Catalyzed Asymmetric C–C Bond Activation/Carbonylation of Cyclobutanones	35
Annulative π-Extension by Cp*Co(III)-Catalyzed Ketone-Directed peri-Annulation: An Approach to Access Fused Arenes	35
Selective C–H Iodination of Weinreb Amides and Benzamides through Iridium Catalysis in Solution and under Mechanochemical Conditions	35
Synthesis of ortho-Methylated Benzamides via Palladium-Catalyzed Denitrogenative Cross-Coupling Reaction of [1,2,3]-Benzotriazin-4(3H)-ones with DABAL-Me3	35
Palladium-Catalyzed 1,2-Alkynylarylation of Vinyl Arenes with Haloalkynes and Arylboronic Acids	35
Hydrazone Activation in the Aminocatalytic Cascade Reaction for the Synthesis of Tetrahydroindolizines	35
Aldehydes as O-Nucleophiles in Cobalt Hydride Hydrogen Atom Transfer Catalysis: Overriding the Innate Somophilicity	35
Correction to “Regioselective Synthesis of Highly Functionalized Pyrazoles from N-Tosylhydrazones”	35
Synthesis of Flavanone and Quinazolinone Derivatives from the Ruthenium-Catalyzed Deaminative Coupling Reaction of 2′-Hydroxyaryl Ketones and 2-Aminobenzamides with Simple Amines	35
AJICAP-M: Traceless Affinity Peptide Mediated Conjugation Technology for Site-Selective Antibody–Drug Conjugate Synthesis	35
Dysambiol, an Anti-inflammatory Secomeroterpenoid from a Dysidea sp. Marine Sponge	34
Biomimetic Asymmetric Reduction of Tetrasubstituted Olefin 2,3-Disubstituted Inden-1-ones with Chiral and Regenerable NAD(P)H Model CYNAM	34
Metal-Free Generation of γ-Cyanoalkyl Radicals by N-Heterocyclic Carbene Catalysis: Assembly of 6-Cyanoalkyl Phenanthridines	34
Organocatalytic Michael Addition of Unactivated α-Branched Nitroalkanes to Afford Optically Active Tertiary Nitrocompounds	34
Neogrisemycin, a Trisulfide-Bridged Angucycline, Produced upon Expressing the Thioangucycline Biosynthetic Gene Cluster in Streptomyces albus J1074	34
[Au]/[Ag]-Catalyzed Glycosidation of Ethynylcyclohexyl Glycosyl Carbonates Enables Direct Stereoselective Synthesis of 2-Azido-2-deoxy-β-mannopyranosides	34
Rhodium-Catalyzed Three-Component Reaction of Alkynes, Arylzinc Chlorides, and Iodomethanes Producing Trisubstituted/Tetrasubstituted Alkenes with/without 1,4-Migration	34
Chemoselective Transformations of Amides: An Approach to Quinolones from β-Amido Ynones	34
Retraction of Activating Imides with Triflic Acid: A General Intramolecular Aldol Condensation Strategy Toward Indolizidine, Quinolizidine, and Valmerin Alkaloids	34
Kinetic Resolution of N-Allylic Pyrazoles via Photoexcited Chiral Copper Complex-Catalyzed Alkene E → Z Isomerization	34
Studies towards the Enantioselective Synthesis of Cryptowolinol via Pd0-Catalyzed C(sp3)–H Arylation/Parallel Kinetic Resolution	34
Rhodium-Catalyzed Trifluoromethoxylation of Allenylic Trichloroacetimidates	34
Organocatalytic Asymmetric Arylation of p-Quinone Phosphonates: A Green Access to Biaryl Monophosphorus Ligands	34
Amino-Based Probe for Natural Products with Covalent Binding Ability to Lysine and Mechanism of Action of Medermycin	34
A Neophyl Palladacycle as an Air- and Thermally Stable Precursor to Oxidative Addition Complexes	33
Asymmetric Synthesis of Bicyclic Isoxazolines via Dearomative Cycloaddition of 4-Nitroisoxazoles with Zwitterionic π-Allyl Palladium Species	33
Oxime Ether Synthesis through O–H Functionalization of Oximes with Diazo Esters under Blue LED Irradiation	33
A Stereoselective Photoinduced Cycloisomerization Inspired by Ophiobolin A	33
Solid-Phase-Based Synthesis of Lactazole-Like Thiopeptides	33
Diastereocontrolled Construction of Spiroindolenines via Hexafluoroisopropanol-Promoted Dearomative Epoxide–Indole Cyclization	33
Synthesis of Enantioenriched gem-Disubstituted 4-Imidazolidinones by Palladium-Catalyzed Decarboxylative Asymmetric Allylic Alkylation	33
Palladium-Catalyzed Coordination-Induced Remote C–H Aryl Etherification/Amination of 8-Amidoquinolines	33
Three-Component, Diastereoselective [6 + 3] Annulation of Tropone, Imino Esters, and Arynes	33
Synthesis of Non- or Antiaromatic Dicarbaamethyrin: [24]Diazulihexaphyrin(0.1.0.0.1.0)	33
Electrocatalysis-Enabled Stereoselective Synthesis of Monofluoroalkenes via Hydrodefluorination of gem-Difluoroakenes	33