Organic Letters

Papers
(The median citation count of Organic Letters is 5. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2021-09-01 to 2025-09-01.)
ArticleCitations
Total Synthesis of (±)-Furanether A85
Construction of Oxo-Bridged Diazocines via Rhodium-Catalyzed (4+3) Cycloaddition of Carbonyl Ylides with Azoalkenes84
Reductive Hydrodehalogenation of Halogenated Carboxylic Acid Derivatives Using a DMSO/HCOONa·2H2O System83
Direct Synthesis of α-Methylated Arylacetamides from Arylacetonitriles via Ir-Catalyzed Cascade α-Methylation and Selective Hydration81
Macrocyclization of Unprotected Peptides via Cycloaddition between o-Diones and Furan-2(3H)-one79
Ascomycotols A–C: Rare Sulfur/Sulfone-Containing Scaffolds from Mushroom Endophytes with Dual Anti-inflammatory and Antirenal Fibrosis Effects77
Visible-Light-Induced Selective α-Fluoroarylation of Secondary N-Alkyl Anilines with Polyfluoroarenes via Direct C–H/C–F Coupling77
Stereoselective Double Spirocyclization of 2-Benzyl-3-alkynyl Chromone with Nitrone via Gold-Catalyzed Cascade Reactions75
Computationally Assisted Analysis of NMR Chemical Shifts as a Tool in Conformational Analysis75
Borylative Cyclization of 1,6-Allenynes Driven by BCl373
Synthesis of γ-Butyrolactones with Chiral Quaternary–Tertiary Stereocenters via Catalytic Asymmetric Mukaiyama–Michael Addition72
Selective C–H Iodination of Weinreb Amides and Benzamides through Iridium Catalysis in Solution and under Mechanochemical Conditions71
Bicyclic Bridgehead Phosphoramidite-Based Hybrid Diphosphorus Ligands: Design, Synthesis, and Application in Catalytic Asymmetric Hydrogenation71
Biocatalytically Generated Library of Chiral Building Blocks Containing a Quaternary Stereocenter70
Synthesis of 3-Benzazepines via Cobalt-Catalyzed C–H Bond Functionalization with CaC2 as the Acetylene Source68
Palladium-Catalyzed Double ipso-Defluoroetherification of Allylic gem-Difluorides with Phenols or Alcohols68
Kinetic Resolution of BINOLs and Biphenols by Atroposelective, Cu–H-Catalyzed Si–O Coupling with Hydrosilanes66
Dichloromethyl(diaryl) Sulfonium Salts as gem-Dichlorocyclopropanation Reagents65
Highly Contorted Rigid Nitrogen-Rich Nanographene with Four Heptagons63
Enantioselective Palladium-Catalyzed Domino Carbonylative Heck Esterification of o-Iodoalkenylbenzenes with Arylboronic Acids61
Chiral Brønsted Acid Catalyzed Enantioselective Synthesis of Spiro-Isoindolinone-Indolines via Formal [3 + 2] Cycloaddition61
Deciphering the δ-Lactam Formation and lron-Reducing Activity of Spinactins from Saccharopolyspora spinosa60
Synthesis of α-Aryl Secondary Amides via Nickel-Catalyzed Reductive Coupling of Redox-Active Esters60
Oxoammonium Salt-Mediated Regioselective Vicinal Dioxidation of Alkenes: Relying on Transient and Persistent Nitroxides59
Nonactivated Aziridine Synthesis by Intermolecular Polarity-Mismatched Carboamination of Unactivated Alkenes with Unactivated Alkyl Halides58
Photocatalytic Strecker-Type Reaction for the Synthesis of Primary α-Aminonitriles58
Spirochrains A–D, Four Caged [5,6,5] Spirocyclic Amides from an Antarctic Fungus Aspergillus ochraceopetaliformis SCSIO 05702 with Anti-RSV Activities57
Nickel-Catalyzed Deaminative Allenylation of Amino Acid Derivatives: Catalytic Activity Enhanced by an Amide-Type NN2 Pincer Ligand57
Dinickel-Catalyzed Asymmetric Allylic Alkylation of Cyclic Ketones with Allylic Amine Derivatives56
Enantioselective Cobalt-Catalyzed Remote Hydroboration of Alkenylboronates56
Kinetic Resolution of Sulfinamides via Asymmetric N-Allylic Alkylation55
Environmentally Friendly Synthesis of Highly Substituted Phenols Using Enallenoates and Grignard Reagents55
Gold-Catalyzed Regioselective Synthesis of Crowded Cyclopentadienes by Migratory Cycloisomerization of Vinylallenes55
Cope-Type Hydroamination of Vinylboronates55
Tosylazide as N1-Synthon: Iron-Catalyzed Nitrogenative Dimerization of Indoles to p-Bisindolopyrazine Derivatives54
Correction to “Access to 6-Deoxy-heptose Constructs by One Carbon Homologation of Hexoses with Malononitrile: Divergent Synthesis of Campylobacter jejuni Strain 81-176 Capsular Trisaccharide Re54
DNA-Compatible Diversification of Indole π-Activated Alcohols via a Direct Dehydrative Coupling Strategy53
Sequential One-Pot Transformation to R–CF2-Embedded 1,5-Diketones Enabled by Nickel: Access to 4-Perfluoroalkylpyridines53
Manipulating Crystal Packing and Self-Assembly by π-Extended and Isomeric Fused Strategies in Thiophene Ring-Terminated Polycyclic Aromatic Hydrocarbons53
Synthesis of 1-Substituted Bicyclo[2.1.1]hexan-2-ones via a Sequential SmI2-Mediated Pinacol Coupling and Acid-Catalyzed Pinacol Rearrangement Reaction52
Collective Syntheses of Corynanthe Alkaloids Based on a Chirality-Tunable Structure Unit52
Gold(I)-Catalyzed Oxidative Amination of β-Amino-ynones to Quaternary Ammonium-olate Salts: The Benefit of a P,N-Bidentate Ligand51
Rh-Catalyzed Carbonylative Cyclization of Propargylic Alcohols with Aryl Boronic Acids51
Asymmetric Synthesis of CF3-Substituted β-Hydroxyketones and 1,3-Diols by Engineered Ketoreductases51
Sequential Strategies to Trigger Mild Dearomative Diels–Alder Cyclizations51
Regiochemical Switching in Ir-Catalyzed C–H Borylation by Altering Ligand Loadings of N,B-Type Diboron Species51
Systematic Route to Construct the 5–5–6 Tricyclic Core of Furanobutenolide-Derived Cembranoids and Norcembranoids51
Chiral Squaramide Catalyzed Asymmetric Spiroketalization toward Aromatic [6,5] Spiroketals50
DalPhos/Nickel-Catalyzed C2–H Arylation of 1,3-Azoles Using a Dual-Base System50
Expanded Access to Fluoroformamidines via a Modular Synthetic Pathway50
Weak-Chelation Assisted Cobalt-Catalyzed C–H Bond Activation: An Approach Toward Regioselective Ethynylation of N-Aryl γ-Lactam49
A Sterically Tuned 2-Fluoropyridinium Salt for the Catalyst-Free, Visible-Light-Mediated Deoxygenation of Alcohols via an Electron Donor–Acceptor Complex49
Radical Alkynylthiolation with Visible-Light-Sensitive S-Alkynylthio Sulfonates49
Palladium-Catalyzed Asymmetric (3 + 2) Cycloaddition of 5-Allenyloxazolidine-2,4-Diones with Barbiturate-Derived Alkenes: Synthesis of Spirobarbiturate-γ-Lactams49
Regioselective Alkylacylation of 1,3-Dienes by Merging N-Heterocyclic Carbene Catalysis with Photoinduced Palladium Catalysis49
Divergent Access to Polycyclic N-Heterocyclic Compounds through Büchner-Type Dearomatization Enabled Cycloisomerization of Diynamides under Gold Catalysis48
Synergistic Copper/Enamine Catalysis for the Regio-, Stereo-, and Enantioselective Intermolecular α-Addition of Aldehydes to Allenamides48
Staudinger Cleavages of Amides on Naphthalene for the Ipsilateral Effect of 1,8-Substituents48
Asymmetric Synthesis of Chiral Aza-macrodiolides via Iridium-Catalyzed Cascade Allylation/Macrolactonization48
From Nitrogen to Sulfur: Investigating the Effect of Core Modification within Azaacene-Fused 21,23-Dithiaporphyrins48
Synthesis of Tertiary Amines through Extrusive Alkylation of Carbamates48
Contractions of 1,4-Diazepines to Pyrroles Triggered by Valence Tautomerization: A One-Pot Approach and Mechanism47
Stereoretentive Decarboxylative Amidation of α,β-Unsaturated Carboxylic Acids to Access Enamides47
Strain-Release Glycosylation of Thio- and Selenoglycosides Enabled by Activation of Donor–Acceptor Oxiranes with Catalytic TfOH47
Organocalcium-Complex-Catalyzed Dehydrogenative Silylation and Mono/Dihydrosilylation Tandem Reactions of Terminal Alkynes47
Mild Installation of Piperidines on 4-Alkylpyridines47
Deciphering Regulatory Proteins of Prenylated Protein via the FRET Technique Using Nitroso-Based Ene-Ligation and Sequential Azidation and Click Reaction47
Deprotonative Generation and Trapping of Haloaryllithium in a Batch Reactor47
Formal Syntheses of (−)-Quinocarcinamide and (−)-Quinocarcin47
Transformation-Guided Genome Mining Provides Access to Brominated Lanthipeptides46
Photocatalytic Synthesis of α-Ketonyl Glycosyl Compounds from Glycosyl Thiols and Silyl Enol Ethers46
Vitamin B12 and Micellar Solution Enable Regioselective Ring Opening of Epoxides and Aziridines with Electrophilic Olefins46
Formation and Rearrangement of a Congested Spiropentane from the Trapping of Dibenzonorcarynyliden(e/oid) by Phencyclone46
My Discovery of Science46
Palladium-Catalyzed Domino Conversion of Aryl–Thianthreniums with Anhydrides: Rapidly Building Highly Functionalized Fluorenones45
Photocatalytic Borylation of Imines and Alkenes via Decarboxylation of Trimethylamine Carboxyborane: A New Approach for Generating Boryl Radicals45
P(O)Me2–Alkenes: From Synthesis to Applications45
Enantioselective [3 + 3] Annulation–Deoxalation Strategy for Rapid Access to δ-Oxoesters via N-Heterocyclic Carbene Catalysis45
Polysubstituted Indole Synthesis via Palladium/Norbornene Cooperative Catalysis of Oxime Esters45
Visible-Light-Induced Three-Component Selenofunctionalization of Alkenes: An Aerobic Selenol Oxidation Approach44
Synthesis and Structural Revision of the Cyclic Hexapeptide Dimers Antatollamides A and B44
Annulative π-Extension by Cp*Co(III)-Catalyzed Ketone-Directed peri-Annulation: An Approach to Access Fused Arenes44
Pd-Catalyzed Asymmetric Intramolecular Dearomatizing Reductive Heck Reaction of Indoles44
Diversity-Oriented Synthesis of ERα Modulators via Mitsunobu Macrocyclization44
DMSO as a C1 Source for [2 + 2 + 1] Pyrazole Ring Construction via Metal-Free Annulation with Enaminones and Hydrazines44
C–C Bond Cleavage-Induced C- to N-Acyl Transfer for Synthesis of Amides44
Ligand-Controlled Diastereodivergency in Propargylic Alkylation of Vinylogous Aza-Enamines: Construction of 1,3-Stereocenters44
Enantioselective Organocatalytic Conjugate Addition of Malonates to β,β-Disubstituted β-Trifluoromethyl Enones under High Pressure44
Syntheses and Properties of Hole-Transporting Biindenofluorenes43
Palladium-Catalyzed Chemo- and Regiocontrolled Tandem Cyclization/Cross-Coupling of 2-Benzyl-3-alkynyl Chromones with Aryl Iodides for the Synthesis of 4H-Furo[3,2-c]chromenes and Xantho43
Visible-Light-Induced NHC-Catalyzed Carboacylation Reaction of Alkenes from Aryl Thianthrenium Salts and Aldehydes43
Electrochemical Desaturation and β-Thiocyanation of Cyclic Amides43
Photochemical Organocatalytic Aerobic Cleavage of C═C Bonds Enabled by Charge-Transfer Complex Formation43
Visible-Light-Induced Photocatalytic Deoxygenative Benzylation of Quinoxalin-2-(1H)-ones with Carboxylic Acid Anhydrides43
Synthesis of Planar Chiral 2-Aryl Aroylferrocenes via Palladium-Catalyzed C–C Bond-Cleavage/Ring-Opening Reaction43
Photoredox-Catalyzed Synthesis of β-Amino Alcohols: Hydroxymethylation of Imines with α-Silyl Ether as Hydroxymethyl Radical Precursor43
Synthesis of ortho-Phosphated (Hetero)Arylamines through Cascade Atherton–Todd Reaction/[3,3]-Rearrangement from Arylhydroxylamines and Dialkyl Phosphites43
Photocatalyzed Aerobic Cross-Dehydrogenative Coupling of Diarylphosphine Oxides with Alcohols and Phenols43
Minisci-Type Dehydrogenative Coupling of C(sp3)–H and N-Heteroaromatics Enabled by Photoelectrochemical Hydrogen Atom Transfer43
Visible-Light-Induced Cascade Cyclization of 3-(2-(Ethynyl)phenyl)quinazolinones to Phosphorylated Quinolino[2,1-b]quinazolinones43
Diarylamine Synthesis via Desulfinylative Smiles Rearrangement42
Nickel-Catalyzed Photoredox Allenylation of Alkyl Halides42
Issue Publication Information42
Rhodium(III)-Catalyzed Synthesis of Diverse Fluorescent Polycyclic Purinium Salts from 6-Arylpurine Nucleosides and Alkynes42
Fluorous Phase-Enhanced Fluorescent Sensitivity for Enantioselective Recognition of Lysine42
Dual 1,2-Migration-Enabled β-Boryl Amide Synthesis42
Visible-Light-Induced Difunctionalization of 3-Butenoic Acid with Bromodifluoromethyl Heteroarylsulfones42
Free Amine-Directed Redox Neutral Ruthenium(II) Catalysis toward Regioselective Synthesis of Heterobiaryls42
Paired Electrocatalysis-Enabled Cross Coupling of Sulfinamides with Olefins toward the Synthesis of Vinyl Sulfoximines42
Total Synthesis of Daphenylline via Diels–Alder Cycloaddition and Rhodium-Catalyzed C–H Alkynylation42
Issue Publication Information42
Total Synthesis of the Phenolic Steroid Myrmenaphthol A42
Issue Editorial Masthead41
Issue Editorial Masthead41
Protecting-Group Free Total Synthesis of β-Levantenolide through Late Stage Bromo-Spirocyclization41
Ring-Enlargement of in Situ Generated Cyclopropanones by the Reaction with Sulfonium Ylides: One-Pot Synthesis of Cyclobutanones41
Issue Publication Information41
Issue Editorial Masthead41
Issue Editorial Masthead41
Boron-Catalyzed Michael Reaction of Donor–Acceptor Carboxylic Acid Pairs Enabling Direct Synthesis of 1,5-Dicarboxylic Acids41
Asymmetric Intramolecular Hydroamination to Construct Diverse N–N/C–N Indole Atropisomers via Cooperative Pd(0) and Chiral Phosphoric Acid Catalysis41
Issue Editorial Masthead41
Issue Publication Information41
Visible-Light-Driven C,N-Selective Heteroarylation of N-Fluoroalkyl Hydroxylamine Reagents with Quinoxalin-2(1H)-ones41
Electrochemical Allylic C(sp3)–H Isothiocyanation via [3,3]-Sigmatropic Rearrangement41
Conformationally Fluxional Pseudo-C2 Symmetric Decaphyrins (1.0.0.0.0.1.0.0.0.0) with Multiple m-Phenylene Subunits and Their Cyclic Bis-BODIPYs41
Asymmetric Organocatalysis Enables Rapid Assembly of Portimine Precursor Chains40
Preparation of 3,5-Methanobenzo[b]azepines: An sp3-Rich Quinolone Isostere40
Charge-Enhanced Reactivity of Esters by a Cationic Substituent40
Iridium-Catalyzed Double Asymmetric Hydrogenation of 2,5-Dialkylienecyclopentanones for the Synthesis of Chiral Cyclopentanones40
Application of Ni/Zr-Mediated Ketone Coupling for the Scalable Synthesis of Homohalichondrin B40
Enantioselective Annulation of α,β-Unsaturated N-Acyliminium Ions with β-Keto Ester Enolates via Cooperative Palladium and Brønsted Acid Catalysis40
Ligand- and Substrate-Controlled para C–H Borylation of Anilines at Room Temperature40
Discovery, Characterization, and Anti-XOD Activity of Calcium Metallophore from Coix lacryma-jobi40
Biomimetic Total Synthesis of Clavicipitic Acid: A DDQ-Mediated Intramolecular Cross-Dehydrogenative Coupling Approach40
Organic Chemistry in Argentina and the Genesis of SAIQO40
Isolation and Total Synthesis of Beru’amide, an Antitrypanosomal Polyketide from a Marine Cyanobacterium Okeania sp.40
Total Synthesis of (+)-Leucolusine and (−)-7-epi-Leucolusine40
Stereoselective Synthesis of Acyclic Tetrasubstituted Alkenes from Anilines by Dearomatization and Trimethylenemethane Cycloaddition40
Chromium-Catalyzed Diastereoselective Synthesis of Conformationally Constrained Spirotetrahydroquinolines39
Pd-Catalyzed Asymmetric Allylic Substitution Cascade of Substituted 4-Hydroxy-2H-pyrones with meso-Allyl Dicarbonates39
Hydrazone Activation in the Aminocatalytic Cascade Reaction for the Synthesis of Tetrahydroindolizines39
Palladium-Catalyzed “Cut-and-Sew” Reaction of C(sp3)–NC: Direct Synthesis of Bulky Nitriles Containing an All-Carbon Quaternary Center39
N-Heterocyclic Carbene Catalysis for Polycyclic Benzazepines Assembly: Regioselective Intramolecular Tandem Radical Cyclization39
Sc-Catalyzed Asymmetric [2 + 2] Annulation of 2-Alkynylnaphthols with Dienes to Access Cyclobutene Frameworks39
Photochemical “Cut and Sew” Transformations of Ethynylbenziodoxolone Reagents and Diazo Compounds39
Palladium-Catalyzed Synthesis of Esters from Arenes through C–H Thianthrenation39
Manganese-Catalyzed Regioselective C–H Lactonization and Hydroxylation of Fatty Acids with H2O239
A Catalytic Enantioselective Suzuki Coupling for the Modular Construction of Axially Chiral BODIPYs with Bright Solid-State Emission39
Ruthenium(II)-Catalyzed C–H Activation/Annulation of 5-Phenyl-pyrroline-2-carboxylates with Alkynes: Synthesis of 2,3-Diphenylspiro-[indene-1,2′pyrrolidine]carboxylate Derivatives39
Intramolecular Friedel–Crafts Reactions of Sulfamoyl Fluorides, Fluorosulfates, and Sulfuramidimidoyl Fluorides39
Diphenylsilylsilanolates Enable the Transfer of a Wide Range of Silyl Groups39
Supramolecular Polymerization of Biphenyl-Cyanostilbenes. Triggering Circularly Polarized Luminescence by Self-Assembly39
Hydrophilic Azide-Containing Amino Acid to Enhance the Solubility of Peptides for SPAAC Reactions39
A Synthetic Strategy for the Preparation of Fused [5,6,5,5]-Tetracyclic Energetic Compounds38
Aromatic Amine and Chiral Phosphoric Acid Synergistic Catalyzed Cascade Reaction of Alkynylnaphthols with Aldehydes38
Light-Induced Activation of C–X Bond via Carbonate-Assisted Anion−π Interactions: Applications to C–P and C–B Bond Formation38
Nickel-Catalyzed Cross-Electrophile Ring Opening/gem-Difluoroallylation of Aziridines38
Triflylpyridinium as Coupling Reagent for Rapid Amide and Ester Synthesis38
Cobalt-Catalyzed Enantioselective Reductive Amination of Ketones with Hydrazides38
Palladium-Catalyzed 1,2-Alkynylarylation of Vinyl Arenes with Haloalkynes and Arylboronic Acids38
Photoinduced Difluoromethylation Cyclization to Generate Medium-Sized Difluoro-benzo[b]azepines38
Isolation and Bioinspired Total Synthesis of Rugosiformisin A, A Skeleton-Rearranged Abietane-Type Diterpenoid from Isodon rugosiformis38
Versatile Access to Tetrasubstituted 2-Amidoacroleins through Formal Silylformylation of Ynamides38
Synthesis of Sulfur-Substituted Bicyclo[1.1.1]pentanes by Iodo-Sulfenylation of [1.1.1]Propellane38
Asymmetric Synthesis of Axially Chiral Arylpyrazole via an Organocatalytic Arylation Reaction38
Photocatalytic Activation of Elemental Sulfur Enables a Chemoselective Three-Component Thioesterification38
Iridium-Catalyzed Regio- and Enantioselective C7-Allylic Alkylation of 4-Aminoindoles38
Ir-Catalyzed Asymmetric Cascade Allylation/Spiroketalization Reaction for Stereoselective Synthesis of Oxazoline-Spiroketals37
Multiselective Diels–Alder Reaction of α-Arylacroleins Catalyzed by Boron Tribromide-Assisted Chiral Phosphoric Acids37
Photochemical Reduction of Quinolines with γ-Terpinene37
AJICAP-M: Traceless Affinity Peptide Mediated Conjugation Technology for Site-Selective Antibody–Drug Conjugate Synthesis37
Copper-Catalyzed Chan–Lam Reaction and Sequential Oxidative Fischer Indole Synthesis to Prepare Indole Derivatives37
Synthesis of ortho-Methylated Benzamides via Palladium-Catalyzed Denitrogenative Cross-Coupling Reaction of [1,2,3]-Benzotriazin-4(3H)-ones with DABAL-Me337
On-DNA Synthesis of Privileged Dihydropteridinones via Diboron-Mediated Cyclizations37
Cobalt/Rhodium-Catalyzed Diversified Amidation of Benzocyclobutenols via C–C Cleavage under Catalyst and Condition Control37
Domino Semipinacol/Iterative Aldol/Iso-Nazarov Cyclization to Triaryl-cyclopentenone: Enantioselective Synthesis of Combretastatin A-4 Analogues37
Asymmetric Synthesis of β-Aminoboronates via Copper-Catalyzed Reductive Coupling of Vinyl Boronates with Imines37
Visible-Light-Promoted Reduction of Epoxides, Hydroxysulfonates, and Halohydrines with Alkyltitanium Alkoxides37
Base Metal-Controlled Chemodivergent Cyclization of Propargylamines for the Atom-Economic Synthesis of Nitrogen Heterocycles37
Electrochemical Cyanation of Alcohols Enabled by an Iodide-Mediated Phosphine P(V/III) Redox Couple37
Solid-Phase Photochemical Decarboxylative Hydroalkylation of Peptides37
Nickel/SKP-Catalyzed Markovnikov Regio- and Enantioselective Hydroamination of Vinylarenes with Hydroxylamines37
Amidophosphine Boranes as Hydroboration Reagents for Nitriles, Alkynes, and Carboxylic Acids37
Exo-Selective and Enantioselective Photoenolization/Diels–Alder Reaction37
Visible-Light Catalyzed Desulfurative Cyclization for Synthesis of 3-Amino-[1,2,4]-triazolo Pyridine37
Photocatalytic Regioselective Alkoxycarbonylation/Cyclization of 3-Aza-1,5-dienes: Access to Ester-Containing Pyrrolin-2-ones36
Copper-Catalyzed Asymmetric Propargylic [3 + 2] Cycloaddition: Synthesis of Enantioenriched Dihydrofuro[3,2-c]coumarins and its Quinolinone and Thiocoumarin Analogues36
Intramolecular Appel Reaction of Trifluoromethylated β-Keto Diazos Enabling Assembly of Trifluoromethylpyrazoles36
Photoredox Catalytic Approach for Difluoroallylation of Electron-Deficient sp3 C–H Bonds36
1,3-Butadiene Dicarbofunctionalization Enabled by the Dual Role of Diaryl Ketone in Photo-HAT/Chromium Catalysis36
Solvent-Driven Room-Temperature Curtius Rearrangements to Access Nucleotides Bearing Substituted Fused Pyridones36
Exploiting Iminoquinones as Electrophilic at Nitrogen “N+” Synthons for C–N Bond Construction36
Aldehydes as O-Nucleophiles in Cobalt Hydride Hydrogen Atom Transfer Catalysis: Overriding the Innate Somophilicity36
Visible-Light-Promoted Selenylative Radical Cyclization of 2-Vinyl-N-Aryl Imines to 3H-Indoles via Oxygen Photosensitization36
Biocatalytic Synthesis of Metaxalone and Its Analogues36
Biosynthesis of Dolastatin 10 in Marine Cyanobacteria, a Prototype for Multiple Approved Cancer Drugs36
Photocatalytic Bicyclization of Indole-Tethered 1,6-Enynes for Diastereoselective Synthesis of Pyrrolo[3,2,1-jk]carbazoles36
Domino Synthesis of Thioindirubin via Aldol Condensation/C–S Cross-Coupling/Cyclization Reaction Using Xanthate as a Sulfur Surrogate36
Nickel-Catalyzed Domino Reaction of α-Aryloxyacetonitriles with Arylboronic Acids: Synthesis of 2-Aroylbenzo[b]furans36
Access to SCF3-Substituted Indolizines via a Photocatalytic Late-Stage Functionalization Protocol36
Photocatalytic Umpolung Strategy for the Synthesis of α-Amino Phosphine Oxides and Deuterated Derivatives36
Tertiary Amine-Mediated Reductions of Phosphine Oxides to Phosphines36
New Approach to Assembling Nucleic Acid Dendrons on a Solid Phase35
A Donor–Acceptor 10-Cycloparaphenylene and Its Use as an Emitter in an Organic Light-Emitting Diode35
Cobalt-Catalyzed Intramolecular [4 + 2] Cycloaddition of Cyclopropyl-Capped Dienes with Alkynes/Alkenes/Allene and Reaction Mechanism35
Environmentally Responsible and Cost-Effective Synthesis of the Antimalarial Drug Pyronaridine35
[Au]/[Ag]-Catalyzed Glycosidation of Ethynylcyclohexyl Glycosyl Carbonates Enables Direct Stereoselective Synthesis of 2-Azido-2-deoxy-β-mannopyranosides35
Solid-Phase Total Synthesis of Plusbacin A335
Synergistic [4 + 1] Spiroannulation and Selective Ring-Opening Strategy toward γ-Spirolactams35
Stereoselective Synthesis of Conjugated Dienes via Aryl-to-Vinyl 1,4-Nickel Migration and Reductive Cross-Coupling35
Rhodium-Catalyzed Selective C(sp2)–H Activation/Annulation of tert-Butyl Benzoyloxycarbamates with 1,3-Diynes: A One Step Access to Alkynylated Isocoumarins and Bis-Isocoumari35
Gold-Catalyzed C–O Cross-Coupling Reactions of Aryl Iodides with Silver Carboxylates35
Studies towards the Enantioselective Synthesis of Cryptowolinol via Pd0-Catalyzed C(sp3)–H Arylation/Parallel Kinetic Resolution35
Ni-Catalyzed Reductive Coupling of Acetals with Anhydrides and Vinyl Triflates via Single-Electron C–O Activation35
Dioxygen-Triggered Oxosulfonylation/Sulfonylation of Terminal Olefins toward β-Keto Sulfones/Sulfones35
Lewis Acid-Catalyzed Annulations of Geminally Disubstituted Cyclopropanes with Aldehydes or 1,3,5-Triazinanes35
Relay Annulation of Ammonium Ylides with Oxindole-Derived α,β-Unsaturated Ketimines: Catalytic Construction of Spiro-polycyclic Oxindoles35
Correction to “Regioselective Synthesis of Highly Functionalized Pyrazoles from N-Tosylhydrazones”35
Rhodium-Catalyzed Three-Component Reaction of Alkynes, Arylzinc Chlorides, and Iodomethanes Producing Trisubstituted/Tetrasubstituted Alkenes with/without 1,4-Migration35
Rhodium-Catalyzed Synthesis of Peptide Polysulfides by Insertion of Sulfur into Unprotected Peptide Disulfides34
Neogrisemycin, a Trisulfide-Bridged Angucycline, Produced upon Expressing the Thioangucycline Biosynthetic Gene Cluster in Streptomyces albus J107434
Retraction of Activating Imides with Triflic Acid: A General Intramolecular Aldol Condensation Strategy Toward Indolizidine, Quinolizidine, and Valmerin Alkaloids34
Bidipyrrin AuIII Complex as a Helical Charged π-Electronic System34
Synthesis of Non- or Antiaromatic Dicarbaamethyrin: [24]Diazulihexaphyrin(0.1.0.0.1.0)34
Light-Initiated Four-Step Domino-Multicomponent Synthesis of Functionalized Alkylidenecyclobutanes34
Organocatalytic Asymmetric Arylation of p-Quinone Phosphonates: A Green Access to Biaryl Monophosphorus Ligands34
Copper-Catalyzed Nucleophilic Cycloisomerization Cascade Constructing Azepinoindolizine34
A Stereoselective Photoinduced Cycloisomerization Inspired by Ophiobolin A34
Palladium-Catalyzed Coordination-Induced Remote C–H Aryl Etherification/Amination of 8-Amidoquinolines34
Stereoselective Synthesis of a Protected Side Chain of Callipeltin A34
Two Bioactive Compounds, Uniformides A and B, Isolated from a Culture of Nocardia uniformis IFM0856T in the Presence of Animal Cells34
Organocatalytic Michael Addition of Unactivated α-Branched Nitroalkanes to Afford Optically Active Tertiary Nitrocompounds34
Water-Mediated Intramolecular Cyclization/Oxidation of α-Carbonyl Sulfur Ylides: Synthesis of Corey–Chaykovsky Reagent Type Heterocycles34
Electrocatalysis-Enabled Stereoselective Synthesis of Monofluoroalkenes via Hydrodefluorination of gem-Difluoroakenes34
Ni-Catalyzed Kumada–Corriu Cross-Coupling Reactions of Tertiary Grignard Reagents and Bromostyrenes34
Bifunctional Lewis Base-Catalyzed (3 + 2) Cycloadditions of Pyrazolone-Derived MBH Carbonates with Arynes33
Correction to “Development of Fmoc-Protected Bis-Amino Acids toward Automated Synthesis of Highly Functionalized Spiroligomers”33
A Visible Light Photoredox Approach for Synthesizing Sulfone-Functionalized Cyclopropenes33
Ni-H-Catalyzed Regioselective Hydroalkylation of Terminal Alkynes with α-Bromo Phosphonates33
Selective Detection of Choline in Pseudophysiological Medium with a Fluorescent Cage Receptor33
Organocatalyzed Enantio- and Diastereoselective Formal Domino 1,3-Dipolar Cycloaddition/Rearrangement: Synthesis of Chiral Pyrrolo-thiazine-2-carbaldehydes33
Syn-Selective Chlorosulfonylation of Alkynes via a Copper-Powder-Initiated Atom Transfer Radical Addition Reaction and Mechanistic Studies33
Pd-Catalyzed Three-Component Coupling of Cyclopropenones via Sequential C–C Bond Activation and Allylation33
Diastereodivergent α-Homoallylation of Cyclic Enones33
Ketenimines as Intermediates To Access Difluoromethoxylated Scaffolds33
Synthesis of N-Fused Triazole–Piperazine–Quinazolinones via One-Pot Tandem Click Reaction and Cross-Dehydrogenative Coupling33
Regioselective Halogenation of Lavanducyanin by a Site-Selective Vanadium-Dependent Chloroperoxidase33
Construction of C(sp2)–Si Bonds via Ligand-Promoted C–C Bonds Cleavage of Unstrained Ketones33
Rh(III)-Catalyzed [4 + 1] Annulation of Benzamides with Vinyl Cyclic Carbonates for the Synthesis of Isoindolinones33
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