OOIR: Observatory of International Research

Papers

(The TQCC of Advanced Synthesis & Catalysis is 9. The table below lists those papers that are above that threshold based on CrossRef citation counts [max. 250 papers]. The publications cover those that have been published in the past four years, i.e., from 2022-05-01 to 2026-05-01.)

Article	Citations
Electrochemical Stereoselective Synthesis of (Z)‐Allyl Aryl Selenides and Sulfides from Baylis‐Hillman Acetates	101
Formal Insertion of a Metal Carbene Complex into a σ‐Carbon‐Carbon Bond. Gold‐Catalyzed Synthesis of 3H‐Indoles	100
Copper‐Catalyzed Oxidative 1,2‐Alkylarylation of Styrenes with Unactivated C(sp³)‐H Alkanes and Electron‐Rich Aromatics via C(sp³)‐H/C(sp²)‐H Func	92
Synthesis of Furfural Sulfides and 4‐Alkylthiopyridines via Heterocyclization of α‐Acyl Ketene Dithioacetals	69
Site‐Selective Direct Intermolecular C(sp³)−H Alkylation of Saccharides and Switching of Reaction Sites by Changing Photocatalysts	55
Selective Formation of 2,3,5‐Trisubstituted Furans from 1,3‐Dicarbonyls and Hydroxyketones	54
	53
Visible‐light‐induced and EDA Complex‐initiated Hydroxyselenization of α‐CF₃ Alkenes: Access to α‐trifluoromethyl‐β‐selanyl tertiary Alcohols	44
Palladium‐Catalyzed Reaction of 2,3‐Allenols with Amines: Synthesis of [3]Dendralenes and 1,3‐Dienes Containing Allylic Amino and Hydroxy Groups	44
Synthesis of 2‐Amino‐3‐arylindoles and their Fused Analogues via Intramolecular C‐Arylation	43
Divergent Reactivity of E/Z‐Azobenzene‐Based Phosphine‐Gold Catalysts: Toward an ON‐ON Catalytic Photoswitch Process	42
	42
Tandem Enantioselective Cycloaromatization/Intramolecular Friedel–Crafts Desymmetrization of Cyclohexadienones	41
Front Cover Picture: Chemo‐ and Regioselective Construction of Functionalized Isocoumarin, Flavone, and Isoquinolinedione via a One‐pot Reaction of o‐Quinol Acetate and Soft Nucleophiles	41
A Lewis Base Hydrogen Bond Donor (LB/HBD) Organocatalytic Approach to Dithiabridged Triarylamine Hetero[4]helicenes	40
Front Cover Picture: Catalytic Asymmetric Arylations of Ketimines (Adv. Synth. Catal. 12/2024)	40
Imidazolium‐Dithiocarboxylate Zwitterions Catalysed Ring‐Opening Additions of Cyclopropenones	40
Front Cover Picture: Filling the Gaps in the Challenging Asymmetric Hydrogenation of Exocyclic Benzofused Alkenes with Ir−P,N Catalysts (Adv. Synth. Catal. 2/2023)	40
Cover Picture: Bench‐Stable Electrophilic Reagents for the Direct Di‐ and Trifluoroethylthiolation of Indoles (Adv. Synth. Catal. 20/2023)	39
Unusual Ring Opening of Bicyclic Terpenes During Pd‐Catalyzed Coupling with Aromatic Halides	39
Gold(I)‐Catalyzed Cascade Cyclization of Nitrogen or Oxygen Containing Nucleophile Tethered‐Vinylidenecyclopropanes to Pyrrole, Furan, Pyrrolidine and Piperidine Skeletons	39
Asymmetric Synthesis of Tricycle‐Fused Dispirooxindoles via Organocatalyzed Three‐Component Cascade Reactions of 2‐Pyrones and Trifluoroethylisatin Ketimines	39
Copper‐Catalyzed Acylhalogenation of 3‐Methylanthranils with Acid Halides: Synthesis of N‐(2‐(2‐Haloyl)phenyl)amides	38
Gold‐Catalyzed Annulation Between 1‐[2‐(Dimethoxymethyl)phenyl]prop‐2‐yn‐1‐yl Acetates and α‐Diazo Esters or Anilines to Form Substituted Naphthoates and Indeno[1,2‐b]quinoline, Respectively	38
Electrochemical Oxidative C−C Bond Functionalization of Methylenecyclopropanes with Diselenides/Ditellurides Leading to 2‐Substituted‐3,4‐Dihydronaphthalenes	37

Regio‐ and Stereoselective, Intramolecular [2+2] Cycloaddition of Allenes, Promoted by Visible Light Photocatalysis	36
Magnesium and Calcium Bisguanidinates: Catalytic Activity in the Hydroboration of Unsaturated Molecules	35
A Gold(I)‐Catalyzed Cyclization/Semipinacol Rearrangement Cascade of 1,6‐Enynes to Access Spiro[4.5]decanes and 7‐Azaspiro[4.5]decanes	35
Witnessing the Birth of Directed Evolution of Stereoselective Enzymes as Catalysts in Organic Chemistry	35
Solvent‐ and Temperature‐Switched Chemoselectivity: Controlled Synthesis of Diverse Pyrazolo[5,1‐a]isoquinolines	35
One Pot Synthesis of 1,2‐Disubstituted Ethanones by Base‐Mediated Reductive Homocoupling of Aldehydes	35
Palladium‐Catalyzed Aryloxycarbonylayion of Aryl Bromides with Phenols Using Inositol Hexaformate as an Efficient CO Source	35
Tandem Asymmetric Cycloaromatization/ Intramolecular Pictet‐Spengler‐Type Reaction. An Entry to Polycyclic Pyrroles	35
Ruthenium (II)‐Catalysed Regioselective C6 Alkylation of Indoles with Maleimides	34
Enzymatic Dimerization of Fungal Natural Products Through Intermolecular Disulfide Bridges	34
Synthesis of 2‐Aminopyridines via Cobalt‐Catalyzed Cycloaddition of Diynes with N‐Substituted and N‐Unsubstituted Cyanamides	34
Access to 2‐Sulfonyl‐4‐arylphenols and 2,6‐Bis‐sulfonyl 5‐Aryl‐4‐arylidene‐2‐cyclohexenones via Metal Triflates‐Catalyzed Domino Cyclocondensation of 1,3‐Bis‐sulfonylacetones and 3‐Arylacroleins	34
Synthesis of 3,4‐Dihydroquinazolinones via Base‐Promoted Formal [4 + 2] Cycloadditions	33
Constructing 5‐Methyl‐2,4‐diaryl‐1H‐imidazoles Using Calcium Carbide as Alkyne Source via A3‐Coupling Cyclization	33
Electrochemical Imidoyl Radical‐Involved Functionalization of Isocyanides to Construct Benzotriazole‐Sulfonamide and Guanidine Derivatives	33
Machine Learning Guided d‐Orbital Electron Modulated Graphene‐Based Catalysts for Enhanced Electrochemical Ammonia Synthesis	33
Harnessing Alkene Radical Anions via Electroreduction Strategy: An Emerging Paradigm for Alkene Functionalization	33
	33
Photoinduced Ligated Boryl Radical‐Mediated Functionalization of Organic Halides	32
SuFEx Reactions When Shaken Not Stirred	31
Regio‐ and Stereospecific Desulfinylative Chlorination of Spiroaziridine Oxindoles at Spiro‐Center for Formal [3+2]‐Cycloaddition with CS₂: Sequential One‐Pot Synthesis of (−)‐Spirobrassini	31
Aryne‐Based Synthesis of Cyclobutadiene‐Containing Oligoacenes and Related Extended Biphenylene Derivatives	31
Martin Silicates as Partners in Photoredox/Ni Dual Catalysis for the Installation of CH₃, CH₂D, CD₂H, CD₃ and ¹³CH₃ Groups onto (Heter	31
Catalyst‐Free, One‐Pot, Three‐Component Synthesis of 3‐Arylsulfonylated Thioflavones	31
N‐Containing Carbon Materials in Metal‐Free and Non‐Noble Metal Liquid Phase Heterogenous Catalysis	30
	30
Cu(III) Trifluoromethyl Complexes with 1,3‐Diketonate Ligands and Their Versatile Reactivity in C−H Trifluoromethylation	30
Silver‐Enabled Inverse Electron Demand Thermal Decarbonylative Skeletal Expansion: A New Gateway to the Synthesis of Multifunctionalized Quinoline	29
Three‐Dimensional Spirobifluorene‐Based COF for Metal‐Free Photocatalytic CH Oxidation Reaction	29
Hypervalent Halogen Compounds in Electrochemical Reactions: Advantages and Prospects	28
Cobalt‐Catalyzed Selective Transformation of Levulinic Acid and Amines into Pyrrolidines and Pyrrolidinones using Hydrogen	28
Enantioselective Synthesis of Five to Eight‐Membered P‐Stereogenic Benzo‐Fused Heterocycles via Copper‐Catalyzed Dynamic Kinetic Resolution	28
Bifunctional Photocatalysts for Asymmetric Epoxidation of Chalcones	28
Cooperative Photocatalysis of 9,10‐Phenanthrenequinone and Sn(OTf) ₂ for Direct Mannich Reaction of Ethers via Hydrogen Atom Transfer Pathway	28
A Combined Halogen‐ and Chalcogen‐Bonding Organocatalyst	27
Nitrosonium Ion Catalyzed Oxidative Bromination of Arenes	27
Bis(oxazoline)–Nickel(II)‐Catalyzed Asymmetric Photochemical Hydroxylation of β‐Keto Esters With Nitrones	26
tert‐Butyl Nitrite Promoted Visible‐Light‐Induced Steric‐Hindrance‐Regulated Concurrent Cross‐Coupling and Regioselective Nitration of 3‐Alkylidene‐2‐oxindoles	26
Recent Advances in Transition Metal Catalysed Dearomatization Toward the Synthesis of Complex Cyclic Compounds	26
Continuous Flow Technology Enabling Photochemistry	26
Monofluorinated C1 Synthon Strategy for the Construction of Fluoromethylene‐Linked Bicyclo[1.1.1]Pentane Derivatives	26
Harnessing the Excited‐State Reactivity of o ‐Nitrobenzyl Alcohols for the Rapid Synthesis of N ‐Substitut	26
Harnessing Carbenoid Reactivity From Imidazoles and Oxiranes	26
Direct Asymmetric Addition of Heteroatom Nucleophiles to Imines	26
Stereoselective Synthesis of Contiguous Cyclopropylaziridines: Enabling the Construction of Versatile Chiral Molecules Including γ‐Lactams via Ring‐Opening Reactions	26
The Novel Strategies for the Construction of Homoallylic Alcohols via Photoredox Catalysis	26
Hypervalent Iodine‐Mediated Regioselective Dearomatization of Non‐Activated Arenes	26
First Bromide‐Catalyzed Selenylation of 2‐Alkyn‐1‐One O‐Methyloximes Enabled the Synthesis of 4‐Selenylated Isoxazoles	26
Enantioselective Syntheses of Multiply Functionalized Six‐Membered Carbocycles from Nitroalkenes and γ,δ‐Unsaturated ß‐Ketoesters using Chiral Catalysts Derived from Cobalt(III) and 1,2‐Diphenylethyle	26
Ring‐Opening Amino Esterification of Cyclic Ketones to Access Distal Amino Acid Derivatives	26

2‐Aminoindoles and 2‐Iminoindolines as Viable Precursors of Indole‐Fused Nitrogenated Polyheterocycles	25
A Redox‐Neutral Organophotocatalytic Cascade: Difluoromethylation and Radical Truce–Smiles ‐Driven C( sp <	25
Silver‐Mediated In‐Situ Generation of Alkynyl Selenium Intramolecular AAC Click Reactions	25
Asymmetric Synthesis of Highly Substituted Spiro[2H‐pyrrole‐2,3‐Succinimide] Derivatives by Copper‐Catalyzed Post‐Ugi Reactions	25
Synthesis of Dihydropyrazoles via Palladium‐Catalyzed Cascade Heterocyclization/Carbonylation/Arylation of β,γ‐Unsaturated N‐Tosyl Hydrazones	25
Copper‐Catalyzed Cross Coupling Reaction of Alkyl Bromides with (DMPU)₂Zn(R_f)₂ Reagent: A Method for the Synthesis of Perfluoroalkylated Compounds	25
K₂S₂O₈‐Mediated Access to Alkylsulfonated Spiro[4,5] Trienones from N‐Arylpropiolamides with the Insertion of Sulfur Dioxide	25
Divergent Synthesis of 3‐Trifluoroethyl Benzofurans Through Rh‐Catalyzed CC Bond Activation Coupled with Transfer Hydrogenation	25
Visible‐Light‐Driven Organocatalyzed Chemoselective Oxidation of Benzylamines	25
Pd‐Catalyzed Ring‐Opening Defluorinative Arylation of gem‐Difluorocyclopropanes with Arylsilanes	25
Multifaceted Domino Knoevenagel‐Cyclization Reactions; Four Movements for 2H‐Chromenes and Chromans	25
Photo‐Catalyzed Stereospecific Synthesis of Trisubstituted Alkenes Incorporating 3,3‐Difluoro‐γ‐Lactams from Morita‐Baylis‐Hillman Acetates and N‐Allylbromodifluoroacetamides	24
N−H Trifluoroethylation of Indoles and other Aromatic N‐Heterocycles with CF₃CHCl₂ by Copper‐Mediated Cross‐Coupling Reaction	24
	24
K₃PO₄–Mediated Synthesis of Chromeno–[3,4‐c]isoxazole from 3–Nitro–2H–chromene and α–Chloro Aldehyde via Michael Addition/C−Cl Bond Cleavage/Deformylation as	24
One‐Pot Synthesis of Quinazolines via Elemental Sulfur‐Mediated Oxidative Condensation of Nitriles and 2‐(Aminomethyl)anilines	24
Visible‐Light Induced Ag‐Palladacycle‐Complex‐Mediated Regioselective C−H Arylation	24
Cobalt(III)‐Catalyzed Aerobic Diamination of α‐Alkyl Styrenes with Anilines	24
Phosphine‐Catalyzed (4+2) Annulation of Alkenes with Acidic Hydrogen‐Tethered Allylic Carbonates	24
Gold‐Catalyzed Redox‐Neutral Reaction of Nitriles with Quinoline N‐Oxides	23
Construction of α‐Pyrones and Enamine Derivatives via Divergent Transformations of β‐Aminoacrylates	23
Indazolones Directed Rh(III)‐Catalyzed C−H Amidation of Arenes	23
Functionalized Alkylidenecyclobutanes from a Cyclopent‐2‐enone Substrate via a Tandem Photochemical Transformation and an Allylic Substitution Protocol	23
Nickel/Copper Co‐catalyzed Enantioselective Reductive Coupling of Oxabenzonorbornadienes with Vinyl Bromides	23
Special Issue Dedicated to Miquel A. Pericàs	23
Front Cover Picture: Redox‐Neutral Vicarious‐Type Nucleophilic Amination of Heterocyclic N‐Oxides with Organic Azides (Adv. Synth. Catal. 19/2024)	23
Total Synthesis of the Myrioneuron Alkaloid (−)‐Schoberine B and Its Enantiomer (+)‐Schoberine B	23
Renewable Platform Chemicals: The Bulk Chemicals of the Future	23
	23
Copper‐Catalyzed Domino Synthesis of Spiropyrazoline Oxindoles via Condensation of Indolin‐2‐One and Phenylhydrazine Derivatives	23
Front Cover Picture: Palladium‐Catalyzed Chemoselective Amination of Chloro(hetero)aryl Triflates Enabled by Alkyl‐Pyrazole‐Based Phosphine Ligands (Adv. Synth. Catal. 7/2024)	22
Bidentate NHC‐Containing Ligands for Copper Catalysed Synthesis of Functionalised Diaryl Ethers	22
Stereoselective Synthesis of Aliphatic α‐Amino Acids by Chemo‐Enzymatic Hydroamination‐Hydrodesulfurisation	22
Visible‐Light‐Induced Controlled C–H Cyanation or Thiocyanation of Indolizines	22
Iron‐Catalyzed Oxyphosphorylation of Styrenes to Access β‐Ketophosphonates and α, β‐Unsaturated Ketones	22
Diarylprolinol with Trifluoromethyl Substituents and Diphenylprolinol‐Derived Perfluoroalkanesulfonamide as Organocatalysts in the Cross‐Aldol Reaction of Aldehydes	22
Palladium‐Catalyzed Denitrative Decarboxylation of Nitroarenes with Alkynyl Carboxylic Acids	22
N,N’‐Difluoro‐2,2’‐bipyridinium Bis(tetrafluoroborate): a New Terminal Oxidant for Iodoarene‐catalyzed Fluorination Reactions	22
An Organocatalytic Route to endo‐Vinylene Carbonates from Carbon Dioxide‐Based exo‐Vinylene Carbonates	22
Gold‐Catalyzed Annulation of Ynamides with Aminocarbonyls as a Route to 2‐Aminoquinolines Diversely Substituted at the 4^th‐Position	22
An Umpolung Route to Amides from α‐Aminonitriles under Metal‐Free Conditions	22
The Chemistry of α‐Enolizable Alkynones: A Comprehensive Review	22
Palladium Catalysis: Dependence of the Efficiency of C−C Bond Formation on Carboxylate Ligand and Alkali Metal Carboxylate or Carboxylic Acid Additive. Part C: The Domino Diarylation and Annelation Re	22
DABCO‐Promoted Selective Photochemical C−N Coupling: Access to Unsymmetrical Azahelicenes	22
A Mild Metal‐Free Approach for the Direct Synthesis of Carbamoyl Azides from Carboxylic Acid Redox Active Esters	22
Pincer‐Ruthenium Catalyzed Oxygen Mediated Dehydrative Etherification of Alcohols and Ortho‐Alkylation of Phenols	21
	21
Front Cover Picture: (Adv. Synth. Catal. 10/2025)	21
	21
Modular Chiral Bithiophene‐2NO Ligands: Synthesis and Application in Asymmetric Palladium(II)‐Catalysed Friedel‐Crafts Alkylation	21
Hydroaminoalkyl Functionalization of Pyrimidin‐2(1H)‐ones by Visible Light Organophotocatalysis: A Radical Approach to Biginelli‐Type Dihydropyrimidines	21
Unexpected Stereoselective Access to 2‐Aminooxazolines from Propargyl Ureas by Silver Salts under Mild Conditions	21
Copper‐Catalyzed α‐Indolmethylation of 2‐Pyridylacetates with 3‐Indoleacetic Acids via Alkylideneindolenine Intermediates	21
Preparation of Mesoporous Cu₂O Nanospheres for Green Synthesis in the Enantioselective Boron Conjugate Addition of α,β‐Unsaturated Chiral Compounds in Aqueous Phase	21
Au(I) and HOTf‐Catalyzed Cascade [5+1]‐Annulations between Allenylacetals and Diazo Esters To Form 1,3‐ and 2,3‐Disubstituted Naphthoates, Respectively	21
Phospholanes via Twofold C‐H‐Addition to Phospholes	21
Well‐Defined [Cp*Co(N,O)I]‐Catalysts for Site‐Selective Intramolecular C−H Amidation	21
Sustainable Photoelectrochemical Geminal α‐Fluorosulfenylation of Diazo Compounds through Carbene Radical Anion Intermediate	21
Peroxidation and Skeletal Rearrangement for the Synthesis of Dioxole‐2‐Carboxamide Derivatives under Continuous‐Flow Conditions	21
	21
1,3‐Iodoesterification of 2‐Substituted Indoles via C_sp2−H/C_sp3−H Retained Dual Functionalization Using Hypervalent Iodine(III)	21
A Mild Reductant N‐Heterocyclic‐Carbene‐Ligated Borane for N ‐Formylation of Amines with CO ₂ under Am	21
Arylation of Secondary Phosphines with Diaryliodonium Salts under Metal‐Free and Non‐Photochemical Conditions	21
Mechanochemically Induced Cross Dehydrogenative Coupling Reactions under Ball Milling	21
Asymmetric CH Functionalization Enabled by a Traceless Oxidizing Chiral Auxiliary	20
Molybdenum‐Catalyzed Direct Synthesis of Pyrroles from Nitroarenes with Glycols as Reductants	20
Synthesis of Deoxysugars from Aliphatic α‐Ketoacids and Aldoses Catalyzed by Thermostable Transketolase Variants from Geobacillus stearothermophilus	20
Corrigendum: Cyclic Sulfoximine and Sulfonimidamide Derivatives by Copper‐Catalyzed Cross‐Coupling Reactions with Elemental Sulfur	20
Metal‐Free Chemoselective Amide Bond Cleavage for the Synthesis of N ‐Acyl Sulfoximines in Batch and Flow	20
Diradical Polar Reactivity Induced by Electricity‐Mediated Ground State Triplet Nitrenium Species	20
Multicomponent Annulative SO₂ Insertion of Heteroatom‐Linked 1,7‐Diynes for Accessing Tricyclic Sulfones	20
Synthesis of 1‐Aryl Isoquinolinones or o‐Diaryl Pyrimidines via Bismuth Triflate‐Mediated Intermolecular Annulation of Arylacetic Acids with Nitroarylaldehydes or Trimethoxybenzene in the Prese	20
One‐Pot Tandem Cyclization of β‐Oxoamides, Primary Amines, and 3‐bromo‐1,1,1‐trifluoroacetone: Synthesis of 2/4‐trifluoromethyl‐substituted dihydropyrrol‐2/4‐ols	20
Halogen Atom Transfer Enabled Radical Fluoroalkyl‐Thiolation of Unactivated Alkenes	20
In Situ Generation of Copper Nanoparticle‐Graphitic Carbon Nitride Composite for Stereoselective Transfer Semihydrogenation of Alkynes: Evaluation of Catalytic Activity Using Fluorescence‐Based	20
Stereoconvergent Access to Z‐Allylborons from E/Z‐Mixed 1,3‐Dienes via Cu‐Guanidine Catalysis	20
Iron‐Catalyzed Regioselective C(sp ² )H Alkylation and Heteroannulation of Hydroxyarenes With 2‐Aryl Aziridines	20
Amide Synthesis via Transaminative Amidation of Aromatic Aldehydes/Ketones: An Entry to ¹⁵ N Isotopologs	20
Mechanistic Insight into Palladium‐Catalyzed Asymmetric Alkylation of Indoles with Diazoesters Employing Bipyridine‐N,N’‐dioxides as Chiral Controllers	20
Dibenzoylperoxide as a Versatile Oxidant for Oxidative Azidations of Phenols Using Quaternary Ammonium Iodides or Bromides.	20

Synthesis of Oxadihydrophenanthroquinolizidinones by Photoinduced Rearrangement of 3‐Biphenyl‐1‐hydroxypropyl‐pyridin‐2(1H)‐ones	20
Asymmetric Hydrogenation of Tetrahydro‐γ‐Carboline Derivatives with Phosphine‐Free Ruthenium Diamine Catalysts	20
Recent Progress of Electron‐Withdrawing‐Group‐Tethered Arenes Involved Asymmetric Nucleophilic Aromatic Functionalizations	20
Enantioselective Synthesis of Triarylmethanes Containing Three Different Aryl/Heteroaryl Moieties by Chiral Phosphoric Acids Catalyzed Friedel−Crafts Reactions	20
Iron Catalyzed Radical Alkylation of Cyclic Ketimines with Olefins via Metal Hydride Atom Transfer	20
Directed Palladium‐Catalyzed pseudo‐Anomeric C−H Functionalization of Glycal‐Type Substrates: Access to Unsymmetrical gem‐Diarylmethyl C‐Glycosides	20
Direct Site‐Selective Deoxygenation of Benzylalcohol Derivatives	19
Visible Light Induced EDA‐mediated Deaminative C‐2 Alkylation of Heterocyclic‐ N ‐Oxides using Katritzky salts	19
Selective Access to Sultams and Spirocyclic Sultams by the Divergent Annulations of (N‐Aryl)‐Alkynyl Sulphonamides	19
DMAP‐promoted [4+2]/[3+3] Annulation Cascade Reaction of Morita–Baylis–Hillman Carbonates with Conjugated Imines to Access Functionalized Benzo[c][2,7]naphthyridine Skeletons	19
Water‐Facilitated Nitromethane‐Mediated Cyclization of 2‐(Phenylvinyl)benzhydrols: Access to 1,3‐Diphenyl‐1H‐indenes with Antitumor Activity	19
Thianthrenium Salts to Arynes: Base Promoted C−N Bond Construction	19
Photoredox and Copper‐Catalyzed Sulfonylphosphorothiolation of Alkenes toward β‐Sulfonyl Phosphorothioates	19
Multicomponent Heteroarylphosphorothiolation of Alkenes for Accessing β‐Phosphorothiolated Quinoxalinones	19
Brønsted Acid‐Catalyzed Enantioselective and Para‐Selective Addition of Phenols to 1‐Alkynylnaphth‐2‐Ols	19
Harnessing Photoredox Catalysis to Access β ‐Ketoamino Esters from 3‐(2‐Isocyanoethyl)indoles	19
Transition‐Metal‐Free Regioselective Direct C2, C4 Difunctionalization and C2, C4, C6 Trifunctionalization of Pyridines	19
Controllable Synthesis of Oxa‐/Thia‐Spirohydroquinolines by [3+(2+1)] Annulation of Aromatic Amines with Bimolecular O/S‐Heterocyclic Ketones	19
N ‐Fluoroalkylthiolation of Amines and Sulfonamides with Fluoroalkyl Sulfoxide as Fluoroalkylthiolating Reagent	19
Stereoselective Organocatalyzed Glycosylation of Glycosyl Trichloroacetimidate Donors: Thiouracil as Brønsted Acid Catalyst	19
Recent Advance in Transition Metal‐Catalyzed Carboxylic Acid Guided B−H Functionalization of Carboranes	19
Photocatalyzed Aerobic Dearomatization of Naphthylamines under Visible‐Light Irradiation	19
Ru(II) Catalyzed Oxidative Dehydrogenative Annulation and Spirocyclization of Isoquinolones with N‐Substituted Maleimides	19
Controllable Access to Furans and Dihydrofurans through Cyclization/Coupling of Internal Acetylenic β‐Ketoesters with Aryl Bromides	19
Front Cover Picture: Mechanochemical Ni‐Catalysed Arylation of ortho‐Hydroxyarylenaminones: Synthesis of Isoflavones (Adv. Synth. Catal. 20/2022)	19
A Sequence‐Controlled Di‐Functionalization of an SO₂‐Surrogate with Amines for the Synthesis of Sulfonamides	19
Ruppert‐Prakash Reagent (TMSCF₃)‐Catalyzed Chemoselective Esterification of Weinreb Amides	18
Copper‐Catalyzed Tandem Cyclization of 2‐(Alkynylaryl)Acetonitriles and Amines: Access to 3‐Hydroxyisoindolinones	18
	18
Manganese‐Mediated Electrooxidative Ring‐Opening Azidation of Cyclobutanol Derivatives with TMSN₃	18
Electrochemical α‐Functionalization of N‐Aryl‐Activated Tertiary Amines	18
Accessing 2‐(Chalcogen)benzothiazoles via Electrochemical Intermolecular Cyclization of Isocyanides with Thiols or Diselenides	18
Front Cover: Gold(I)‐Catalyzed Enantioselective Cycloisomerization of 1,6‐Oxygenated Enynes: An Entry to Hedonic Derivatives (Adv. Synth. Catal. 19/2025)	18
C−N Coupling between Aryl Azides and Cyclopropanols by Photoredox/Copper Dual Catalysis	18
	18
Visible‐Light‐Induced Oxidative Carboazidation of Arylacrylamides	18
A Solely Fe‐Catalyzed Sonogashira‐Type Coupling of non‐Activated Secondary Alkyl Iodides with Terminal Alkynes	18
TEMPO Mediated Cyclopropanols Ring Opening C−N Cross‐Coupling with Nitrogen Nucleophiles	18
Rhodium(III)‐Catalyzed Redox‐Neutral Synthesis of Indenones from 2‐Aryl‐3‐nitrosoindoles with Alkynes	18
Modular Synthesis of 2,3,4,6‐Tetrasubstituted Thieno[2,3‐c]furans Based on Formal [3+2] Cycloaddition Utilizing [1,2]‐Phospha‐Brook Rearrangement / Brønsted Base‐Mediated Cyclization Strategy	18
Silver‐Catalyzed [3+2] Cycloaddition for the Diastereoselective Synthesis of anti‐3‐Substituted Hydroindolin‐2‐Imines	18
Iron‐Catalyzed C−C and C−N Bond‐Forming Tandem Amidation Offering Access to 3‐Amino‐3‐Aminomethyl‐2‐Oxindole Frameworks	18
Modular Photochemical Flow Synthesis of Structurally Diverse Benzyne and Triazine Precursors	18
Electrochemical Decarboxylative Coupling of N‐Substituted Glycines under Air: Access to C3‐Aminomethylated Imidazo[1,2‐a]pyridines	18
An Acid Promoted, Domino Approach for the Selective Synthesis of Spirocyclic Systems^#	18
Palladium‐Catalyzed Chemoselective Amination of Chloro(hetero)aryl Triflates Enabled by Alkyl‐Pyrazole‐Based Phosphine Ligands	17
Asymmetric Boracarboxylation of Styrenes Using Carbon Dioxide	17
Solvent‐Switchable Regiodivergent Chlorination of Quinone Monoacetals: A Practical Route to 2‐ and 3‐Chlorophenols	17
Recent Advances in the 1,2‐Diarylation of Alkenes	17
Noncovalent‐Interaction‐Dictated Product Selectivity in Intermolecular and Intramolecular Controllable Oxidation of Aromatic Amines Using 2,2′‐Diperoxyphenic Acid	17
Regioselective Construction of Indolylated Cyclic Tetrasubstituted Carbon Centers through Brønsted Acid‐Catalyzed Dearomative Skeletal Rearrangement of Azofurans	17
Visible‐Light Photoredox‐Catalyzed Tandem One‐Pot Construction of C4‐Difluoroalkylated Phthalazin‐1(2H)‐Ones	17
Synthesis of Functionalized 3‐(1H‐Isochromen)‐chromones via Ag₂O‐Catalyzed Cascade Cyclization Reaction of o‐Hydroxyarylenaminones with o‐Alkynylbenzaldehydes	17
Maleimide‐Controlled Formation of Indanonylpyrrolinediones and Spiroindanonylpyrrolinediones via Rh(III)‐Catalyzed C−H Activation of Sulfoxonium Ylides	17
[(5+1)−1] Cyclization of Nitroepoxides to Pyridinium 1,4‐Zwitterionic Thiolates for the Synthesis of Indolizine Derivatives	17
Visible‐Light‐Induced Stereoselective C(sp³)−C(sp³)−H Glycosylation for the Synthesis of C‐Glycoamino Acid Derivatives	17
Deoxygenative Coupling Between Morita–Baylis–Hillman Acetates and Unprotected Cycloketone Oximes Enabled by Photoredox/Ti Dual Catalysis	17
Strategies and Methods for the Synthesis of 2‐Pyrazolines: Recent Developments (2012–2022)	17
Synthesis of 2‐Aryl‐2H‐1,2,3‐triazoles via P(OMe)₃‐Promoted Intramolecular Transannulation of 4‐Diazenylisoxazol‐5(4H)‐ones	17
Synthesis of 3‐Arylazoindoles through Iron(III)‐Catalyzed C−H Azolation of Indoles and Arylhydrazines	17
Electrosynthesis of 2,5‐Disubstituted Furans through a CC Double Bond Cleavage Radical Cascade	17
Heterogeneous Copper‐Catalyzed 1,4‐Conjugate Additions of Grignard Reagents to Cyclic and Linear Enones	17
Electrochemically‐Driven Organocatalytic Enantioselective Oxidative Coupling of Tetrahydroisoquinolines and Acrylaldehyde	17
Cu(I) Catalyzed Germyl S ‐Phosphorothiolation of Electron‐Deficient Alkene	17
Visible‐Light‐Enabled Photosensitizer‐ and Additive‐Free Decarboxylative Coupling Cyclization of Enaminone with N‐Arylglycine for 3‐Aminoalkyl Chromones	17
Facile Access to 2‐Substituted‐1,2,3,4‐Tetrahydroquinoxalines via Borane‐Catalyzed One‐Pot Tandem Cyclization/Hydrosilylation	17
Photocatalytic Silacyclization of 1,7‐Enynes via Selective Functionalization of Si‐H/Silyl C(sp ³ )‐H Bonds: Access to Densely Functionalized Silacyc	17
Synthesis of Monofluorocyclohexene via Photocatalytic Defluorinative [4+2] Annulation of gem‐Difluoroalkenes with Unactivated Alkenes	17
γ‐Terpinene: Biorenewable Reductant for the Molybdenum‐Catalyzed Reduction of Sulfoxides, N ‐Oxides and Nitroarenes	17
Synthesis of 4‐Phosphinylpyrrolidin‐3‐ones via [3+2] Cycloaddition of Nitrones with Phosphinylallenes	17
Photoinduced Transition‐Metal‐Free Chemodivergent Phosphorylation‐Peroxidation and Oxyphosphorylation of Alkenes	17
Corrigendum: Mechanistic Insights on the Enantioselective (4+3) cycloaddition between Oxyallylcations and Furans Catalyzed by BINOL‐based Phosphoramides	17
Molecular Oxygen‐Induced Transamidation of Unactivated Amides in Diethyl Carbonate in the Presence of a Palladium Catalyst	16
Copper‐Catalyzed Olefinic C(sp²)−H Activation/Carbene Insertion/Ester Hydrolysis/Cyclization with Aryl Diazo Esters for the Synthesis of Multisubstituted Furanones	16
Rh(II)‐Catalyzed Homocoupling/[4+1] Cycloaddition Cascade of Diazobarbiturates with Diazopyrazolones to Prepare Spirobarbiturates	16
Synthesis of 3‐(2‐Hydroxyaryl)indazole Derivatives through Radical O‐Arylation and [3,3]‐Rearrangement from N‐Hydroxyindazoles and Diaryliodonium Salts	16
Palladium‐Catalysed Amide‐Directed Ligand Free C8‐Olefination of 1‐Naphthamides for the synthesis of 2,3‐dihydro‐1H‐benzo[de]isoquinolin‐1‐ones	16
Nucleophile Promoted Functionalization of Cross‐Conjugated Enynone Gives Sulfonylated Furan	16
Visible Light Induced Difunctional Hetero‐Annulation of Unsaturated C−C Bonds	16
Carboxylic acids as enabling directing groups in C−H activation and functionalization: A decade review	16
Synthesis of Functionalized Benzo[f]chromanes and Hydroxyalkyl Naphthols: Catalytic Coupling of Naphthols and Allylic Alcohols	16
Liquid‐Liquid‐Gas Triphasic Hydrogenation of Bicarbonate to Formate in a Continuous Flow Tubular Reactor	16
Electrochemical Oxidative Functionalization of Pyrazolin‐5‐Ones: Access to 4‐Quinoxalinone‐Substistuted Pyrazoles	16
Palladium‐Catalyzed Two‐fold Annulation Reaction of 2,6‐Dihalogenobiphenyls with o‐Chloroaromatic Carboxylic Acids to Access (Aza)dibenzo[fg,op]tetracenes	16
Accessing SuFExable Cyclobutane‐Fused Indolines via Photocatalytic Intermolecular [2+2] Cycloaddition of Indoles	16
Zinc Hydride Complexes Stabilized by Anionic N ‐Heterocyclic Carbenes for Hydrosilylation of Aldehydes and Ketones	16
Palladium‐Catalyzed [4+2] Cycloaddition of Hydroxy‐Tethered Allylic Carbonates with Alkenes: Synthesis of Functionalized Tetrahydropyrans	16
Deconstructive Alkynylation of Spiro‐Dihydroquinazolinones via Aromatization‐Driven Ring Opening Under Visible Light Irradiation	16
A Direct Silver‐Catalyzed Three‐Component Approach to Trifluoromethylated Cyanopyrazoles and Cyanopyrazolines	16
Quaternary Ammonium Salts: Catalysts for Hydrosilylation of Alkynes with Hydrosilanes	16
Total Synthesis of (−)‐Daphenylline by Gold‐Catalyzed Intramolecular Dearomatization Reaction of Methoxynaphthalene	16
Ring Closure of Nitroalkylmalonates for the Synthesis of Isoxazolines under the Acylation Conditions	16
Direct Assembly of Polysubstituted Furans with Dimethyl Sulfoxide as a Multipurpose Precursor via β‐C(sp³)−H Functionalization of Saturated Ketones	16
AgNO₃‐Catalyzed Regio‐selective Bis‐heteroannulation of o‐Hydroxyphenyl Enaminones and Yne‐enones: A Facile synthesis of Functionalized 3‐(Furan‐3‐ylmethyl) Chromones	16
Advances of Chiral Metal Complexes as Standalone Photocatalyst for Asymmetric Organic Transformations	16