Future Medicinal Chemistry

Article	Citations
Sulfonamide-salicylaldehyde Imines Active Against methicillin- and trimethoprim/sulfonamide-resistant Staphylococci	58
Super-Conserved Receptors Expressed in the Brain: Biology and Medicinal Chemistry Efforts	57
Novel Set of Highly Substituted Bis-Pyridines: Synthesis, Molecular Docking and Drug-Resistant Antibacterial Profile	57
In vivo evaluation of novel synthetic pyrazolones as CDK9 inhibitors with enhanced pharmacokinetic properties	52
Design of SARS-CoV-2 Mpro, PLpro Dual-Target Inhibitors Based on Deep Reinforcement Learning and Virtual Screening	51
Combining EGFR Inhibitors With SHP2 Or LSD1 Inhibitors to Overcome Multidrug Resistance in Cancer	44
Biological and computational evaluation of novel benzofuranyl derivatives as acetylcholinesterase and butyrylcholinesterase inhibitors	44
Identification of Sulfonamide-Based Butyrylcholinesterase Inhibitors Using Machine Learning	42
Citrate Transporter Inhibitors: Possible New Anticancer Agents	40
Therapeutic N -Heterocyclic Carbenes: An Interview With Alejandro Bugarin	39
The Connection Between PARP14 and SARS-CoV-2	38
Targeting Tuberculosis – An Interview With Robert Abramovitch	36
Development of 5-hydroxybenzothiophene derivatives as multi-kinase inhibitors with potential anti-cancer activity	34
Selection of SARS-CoV-2 Main Protease Inhibitor Using Structure-Based Virtual Screening	34
Investigations of New N 1 -Substituted Pyrazoles as Anti-Inflammatory and Analgesic Agents having COX Inhibitory Act	31
Design and synthesis of new nicotinamides as immunomodulatory VEGFR-2 inhibitors and apoptosis inducers	28
Combining Structure-Based and 3D QSAR Pharmacophore Models to Discover Diverse Ligands Against EGFR in Oral Cancer	28
5,7,3′,4′-Tetramethoxyflavone Ameliorates Cholesterol Dysregulation by Mediating SIRT1/FOXO3a/ABCA1 Signaling in Osteoarthritis Chondrocytes	28
Barbiturate–sulfonate hybrids as potent cholinesterase inhibitors: design, synthesis and molecular modeling studies	27
HDAC8 As an Emerging Target in Drug Discovery With Special Emphasis on Medicinal Chemistry	26
Rh(III) and Ru(II) Complexes With Phosphanyl–Alkylamines: Inhibition of DNA Synthesis Induced By Anticancer Rh Complex	23
Synergistic effect of new pyrimidine derivative with oxacilin against methicillin-resistant Staphylococcus aureus	23
Computational Insights Into Novel Inhibitor Indole-Heterocycle Specific Against Glycogen Phosphorylase Isoenzymes Interaction Mechanism	22
Advances in AR-Targeting Chimeras: A Case Study of proteolysis-targeting Chimeras From Bench to Bedside	22
Design, synthesis and inhibition evaluation of novel chalcone amide α-glucosidase inhibitors	22

Synthesis, in vitro and in silico anticancer evaluation of novel pyridin-2-yl estra-1,3,5(10)-triene derivatives	21
Propargylamine: an Important Moiety in Drug Discovery	20
Diaminomaleonitrile Derivatives as new Potential Antichagasic Compounds: A Study of Structure–Activity Relationships	20
Discovery of Novel Covalent Inhibitors of DJ-1 Through Hybrid Virtual Screening	20
Novel Xylenyl-Spaced Bis-Thiazoles/Thiazines: Synthesis, Biological Profile as Herpes Simplex Virus Type 1 Inhibitors and in Silico Simulations	19
Synthesis, antimicrobial evaluation, HPLC-based compound accumulation and docking studies of 2-methoxybenzoyl thioureas	18
Synthesis of Hydrazinyl–Thiazole Ester Derivatives, in Vitro Trypanocidal and Leishmanicidal Activities	18
Basic nitrogen (BaN): a ‘privileged element’ in medicinal chemistry	18
New pyrrolopyridine-based Thiazolotriazoles As Diabetics Inhibitors: Enzymatic Kinetics and In Silico Study	18
Management of Adenocarcinoma With Honokiol: Progress So Far and the Way Forward	17
Keto-Bridged Dual Triazole-Linked Benzenesulfonamides As Potent Carbonic Anhydrase and Cathepsin B Inhibitors	17
γ-Secretase As a Drug Target for Familial Alzheimer's Disease: The Road Less Traveled	17
Unlocking the power of imidazoquinolines: recent advances in anticancer and immunotherapeutic strategies	17
Medicinal Chemistry in Big Pharma has a Gender Diversity Problem	16
Potent α-glucosidase inhibitors with benzimidazole-propionitrile hybridization; synthesis, bioassay and docking study	16
Recent Advancements in the Discovery of Cereblon-Based Protease-Targeted Chimeras With Potential for Therapeutic Intervention	16
GANT61 Elevates Chemosensitivity to Cisplatin Through Regulating the Hedgehog, AMPK and cAMP Pathways in Ovarian Cancer	15
Computational Repurposing of Benzimidazole Anthelmintic Drugs As Potential Colchicine Binding Site Inhibitors	15
HIV-1 Capsid Inhibitors: A Sword to Destroy the Virus	15
Machine Learning and Deep Learning in Data-Driven Decision Making of Drug Discovery and Challenges in High-Quality Data Acquisition in the Pharmaceutical Industry	15
How does machine learning augment alchemical binding free energy calculations?	14
Copper(II) complexes of 2-hydroxy-1-naphthaldehyde Schiff bases: synthesis, in vitro activity and computational studies	14
Autophagy degradation: a promising dimension in drug discovery for neurodegenerative diseases	14
The versatility of phenothiazines as an anticancer drug scaffold	14
Targeting TGF-β: Triumphs and Challenges	14
Synthesis of Novel Furan-Based Chalcone Derivatives As Anti-Tuberculosis Agents: In Vitro , Cytotoxicity Assessment and In Silico	13
Novel bis-benzimidazole-triazole hybrids: anticancer study, in silico approaches, and mechanistic investigation	13
Palbociclib-derived multifunctional molecules for lysosomal targeting and diagnostic-therapeutic integration	13
Latest developments in photosensitizers: improving stability, specificity and responsiveness	13
Synthesis of indole-functionalized isoniazid conjugates with potent antimycobacterial and antioxidant efficacy	13
Synovial Mesenchymal Stem Cell-Derived Exosomal miR-320c Enhances Chondrogenesis By Targeting ADAM19	13
E3 Ligases: a Potential Multi-Drug Target for Different Types of Cancers and Neurological Disorders	13
Design, Synthesis and Antitumor Activity of Novel pyran-functionalized Uracil Derivatives: Docking Studies	13
Proteolysis Targeting Chimeras in Antiviral Research	13
Synthesis and Characterization of Potent RIPK3 Inhibitors Based on a Tricyclic Scaffold	12
Treating Neurodegenerative Diseases with Multitarget Drugs: An Interview With Maria João Matos	12
NeuroClick: Software for Mimicking Click Reaction to Generate Drug-Like Molecules Permeating the Blood–Brain Barrier	12
Piperazine-1,2,3-triazole Scaffolds: design, synthesis, Anticancer and Antimicrobial Evaluation	12
Novel Effective Small-Molecule Inhibitors of Protein Kinases Related to Tau Pathology in Alzheimer's Disease	12
New Theobromine Derivatives Inhibiting VEGFR-2: Design, Synthesis, Antiproliferative, Docking and Molecular Dynamics Simulations	11
Recent advances in the investigation of the quinazoline nucleus and derivatives with potential anticancer activities	11
The current landscape of indole hybrids with in vivo antitumor potential	11
New Indole Derivatives As Multitarget anti-Alzheimer's Agents: synthesis, Biological Evaluation and Molecular Dynamics	11
Design, Synthesis and Bio-Evaluation of Indolin-2-Ones As Potential Antidiabetic Agents	10
Refinement of MEK inhibitors	10
Design, Synthesis and Biological Evaluation of Novel Selective PI3Kδ Inhibitors Containing Pyridopyrimidine Scaffold	10
Levamisole Derivatives As Immune Modulators for the Treatment of Amyotrophic Lateral Sclerosis (ALS)	10
Explainable Machine Learning for Medicinal Chemistry: Exploring Multi-Target Compounds	10
19 Schiff Bases as Antimycobacterial Agents: Synthesis, Molecular Docking and a Plausible Mechanism of Action	10
Novel 2-Indolinone Derivatives as Promising Agents against Respiratory Syncytial and Yellow Fever Viruses	9

In vitro anti-breast cancer study of hybrid cinnamic acid derivatives bearing 2-thiohydantoin moiety	9
One-pot synthesis and pharmacological evaluation of new quinoline/pyrimido-diazepines as pulmonary antifibrotic agents	9
Novel Benzochromenes: Design, Synthesis, Cytotoxicity, Molecular Docking and Mechanistic Investigations	9
Novel Carbonic Anhydrase Inhibitors	9
Advances of Biphenyl Small-Molecule Inhibitors Targeting PD-1/PD-L1 Interaction in Cancer Immunotherapy	9
Selenium: The Emerging Element in the Medicinal Chemist’s Toolkit	9
Novel Diamides Inspired By Protein Kinase Inhibitors As Anti- Trypanosoma Cruzi Agents: In Vitro and In Vivo	8
Clinical Progress of KRAS-targeted Therapies: What next?	8
Targeted small molecule therapy and inhibitors for lymphoma	8
Mucin Glycosylation: A Potential Target for Prostate Cancer Management	8
Novel Pyrimidine-1,3,4-Oxadiazole Hybrids and Their Precursors As Potential Antimycobacterial Agents	8
Transition metal complexes: next-generation photosensitizers for combating Gram-positive bacteria	8
Development of indole hybrids for potential lung cancer treatment-part I: nitrogen-containing six-membered aromatic heterocycles	8
Molecular Glues Targeting Protein Degradation Pathways for Drug Discovery	8
Candesartan, Losartan and Valsartan Zn(II) Complexes Interactions With Bovine Serum Albumin	8
Advancement of Targeted Protein Degradation Strategies As Therapeutics for Undruggable Disease Targets	7
Dorzolamide Suppresses PKCδ -TIRAP-p38 MAPK Signaling Axis to Dampen the Inflammatory Response	7
Recent Advances of Cannabidiol Studies in Medicinal chemistry, Pharmacology and Therapeutics	7
Kynomycin: A Beacon of Hope in the Battle Against Antibiotic Resistance	7
Synthesis of Hydrazinylthiazole Carboxylates: A Mechanistic Approach for Treatment of Diabetes and Its Complications	7
Research Progress on Tamoxifen and Its Analogs Associated With Nuclear Receptors	7
Network Analysis and Ligand-Based Pharmacophore Modeling for Discovery of Small Molecule Against Glioblastoma Multiforme	7
Novel coumarin linked pyrazoles, thiazoles, and thiadiazoles: synthetic strategies and in vitro antimicrobial investigation	7
CK1 Delta Inhibition: An Emerging Strategy to Combat Neurodegenerative Diseases	7
Recent Advances in dehydroacetic acid-clubbed pyridine conjugates: design, synthesis, characterization, molecular docking investigations and evaluation of anti-cancer efficacy	7
New thiazolidin-4-ones as anti-cervical cancer agents targeting EGFR: design, synthesis, and computational studies	7
In-vitro and in-silico assessment of thiazole-thiazolidinone derivatives as selective inhibitors of urease and α-glucosidase	7
Organoselenium compounds beyond antioxidants	7
Novel 4-Aminoquinoline Analogs Targeting the HIF-1α Signaling Pathway	7
The antibreast cancer therapeutic potential of quinazoline hybrids–Part I	7
Corrigendum	7
Welcome to the 16th Volume of Future Medicinal Chemistry	7
The emerging field of senotherapeutic drugs	7
From clove oil to bioactive agents: synthetic routes, antimicrobial and antiparasitic activities of eugenol derivatives	7
Thiazolidinedione–Triazole Conjugates: Design, Synthesis and Probing of the α-Amylase Inhibitory Potential	7
BioPrint Meets the AI Age: Development of Artificial Intelligence-Based ADMET Models for the Drug-Discovery Platform SAFIRE	7
Design, synthesis and mechanistic exploration of anti-plasmodial Indolo[2,3- b ]quinoxaline-7-chloroquinoline hybrids	7
Benzimidazole-acrylonitrile hybrid derivatives act as potent urease inhibitors with possible fungicidal activity	7
COVID-19 Diagnostic Assay Sensitivity: Lessons for the Upcoming Wave Or Next Pandemic	7
Design and Synthesis of Selective FLT3 Inhibitors Via Exploration of Back Pocket II	7
Optimizing selective estrogen receptor degraders for anticancer drug development	7
Expanding potential of quinoline hydrazide/hydrazone derivatives as anticancer agents	6
Synthesis, characterization and biological evaluation of aurones as potential neuroprotective agents	6
Ultrasonic-assisted synthesis and antitumor evaluation of novel variant heterocyclic compounds based on piperidine ring	6
Antimicrobial, Anticancer and Immunomodulatory Potential of New Quinazolines Bearing Benzenesulfonamide Moiety	6
Pyrazine-based small molecule kinase inhibitors: clinical applications and patent review (2019–2023)	6
Virtual and Augmented Reality Applications in Medicinal Chemistry	6
Human Sirtuin 2 inhibitors, Their Mechanisms and Binding Modes	6
Establishment of Models for Reliability Evaluation of 3CLpro Ligand-Receptor Complexes With Different Binding Sites	6
Design and synthesis of newer 5-aryl- N -(naphthalen-2-yl)-1,3,4-oxadiazol-2-amine analogues as anticancer agents	6
Tetrahydroquinoline: An Efficient Scaffold As mTOR Inhibitor for the Treatment of Lung Cancer	6
Benzo[ d ]thiazole-2-Carboxamides As New Antituberculosis Chemotypes Inhibiting Mycobacterial ATP Phosphoribosyl Transferase	6
Evidence-based drug discovery	6
Proteolysis-Targeting Chimera Molecules Targeting SHP2	6
Synthesis and antiproliferative evaluation of novel 3,5,8-trisubstituted coumarins against breast cancer	6
The anticancer therapeutic potential of pyrimidine–sulfonamide hybrids	6
Therapeutic targeting of neuroinflammation in methamphetamine use disorder	6
Cyclin-Dependent Kinases As Potential Targets for Colorectal Cancer: Past, Present and Future	6
Design, Synthesis and Anticancer Evaluation of Some Novel 7-Hydroxy-4-Methyl-3-Substituted Benzopyran-2-One Derivatives	6
Therapeutic potential of chalcone-1,2,3-triazole hybrids as anti-tumour agents: a systematic review and SAR studies	6
Coumarin hybrids: dual-target candidates for future antimicrobial and antitubercular therapies	6
Synthesis and Anti-Ovarian Cancer Effects of Benzimidazole-2-Substituted Pyridine and Phenyl Propenone Derivatives	6
Dual VEGFR-2 and EGFR T790M inhibitors of phenyldiazenes: anticancer evaluations, ADMET, docking, design and synthesis	6
Development of Small Macrocyclic Kinase Inhibitors	6
Key developments in fluorinated heterocycles	6
Designing molecular hybrids as novel breast cancer therapeutics	6
Our New Year's (re)solution: Welcome to the 15th Volume of Future Medicinal Chemistry	6
Challenging Breast Cancer Through Novel sulfonamide–pyridine Hybrids: design, synthesis, Carbonic Anhydrase IX Inhibition and Induction of Apoptosis	6
Recent developments in matrine as a versatile molecular scaffold in small molecule drug discovery	6
Environment benign synthesis of 5-acyl-4-hydroxypyridin-2(1 H )-one derivatives as antioxidant and α -amylase inhibitors	5
Exploring the therapeutic potential and chemical properties of trans-chalcone: a comprehensive review	5
Design, synthesis, and molecular docking studies of thiazole derivatives against phospholipase A 2 ( Naja oxiana ) venom	5
Glyco Disulfide Capped Gold Nanoparticle Synthesis: Cytotoxicity Studies and Effects on Lung Cancer A549 Cells	5
Semicarbazone, thiosemicarbazone tailed isoxazoline-pyrazole: synthesis, DFT, biological and computational assessment	5
Development of indole hybrids for potential lung cancer treatment - part II	5
Design and Synthesis of Novel Aza-Ursolic Acid Derivatives: In Vitro Cytotoxicity and Nitric Oxide Release Inhibitory Activity	5
Design, semi-synthesis and bioevaluation of koumine-like derivatives as potential antitumor agents in vitro and in vivo	5
Sirtuin Modulators: Past, Present, and Future Perspectives	5
Recent Progress of Palmitoyl Transferase DHHC3 As a Novel Antitumor Target	5
New and potential boron-containing compounds for treatment of Alzheimer's disease and cancers	5

Regulation of post-translational modification of PD-L1 and associated opportunities for novel small-molecule therapeutics	5
Urea-sugar and thiourea-sugar diastereomers: synthesis, crystal structure and biological activities	5
Enoxacin-Based Derivatives: Antimicrobial and Antibiofilm Agent: A Biology-Oriented Drug Synthesis (BIODS) Approach	5
Design, Synthesis and Structure–Activity Relationship Studies of Novel Spirochromanone Hydrochloride Analogs As Anticancer Agents	5
Targeting STK33: From Inhibition to Degradation	5
Unveiling the potential of HS-1793: a review of its anticancer properties and therapeutic promise	5
Advances in Research With Rutin-Loaded Nanoformulations in Mitigating Lung Diseases	5
Conjugated Carbon Monoxide-Releasing Molecules have Broad-Spectrum Antimicrobial Activity	5
Recent advances in targeted degradation in the RAS pathway	5
Synthesis, cytotoxicity and 99m Tc-MIBI tumor cell uptake evaluation of 2-phenylbenzothiazole tagged triazole derivatives	5
Gold: Not Just jewelry…	5
A novel class of potent antiangiogenic and antioxidant pyrazoles: synthesis, bioactivity, docking and ADMET studies	5
Combining Virtual Screening and In Vitro Evaluation for the Discovery of Potential CYP11B2 Inhibitors	5
Prioritizing oral bioavailability in drug development strategies	5
Innovative virtual screening of PD-L1 inhibitors: the synergy of molecular similarity, neural networks and GNINA docking	5
Recent development of azole–sulfonamide hybrids with the anticancer potential	5
Novel Sulfonamide Derivatives as a Tool to Combat Methicillin-Resistant Staphylococcus Aureus	5
Antimicrobial Potential of Quaternary Phosphonium Salt Compounds: a Review	4
Epigenetic therapy meets targeted protein degradation: HDAC-PROTACs in cancer treatment	4
TSPYL2 Reduced Gefitinib Resistance and DNA Damage Repair Via Suppressing SIRT1-Mediated FOXO3 Deacetylation	4
Protein–Protein Interactions By Influenza Polymerase Subunits As Drug Targets	4
Preclinical characterization of a water-soluble low-impact ampakine prodrug, CX1942 and its active moiety, CX1763	4
Application of Iron Oxide Nanoparticles to Control the Release of Minocycline for the Treatment of Glioblastoma	4
Application of a Fluorescent H 2 S Probe Based on Excited-State Intramolecular Proton Transfer for Detecting Latent Mechanism of H 2	4
Can Dextran-Based Nanoparticles Mitigate Inflammatory Lung diseases?	4
Recent advances and future perspectives in small molecule JAK2 inhibitors	4
Emerging Therapeutic Approaches of SHP2-Targeted Modulators	4
Application of parallel artificial membrane permeability assay technique and chemometric modeling for blood–brain barrier permeability prediction of protein kinase inhibitors	4
Sweet Targets: Sugar Nucleotide Biosynthesis Inhibitors	4
Medicinal Chemistry Approaches for the Discovery of Plasmodium Falciparum Dihydroorotate Dehydrogenase Inhibitors as Antimalarial Agents	4
Synthesis of Novel Benzothiophene Derivatives As Protectors Against Cranial Irradiation-Induced Neuroinflammation	4
Therapeutic potential of a novel pyrazolyl-pyridine derivative in the treatment of experimental colitis	4
Recent Advances in ATM Inhibitors As Potential Therapeutic Agents	4
Synthesis of 2,4-dihydroxyacetophenone derivatives as potent PDE-1 and -3 inhibitors: in vitro and in silico insights	4
Exploring the antimicrobial and cytotoxic potential of novel chloroquine analogues	4
Exploring digestive enzymes’ differential affectivity of synthesized 2-thienyl-based chalcones	4
Protein-protein interactions in cGAS-STING pathway: a medicinal chemistry perspective	4
Design, Synthesis and Bioevaluation of Novel Trifluoromethylquinoline Derivatives As Tubulin Polymerization Inhibitors	4
Norfloxacin Derivatives as DNA Gyrase and Urease Inhibitors: Synthesis, Biological Evaluation and Molecular Docking	4
Xanthohumol Alleviates T2DM-induced Liver Steatosis and Fibrosis by Mediating the NRF2/RAGE/NF-κB Signaling Pathway	4
A Hybrid Resampling Algorithms SMOTE and ENN Based Deep Learning Models for Identification of Marburg Virus Inhibitors	4
The Diverse Bioactivity of α-mangostin and Its Therapeutic Implications	4
Exploring New Imines as Anti-Inflammatory COX and 5-LOX Inhibitors with an Improved Pharmacokinetic Profile	4
Advances of deep Neural Networks (DNNs) in the development of peptide drugs	4
Phthalimides as anti-inflammatory agents	4
An Interpretable Machine Learning Model for Selectivity of Small-Molecules Against Homologous Protein Family	4
Structure–Activity Relationships of Novel N -Imidazoylpiperazines with Potent Anti- Trypanosoma Cruzi Activity	4
RNA-targeting therapeutics: drugging the undruggable	4
Pharmacokinetic Correlation of Structurally Modified Chalcone Derivatives As Promising Leads to Treat Tuberculosis	4
Cu(II) complexes based on benzimidazole ligands: synthesis, characterization, DFT, molecular docking & bioactivity study	4
Exploration of pyrazole-based pyridine-4-carbohydrazide derivatives as drug-resistant Mtb agents: design, synthesis, biological evaluation, and in-silico<	4
Design, synthesis and biological evaluation of sulfamethazine derivatives as potent neuraminidase inhibitors	4
Thiourea-functionalized aminoglutethimide derivatives as anti-leishmanial agents	4
Design, synthesis and biological evaluation of novel pyrazole-based compounds as potential chemotherapeutic agents	4
Mitigating Inflammation Using Advanced Drug Delivery By Targeting TNF-α in Lung Diseases	4
Calcium Complexes of Oxicams: New Dimensions in Rheumatoid Arthritis Treatment	4
Breaker Peptides Against amyloid-β Aggregation: a Potential Therapeutic Strategy for Alzheimer’s Disease	4
Discovery of bis -chalcones and bis -pyrimidines as potential urease inhibitors: from synthesis to computational insights	4
Exploring ACSL4/LPCAT3/ALOX15 and SLC7A11/GPX4/NFE2L2 as Potential Targets in Ferroptosis-Based Cancer Therapy	4
Structure–activity relationships study of N -ethylene glycol-comprising alkyl heterocyclic carboxamides against A549 lung cancer cells	4
Progress and challenges in the development of triazole antimicrobials	3
Inhibition of α-glucosidase Enzyme By ‘click'-inspired Pharmacophore Framework 1,3,4-thiadiazole–1,2,3-triazole Hybrids	3
Virtual Screening Identifies Tipranavir As a SIRT1 Inhibitor With anti-hepatocarcinoma Effect	3
Insights into direct KRAS inhibition strategies for cancer treatment	3
Design, synthesis, docking studies and bioactivity evaluation of 1,2,3-triazole eugenol derivatives	3
In silico studies, synthesis, characterization and in vitro studies of levosulpiride derivatives	3
Synthesis of Ponatinib Analogues As Novel Inhibitors of Leukemia Stem Cells	3
Special Focus Issue – Targeted Protein Degradation: A New Paradigm in Medicinal Chemistry	3
Repurposing Dyphylline as a Pan-Coronavirus Antiviral Therapy	3
Versatile Tools of Synthetic Biology Applied to Drug Discovery and Production	3
Leishmanicidal Activity and 4D Quantitative Structure–Activity Relationship and Molecular Docking Studies of Vanillin-Containing 1,2,3-Triazole Derivatives	3
Recent Advances in Oxazolidinones as Antituberculosis Agents	3
Recent Advances in Anti-Coxsackievirus A16 Viral Drug Research	3
Recent advances in quinazolinone derivatives: structure, design and therapeutic potential	3
Biological and Computational Investigation of Transition metal(II) Complexes of 2-phenoxyaniline-based Ligands	3
Pyrimido[4,5-b]indole Derivatives Bearing 1,2,4-oxadiazole Moiety As MDM2 Inhibitor Candidates in Cancer Treatment	3
Long-acting Biodegradable Implants for Osteoporosis Management: Transforming the Landscape of Bisphosphonates Delivery	3
Curcumin-based Nanoformulations As an Emerging Therapeutic Strategy for Inflammatory Lung Diseases	3
Discovery of novel ULK1 inhibitors through machine learning-guided virtual screening and biological evaluation	3
Discovery of New thieno[2,3- d ]pyrimidines as EGFR Tyrosine Kinase Inhibitors for Cancer Treatment	3
Synthesis, in Vitro Bio-Evaluation and in Silico Molecular Docking Studies of Thiadiazole-Based Schiff Base Derivatives	3
New immunomodulatory anticancer quinazolinone-based thalidomide analogs: design, synthesis and biological evaluation	3
Benzimidazole derivatives as potent α -amylase inhibitors: synthesis, characterization and in vitro α -amylase inhibition	3
Fluorinated building blocks in drug design: new pathways and targets	3
Hitting Drug-Resistant Malaria Infection With Triazole-Linked Flavonoid–Chloroquine Hybrid Compounds	3
In vitro α-glucosidase, docking and density functional theory studies on novel azide metal complexes	3
Design, synthesis and biological evaluation of non-glucosidal based 1,3,4-thiadiazoles as SGLT-2 inhibitors	3
Anti-proliferation evaluation of new derivatives of indole-6-carboxylate ester as receptor tyrosine kinase inhibitors	3
A comprehensive insight into naphthalimides as novel structural skeleton of multitargeting promising antibiotics	3
Literature-Based Drug–Drug Similarity for Drug Repurposing: Impact of Medical Subject Headings Term Refinement and Hierarchical Clustering	3
Rapidly Evolving First-Line Therapy Using Checkpoint Inhibitors in Metastatic Renal Cell Cancer	3
New Thiouracil Derivatives As Histone Deacetylase Inhibitors and Apoptosis Inducers: Design, Synthesis and Anticancer Evaluation	3
Latest Advances in Specific Inhibition of Tumor-Associated Carbonic Anhydrases	3
Challenges and Opportunities for In Vivo PROTAC Delivery	3
The Role of microRNA-21 in the Onset and Progression of Cancer	3