Future Medicinal Chemistry

Article	Citations
Novel coumarin linked pyrazoles, thiazoles, and thiadiazoles: synthetic strategies and in vitro antimicrobial investigation	57
Advancements in PROTAC-based therapies for neurodegenerative diseases	50
Biochemical evaluation of novel thiazolone derivatives as dual α-glucosidase/α-amylase inhibitors, anti-inflammatory agents	45
Dual VEGFR-2 and EGFR T790M inhibitors of phenyldiazenes: anticancer evaluations, ADMET, docking, design and synthesis	45
Chemical and Biological Versatility of Pyrazolo[3,4- d ]Pyrimidines: One Scaffold, Multiple Modes of Action	42
Panantiviral Agents: Implications for Treating Cancers Associated With Oncoviruses	37
Enhancing the Affinity of Novel GLS1 Allosteric Inhibitors By Targeting Key Residue Lys320	37
Chemical Language Models for Applications in Medicinal Chemistry	37
New Thiouracil Derivatives As Histone Deacetylase Inhibitors and Apoptosis Inducers: Design, Synthesis and Anticancer Evaluation	36
Targeting LRRK2 Mutations in Parkinson's Disease	32
Advances in Non-Covalent Based Inhibitors Targeting Myc: A Promising Approach for Cancer Treatment	31
Welcome to the 16th Volume of Future Medicinal Chemistry	31
PPARγ Transcription Effect on Naturally Occurring O -Prenyl Cinnamaldehydes and Cinnamyl Alcohol Derivatives	29
P2Y14R for Inflammation Therapy: Is It a Promising target?	28
Discovery of α-Helix-Mimicking Sulfono-γ-AApeptides as p53−MDM2 Inhibitors	25
Synthetic Corticosteroids As Tryptophan Hydroxylase Stabilizers	24
Unsymmetrical Thiourea Derivatives: Synthesis and Evaluation as Promising Antioxidant and Enzyme Inhibitors	24
COVID-19 Diagnostic Assay Sensitivity: Lessons for the Upcoming Wave Or Next Pandemic	24
Citrate Transporter Inhibitors: Possible New Anticancer Agents	22
Therapeutic Potential of Vitamin B 1 Derivative Benfotiamine From Diabetes to COVID-19	22
Welcome to Volume 14 of Future Medicinal Chemistry	22
Therapeutic N -Heterocyclic Carbenes: An Interview With Alejandro Bugarin	21
Multicomponent Reactions As a Privileged Tool for Multitarget-Directed Ligand Strategies in Alzheimer’s Disease Therapy	20
Virtual and Augmented Reality Applications in Medicinal Chemistry	20
Investigations of New N 1 -Substituted Pyrazoles as Anti-Inflammatory and Analgesic Agents having COX Inhibitory Act	19

Cheminformatics-driven Discovery of Hit Compounds Against Paracoccidioides spp.	19
Identification of Sulfonamide-Based Butyrylcholinesterase Inhibitors Using Machine Learning	18
Targeting Tuberculosis – An Interview With Robert Abramovitch	18
Advanced Drug Delivery Systems Targeting NF-κB in Respiratory Diseases	18
The Connection Between PARP14 and SARS-CoV-2	18
Super-Conserved Receptors Expressed in the Brain: Biology and Medicinal Chemistry Efforts	18
Design, Synthesis and In Vitro Antiproliferation Activity of Some 2-aryl and -heteroaryl Benzoxazole Derivatives	18
Combining Structure-Based and 3D QSAR Pharmacophore Models to Discover Diverse Ligands Against EGFR in Oral Cancer	18
Antimicrobial, Anticancer and Immunomodulatory Potential of New Quinazolines Bearing Benzenesulfonamide Moiety	17
Synthesis and antiproliferative evaluation of novel 3,5,8-trisubstituted coumarins against breast cancer	16
An Emerging Role of KRAS in Biogenesis, Cargo Sorting and Uptake of Cancer-Derived Extracellular Vesicles	16
The anticancer therapeutic potential of pyrimidine–sulfonamide hybrids	16
Pyrazine-based small molecule kinase inhibitors: clinical applications and patent review (2019–2023)	15
Sulfonamide-salicylaldehyde Imines Active Against methicillin- and trimethoprim/sulfonamide-resistant Staphylococci	15
Synthesis, biological and computational evaluation of benzoxazole hybrid analogs as potential anti-Alzheimer's agents	15
Mitochondrial Dysfunctions Associated With Chronic Respiratory Diseases and Their Targeted Therapies: an Update	15
Isocoumarins incorporating chalcone moieties act as isoform selective tumor-associated carbonic anhydrase inhibitors	15
Ultrasonic-assisted synthesis and antitumor evaluation of novel variant heterocyclic compounds based on piperidine ring	15
In Vitro Cytotoxic Investigation of Some Synthesized 1,6-Disubstituted-1-Azacoumarin Derivatives as Anticancer Agents	15
Design and synthesis of new nicotinamides as immunomodulatory VEGFR-2 inhibitors and apoptosis inducers	14
The Role of microRNA-21 in the Onset and Progression of Cancer	14
Facile synthesis, antimicrobial activity, and molecular docking analysis of 8-hydroxyquinoline-4-thiazolidinone hybrids	13
Small-Molecule Oligonucleotides As Smart Modality for Antiviral Therapy: A Medicinal Chemistry Perspective	13
Novel Pyrimido-Pyridazine Derivatives: Design, Synthesis, Anticancer Evaluation and In Silico Studies	13
Novel inhibitors of PARP1 and PARP14: design, synthesis, and potentiation of cisplatin efficacy in cancer	13
Design and Synthesis of Selective FLT3 Inhibitors Via Exploration of Back Pocket II	13
Selection of SARS-CoV-2 Main Protease Inhibitor Using Structure-Based Virtual Screening	13
The Structural Basis of Effective LOX-1 Inhibition	13
FAK Inhibitors As Promising Anticancer Targets: Present and Future Directions	13
Novel 3-substituted coumarins inspire a custom pharmacology prediction pipeline: an anticancer discovery adventure	12
Design, synthesis and evaluation of novel norfloxacin analogs as potent anticancer and antioxidant agents	12
Repurposing Dyphylline as a Pan-Coronavirus Antiviral Therapy	12
Novel Amodiaquine Analogues to Treat Cervical Cancer and Microbial Infection in the Future	12
One-step synthesis of diaryloxadiazoles as potent inhibitors of BCRP	11
Using Novel Click Chemistry Algorithm to Design D3R Inhibitors As Blood–Brain Barrier Permeants	11
The Story of EGFR: From Signaling Pathways to a Potent Anticancer Target	11
Structure-Based Discovery of Thiosemicarbazones As SARS-CoV-2 Main Protease Inhibitors	11
Biological and computational evaluation of novel benzofuranyl derivatives as acetylcholinesterase and butyrylcholinesterase inhibitors	11
Leishmanicidal Activity and 4D Quantitative Structure–Activity Relationship and Molecular Docking Studies of Vanillin-Containing 1,2,3-Triazole Derivatives	11
Treatment of Rheumatoid Arthritis With Curcumin Analog 3,5-bis(arylidene)-4-piperidone	10
The Synthesis and Effects of a Novel TRPC6 inhibitor, BP3112, on Hepatocellular Carcinoma	10
Novel candidates synthesis of indenopyrazole, indenoazine and indenothiophene, with anticancer and in silico studies	10
Combining EGFR Inhibitors With SHP2 Or LSD1 Inhibitors to Overcome Multidrug Resistance in Cancer	10
Development of Small Macrocyclic Kinase Inhibitors	10
Benzimidazole-acrylonitrile hybrid derivatives act as potent urease inhibitors with possible fungicidal activity	10
Synthesis, characterization and biological evaluation of aurones as potential neuroprotective agents	10
CK1 Delta Inhibition: An Emerging Strategy to Combat Neurodegenerative Diseases	9
Latest Progress in the Development of Cyclooxygenase-2 Pathway Inhibitors Targeting Microsomal Prostaglandin E 2 Synthase-1	9
Novel Anthraquinone Derivatives Trigger Endoplasmic Reticulum Stress Response and Induce Apoptosis	9
In Silico Multiscale Drug Design to Discover Key Structural Features of Potential JAK2 Inhibitors	9

Novel Hydroxy- and Amidino-Substituted Benzimidazoles and Benzothiazoles as Antibacterial and Antiproliferative Agents	9
Potential Strategies for the Management of Adenocarcinoma: a Perspective	9
New Kinase and HDAC Hybrid Inhibitors: Recent Advances and Perspectives	9
STING Upregulation Strategies to Potentiate STING Immunotherapy	9
Discovery of 1,5-diaryl-1,2,4-triazole Derivatives as Myoferlin Inhibitors and Their Antitumor Effects in Pancreatic Cancer	9
Proteolysis-Targeting Chimera Molecules Targeting SHP2	9
Research Progress on Tamoxifen and Its Analogs Associated With Nuclear Receptors	8
Development of 5-hydroxybenzothiophene derivatives as multi-kinase inhibitors with potential anti-cancer activity	8
Synthesis and Molecular Modeling Studies of 1-Benzyl-2-Indolinones As Selective AChE Inhibitors	8
Synthesis and Biological Evaluation of New Antiseizure Compounds Derived From Valproic Acid	8
Medicinal chemistry aspects of fat mass and obesity associated protein: structure, function and inhibitors	8
Novel 4-Aminoquinoline Analogs Targeting the HIF-1α Signaling Pathway	8
Sulfonic Acid: Key Drug Design Elements With potent, broad-ranging Pharmacological Activities	8
A novel chromone-based as a potential inhibitor of ULK1 that modulates autophagy and induces apoptosis in colon cancer	8
Exploitation of a Novel Allosteric Binding Region in DNA Gyrase and its Implications for Antibacterial Drug Discovery	7
Structure-Based Molecular Insights Into Matrix Metalloproteinase Inhibitors in Cancer Treatments	7
Synergistic anti-inflammatory and anti-tb effects of Au-Pt-Cu nanofluids: experimental and computational insights	7
Optimizing selective estrogen receptor degraders for anticancer drug development	7
Naphthoquinone fused diazepines targeting hyperamylasemia: potential therapeutic agents for diabetes and cancer	7
Leading designs of peptide-based chemical probes for medical imaging– the dawn of precision diagnostics	7
Rational Design of Peptide Inhibitors Targeting HSP90–CDC37 Protein–Protein Interaction	7
A Review of Current and Promising Nontuberculous Mycobacteria Antibiotics	7
A comprehensive review on the latest advances of dimeric anticancer prodrugs	7
Network Analysis and Ligand-Based Pharmacophore Modeling for Discovery of Small Molecule Against Glioblastoma Multiforme	7
Design, Synthesis and Exploration of Novel Triazinoindoles as Potent Quorum-Sensing Inhibitors and Radical Quenchers	7
Exploring biological activities of novel Schiff bases derived from amlodipine and in silico molecular modeling studies	7
Synthesis, Molecular Modeling and Cholinesterase Inhibitory Effects of 2-Indolinone-Based Hydrazinecarbothioamides	7
Corrigendum	7
Novel Set of Highly Substituted Bis-Pyridines: Synthesis, Molecular Docking and Drug-Resistant Antibacterial Profile	7
Expecting medication misuse: a proactive approach to drug discovery to prevent fatal overdose	7
A Systematic Review of carbohydrate-based Bioactive Molecules for Alzheimer’s Disease	7
Organotellurium (IV) complexes as anti-malarial agents: synthesis, characterization and computational insights	7
The emerging field of senotherapeutic drugs	7
Design of SARS-CoV-2 Mpro, PLpro Dual-Target Inhibitors Based on Deep Reinforcement Learning and Virtual Screening	6
Pyrazole: an Emerging Privileged Scaffold in Drug Discovery	6
In vivo evaluation of novel synthetic pyrazolones as CDK9 inhibitors with enhanced pharmacokinetic properties	6
Design, synthesis and inhibition evaluation of novel chalcone amide α-glucosidase inhibitors	6
Design and application of CCR8 antagonists	6
Advances in AR-Targeting Chimeras: A Case Study of proteolysis-targeting Chimeras From Bench to Bedside	6
Novel Benzimidazole Derivatives as Effective Inhibitors of Prolyl Oligopeptidase: Synthesis, in Vitro and in Silico Analysis	6
New pyrano-pyridine conjugates as potential anticancer agents: design, synthesis and computational studies	6
Targeting Mucin Hypersecretion in COVID-19 Therapy	6
Cyclin-Dependent Kinases As Potential Targets for Colorectal Cancer: Past, Present and Future	6
Targeting cyclin-dependent kinase 2 (CDK2) interactions with cyclins and Speedy 1 (Spy1) for cancer and male contraception	6
Challenges and Opportunities for In Vivo PROTAC Delivery	6
New (S)-verbenone-isoxazoline-1,3,4-thiadiazole Hybrids: Synthesis, Anticancer Activity and Apoptosis-Inducing Effect	6
New Horizons in Lung Cancer Management Through ATR/CHK1 Pathway Modulation	6
Inhibiting the Metallo-β-lactamases: Challenges and Strategies to Overcome Bacterial β-lactam Resistance	6
Establishment of Models for Reliability Evaluation of 3CLpro Ligand-Receptor Complexes With Different Binding Sites	6
Synthesis and in vitro antitrypanosomatid activity of novel 5-nitroindole-rhodanine conjugates	6
Challenging Breast Cancer Through Novel sulfonamide–pyridine Hybrids: design, synthesis, Carbonic Anhydrase IX Inhibition and Induction of Apoptosis	5
Novel Antimicrobial Iodo-Dihydro-Pyrrole-2-One Compounds	5
Current landscape of tropomyosin receptor tyrosine kinase inhibitors	5
Comprehensive drug-like assessment of pyridine carbothioamide analogs: from molecular modeling to in-vivo evaluation	5
H 2 S-releasing Molecules in Pharmaceutical Development	5
Docking and Antibacterial Activity of Novel Nontoxic 5-Arylidenepyrimidine-Triones as Inhibitors of NDM-1 and MetAP-1	5
Synthesis of new coumarin derivatives and assessment of their antimicrobial efficacy	5
Key developments in fluorinated heterocycles	5
Evaluation of Synthetic Aminoquinoline Derivatives As Urease Inhibitors: In Vitro , In Silico and Kinetic Studies	5
Targeting undruggable protein KRAS for cancer therapy: novel opportunities and challenges	5
Novel HIF-1α Inhibitor CDMP-TQZ for Cancer Therapy	5
Serendipitous Identification of Phenylhydrazine Derivatives As Potent Inhibitors of carbapenem-resistant Acinetobacter Baumannii	5
HDAC8 As an Emerging Target in Drug Discovery With Special Emphasis on Medicinal Chemistry	5
The design and development of LRRK2 inhibitors as novel therapeutics for Parkinson’s disease	5
Minimal Screening Requirements for Identifying Highly Promiscuous Kinase Inhibitors	5
Design, Synthesis and Anticancer Evaluation of Some Novel 7-Hydroxy-4-Methyl-3-Substituted Benzopyran-2-One Derivatives	5
Rapidly Evolving First-Line Therapy Using Checkpoint Inhibitors in Metastatic Renal Cell Cancer	5
Special Focus Issue – Targeted Protein Degradation: A New Paradigm in Medicinal Chemistry	5
Discovery of novel ULK1 inhibitors through machine learning-guided virtual screening and biological evaluation	5
A comprehensive insight into naphthalimides as novel structural skeleton of multitargeting promising antibiotics	5
Development of Novel Anti-Infective and Antioxidant Azole Hybrids using a Wet and Dry Approach	5
Current Development of Pyrazole–Azole Hybrids With Anticancer Potential	5
Computational Insights Into Novel Inhibitor Indole-Heterocycle Specific Against Glycogen Phosphorylase Isoenzymes Interaction Mechanism	5
Synthesis of Quercetin–Iron (Fe) Complex and Its In Silico and In Vitro Confirmation Towards Antibacterial Activity	5
Synthesis of Ponatinib Analogues As Novel Inhibitors of Leukemia Stem Cells	5
Therapeutic targeting of neuroinflammation in methamphetamine use disorder	5
A New Class of 5-HT 1A Receptor Antagonists With Procognitive and Antidepressant Properties	5
Literature-Based Drug–Drug Similarity for Drug Repurposing: Impact of Medical Subject Headings Term Refinement and Hierarchical Clustering	5
Molecular docking, derivatization, characterization and biological assays of amantadine	5
Synthesis, anticancer activity, docking and computational studies of new pyridyl-glycosyl hybrids and acyclic analogs	5

Synthetic benzofuran-linked Chalcones With Dual Actions: a Potential Therapeutic Approach to Manage Diabetes Mellitus	5
New pyrrolopyridine-based Thiazolotriazoles As Diabetics Inhibitors: Enzymatic Kinetics and In Silico Study	5
α -amylase Inhibition and In Silico Studies of Novel Naphtho[2,3- d ]imidazole-4,9-Dione Linked N	5
Synthesis and Anti-Ovarian Cancer Effects of Benzimidazole-2-Substituted Pyridine and Phenyl Propenone Derivatives	5
Exploring of novel oxazolones and imidazolones as anti-inflammatory and analgesic candidates with cyclooxygenase inhibitory action	4
Insight on novel oxindole conjugates adopting different anti-inflammatory investigations and quantitative evaluation	4
The Discovery and Development of Transthyretin Amyloidogenesis Inhibitors: What are the Lessons?	4
Fluorinated building blocks in drug design: new pathways and targets	4
Structure-Guided Discovery of Adenosine Triphosphate-Competitive Casein Kinase 2 Inhibitors	4
Synergistic effect of new pyrimidine derivative with oxacilin against methicillin-resistant Staphylococcus aureus	4
Rh(III) and Ru(II) Complexes With Phosphanyl–Alkylamines: Inhibition of DNA Synthesis Induced By Anticancer Rh Complex	4
G-quadruplex Ligands As Therapeutic Agents Against cancer, Neurological Disorders and Viral Infections	4
Discovery of New thieno[2,3- d ]pyrimidines as EGFR Tyrosine Kinase Inhibitors for Cancer Treatment	4
Novel Inhibitors of the Renal Inward Rectifier Potassium Channel of the Mosquito Vector Aedes Aegypti	4
Discovery of Novel Covalent Inhibitors of DJ-1 Through Hybrid Virtual Screening	4
Restoration of p53 Functions By Suppression of mortalin–p53 Sequestration: an Emerging Target in Cancer Therapy	4
Synthesis of quercetin derivatives as cytotoxic against breast cancer MCF-7 cell line in vitro and in silico studies	4
Synthesis, crystal structure, biological and docking studies of 5-hydroxy-2-{[(2-methylpropyl)iminio]methyl}phenolate	4
Harnessing molecular hybridization approach to discover novel quinoline EGFR-TK inhibitors for cancer treatment	4
Barbiturate–sulfonate hybrids as potent cholinesterase inhibitors: design, synthesis and molecular modeling studies	4
Structural Insight Into SSE15206 in Complex With Tubulin Provides a Rational Design for Pyrazolinethioamides As Tubulin Polymerization Inhibitors	4
Synthesis of Hydrazinyl–Thiazole Ester Derivatives, in Vitro Trypanocidal and Leishmanicidal Activities	4
KSHV-Specific Antivirals Targeting the Protein–DNA Interaction of the Latency-Associated Nuclear Antigen	4
Expanding potential of quinoline hydrazide/hydrazone derivatives as anticancer agents	4
Thiosemicarbazones Reprogram Pancreatic Cancer Bidirectional Oncogenic Signaling Between Cancer Cells and Stellate Cells to Suppress Desmoplasia	4
Synthesis and In Vitro Studies for Structure-Based Design of Novel Chalcones As Antitubercular Agents Targeting InhA	4
Targeting FGL2, a Molecular Drug Target for Glioblastoma, With Natural Compounds Through Virtual Screening Method	4
Benzo[ d ]thiazole-2-Carboxamides As New Antituberculosis Chemotypes Inhibiting Mycobacterial ATP Phosphoribosyl Transferase	4
Resistant Starch: Ideal Candidate for the Enteric Coating of NSAIDs?	4
Functional Characterization of HIC, a P2Y1 agonist, As a p53 Stabilizer for Prostate Cancer Cell Death Induction	4
Synthesis and interest in medicinal chemistry of β-phenylalanine derivatives (β-PAD): an update (2010–2022)	4
Synthesis, in vitro and in silico anticancer evaluation of novel pyridin-2-yl estra-1,3,5(10)-triene derivatives	4
New 1,3,4-thiadiazoles Derivatives: Synthesis, Antiproliferative Activity, Molecular Docking and Molecular Dynamics	4
Identification of a Novel Antifungal Backbone of Naphthalimide Thiazoles with Synergistic Potential for Chemical and Dynamic Treatment	4
Salvianolic Acid B Noncovalently Interacts With Disordered c-Myc: A Computational and Spectroscopic-Based Study	4
Bacterial Carbonic Anhydrases: Underexploited Antibacterial Therapeutic Targets	4
Exploring the therapeutic potential of cinnamoyl derivatives in attenuating inflammation in lipopolysaccharide-induced Caco-2 cells	4
Propargylamine: an Important Moiety in Drug Discovery	4
Design, Synthesis and Biological Evaluation of Novel Indanones Derivatives As Potent Acetylcholinesterase/Monoamine Oxidase B Inhibitors	4
Epigenetics: rethinking of drug research and development	4
Discovery of Novel STAT3 DNA Binding Domain Inhibitors	4
One-Pot Multicomponent Synthesis of Novel Pyridine Derivatives for Antidiabetic and Antiproliferative Activities	4
A series of benzensulfonamide derivatives as new potent carbonic anhydrase IX and XII inhibitors	4
An Insight Into the Structure–Activity Relationship Studies of Anticancer Medicinal Attributes of 7-Azaindole Derivatives: A Review	4
Chitosan–maleic Acid Conjugate As Potential Excipient Candidate for Oral Drug delivery?	3
Hitting Drug-Resistant Malaria Infection With Triazole-Linked Flavonoid–Chloroquine Hybrid Compounds	3
Zn (II) complex with vanillin derived Schiff base: antifungal, antibacterial, antioxidant and anticholinesterase activities	3
Discovery of Reversible Selective Monoamine Oxidase B Inhibitors With anti-acetylcholinesterase Activity Derived From 4-oxo-N-4-diphenyl Butanamides	3
PROTAC Cell Permeability and Oral Bioavailability: A Journey Into Uncharted Territory	3
Antimicrobial Activity of Carvacrol and Its Derivatives on Mycobacterium Spp.: Systematic Review of Preclinical Studies	3
Discovery of New VEGFR-2 Inhibitors and Apoptosis inducer-based thieno[2,3- d ]pyrimidine	3
Key molecular scaffolds in the development of clinically viable α-amylase inhibitors	3
Tetrahydroquinoline: An Efficient Scaffold As mTOR Inhibitor for the Treatment of Lung Cancer	3
Recent Advances in Quinolone Hybrids With Potential Antibacterial Activity Against drug-resistant Bacteria	3
Our New Year's (re)solution: Welcome to the 15th Volume of Future Medicinal Chemistry	3
Gold: Not Just jewelry…	3
Versatile Tools of Synthetic Biology Applied to Drug Discovery and Production	3
Combining Virtual Screening and In Vitro Evaluation for the Discovery of Potential CYP11B2 Inhibitors	3
Designing molecular hybrids as novel breast cancer therapeutics	3
The other side of the coin: protein deubiquitination by Ubiquitin-Specific Protease 1 in cancer progression and therapy	3
Artificial intelligence-guided Approach for Efficient Virtual Screening of Hits Against Schistosoma Mansoni	3
Recent Advances in the Synthesis and Medicinal Perspective of Pyrazole-Based α-Amylase Inhibitors as Antidiabetic Agents	3
5,7,3′,4′-Tetramethoxyflavone Ameliorates Cholesterol Dysregulation by Mediating SIRT1/FOXO3a/ABCA1 Signaling in Osteoarthritis Chondrocytes	3
Transition metal complexes: a new generation of anticancer drugs	3
Curcumin-based Nanoformulations As an Emerging Therapeutic Strategy for Inflammatory Lung Diseases	3
Selective CDK9 Degradation Using a Proteolysis-Targeting Chimera (PROTAC) Strategy	3
Therapeutic potential of chalcone-1,2,3-triazole hybrids as anti-tumour agents: a systematic review and SAR studies	3
Human Sirtuin 2 inhibitors, Their Mechanisms and Binding Modes	3
Pyrazoline Scaffold: Hit Identification to Lead Synthesis and Biological Evaluation As Antidiabetic Agents	3
Novel Xylenyl-Spaced Bis-Thiazoles/Thiazines: Synthesis, Biological Profile as Herpes Simplex Virus Type 1 Inhibitors and in Silico Simulations	3
Inhibition of α-glucosidase Enzyme By ‘click'-inspired Pharmacophore Framework 1,3,4-thiadiazole–1,2,3-triazole Hybrids	3
The Key New Techniques in the Medicinal Chemist’s Toolkit to Prioritize Solubility During Drug Design	3
Development and Implementation of an enterprise-wide Predictive Model for Early absorption, distribution, Metabolism and Excretion Properties	3
Targeting STK33: From Inhibition to Degradation	3
Basic nitrogen (BaN): a ‘privileged element’ in medicinal chemistry	3
Copper(II) complexes of 2-hydroxy-1-naphthaldehyde Schiff bases: synthesis, in vitro activity and computational studies	3
EGFR molecular degraders: preclinical successes and the road ahead	3
Recent Advances in Anti-Coxsackievirus A16 Viral Drug Research	3
PROTACs in the treatment of viral diseases	3
Recent Advances in Oxazolidinones as Antituberculosis Agents	3
Diaminomaleonitrile Derivatives as new Potential Antichagasic Compounds: A Study of Structure–Activity Relationships	3
Camptothecin: a key building block in the design of anti-tumor agents	3
Pharmaceutical technological trends containing flavonoids: a patent review	3
Latest Advances in Specific Inhibition of Tumor-Associated Carbonic Anhydrases	3
Machine Learning Study: From the Toxicity Studies to Tetrahydrocannabinol Effects on Parkinson's Disease	3
Thio-substituted Derivatives of 4-amino-pyrazolo[3,4-d]pyrimidine-6-thiol As Antiproliferative Agents	3
Engineering ‘Enzymelink’ for Screening Lead Compounds to Inhibit mPGES-1 while Maintaining Prostacyclin Synthase Activity	3
Recent Advancements in the Discovery of Cereblon-Based Protease-Targeted Chimeras With Potential for Therapeutic Intervention	3
Synthesis and Antimicrobial Activity of Thiophene-Based Heterocycles Derived from Thiophene-2-Carbohydrazide	3
Long-acting Biodegradable Implants for Osteoporosis Management: Transforming the Landscape of Bisphosphonates Delivery	3
Design, synthesis and biological evaluation of non-glucosidal based 1,3,4-thiadiazoles as SGLT-2 inhibitors	2
Multitarget Therapeutic Approaches for Alzheimer's and Parkinson's Diseases: An Opportunity or an illusion?	2
Novel Trypanocidal Thiophen-Chalcone Cruzain Inhibitors: Structure- and Ligand-Based Studies	2
Benzimidazole-based small molecules as anticancer agents targeting telomeric G-quadruplex and inhibiting telomerase enzyme	2
Latest Advancements in the Study of the Relationship Between NSAIDs and Three Prostaglandin E2 Synthases	2