Beilstein Journal of Organic Chemistry

Article	Citations
Deciphering the mechanism of γ-cyclodextrin’s hydrophobic cavity hydration: an integrated experimental and theoretical study	57
Asymmetric synthesis of a stereopentade fragment toward latrunculins	50
Recent advances in electrochemical copper catalysis for modern organic synthesis	39
Facile approach to N,O,S-heteropentacycles via condensation of sterically crowded 3H-phenoxazin-3-one with ortho-substituted anilines	38
Anion-dependent ion-pairing assemblies of triazatriangulenium cation that interferes with stacking structures	30
A novel recyclable organocatalyst for the gram-scale enantioselective synthesis of (S)-baclofen	30
Entry to 2-aminoprolines via electrochemical decarboxylative amidation of N‑acetylamino malonic acid monoesters	29
Redox-active molecules as organocatalysts for selective oxidative transformations – an unperceived organocatalysis field	29
A new analog of dihydroxybenzoic acid from Saccharopolyspora sp. KR21-0001	28
Finding the most potent compounds using active learning on molecular pairs	27
A recent overview on the synthesis of 1,4,5-trisubstituted 1,2,3-triazoles	26
Correction: One-pot multicomponent green Hantzsch synthesis of 1,2-dihydropyridine derivatives with antiproliferative activity	24
AlBr3-Promoted stereoselective anti-hydroarylation of the acetylene bond in 3-arylpropynenitriles by electron-rich arenes: synthesis of 3,3-diarylpropenenitriles	22
Modular synthesis of 2-furyl carbinols from 3-benzyldimethylsilylfurfural platforms relying on oxygen-assisted C–Si bond functionalization	20
Computational model predicts protein binding sites of a luminescent ligand equipped with guanidiniocarbonyl-pyrrole groups	19
Enzymes in biosynthesis	19
Antiviral therapy in shrimp through plant virus VLP containing VP28 dsRNA against WSSV	18
Mechanochemical halogenation of unsymmetrically substituted azobenzenes	18
Efficacy of radical reactions of isocyanides with heteroatom radicals in organic synthesis	18
Biobased carbon dots as photoreductants – an investigation by using triarylsulfonium salts	18
N-Boc-α-diazo glutarimide as efficient reagent for assembling N-heterocycle-glutarimide diads via Rh(II)-catalyzed N–H insertion reaction	18
Cyclization of 1-aryl-4,4,4-trichlorobut-2-en-1-ones into 3-trichloromethylindan-1-ones in triflic acid	18
Electrochemical and spectroscopic properties of twisted dibenzo[g,p]chrysene derivatives	17
Synthesis of extended fluorinated tripeptides based on the tetrahydropyridazine scaffold	17
Preparation of an advanced intermediate for the synthesis of leustroducsins and phoslactomycins by heterocycloaddition	17

Domino reactions of chromones with activated carbonyl compounds	17
Efficient synthesis of fluorinated triphenylenes with enhanced arene–perfluoroarene interactions in columnar mesophases	17
Hydrogen-bond activation enables aziridination of unactivated olefins with simple iminoiodinanes	17
Synthesis of N-acetyl diazocine derivatives via cross-coupling reaction	17
Synthesis, α-mannosidase inhibition studies and molecular modeling of 1,4-imino-ᴅ-lyxitols and their C-5-altered N-arylalkyl derivatives	16
Recent advances in the syntheses of anthracene derivatives	16
Green and sustainable approaches for the Friedel–Crafts reaction between aldehydes and indoles	16
Sustainable tandem acylation/Diels–Alder reaction toward versatile tricyclic epoxyisoindole-7-carboxylic acids in renewable green solvents	16
Novel truxene-based dipyrromethanes (DPMs): synthesis, spectroscopic characterization and photophysical properties	16
Recent advances in the tandem annulation of 1,3-enynes to functionalized pyridine and pyrrole derivatives	16
Two-fold addition reaction of silylene to C60: structural and electronic properties of a bis-adduct	16
Reactivity of hypervalent iodine(III) reagents bearing a benzylamine with sulfenate salts	15
Multi-redox indenofluorene chromophores incorporating dithiafulvene donor and ene/enediyne acceptor units	15
N-Sulfinylpyrrolidine-containing ureas and thioureas as bifunctional organocatalysts	15
Organocatalytic asymmetric Michael/acyl transfer reaction between α-nitroketones and 4-arylidenepyrrolidine-2,3-diones	14
Copper-catalyzed N-arylation of amines with aryliodonium ylides in water	14
Photocatalytic sequential C–H functionalization expediting acetoxymalonylation of imidazo heterocycles	14
Synthesis of disulfides and 3-sulfenylchromones from sodium sulfinates catalyzed by TBAI	14
Polymer chemistry: fundamentals and applications	14
In-depth characterization of self-healing polymers based on π–π nteractions	13
Synthesis of novel alkynyl imidazopyridinyl selenides: copper-catalyzed tandem selenation of selenium with 2-arylimidazo[1,2-a]pyridines and terminal alkynes	13
1-Butyl-3-methylimidazolium tetrafluoroborate as suitable solvent for BF3: the case of alkyne hydration. Chemistry vs electrochemistry	13
Ready access to 7,8-dihydroindolo[2,3-d][1]benzazepine-6(5H)-one scaffold and analogues via early-stage Fischer ring-closure reaction	12
A study of the DIBAL-promoted selective debenzylation of α-cyclodextrin protected with two different benzyl groups	12
Diametric calix[6]arene-based phosphine gold(I) cavitands	12
Design, synthesis, and evaluation of chiral thiophosphorus acids as organocatalysts	12
Synthesis of protected precursors of chitin oligosaccharides by electrochemical polyglycosylation of thioglycosides	12
Development and mechanistic studies of calcium–BINOL phosphate-catalyzed hydrocyanation of hydrazones	11
Bromination of endo-7-norbornene derivatives revisited: failure of a computational NMR method in elucidating the configuration of an organic structure	11
Palladium-catalyzed three-component radical-polar crossover carboamination of 1,3-dienes or allenes with diazo esters and amines	11
Inclusion complexes of the steroid hormones 17β-estradiol and progesterone with β- and γ-cyclodextrin hosts: syntheses, X-ray structures, thermal analyses and API solubility enhancements	11
Photochemically assisted synthesis of phenacenes fluorinated at the terminal benzene rings and their electronic spectra	11
HFIP as a versatile solvent in resorcin[n]arene synthesis	11
Ring opening of photogenerated azetidinols as a strategy for the synthesis of aminodioxolanes	11
Methodology for awakening the potential secondary metabolic capacity in actinomycetes	11
Synthesis of 1,4-azaphosphinine nucleosides and evaluation as inhibitors of human cytidine deaminase and APOBEC3A	11
Photoredox catalysis in nickel-catalyzed C–H functionalization	11
Ugi bisamides based on pyrrolyl-β-chlorovinylaldehyde and their unusual transformations	11
Catalytic aza-Nazarov cyclization reactions to access α-methylene-γ-lactam heterocycles	11
Photoluminescence color-tuning with polymer-dispersed fluorescent films containing two fluorinated diphenylacetylene-type fluorophores	11
Mild and efficient synthesis and base-promoted rearrangement of novel isoxazolo[4,5-b]pyridines	11
Copper-promoted C5-selective bromination of 8-aminoquinoline amides with alkyl bromides	11
Electrophotochemical metal-catalyzed synthesis of alkylnitriles from simple aliphatic carboxylic acids	11
Synthesis of π-conjugated polycyclic compounds by late-stage extrusion of chalcogen fragments	10
Harnessing tethered nitreniums for diastereoselective amino-sulfonoxylation of alkenes	10
Advancements in hydrochlorination of alkenes	10
Three-component N-alkenylation of azoles with alkynes and iodine(III) electrophile: synthesis of multisubstituted N-vinylazoles	10
Characterization of a new fusicoccane-type diterpene synthase and an associated P450 enzyme	10
Isolation and characterization of new phenolic siderophores with antimicrobial properties from Pseudomonas sp. UIAU-6B	10
Copper-catalyzed monoselective C–H amination of ferrocenes with alkylamines	10

Access to cyclopropanes with geminal trifluoromethyl and difluoromethylphosphonate groups	10
Synthesis of the aggregation pheromone of Tribolium castaneum	10
Computational studies of Brønsted acid-catalyzed transannular cycloadditions of cycloalkenone hydrazones	10
Synthesis of α-(perfluoroalkylsulfonyl)propiophenones: a new set of reagents for the light-mediated perfluoroalkylation of aromatics	10
Chitosan-supported CuI-catalyzed cascade reaction of 2-halobenzoic acids and amidines for the synthesis of quinazolinones	10
Palladium-catalyzed enantioselective three-component synthesis of α-arylglycine derivatives from glyoxylic acid, sulfonamides and aryltrifluoroborates	10
Multi-faceted reactivity of N-fluorobenzenesulfonimide (NFSI) under mechanochemical conditions: fluorination, fluorodemethylation, sulfonylation, and amidation reactions	10
Quantifying the ability of the CF2H group as a hydrogen bond donor	10
N-Glycosides of indigo, indirubin, and isoindigo: blue, red, and yellow sugars and their cancerostatic activity	10
Dissecting Mechanochemistry III	10
Synthesis of novel [1,2,4]triazolo[1,5-b][1,2,4,5]tetrazines and investigation of their fungistatic activity	10
Synthesis and biological profile of 2,3-dihydro[1,3]thiazolo[4,5-b]pyridines, a novel class of acyl-ACP thioesterase inhibitors	9
One-pot nucleophilic substitution–double click reactions of biazides leading to functionalized bis(1,2,3-triazole) derivatives	9
Metal catalyst-free N-allylation/alkylation of imidazole and benzimidazole with Morita–Baylis–Hillman (MBH) alcohols and acetates	9
Applications of microscopy and small angle scattering techniques for the characterisation of supramolecular gels	9
Chemical and chemoenzymatic routes to bridged homoarabinofuranosylpyrimidines: Bicyclic AZT analogues	9
Electrogenerated base-promoted cyclopropanation using alkyl 2-chloroacetates	9
Rhodium-catalyzed homo-coupling reaction of aryl Grignard reagents and its application for the synthesis of an integrin inhibitor	9
Navigating and expanding the roadmap of natural product genome mining tools	9
Organocatalytic asymmetric nitroso aldol reaction of α-substituted malonamates	9
Total synthesis: an enabling science	9
C3-Alkylation of furfural derivatives by continuous flow homogeneous catalysis	9
Kinetically stabilized 1,3-diarylisobenzofurans and the possibility of preparing large, persistent isoacenofurans with unusually small HOMO–LUMO gaps	9
Synthesis of cyclic β-1,6-oligosaccharides from glucosamine monomers by electrochemical polyglycosylation	9
(Bio)isosteres of ortho- and meta-substituted benzenes	8
Regioselective quinazoline C2 modifications through the azide–tetrazole tautomeric equilibrium	8
Oxidative hydrolysis of aliphatic bromoalkenes: scope study and reactivity insights	8
A novel spirocyclic scaffold accessed via tandem Claisen rearrangement/intramolecular oxa-Michael addition	8
New azodyrecins identified by a genome mining-directed reactivity-based screening	8
Recent advances in the application of isoindigo derivatives in materials chemistry	8
Efficient synthesis of ethyl 2-(oxazolin-2-yl)alkanoates via ethoxycarbonylketene-induced electrophilic ring expansion of aziridines	8
The unique reactivity of 5,6-unsubstituted 1,4-dihydropyridine in the Huisgen 1,4-diploar cycloaddition and formal [2 + 2] cycloaddition	8
Synthetic strategies for the preparation of γ-phostams: 1,2-azaphospholidine 2-oxides and 1,2-azaphospholine 2-oxides	8
Chemical structure metagenomics of microbial natural products: surveying nonribosomal peptides and beyond	8
Orthogonal photoswitching of heterobivalent azobenzene glycoclusters: the effect of glycoligand orientation in bacterial adhesion	8
An efficient metal-free and catalyst-free C–S/C–O bond-formation strategy: synthesis of pyrazole-conjugated thioamides and amides	8
Four bioactive new steroids from the soft coral Lobophytum pauciflorum collected in South China Sea	8
Selective and scalable oxygenation of heteroatoms using the elements of nature: air, water, and light	8
Ligand effects, solvent cooperation, and large kinetic solvent deuterium isotope effects in gold(I)-catalyzed intramolecular alkene hydroamination	8
Cycloaddition reactions of heterocyclic azides with 2-cyanoacetamidines as a new route to C,N-diheteroarylcarbamidines	8
Studies on the syntheses of β-carboline alkaloids brevicarine and brevicolline	8
Stereoselective mechanochemical synthesis of thiomalonate Michael adducts via iminium catalysis by chiral primary amines	8
A novel bis-triazole scaffold accessed via two tandem [3 + 2] cycloaddition events including an uncatalyzed, room temperature azide–alkyne click reaction	7
A novel methodology for the efficient synthesis of 3-monohalooxindoles by acidolysis of 3-phosphate-substituted oxindoles with haloid acids	7
Mechanistic investigations of polyaza[7]helicene in photoredox and energy transfer catalysis	7
Effect of substitution position of aryl groups on the thermal back reactivity of aza-diarylethene photoswitches and prediction by density functional theory	7
Mechanochemical difluoromethylations of ketones	7
Efficient synthesis of polyfunctionalized carbazoles and pyrrolo[3,4-c]carbazoles via domino Diels–Alder reaction	7
Ortho-ester-substituted diaryliodonium salts enabled regioselective arylocyclization of naphthols toward 3,4-benzocoumarins	7
Chiral phosphoric acid-catalyzed transfer hydrogenation of 3,3-difluoro-3H-indoles	7
Manganese-catalyzed C–C and C–N bond formation with alcohols via borrowing hydrogen or hydrogen auto-transfer	7
Functions of enzyme domains in 2-methylisoborneol biosynthesis and enzymatic synthesis of non-natural analogs	7
Synthesis and reactivity of the di(9-anthryl)methyl radical	7
Three-component reactions of conjugated dienes, CH acids and formaldehyde under diffusion mixing conditions	7
Photoredox catalysis enabling decarboxylative radical cyclization of γ,γ-dimethylallyltryptophan (DMAT) derivatives: formal synthesis of 6,7-secoagroclavine	7
Acetaldehyde in the Enders triple cascade reaction via acetaldehyde dimethyl acetal	7
Intramolecular C–H arylation of pyridine derivatives with a palladium catalyst for the synthesis of multiply fused heteroaromatic compounds	7
Recent advances in controllable/divergent synthesis	7
Double-headed nucleosides: Synthesis and applications	7
Synthesis of benzo[f]quinazoline-1,3(2H,4H)-diones	7
1,2-Naphthoquinone-4-sulfonic acid salts in organic synthesis	7
4,6-Diaryl-5,5-difluoro-1,3-dioxanes as chiral dopants for liquid crystal compositions	7
Tandem diazotization/cyclization approach for the synthesis of a fused 1,2,3-triazinone-furazan/furoxan heterocyclic system	7
Progress and challenges in the synthesis of sequence controlled polysaccharides	7
New cembrane-type diterpenoids with anti-inflammatory activity from the South China Sea soft coral Sinularia sp.	7
Enhanced reactivity of Li+@C60 toward thermal [2 + 2] cycloaddition by encapsulated Li+ Lewis acid	7
Solid-phase total synthesis and structural confirmation of antimicrobial longicatenamide A	7
Efficient production of clerodane and ent-kaurane diterpenes through truncated artificial pathways in Escherichia coli	7
Long oligodeoxynucleotides: chemical synthesis, isolation via catching-by-polymerization, verification via sequencing, and gene expression demonstration	7
Tenacibactins K–M, cytotoxic siderophores from a coral-associated gliding bacterium of the genus Tenacibaculum	7
Facile access to 3-sulfonylquinolines via Knoevenagel condensation/aza-Wittig reaction cascade involving ortho-azidobenzaldehydes and β-ketosulfonamides and sulfones	7
Biphenylene-containing polycyclic conjugated compounds	7
Synthesis of sulfur karrikin bioisosteres as potential neuroprotectives	7
Beyond symmetric self-assembly and effective molarity: unlocking functional enzyme mimics with robust organic cages	6
Digyalipopeptide A, an antiparasitic cyclic peptide from the Ghanaian Bacillus sp. strain DE2B	6
Divergent role of PIDA and PIFA in the AlX3 (X = Cl, Br) halogenation of 2-naphthol: a mechanistic study	6
Anomeric 1,2,3-triazole-linked sialic acid derivatives show selective inhibition towards a bacterial neuraminidase over a trypanosome trans-sialidase	6
On drug discovery against infectious diseases and academic medicinal chemistry contributions	6
Discrimination of β-cyclodextrin/hazelnut (Corylus avellana L.) oil/flavonoid glycoside and flavonolignan ternary complexes by Fourier-transform infrared spectroscopy coupled with principal com	6
Mechanisms for radical reactions initiating from N-hydroxyphthalimide esters	6

Cage-like microstructures via sequential Ugi reactions in aqueous emulsions	6
On the application of 3d metals for C–H activation toward bioactive compounds: The key step for the synthesis of silver bullets	6
Rapid construction of tricyclic tetrahydrocyclopenta[4,5]pyrrolo[2,3-b]pyridine via isocyanide-based multicomponent reaction	6
Advances in the use of metal-free tetrapyrrolic macrocycles as catalysts	6
Synthesis of polycyclic aromatic quinones by continuous flow electrochemical oxidation: anodic methoxylation of polycyclic aromatic phenols (PAPs)	6
4-(1-Methylamino)ethylidene-1,5-disubstituted pyrrolidine-2,3-diones: synthesis, anti-inflammatory effect and in silico approaches	6
Transition-metal-catalyzed C–H bond activation as a sustainable strategy for the synthesis of fluorinated molecules: an overview	6
Discovery and biosynthesis of bacterial drimane-type sesquiterpenoids from Streptomyces clavuligerus	6
Identification and determination of the absolute configuration of amorph-4-en-10β-ol, a cadinol-type sesquiterpene from the scent glands of the African reed frog Hyperolius cinnamomeoventris	6
A myo-inositol dehydrogenase involved in aminocyclitol biosynthesis of hygromycin A	6
The ethoxycarbonyl group as both activating and protective group in N-acyl-Pictet–Spengler reactions using methoxystyrenes. A short approach to racemic 1-benzyltetrahydroisoquinoline alkaloids	6
Practical synthesis of isocoumarins via Rh(III)-catalyzed C–H activation/annulation cascade	6
Mechanochemical bottom-up synthesis of phosphorus-linked, heptazine-based carbon nitrides using sodium phosphide	6
Electroreductive coupling of 2-acylbenzoates with α,β-unsaturated carbonyl compounds: density functional theory study on product selectivity	6
Synthesis of substituted 8H-benzo[h]pyrano[2,3-f]quinazolin-8-ones via photochemical 6π-electrocyclization of pyrimidines containing an allomaltol fragment	6
Harnessing unprotected deactivated amines and arylglyoxals in the Ugi reaction for the synthesis of fused complex nitrogen heterocycles	6
Synthetic strategies toward 1,3-oxathiolane nucleoside analogues	6
Chemoselective N-acylation of indoles using thioesters as acyl source	6
Synthesis of tetrahydrofuro[3,2-c]pyridines via Pictet–Spengler reaction	6
Mechanochemical solid state synthesis of copper(I)/NHC complexes with K3PO4	6
Synthesis and antimycotic activity of new derivatives of imidazo[1,2-a]pyrimidines	6
Asymmetric tandem conjugate addition and reaction with carbocations on acylimidazole Michael acceptors	6
Modern flow chemistry – prospect and advantage	5
Synthesis of a novel aminobenzene-containing hemicucurbituril and its fluorescence spectral properties with ions	5
Synthesis of new representatives of A3B-type carboranylporphyrins based on meso-tetra(pentafluorophenyl)porphyrin transformations	5
Synthesis and antimicrobial activity of 1H-1,2,3-triazole and carboxylate analogues of metronidazole	5
Primary amine-catalyzed enantioselective 1,4-Michael addition reaction of pyrazolin-5-ones to α,β-unsaturated ketones	5
Direct C–H amination reactions of arenes with N-hydroxyphthalimides catalyzed by cuprous bromide	5
Cu–Bpin-mediated dimerization of 4,4-dichloro-2-butenoic acid derivatives enables the synthesis of densely functionalized cyclopropanes	5
Oxa-Michael-initiated cascade reactions of levoglucosenone	5
Organophosphorus chemistry: from model to application	5
Controlled oligomerization of [1.1.1]propellane through radical polarity matching: selective synthesis of SF5- and CF3SF4-containing [2]staffanes	5
Semisynthetic derivatives of massarilactone D with cytotoxic and nematicidal activities	5
Synthesis of spiroindolenines through a one-pot multistep process mediated by visible light	5
Synthesis of electrophile-tethered preQ1 analogs for covalent attachment to preQ1 RNA	5
Optimizing reaction conditions for the light-driven hydrogen evolution in a loop photoreactor	5
Bioinspired tetraamino-bisthiourea chiral macrocycles in catalyzing decarboxylative Mannich reactions	5
1,2-Difluoroethylene (HFO-1132): synthesis and chemistry	5
One-pot synthesis of 2-arylated and 2-alkylated benzoxazoles and benzimidazoles based on triphenylbismuth dichloride-promoted desulfurization of thioamides	5
Bifunctional thiourea-catalyzed asymmetric [3 + 2] annulation reactions of 2-isothiocyanato-1-indanones with barbiturate-based olefins	5
Correction: Amine–borane complex-initiated SF5Cl radical addition on alkenes and alkynes	5
Synthesis of fluorinated acid-functionalized, electron-rich nickel porphyrins	5
Cationic oligonucleotide derivatives and conjugates: A favorable approach for enhanced DNA and RNA targeting oligonucleotides	5
Copper-mediated oxidative C−H/N−H activations with alkynes by removable hydrazides	5
Flow synthesis of oxadiazoles coupled with sequential in-line extraction and chromatography	5
Cell-free protein synthesis with technical additives – expanding the parameter space of in vitro gene expression	5
Mining raw plant transcriptomic data for new cyclopeptide alkaloids	5
Phenanthridine–pyrene conjugates as fluorescent probes for DNA/RNA and an inactive mutant of dipeptidyl peptidase enzyme	5
Confirmation of the stereochemistry of spiroviolene	5
First series of N-alkylamino peptoid homooligomers: solution phase synthesis and conformational investigation	5
Selective construction of dispiro[indoline-3,2'-quinoline-3',3''-indoline] and dispiro[indoline-3,2'-pyrrole-3',3''-indoline] via three-component reaction	5
Revisiting the bromination of 3β-hydroxycholest-5-ene with CBr4/PPh3 and the subsequent azidolysis of the resulting bromide, disparity in stereochemical behavior	5
GlAIcomics: a deep neural network classifier for spectroscopy-augmented mass spectrometric glycans data	5
Red light excitation: illuminating photocatalysis in a new spectrum	5
Synthesis, structure, ionochromic and cytotoxic properties of new 2-(indolin-2-yl)-1,3-tropolones	5
Strategies for the synthesis of brevipolides	5
Five new sesquiterpenoids from agarwood of Aquilaria sinensis	5
Trichloroacetic acid fueled practical amine purifications	5
2,4-Bis(arylethynyl)-9-chloro-5,6,7,8-tetrahydroacridines: synthesis and photophysical properties	5
Introducing a new 7-ring fused diindenone-dithieno[3,2-b:2',3'-d]thiophene unit as a promising component for organic semiconductor materials	5
Heteroannulations of cyanoacetamide-based MCR scaffolds utilizing formamide	5
Charge carrier transport in perylene-based and pyrene-based columnar liquid crystals	5
Insight into oral amphiphilic cyclodextrin nanoparticles for colorectal cancer: comprehensive mathematical model of drug release kinetic studies and antitumoral efficacy in 3D spheroid colon tumors	5
Bismuth(III) triflate: an economical and environmentally friendly catalyst for the Nazarov reaction	5
Molecular diversity of the reactions of MBH carbonates of isatins and various nucleophiles	5