Beilstein Journal of Organic Chemistry

Article	Citations
Cyclization of 1-aryl-4,4,4-trichlorobut-2-en-1-ones into 3-trichloromethylindan-1-ones in triflic acid	43
Deciphering the mechanism of γ-cyclodextrin’s hydrophobic cavity hydration: an integrated experimental and theoretical study	32
Anion-dependent ion-pairing assemblies of triazatriangulenium cation that interferes with stacking structures	32
Facile approach to N,O,S-heteropentacycles via condensation of sterically crowded 3H-phenoxazin-3-one with ortho-substituted anilines	32
Redox-active molecules as organocatalysts for selective oxidative transformations – an unperceived organocatalysis field	30
Entry to 2-aminoprolines via electrochemical decarboxylative amidation of N‑acetylamino malonic acid monoesters	29
A novel recyclable organocatalyst for the gram-scale enantioselective synthesis of (S)-baclofen	28
A new analog of dihydroxybenzoic acid from Saccharopolyspora sp. KR21-0001	28
Photoredox-catalyzed arylation of isonitriles by diaryliodonium salts towards benzamides	28
Finding the most potent compounds using active learning on molecular pairs	21
AlBr3-Promoted stereoselective anti-hydroarylation of the acetylene bond in 3-arylpropynenitriles by electron-rich arenes: synthesis of 3,3-diarylpropenenitriles	20
Correction: One-pot multicomponent green Hantzsch synthesis of 1,2-dihydropyridine derivatives with antiproliferative activity	20
Computational model predicts protein binding sites of a luminescent ligand equipped with guanidiniocarbonyl-pyrrole groups	19
Enzymes in biosynthesis	19
Modular synthesis of 2-furyl carbinols from 3-benzyldimethylsilylfurfural platforms relying on oxygen-assisted C–Si bond functionalization	19
Biobased carbon dots as photoreductants – an investigation by using triarylsulfonium salts	19
Synthesis of N-acetyl diazocine derivatives via cross-coupling reaction	18
N-Boc-α-diazo glutarimide as efficient reagent for assembling N-heterocycle-glutarimide diads via Rh(II)-catalyzed N–H insertion reaction	18
Efficacy of radical reactions of isocyanides with heteroatom radicals in organic synthesis	18
Hydrogen-bond activation enables aziridination of unactivated olefins with simple iminoiodinanes	18
Mechanochemical halogenation of unsymmetrically substituted azobenzenes	18
Asymmetric synthesis of a stereopentade fragment toward latrunculins	18
Electrochemical and spectroscopic properties of twisted dibenzo[g,p]chrysene derivatives	18
Recent advances in electrochemical copper catalysis for modern organic synthesis	18
Green and sustainable approaches for the Friedel–Crafts reaction between aldehydes and indoles	17

Synthesis, α-mannosidase inhibition studies and molecular modeling of 1,4-imino-ᴅ-lyxitols and their C-5-altered N-arylalkyl derivatives	17
Efficient synthesis of fluorinated triphenylenes with enhanced arene–perfluoroarene interactions in columnar mesophases	17
Domino reactions of chromones with activated carbonyl compounds	16
Two-fold addition reaction of silylene to C60: structural and electronic properties of a bis-adduct	16
Preparation of an advanced intermediate for the synthesis of leustroducsins and phoslactomycins by heterocycloaddition	16
Synthesis of extended fluorinated tripeptides based on the tetrahydropyridazine scaffold	16
Sustainable tandem acylation/Diels–Alder reaction toward versatile tricyclic epoxyisoindole-7-carboxylic acids in renewable green solvents	16
Recent advances in the syntheses of anthracene derivatives	16
Gold extraction at the molecular level using α- and β-cyclodextrins	15
Novel truxene-based dipyrromethanes (DPMs): synthesis, spectroscopic characterization and photophysical properties	15
Ambident reactivity of enolizable 5-mercapto-1H-tetrazoles in trapping reactions with in situ-generated thiocarbonyl S-methanides derived from sterically crowded cycloaliphatic thioketon	15
Recent advances in the tandem annulation of 1,3-enynes to functionalized pyridine and pyrrole derivatives	15
Multi-redox indenofluorene chromophores incorporating dithiafulvene donor and ene/enediyne acceptor units	14
Reactivity of hypervalent iodine(III) reagents bearing a benzylamine with sulfenate salts	14
Catalytic aza-Nazarov cyclization reactions to access α-methylene-γ-lactam heterocycles	14
N-Sulfinylpyrrolidine-containing ureas and thioureas as bifunctional organocatalysts	13
Polymer chemistry: fundamentals and applications	13
Synthesis of disulfides and 3-sulfenylchromones from sodium sulfinates catalyzed by TBAI	13
1-Butyl-3-methylimidazolium tetrafluoroborate as suitable solvent for BF3: the case of alkyne hydration. Chemistry vs electrochemistry	12
Ready access to 7,8-dihydroindolo[2,3-d][1]benzazepine-6(5H)-one scaffold and analogues via early-stage Fischer ring-closure reaction	12
Diametric calix[6]arene-based phosphine gold(I) cavitands	12
Photocatalytic sequential C–H functionalization expediting acetoxymalonylation of imidazo heterocycles	12
A study of the DIBAL-promoted selective debenzylation of α-cyclodextrin protected with two different benzyl groups	12
Design, synthesis, and evaluation of chiral thiophosphorus acids as organocatalysts	12
Synthesis of novel alkynyl imidazopyridinyl selenides: copper-catalyzed tandem selenation of selenium with 2-arylimidazo[1,2-a]pyridines and terminal alkynes	12
Mild and efficient synthesis and base-promoted rearrangement of novel isoxazolo[4,5-b]pyridines	12
Bromination of endo-7-norbornene derivatives revisited: failure of a computational NMR method in elucidating the configuration of an organic structure	12
Inclusion complexes of the steroid hormones 17β-estradiol and progesterone with β- and γ-cyclodextrin hosts: syntheses, X-ray structures, thermal analyses and API solubility enhancements	11
Palladium-catalyzed three-component radical-polar crossover carboamination of 1,3-dienes or allenes with diazo esters and amines	11
Ring opening of photogenerated azetidinols as a strategy for the synthesis of aminodioxolanes	11
Photochemically assisted synthesis of phenacenes fluorinated at the terminal benzene rings and their electronic spectra	11
In-depth characterization of self-healing polymers based on π–π nteractions	11
Methodology for awakening the potential secondary metabolic capacity in actinomycetes	11
Copper-catalyzed N-arylation of amines with aryliodonium ylides in water	11
Copper-promoted C5-selective bromination of 8-aminoquinoline amides with alkyl bromides	11
Electrophotochemical metal-catalyzed synthesis of alkylnitriles from simple aliphatic carboxylic acids	11
Photoluminescence color-tuning with polymer-dispersed fluorescent films containing two fluorinated diphenylacetylene-type fluorophores	11
Synthesis of protected precursors of chitin oligosaccharides by electrochemical polyglycosylation of thioglycosides	11
Development and mechanistic studies of calcium–BINOL phosphate-catalyzed hydrocyanation of hydrazones	11
HFIP as a versatile solvent in resorcin[n]arene synthesis	11
Isolation and characterization of new phenolic siderophores with antimicrobial properties from Pseudomonas sp. UIAU-6B	10
N-Glycosides of indigo, indirubin, and isoindigo: blue, red, and yellow sugars and their cancerostatic activity	10
Photoredox catalysis in nickel-catalyzed C–H functionalization	10
Multi-faceted reactivity of N-fluorobenzenesulfonimide (NFSI) under mechanochemical conditions: fluorination, fluorodemethylation, sulfonylation, and amidation reactions	10
Synthesis of π-conjugated polycyclic compounds by late-stage extrusion of chalcogen fragments	10
Synthesis of cyclic β-1,6-oligosaccharides from glucosamine monomers by electrochemical polyglycosylation	10
N-Salicyl-amino acid derivatives with antiparasitic activity from Pseudomonas sp. UIAU-6B	10
Synthesis and biological profile of 2,3-dihydro[1,3]thiazolo[4,5-b]pyridines, a novel class of acyl-ACP thioesterase inhibitors	10
Ugi bisamides based on pyrrolyl-β-chlorovinylaldehyde and their unusual transformations	10
Palladium-catalyzed enantioselective three-component synthesis of α-arylglycine derivatives from glyoxylic acid, sulfonamides and aryltrifluoroborates	10

Orthogonal photoswitching of heterobivalent azobenzene glycoclusters: the effect of glycoligand orientation in bacterial adhesion	10
Efficient synthesis of ethyl 2-(oxazolin-2-yl)alkanoates via ethoxycarbonylketene-induced electrophilic ring expansion of aziridines	10
Access to cyclopropanes with geminal trifluoromethyl and difluoromethylphosphonate groups	10
Three-component N-alkenylation of azoles with alkynes and iodine(III) electrophile: synthesis of multisubstituted N-vinylazoles	10
Synthesis of 1,4-azaphosphinine nucleosides and evaluation as inhibitors of human cytidine deaminase and APOBEC3A	10
Copper-catalyzed monoselective C–H amination of ferrocenes with alkylamines	10
Harnessing tethered nitreniums for diastereoselective amino-sulfonoxylation of alkenes	10
Reactions of acryl thioamides with iminoiodinanes as a one-step synthesis of N-sulfonyl-2,3-dihydro-1,2-thiazoles	10
New azodyrecins identified by a genome mining-directed reactivity-based screening	9
Chitosan-supported CuI-catalyzed cascade reaction of 2-halobenzoic acids and amidines for the synthesis of quinazolinones	9
Characterization of a new fusicoccane-type diterpene synthase and an associated P450 enzyme	9
Electrogenerated base-promoted cyclopropanation using alkyl 2-chloroacetates	9
An efficient metal-free and catalyst-free C–S/C–O bond-formation strategy: synthesis of pyrazole-conjugated thioamides and amides	9
Quantifying the ability of the CF2H group as a hydrogen bond donor	9
Computational studies of Brønsted acid-catalyzed transannular cycloadditions of cycloalkenone hydrazones	9
Synthesis of α-(perfluoroalkylsulfonyl)propiophenones: a new set of reagents for the light-mediated perfluoroalkylation of aromatics	9
Total synthesis: an enabling science	9
Studies on the syntheses of β-carboline alkaloids brevicarine and brevicolline	9
Synthesis of the aggregation pheromone of Tribolium castaneum	9
Dissecting Mechanochemistry III	9
Synthesis of novel [1,2,4]triazolo[1,5-b][1,2,4,5]tetrazines and investigation of their fungistatic activity	9
Stereoselective mechanochemical synthesis of thiomalonate Michael adducts via iminium catalysis by chiral primary amines	8
Organocatalytic asymmetric nitroso aldol reaction of α-substituted malonamates	8
Metal catalyst-free N-allylation/alkylation of imidazole and benzimidazole with Morita–Baylis–Hillman (MBH) alcohols and acetates	8
Chemical and chemoenzymatic routes to bridged homoarabinofuranosylpyrimidines: Bicyclic AZT analogues	8
Advancements in hydrochlorination of alkenes	8
Regioselective quinazoline C2 modifications through the azide–tetrazole tautomeric equilibrium	8
A novel spirocyclic scaffold accessed via tandem Claisen rearrangement/intramolecular oxa-Michael addition	8
Kinetically stabilized 1,3-diarylisobenzofurans and the possibility of preparing large, persistent isoacenofurans with unusually small HOMO–LUMO gaps	8
Applications of microscopy and small angle scattering techniques for the characterisation of supramolecular gels	8
C3-Alkylation of furfural derivatives by continuous flow homogeneous catalysis	8
Facile synthesis of hydantoin/1,2,4-oxadiazoline spiro-compounds via 1,3-dipolar cycloaddition of nitrile oxides to 5-iminohydantoins	8
(Bio)isosteres of ortho- and meta-substituted benzenes	8
Oxidative hydrolysis of aliphatic bromoalkenes: scope study and reactivity insights	8
Chemical structure metagenomics of microbial natural products: surveying nonribosomal peptides and beyond	8
Navigating and expanding the roadmap of natural product genome mining tools	8
Correction: Diastereoselective synthesis of highly substituted cyclohexanones and tetrahydrochromene-4-ones via conjugate addition of curcumins to arylidenemalonates	8
One-pot nucleophilic substitution–double click reactions of biazides leading to functionalized bis(1,2,3-triazole) derivatives	8
Rhodium-catalyzed homo-coupling reaction of aryl Grignard reagents and its application for the synthesis of an integrin inhibitor	8
Four bioactive new steroids from the soft coral Lobophytum pauciflorum collected in South China Sea	8
Synthetic strategies for the preparation of γ-phostams: 1,2-azaphospholidine 2-oxides and 1,2-azaphospholine 2-oxides	8
Recent advances in amidyl radical-mediated photocatalytic direct intermolecular hydrogen atom transfer	7
1,2-Naphthoquinone-4-sulfonic acid salts in organic synthesis	7
Ortho-ester-substituted diaryliodonium salts enabled regioselective arylocyclization of naphthols toward 3,4-benzocoumarins	7
Tandem diazotization/cyclization approach for the synthesis of a fused 1,2,3-triazinone-furazan/furoxan heterocyclic system	7
Mechanochemical difluoromethylations of ketones	7
Effect of substitution position of aryl groups on the thermal back reactivity of aza-diarylethene photoswitches and prediction by density functional theory	7
Photoredox catalysis enabling decarboxylative radical cyclization of γ,γ-dimethylallyltryptophan (DMAT) derivatives: formal synthesis of 6,7-secoagroclavine	7
Ligand effects, solvent cooperation, and large kinetic solvent deuterium isotope effects in gold(I)-catalyzed intramolecular alkene hydroamination	7
Cycloaddition reactions of heterocyclic azides with 2-cyanoacetamidines as a new route to C,N-diheteroarylcarbamidines	7
Chiral phosphoric acid-catalyzed transfer hydrogenation of 3,3-difluoro-3H-indoles	7
Synthesis of benzo[f]quinazoline-1,3(2H,4H)-diones	7
Synthesis of sulfur karrikin bioisosteres as potential neuroprotectives	7
Enhanced reactivity of Li+@C60 toward thermal [2 + 2] cycloaddition by encapsulated Li+ Lewis acid	7
Solid-phase total synthesis and structural confirmation of antimicrobial longicatenamide A	7
Mechanistic investigations of polyaza[7]helicene in photoredox and energy transfer catalysis	7
A novel methodology for the efficient synthesis of 3-monohalooxindoles by acidolysis of 3-phosphate-substituted oxindoles with haloid acids	7
Facile access to 3-sulfonylquinolines via Knoevenagel condensation/aza-Wittig reaction cascade involving ortho-azidobenzaldehydes and β-ketosulfonamides and sulfones	7
4,6-Diaryl-5,5-difluoro-1,3-dioxanes as chiral dopants for liquid crystal compositions	7
Functions of enzyme domains in 2-methylisoborneol biosynthesis and enzymatic synthesis of non-natural analogs	7
Three-component reactions of conjugated dienes, CH acids and formaldehyde under diffusion mixing conditions	7
Selective and scalable oxygenation of heteroatoms using the elements of nature: air, water, and light	7
The unique reactivity of 5,6-unsubstituted 1,4-dihydropyridine in the Huisgen 1,4-diploar cycloaddition and formal [2 + 2] cycloaddition	7
Acetaldehyde in the Enders triple cascade reaction via acetaldehyde dimethyl acetal	7
Synthesis and reactivity of the di(9-anthryl)methyl radical	6
Asymmetric tandem conjugate addition and reaction with carbocations on acylimidazole Michael acceptors	6
4-(1-Methylamino)ethylidene-1,5-disubstituted pyrrolidine-2,3-diones: synthesis, anti-inflammatory effect and in silico approaches	6
Advances in the use of metal-free tetrapyrrolic macrocycles as catalysts	6
Long oligodeoxynucleotides: chemical synthesis, isolation via catching-by-polymerization, verification via sequencing, and gene expression demonstration	6
High-pressure activation for the solvent- and catalyst-free syntheses of heterocycles, pharmaceuticals and esters	6
Digyalipopeptide A, an antiparasitic cyclic peptide from the Ghanaian Bacillus sp. strain DE2B	6
Mechanochemical bottom-up synthesis of phosphorus-linked, heptazine-based carbon nitrides using sodium phosphide	6
Synthesis of polycyclic aromatic quinones by continuous flow electrochemical oxidation: anodic methoxylation of polycyclic aromatic phenols (PAPs)	6
Discrimination of β-cyclodextrin/hazelnut (Corylus avellana L.) oil/flavonoid glycoside and flavonolignan ternary complexes by Fourier-transform infrared spectroscopy coupled with principal com	6
Manganese-catalyzed C–C and C–N bond formation with alcohols via borrowing hydrogen or hydrogen auto-transfer	6
A novel bis-triazole scaffold accessed via two tandem [3 + 2] cycloaddition events including an uncatalyzed, room temperature azide–alkyne click reaction	6
Recent advances in controllable/divergent synthesis	6
Practical synthesis of isocoumarins via Rh(III)-catalyzed C–H activation/annulation cascade	6
Anomeric 1,2,3-triazole-linked sialic acid derivatives show selective inhibition towards a bacterial neuraminidase over a trypanosome trans-sialidase	6
Identification and determination of the absolute configuration of amorph-4-en-10β-ol, a cadinol-type sesquiterpene from the scent glands of the African reed frog Hyperolius cinnamomeoventris	6

Transition-metal-catalyzed C–H bond activation as a sustainable strategy for the synthesis of fluorinated molecules: an overview	6
Efficient synthesis of polyfunctionalized carbazoles and pyrrolo[3,4-c]carbazoles via domino Diels–Alder reaction	6
Rapid construction of tricyclic tetrahydrocyclopenta[4,5]pyrrolo[2,3-b]pyridine via isocyanide-based multicomponent reaction	6
Efficient production of clerodane and ent-kaurane diterpenes through truncated artificial pathways in Escherichia coli	6
Divergent role of PIDA and PIFA in the AlX3 (X = Cl, Br) halogenation of 2-naphthol: a mechanistic study	6
Electroreductive coupling of 2-acylbenzoates with α,β-unsaturated carbonyl compounds: density functional theory study on product selectivity	6
Advances in nitrogen-containing helicenes: synthesis, chiroptical properties, and optoelectronic applications	6
Progress and challenges in the synthesis of sequence controlled polysaccharides	6
Intramolecular C–H arylation of pyridine derivatives with a palladium catalyst for the synthesis of multiply fused heteroaromatic compounds	6
Biphenylene-containing polycyclic conjugated compounds	6
Discovery and biosynthesis of bacterial drimane-type sesquiterpenoids from Streptomyces clavuligerus	6
Chemoselective N-acylation of indoles using thioesters as acyl source	6
Beyond symmetric self-assembly and effective molarity: unlocking functional enzyme mimics with robust organic cages	6
Synthesis of β-ketophosphonates through aerobic copper(II)-mediated phosphorylation of enol acetates	6
On drug discovery against infectious diseases and academic medicinal chemistry contributions	6
Harnessing unprotected deactivated amines and arylglyoxals in the Ugi reaction for the synthesis of fused complex nitrogen heterocycles	6
Synthesis and antimycotic activity of new derivatives of imidazo[1,2-a]pyrimidines	6
Synthesis of substituted 8H-benzo[h]pyrano[2,3-f]quinazolin-8-ones via photochemical 6π-electrocyclization of pyrimidines containing an allomaltol fragment	6
New cembrane-type diterpenoids with anti-inflammatory activity from the South China Sea soft coral Sinularia sp.	6
Tenacibactins K–M, cytotoxic siderophores from a coral-associated gliding bacterium of the genus Tenacibaculum	6
Selective construction of dispiro[indoline-3,2'-quinoline-3',3''-indoline] and dispiro[indoline-3,2'-pyrrole-3',3''-indoline] via three-component reaction	5
Synthesis of electrophile-tethered preQ1 analogs for covalent attachment to preQ1 RNA	5
GlAIcomics: a deep neural network classifier for spectroscopy-augmented mass spectrometric glycans data	5
Optimizing reaction conditions for the light-driven hydrogen evolution in a loop photoreactor	5
Synthesis of spiroindolenines through a one-pot multistep process mediated by visible light	5
A myo-inositol dehydrogenase involved in aminocyclitol biosynthesis of hygromycin A	5
Bioinspired tetraamino-bisthiourea chiral macrocycles in catalyzing decarboxylative Mannich reactions	5
1,2-Difluoroethylene (HFO-1132): synthesis and chemistry	5
Mechanochemical solid state synthesis of copper(I)/NHC complexes with K3PO4	5
Red light excitation: illuminating photocatalysis in a new spectrum	5
Controlled oligomerization of [1.1.1]propellane through radical polarity matching: selective synthesis of SF5- and CF3SF4-containing [2]staffanes	5
First series of N-alkylamino peptoid homooligomers: solution phase synthesis and conformational investigation	5
Introducing a new 7-ring fused diindenone-dithieno[3,2-b:2',3'-d]thiophene unit as a promising component for organic semiconductor materials	5
Synthesis of fluorinated acid-functionalized, electron-rich nickel porphyrins	5
Phenanthridine–pyrene conjugates as fluorescent probes for DNA/RNA and an inactive mutant of dipeptidyl peptidase enzyme	5
Organophosphorus chemistry: from model to application	5
Synthesis of a novel aminobenzene-containing hemicucurbituril and its fluorescence spectral properties with ions	5
Mining raw plant transcriptomic data for new cyclopeptide alkaloids	5
Mechanisms for radical reactions initiating from N-hydroxyphthalimide esters	5
Cell-free protein synthesis with technical additives – expanding the parameter space of in vitro gene expression	5
Revisiting the bromination of 3β-hydroxycholest-5-ene with CBr4/PPh3 and the subsequent azidolysis of the resulting bromide, disparity in stereochemical behavior	5
The ethoxycarbonyl group as both activating and protective group in N-acyl-Pictet–Spengler reactions using methoxystyrenes. A short approach to racemic 1-benzyltetrahydroisoquinoline alkaloids	5
Heteroannulations of cyanoacetamide-based MCR scaffolds utilizing formamide	5
Insight into oral amphiphilic cyclodextrin nanoparticles for colorectal cancer: comprehensive mathematical model of drug release kinetic studies and antitumoral efficacy in 3D spheroid colon tumors	5
Five new sesquiterpenoids from agarwood of Aquilaria sinensis	5
Trichloroacetic acid fueled practical amine purifications	5
Elucidating the glycan-binding specificity and structure of Cucumis melo agglutinin, a new R-type lectin	5
Molecular diversity of the reactions of MBH carbonates of isatins and various nucleophiles	5
Cu–Bpin-mediated dimerization of 4,4-dichloro-2-butenoic acid derivatives enables the synthesis of densely functionalized cyclopropanes	5
One-pot synthesis of 2-arylated and 2-alkylated benzoxazoles and benzimidazoles based on triphenylbismuth dichloride-promoted desulfurization of thioamides	5
Bismuth(III) triflate: an economical and environmentally friendly catalyst for the Nazarov reaction	5
Synthesis of new representatives of A3B-type carboranylporphyrins based on meso-tetra(pentafluorophenyl)porphyrin transformations	5
Cage-like microstructures via sequential Ugi reactions in aqueous emulsions	5
Confirmation of the stereochemistry of spiroviolene	5
Modern flow chemistry – prospect and advantage	5
Synthetic strategies toward 1,3-oxathiolane nucleoside analogues	5
Bifunctional thiourea-catalyzed asymmetric [3 + 2] annulation reactions of 2-isothiocyanato-1-indanones with barbiturate-based olefins	5
Synthesis of tetrahydrofuro[3,2-c]pyridines via Pictet–Spengler reaction	5
Semisynthetic derivatives of massarilactone D with cytotoxic and nematicidal activities	5
Direct C–H amination reactions of arenes with N-hydroxyphthalimides catalyzed by cuprous bromide	5
Oxa-Michael-initiated cascade reactions of levoglucosenone	5
Azide–alkyne cycloaddition (click) reaction in biomass-derived solvent CyreneTM under one-pot conditions	5
Charge carrier transport in perylene-based and pyrene-based columnar liquid crystals	5