Beilstein Journal of Organic Chemistry

Article	Citations
Synthetic reactions driven by electron-donor–acceptor (EDA) complexes	92
Activated carbon as catalyst support: precursors, preparation, modification and characterization	90
Photocatalysis with organic dyes: facile access to reactive intermediates for synthesis	87
Recent developments in enantioselective photocatalysis	80
Recent applications of porphyrins as photocatalysts in organic synthesis: batch and continuous flow approaches	71
When metal-catalyzed C–H functionalization meets visible-light photocatalysis	68
Heterogeneous photocatalysis in flow chemical reactors	57
19F NMR as a tool in chemical biology	49
Dawn of a new era in industrial photochemistry: the scale-up of micro- and mesostructured photoreactors	46
Development of N-F fluorinating agents and their fluorinations: Historical perspective	41
Oxime radicals: generation, properties and application in organic synthesis	40
A comprehensive review of flow chemistry techniques tailored to the flavours and fragrances industries	38
Chemical approaches to discover the full potential of peptide nucleic acids in biomedical applications	37
An overview on disulfide-catalyzed and -cocatalyzed photoreactions	36
Photosensitized direct C–H fluorination and trifluoromethylation in organic synthesis	33
A recent overview on the synthesis of 1,4,5-trisubstituted 1,2,3-triazoles	32
Fabclavine diversity in Xenorhabdus bacteria	31
Anthelmintic drug discovery: target identification, screening methods and the role of open science	31
Microwave-assisted multicomponent reactions in heterocyclic chemistry and mechanistic aspects	30
Valorisation of plastic waste via metal-catalysed depolymerisation	29
Mechanochemical green synthesis of hyper-crosslinked cyclodextrin polymers	29
The preparation and properties of 1,1-difluorocyclopropane derivatives	29
A cyclopeptide and three oligomycin-class polyketides produced by an underexplored actinomycete of the genus Pseudosporangium	24
Photoredox catalysis in nickel-catalyzed C–H functionalization	23
Prins cyclization-mediated stereoselective synthesis of tetrahydropyrans and dihydropyrans: an inspection of twenty years	23

Synthetic approaches to bowl-shaped π-conjugated sumanene and its congeners	23
Cryogels: recent applications in 3D-bioprinting, injectable cryogels, drug delivery, and wound healing	21
Recent advances in the tandem annulation of 1,3-enynes to functionalized pyridine and pyrrole derivatives	21
Recent advances in organocatalytic asymmetric aza-Michael reactions of amines and amides	21
Amine–borane complex-initiated SF5Cl radical addition on alkenes and alkynes	21
Copper-based fluorinated reagents for the synthesis of CF2R-containing molecules (R ≠ F)	21
One-pot synthesis of isosorbide from cellulose or lignocellulosic biomass: a challenge?	20
N-tert-Butanesulfinyl imines in the asymmetric synthesis of nitrogen-containing heterocycles	20
Insight into functionalized-macrocycles-guided supramolecular photocatalysis	20
Natural dolomitic limestone-catalyzed synthesis of benzimidazoles, dihydropyrimidinones, and highly substituted pyridines under ultrasound irradiation	20
Visible-light-mediated copper photocatalysis for organic syntheses	20
Beyond ribose and phosphate: Selected nucleic acid modifications for structure–function investigations and therapeutic applications	20
How and why plants and human N-glycans are different: Insight from molecular dynamics into the “glycoblocks” architecture of complex carbohydrates	19
Photocatalyzed syntheses of phenanthrenes and their aza-analogues. A review	19
pH- and concentration-dependent supramolecular self-assembly of a naturally occurring octapeptide	19
Recent synthesis of thietanes	19
Using multiple self-sorting for switching functions in discrete multicomponent systems	19
Photocatalytic trifluoromethoxylation of arenes and heteroarenes in continuous-flow	19
Progress and challenges in the synthesis of sequence controlled polysaccharides	18
On the application of 3d metals for C–H activation toward bioactive compounds: The key step for the synthesis of silver bullets	18
Recent advances in the asymmetric phosphoric acid-catalyzed synthesis of axially chiral compounds	18
Secondary metabolites of Bacillus subtilis impact the assembly of soil-derived semisynthetic bacterial communities	17
Synthesis of N-perfluoroalkyl-3,4-disubstituted pyrroles by rhodium-catalyzed transannulation of N-fluoroalkyl-1,2,3-triazoles with terminal alkynes	17
Biochemistry of fluoroprolines: the prospect of making fluorine a bioelement	16
Incorporation of a metal-mediated base pair into an ATP aptamer – using silver(I) ions to modulate aptamer function	16
Regiodivergent synthesis of functionalized pyrimidines and imidazoles through phenacyl azides in deep eutectic solvents	16
Ferrocenyl-substituted tetrahydrothiophenes via formal [3 + 2]-cycloaddition reactions of ferrocenyl thioketones with donor–acceptor cyclopropanes	16
Enhanced target cell specificity and uptake of lipid nanoparticles using RNA aptamers and peptides	16
Leveraging glycomics data in glycoprotein 3D structure validation with Privateer	16
Halides as versatile anions in asymmetric anion-binding organocatalysis	15
The McKenna reaction – avoiding side reactions in phosphonate deprotection	15
Computational tools for drawing, building and displaying carbohydrates: a visual guide	14
All-carbon [3 + 2] cycloaddition in natural product synthesis	14
Effective microwave-assisted approach to 1,2,3-triazolobenzodiazepinones via tandem Ugi reaction/catalyst-free intramolecular azide–alkyne cycloaddition	14
Fluorinated phenylalanines: synthesis and pharmaceutical applications	14
Towards new NIR dyes for free radical photopolymerization processes	14
Constrained thermoresponsive polymers – new insights into fundamentals and applications	14
CF3-substituted carbocations: underexploited intermediates with great potential in modern synthetic chemistry	13
Sustainable manganese catalysis for late-stage C–H functionalization of bioactive structural motifs	13
Suzuki–Miyaura cross coupling is not an informative reaction to demonstrate the performance of new solvents	13
Lipophilicity trends upon fluorination of isopropyl, cyclopropyl and 3-oxetanyl groups	13
Earth-abundant 3d transition metals on the rise in catalysis	13
A consensus-based and readable extension of Linear Code for Reaction Rules (LiCoRR)	13
Pauson–Khand reaction of fluorinated compounds	13
Synthesis of 1,4-benzothiazinones from acylpyruvic acids or furan-2,3-diones and o-aminothiophenol	12
Molecular basis for protein–protein interactions	12
BINOL as a chiral element in mechanically interlocked molecules	12
Synthesis of 3(2)-phosphonylated thiazolo[3,2-a]oxopyrimidines	12
Design, synthesis and photophysical properties of novel star-shaped truxene-based heterocycles utilizing ring-closing metathesis, Clauson–Kaas, Van Leusen and Ullmann-type reactions as key tools	12
Polarity effects in 4-fluoro- and 4-(trifluoromethyl)prolines	12

Design, synthesis and application of carbazole macrocycles in anion sensors	12
Heteroleptic metallosupramolecular aggregates/complexation for supramolecular catalysis	12
Synthetic accesses to biguanide compounds	12
Metal-free synthesis of phosphinoylchroman-4-ones via a radical phosphinoylation–cyclization cascade mediated by K2S2O8	12
Selective and reversible 1,3-dipolar cycloaddition of 6-aryl-1,5-diazabicyclo[3.1.0]hexanes with 1,3-diphenylprop-2-en-1-ones under microwave irradiation	11
Synthesis of trifluoromethyl ketones by nucleophilic trifluoromethylation of esters under a fluoroform/KHMDS/triglyme system	11
Nomimicins B–D, new tetronate-class polyketides from a marine-derived actinomycete of the genus Actinomadura	11
Synthesis and investigation of quadruplex-DNA-binding, 9-O-substituted berberine derivatives	11
Antiviral therapy in shrimp through plant virus VLP containing VP28 dsRNA against WSSV	11
Photoredox catalysis harvesting multiple photon or electrochemical energies	11
Tools for generating and analyzing glycan microarray data	11
Unsaturated fatty acids and a prenylated tryptophan derivative from a rare actinomycete of the genus Couchioplanes	11
Synthesis of (Z)-3-[amino(phenyl)methylidene]-1,3-dihydro-2H-indol-2-ones using an Eschenmoser coupling reaction	10
A new glance at the chemosphere of macroalgal–bacterial interactions: In situ profiling of metabolites in symbiosis by mass spectrometry	10
Azo-dimethylaminopyridine-functionalized Ni(II)-porphyrin as a photoswitchable nucleophilic catalyst	10
Activation of pentafluoropropane isomers at a nanoscopic aluminum chlorofluoride: hydrodefluorination versus dehydrofluorination	10
Selected peptide-based fluorescent probes for biological applications	10
Copper-catalysed alkylation of heterocyclic acceptors with organometallic reagents	10
Efficient production of clerodane and ent-kaurane diterpenes through truncated artificial pathways in Escherichia coli	10
Nocarimidazoles C and D, antimicrobial alkanoylimidazoles from a coral-derived actinomycete Kocuria sp.: application of 1JC,H coupling constants for the unequivocal	10
Synthesis and anticancer activity of bis(2-arylimidazo[1,2-a]pyridin-3-yl) selenides and diselenides: the copper-catalyzed tandem C–H selenation of 2-arylimidazo[1,2-a]pyridine with sele	10
Stereoselective Biginelli-like reaction catalyzed by a chiral phosphoric acid bearing two hydroxy groups	10
A complementary approach to conjugated N-acyliminium formation through photoredox-catalyzed intermolecular radical addition to allenamides and allencarbamates	10
Tetraphenylethylene-embedded pillar[5]arene-based orthogonal self-assembly for efficient photocatalysis in water	10
Deoxygenative C2-heteroarylation of quinoline N-oxides: facile access to α-triazolylquinolines	10
Deoxyfluorination of acyl fluorides to trifluoromethyl compounds by FLUOLEAD®/Olah’s reagent under solvent-free conditions	10
DNA with zwitterionic and negatively charged phosphate modifications: Formation of DNA triplexes, duplexes and cell uptake studies	10
Antibacterial scalarane from Doriprismatica stellata nudibranchs (Gastropoda, Nudibranchia), egg ribbons, and their dietary sponge Spongia cf. agaricina (Demospongiae, Dictyocerat	10
Natural products in the predatory defence of the filamentous fungal pathogen Aspergillus fumigatus	10
Et3N/DMSO-supported one-pot synthesis of highly fluorescent β-carboline-linked benzothiophenones via sulfur insertion and estimation of the photophysical properties	10
Palladium-catalyzed solid-state borylation of aryl halides using mechanochemistry	10
Controlled decomposition of SF6 by electrochemical reduction	10
A sustainable strategy for the straightforward preparation of 2H-azirines and highly functionalized NH-aziridines from vinyl azides using a single solvent flow-batch approach	10
One-pot multicomponent green Hantzsch synthesis of 1,2-dihydropyridine derivatives with antiproliferative activity	10
Menadione: a platform and a target to valuable compounds synthesis	10
Palladium nanoparticles supported on chitin-based nanomaterials as heterogeneous catalysts for the Heck coupling reaction	10
The charge-assisted hydrogen-bonded organic framework (CAHOF) self-assembled from the conjugated acid of tetrakis(4-aminophenyl)methane and 2,6-naphthalenedisulfonate as a new class of recyclable Brøn	10
Synthetic strategies for the preparation of γ-phostams: 1,2-azaphospholidine 2-oxides and 1,2-azaphospholine 2-oxides	10
Cytochrome P450 monooxygenase-mediated tailoring of triterpenoids and steroids in plants	9
Ionic multiresonant thermally activated delayed fluorescence emitters for light emitting electrochemical cells	9
Radical cation Diels–Alder reactions of arylidene cycloalkanes	9
Iron-catalyzed domino coupling reactions of π-systems	9
Diels–Alder reaction of β-fluoro-β-nitrostyrenes with cyclic dienes	9
Recent advances in the syntheses of anthracene derivatives	9
Synthesis of novel fluorinated building blocks via halofluorination and related reactions	9
Synthesis of new dihydroberberine and tetrahydroberberine analogues and evaluation of their antiproliferative activity on NCI-H1975 cells	9
Disposable cartridge concept for the on-demand synthesis of turbo Grignards, Knochel–Hauser amides, and magnesium alkoxides	9
Synthesis and antimicrobial activity of 1H-1,2,3-triazole and carboxylate analogues of metronidazole	9
Conformational preferences of fluorine-containing agrochemicals and their implications for lipophilicity prediction	9
Continuous flow synthesis of azobenzenes via Baeyer–Mills reaction	9
Asymmetric organocatalyzed synthesis of coumarin derivatives	9
Metal-free nucleophilic trifluoromethylselenolation via an iodide-mediated umpolung reactivity of trifluoromethylselenotoluenesulfonate	9
Synthesis of esters of diaminotruxillic bis-amino acids by Pd-mediated photocycloaddition of analogs of the Kaede protein chromophore	9
One-pot synthesis of oxazolidinones and five-membered cyclic carbonates from epoxides and chlorosulfonyl isocyanate: theoretical evidence for an asynchronous concerted pathway	9
Recent advances in the application of isoindigo derivatives in materials chemistry	9
Substituted nitrogen-bridged diazocines	9
Synthesis of functionalized imidazo[4,5-e]thiazolo[3,2-b]triazines by condensation of imidazo[4,5-e]triazinethiones with DMAD or DEAD and rearrangement to imidazo[4,5-e]thi	9
Cerium-photocatalyzed aerobic oxidation of benzylic alcohols to aldehydes and ketones	9
Synthesis of pyrrolidinedione-fused hexahydropyrrolo[2,1-a]isoquinolines via three-component [3 + 2] cycloaddition followed by one-pot N-allylation and intramolecular Heck reactions	9
Inline purification in continuous flow synthesis – opportunities and challenges	8
A study of the photochemical behavior of terarylenes containing allomaltol and pyrazole fragments	8
Fluorine effect in nucleophilic fluorination at C4 of 1,6-anhydro-2,3-dideoxy-2,3-difluoro-β-D-hexopyranose	8
Transition-metal-catalyzed domino reactions of strained bicyclic alkenes	8
[2 + 1] Cycloaddition reactions of fullerene C60 based on diazo compounds	8
Regioselective N-alkylation of the 1H-indazole scaffold; ring substituent and N-alkylating reagent effects on regioisomeric distribution	8
In-depth characterization of self-healing polymers based on π–π nteractions	8
New efficient synthesis of polysubstituted 3,4-dihydroquinazolines and 4H-3,1-benzothiazines through a Passerini/Staudinger/aza-Wittig/addition/nucleophilic substitution sequence	8
Host–guest interaction of cucurbit[8]uril with oroxin A and its effect on the properties of oroxin A	8
Synthesis and characterization of S,N-heterotetracenes	8
B–N/B–H Transborylation: borane-catalysed nitrile hydroboration	8
3-Acetoxy-fatty acid isoprenyl esters from androconia of the ithomiine butterfly Ithomia salapia	8
The synthesis of chiral β-naphthyl-β-sulfanyl ketones via enantioselective sulfa-Michael reaction in the presence of a bifunctional cinchona/sulfonamide organocatalyst	8
Electron-rich triarylphosphines as nucleophilic catalysts for oxa-Michael reactions	8
A new and efficient methodology for olefin epoxidation catalyzed by supported cobalt nanoparticles	8
Heterogeneous photocatalytic cyanomethylarylation of alkenes with acetonitrile: synthesis of diverse nitrogenous heterocyclic compounds	8
Chemical syntheses and salient features of azulene-containing homo- and copolymers	8
Regioselective cobalt(II)-catalyzed [2 + 3] cycloaddition reaction of fluoroalkylated alkynes with 2-formylphenylboronic acids: easy access to 2-fluoroalkylated indenols	8
A Se···O bonding catalysis approach to the synthesis of calix[4]pyrroles	8
Germacrene B – a central intermediate in sesquiterpene biosynthesis	8
Synthesis, crystal structures and properties of carbazole-based [6]helicenes fused with an azine ring	8

Inductive heating and flow chemistry – a perfect synergy of emerging enabling technologies	7
UV resonance Raman spectroscopy of the supramolecular ligand guanidiniocarbonyl indole (GCI) with 244 nm laser excitation	7
Inclusion complexes of the steroid hormones 17β-estradiol and progesterone with β- and γ-cyclodextrin hosts: syntheses, X-ray structures, thermal analyses and API solubility enhancements	7
DDQ in mechanochemical C–N coupling reactions	7
Particle size effect in the mechanically assisted synthesis of β-cyclodextrin mesitylene sulfonate	7
Synthesis of novel multifunctional carbazole-based molecules and their thermal, electrochemical and optical properties	7
The PIFA-initiated oxidative cyclization of 2-(3-butenyl)quinazolin-4(3H)-ones – an efficient approach to 1-(hydroxymethyl)-2,3-dihydropyrrolo[1,2-a]quinazolin-5(1H)-ones	7
GlypNirO: An automated workflow for quantitative N- and O-linked glycoproteomic data analysis	7
Pd-catalyzed asymmetric Suzuki–Miyaura coupling reactions for the synthesis of chiral biaryl compounds with a large steric substituent at the 2-position	7
Recent developments and trends in the iron- and cobalt-catalyzed Sonogashira reactions	7
Glycosylated coumarins, flavonoids, lignans and phenylpropanoids from Wikstroemia nutans and their biological activities	7
Cholyl 1,3,4-oxadiazole hybrid compounds: design, synthesis and antimicrobial assessment	7
Naphthalonitriles featuring efficient emission in solution and in the solid state	7
Fluorohydration of alkynes via I(I)/I(III) catalysis	7
Annulation of a 1,3-dithiole ring to a sterically hindered o-quinone core. Novel ditopic redox-active ligands	7
Targeting active site residues and structural anchoring positions in terpene synthases	7
Accelerating fragment-based library generation by coupling high-performance photoreactors with benchtop analysis	7
Manganese/bipyridine-catalyzed non-directed C(sp3)–H bromination using NBS and TMSN3	7
A novel and robust heterogeneous Cu catalyst using modified lignosulfonate as support for the synthesis of nitrogen-containing heterocycles	7
Navigating and expanding the roadmap of natural product genome mining tools	7
Vicinal difluorination as a C=C surrogate: an analog of piperine with enhanced solubility, photostability, and acetylcholinesterase inhibitory activity	7
Benzothiazolium salts as reagents for the deoxygenative perfluoroalkylthiolation of alcohols	7
Synthesis of dibenzosuberenone-based novel polycyclic π-conjugated dihydropyridazines, pyridazines and pyrroles	7
Syntheses of spliceostatins and thailanstatins: a review	7
Microwave-assisted efficient one-pot synthesis of N2-(tetrazol-5-yl)-6-aryl/heteroaryl-5,6-dihydro-1,3,5-triazine-2,4-diamines	7
One-pot synthesis of 1,3,5-triazine-2,4-dithione derivatives via three-component reactions	7
A systems-based framework to computationally describe putative transcription factors and signaling pathways regulating glycan biosynthesis	7
Recent advances in palladium-catalysed asymmetric 1,4–additions of arylboronic acids to conjugated enones and chromones	7
Automated high-content imaging for cellular uptake, from the Schmuck cation to the latest cyclic oligochalcogenides	7
Semiautomated glycoproteomics data analysis workflow for maximized glycopeptide identification and reliable quantification	7
Thermodynamic and electrochemical study of tailor-made crown ethers for redox-switchable (pseudo)rotaxanes	7
Clickable azide-functionalized bromoarylaldehydes – synthesis and photophysical characterization	7
Enantioenriched α-substituted glutamates/pyroglutamates via enantioselective cyclopropenimine-catalyzed Michael addition of amino ester imines	7
Unexpected rearrangements and a novel synthesis of 1,1-dichloro-1-alkenones from 1,1,1-trifluoroalkanones with aluminium trichloride	6
Mechanochemical halogenation of unsymmetrically substituted azobenzenes	6
Synergy between supported ionic liquid-like phases and immobilized palladium N-heterocyclic carbene–phosphine complexes for the Negishi reaction under flow conditions	6
1,2,3-Triazoles as leaving groups in SNAr–Arbuzov reactions: synthesis of C6-phosphonated purine derivatives	6
Reactions of 3-aryl-1-(trifluoromethyl)prop-2-yn-1-iminium salts with 1,3-dienes and styrenes	6
Efficient synthesis of ethyl 2-(oxazolin-2-yl)alkanoates via ethoxycarbonylketene-induced electrophilic ring expansion of aziridines	6
One-step route to tricyclic fused 1,2,3,4-tetrahydroisoquinoline systems via the Castagnoli–Cushman protocol	6
Regioselective synthesis of heterocyclic N-sulfonyl amidines from heteroaromatic thioamides and sulfonyl azides	6
Clustering and curation of electropherograms: an efficient method for analyzing large cohorts of capillary electrophoresis glycomic profiles for bioprocessing operations	6
Chemoselective N-acylation of indoles using thioesters as acyl source	6
Electrocatalytic C(sp3)–H/C(sp)–H cross-coupling in continuous flow through TEMPO/copper relay catalysis	6
Regioselective synthesis of methyl 5-(N-Boc-cycloaminyl)-1,2-oxazole-4-carboxylates as new amino acid-like building blocks	6
Double-headed nucleosides: Synthesis and applications	6
Water-soluble host–guest complexes between fullerenes and a sugar-functionalized tribenzotriquinacene assembling to microspheres	6
A novel methodology for the efficient synthesis of 3-monohalooxindoles by acidolysis of 3-phosphate-substituted oxindoles with haloid acids	6
β-Lactamase inhibition profile of new amidine-substituted diazabicyclooctanes	6
Correction: Amine–borane complex-initiated SF5Cl radical addition on alkenes and alkynes	6
Cationic oligonucleotide derivatives and conjugates: A favorable approach for enhanced DNA and RNA targeting oligonucleotides	6
Multi-faceted reactivity of N-fluorobenzenesulfonimide (NFSI) under mechanochemical conditions: fluorination, fluorodemethylation, sulfonylation, and amidation reactions	6
The B & B approach: Ball-milling conjugation of dextran with phenylboronic acid (PBA)-functionalized BODIPY	6
A straightforward conversion of 1,4-quinones into polycyclic pyrazoles via [3 + 2]-cycloaddition with fluorinated nitrile imines	6
Efficient synthesis of polyfunctionalized carbazoles and pyrrolo[3,4-c]carbazoles via domino Diels–Alder reaction	6
Tenacibactins K–M, cytotoxic siderophores from a coral-associated gliding bacterium of the genus Tenacibaculum	6
Synthesis of imidazo[1,5-a]pyridines via cyclocondensation of 2-(aminomethyl)pyridines with electrophilically activated nitroalkanes	6
Synthesis and properties of quinazoline-based versatile exciplex-forming compounds	6
Metal-free glycosylation with glycosyl fluorides in liquid SO2	6
Bipyrrole boomerangs via Pd-mediated tandem cyclization–oxygenation. Controlling reaction selectivity and electronic properties	6
Recent progress in the synthesis of homotropane alkaloids adaline, euphococcinine and N-methyleuphococcinine	6
Synthesis of O6-alkylated preQ1 derivatives	6
Synthesis of new fluorescent molecules having an aggregation-induced emission property derived from 4-fluoroisoxazoles	6
Post-functionalization of drug-loaded nanoparticles prepared by polymerization-induced self-assembly (PISA) with mitochondria targeting ligands	6
Synthesis of phenanthridines via a novel photochemically-mediated cyclization and application to the synthesis of triphaeridine	6
Designed whole-cell-catalysis-assisted synthesis of 9,11-secosterols	6